A Study to Evaluate the Effect of GDC-4198 Alone and in Combination With Giredestrant Versus Abemaciclib and Giredestrant in Participants With Locally Advanced or Metastatic Estrogen Receptor-Positive (ER+), Human Epidermal Growth Factor Receptor-Negative (HER2-) Breast Cancer

NCT ID: NCT07100106

Last Updated: 2026-01-16

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

RECRUITING

Clinical Phase

PHASE1/PHASE2

Total Enrollment

285 participants

Study Classification

INTERVENTIONAL

Study Start Date

2025-10-07

Study Completion Date

2030-07-31

Brief Summary

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The purpose of this study is to assess the safety of GDC-4198 alone and in combination with giredestrant and also the efficacy of GDC-4198 + giredestrant versus abemaciclib + giredestrant in participants with locally advanced or metastatic ER+, HER2- breast cancer. The study consists of 2 phases: Phase Ib and Phase II. Phase Ib will evaluate the safety and pharmacokinetics (PK) of GDC-4198 alone and in combination with giredestrant. Phase II stage will compare the activity and safety of GDC-4198 and giredestrant with abemaciclib and giredestrant.

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Detailed Description

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Conditions

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Breast Cancer

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

SEQUENTIAL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Phase Ib: Dose-Finding Stage

Participants will receive GDC-4198 as monotherapy and in combination with giredestrant, 30 milligrams (mg), orally, daily, as per a pre-defined dosing regimen during each cycle until unacceptable toxicity or disease progression and/or loss of clinical benefit. (1 cycle=28 days).

Group Type EXPERIMENTAL

GDC-4198

Intervention Type DRUG

GDC-4198 will be administered orally.

Giredestrant

Intervention Type DRUG

Giredestrant will be administered orally.

Phase II: Arm A

Participants will receive GDC-4198, higher dose, in combination with giredestrant, 30 mg, orally, daily, as per a pre-defined dosing regimen during each cycle until unacceptable toxicity or disease progression and/or loss of clinical benefit. (1 cycle=28 days).

Group Type EXPERIMENTAL

GDC-4198

Intervention Type DRUG

GDC-4198 will be administered orally.

Giredestrant

Intervention Type DRUG

Giredestrant will be administered orally.

Phase II: Arm B

Participants will receive GDC-4198, lower dose, in combination with giredestrant, 30 mg, orally, daily, as per a pre-defined dosing regimen during each cycle until unacceptable toxicity or disease progression and/or loss of clinical benefit. (1 cycle=28 days).

Group Type EXPERIMENTAL

GDC-4198

Intervention Type DRUG

GDC-4198 will be administered orally.

Giredestrant

Intervention Type DRUG

Giredestrant will be administered orally.

Phase II: Arm C

Participants will receive abemaciclib, 150 mg twice daily, in combination with giredestrant, 30 mg, orally, daily, as per a pre-defined dosing regimen during each cycle until unacceptable toxicity or disease progression and/or loss of clinical benefit. (1 cycle=28 days).

Group Type EXPERIMENTAL

Giredestrant

Intervention Type DRUG

Giredestrant will be administered orally.

Abemaciclib

Intervention Type DRUG

Abemaciclib will be administered orally.

Interventions

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GDC-4198

GDC-4198 will be administered orally.

Intervention Type DRUG

Giredestrant

Giredestrant will be administered orally.

Intervention Type DRUG

Abemaciclib

Abemaciclib will be administered orally.

Intervention Type DRUG

Other Intervention Names

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RGT-419B RO7840734 GDC-9545 RO7197597

Eligibility Criteria

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Inclusion Criteria

* Histologically and/or cytologically confirmed adenocarcinoma of the breast that is locally advanced or metastatic.
* Previously documented ER+ and HER2- tumor according to American Society of Clinical Oncology (ASCO)/ College of American Pathologists (CAP) or European Society of Medical Oncology (ESMO) guidelines or any national guidelines with criteria conforming to ASCO/CAP or ESMO guidelines.
* Disease progression during or after treatment with an approved cyclin-dependent kinase 4/6 (CDK4/6) inhibitor and endocrine therapy (ET) in the locally advanced or metastatic setting.
* Measurable or non-measurable evaluable, disease per Response Evaluation Criteria in Solid Tumors version 1.1 (RECIST v1.1)
* Eastern Cooperative Oncology Group (ECOG) Performance Status of 0 or 1
* Life expectancy ≥ 6 months

Exclusion Criteria

* Advanced, symptomatic, visceral spread that is at risk of life-threatening complications in the short term appropriate for treatment with cytotoxic chemotherapy at time of entry into the study, as per national or local treatment guidelines.
* Have received more than one-line of therapy for locally advanced or metastatic disease.
* Have received prior chemotherapy for metastatic breast cancer
* Treatment with anti-cancer therapies, including investigational therapies, within 28 days or 5 drug elimination half -lives, whichever is shorter, prior to initiation of study drug. Treatment with an approved oral endocrine therapy (ET) within 7 days prior to initiation of study drug; treatment with fulvestrant or an approved CDK4/6 inhibitor within 21 days prior to initiation of study drug.
* Poor peripheral venous access
* Malabsorption condition or other gastrointestinal (GI) conditions/surgeries that the investigator assesses may significantly interfere with enteral absorption
* History of malignancy within 3 years prior to screening, except for cancer under investigation in this study and malignancies with a negligible risk of metastasis or death.
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Roche (China) Holding Ltd.

UNKNOWN

Sponsor Role collaborator

Genentech, Inc.

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Clinical Trials

Role: STUDY_DIRECTOR

Hoffmann-La Roche

Locations

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City of Hope

Duarte, California, United States

Site Status RECRUITING

City of Hope - Orange County Lennar Foundation Cancer Center

Irvine, California, United States

Site Status RECRUITING

Moffitt Cancer Center

Tampa, Florida, United States

Site Status RECRUITING

Winship Cancer Institute of Emory University

Atlanta, Georgia, United States

Site Status RECRUITING

City of Hope® Cancer Center Chicago

Zion, Illinois, United States

Site Status RECRUITING

Barbara Ann Karmanos Cancer Institute

Detroit, Maine, United States

Site Status RECRUITING

Rutgers Cancer Institute of New Jersey

New Brunswick, New Jersey, United States

Site Status RECRUITING

New York Cancer & Blood Specialists

East Patchogue, New York, United States

Site Status RECRUITING

St Vincent's Hospital Sydney

Darlinghurst, New South Wales, Australia

Site Status RECRUITING

Cancer Research SA

Adelaide, South Australia, Australia

Site Status RECRUITING

Princess Margaret Hospital

Toronto, Ontario, Canada

Site Status RECRUITING

Institut Jean Godinot

Reims, Champagne-Ardenne, France

Site Status RECRUITING

Hospital Beata Maria Ana

Madrid, , Spain

Site Status RECRUITING

Hospital Universitario 12 de Octubre

Madrid, , Spain

Site Status RECRUITING

Countries

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United States Australia Canada France Spain

Central Contacts

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Reference Study ID Number: GO46021 https://forpatients.roche.com/

Role: CONTACT

888-662-6728 (U.S. Only)

Other Identifiers

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2025-521128-31-00

Identifier Type: CTIS

Identifier Source: secondary_id

GO46021

Identifier Type: -

Identifier Source: org_study_id

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