A Clinical Study of Patritumab Deruxtecan to Treat Breast Cancer (MK-1022-016)

NCT ID: NCT07060807

Last Updated: 2025-12-24

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

RECRUITING

Clinical Phase

PHASE3

Total Enrollment

1000 participants

Study Classification

INTERVENTIONAL

Study Start Date

2025-07-21

Study Completion Date

2033-07-14

Brief Summary

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Researchers are looking for other ways to treat breast cancer (BC) that is hormone receptor-positive and human epidermal growth factor receptor 2-negative (HR+/HER2-) and either unresectable locally advanced or metastatic.

* HR positive (HR+) means the cancer cells have proteins that attach to estrogen or progesterone (hormones) which help the cancer to grow and spread
* HER2 negative (HER2-) means the cancer cells have a low amount of a protein called HER2
* Unresectable locally advanced means the cancer cannot be completely removed by surgery and has spread into nearby tissue or muscles
* Metastatic means the cancer has spread to other parts of the body

Treatment for this type of breast cancer usually includes endocrine therapy (ET) and sometimes a second treatment. The main goal of this study is to learn if people who receive patritumab deruxtecan (also known as HER3-DXd and MK-1022) live longer overall or without the cancer growing/spreading, compared to people who receive chemotherapy or a different drug called trastuzumab deruxtecan.

Detailed Description

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Conditions

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Breast Neoplasms

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Patritumab Deruxtecan

Participants receive patritumab deruxtecan via intravenous (IV) infusion every 3 weeks (Q3W) for approximately 13 months.

Group Type EXPERIMENTAL

Patritumab deruxtecan

Intervention Type BIOLOGICAL

Administered via intravenous (IV) infusion

Treatment of Physician's Choice

Participants receive treatment of physician's choice (TPC) for up to 13 months. The TPC may be any of the following options: Paclitaxel (80 mg/m\^2) on Days 1, 8, 15, and 22 of each 4-week cycle; Paclitaxel (90 mg/m\^2) on Days 1, 8, and 15 of each 4-week cycle; Nab-paclitaxel (100 mg/m\^2) on Days 1, 8, and 15 of each 4-week cycle; Capecitabine (1000 mg/m\^2) bid on Days 1 to 14 of each 3-week cycle; Liposomal doxorubicin (50 mg/m\^2) on Day 1 of each 4-week cycle; or trastuzumab deruxtecan (T-DXd) (5.4 mg/kg) Q3W.

Group Type ACTIVE_COMPARATOR

Paclitaxel

Intervention Type DRUG

Administered via IV infusion

Nab-paclitaxel

Intervention Type DRUG

Administered via IV infusion

Capecitabine

Intervention Type DRUG

Administered via oral tablets

Liposomal doxorubicin

Intervention Type DRUG

Administered via IV infusion

Trastuzumab deruxtecan

Intervention Type BIOLOGICAL

Administered via IV infusion

Interventions

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Patritumab deruxtecan

Administered via intravenous (IV) infusion

Intervention Type BIOLOGICAL

Paclitaxel

Administered via IV infusion

Intervention Type DRUG

Nab-paclitaxel

Administered via IV infusion

Intervention Type DRUG

Capecitabine

Administered via oral tablets

Intervention Type DRUG

Liposomal doxorubicin

Administered via IV infusion

Intervention Type DRUG

Trastuzumab deruxtecan

Administered via IV infusion

Intervention Type BIOLOGICAL

Other Intervention Names

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MK-1022 HER3-DXd U3-1402 TAXOL® ONXAL® Abraxane® XELODA® Doxil® T-DXd Enhertu®

Eligibility Criteria

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Inclusion Criteria

* Has a diagnosis of hormone receptor positive (HR+)/human epidermal growth factor receptor 2 (HER2)- invasive breast carcinoma that is either locally advanced disease not amenable to resection with curative intent (herein called unresectable) or metastatic disease not treatable with curative intent
* Has centrally-confirmed HR+ and HER2- results and human epidermal growth factor receptor 3 (HER3) evaluable results from a biopsy obtained from a distant metastatic site or a locally advanced lesion on or after the most recent line of therapy (with certain exceptions)
* Must have had progression or recurrence on prior cyclin-dependent kinase (CDK)4/6 inhibitor + endocrine therapy (ET) with one of the following:

* Radiographic disease progression, as assessed by the investigator, on CDK4/6 inhibitor + ET as 1L for treatment of unresectable locally advanced or metastatic HR+/HER2- breast cancer. CDK4/6 inhibitor + ET must be the only line of therapy received in the advanced setting, or
* Disease recurrence, either radiographic and/or confirmed histologically via biopsy as assessed by the investigator, while on adjuvant ET in combination with a CDK4/6 inhibitor OR within 24 months from the date of last dose of adjuvant CDK4/6 inhibitor
* Has measurable disease per RECIST 1.1 as assessed by the local site investigator/radiology
* Human immunodeficiency virus (HIV)-infected participants must have well controlled HIV on antiretroviral therapy
* Has an Eastern Cooperative Oncology Group performance status of 0 or 1 assessed within 7 days before randomization

Exclusion Criteria

* Has breast cancer amenable to treatment with curative intent
* Is eligible to receive additional endocrine-based treatment in the advanced setting as determined by the investigator
* Has a known germline breast cancer gene (BRCA) mutation (deleterious or suspected deleterious) where poly (ADP-ribose) polymerase (PARP) inhibitor(s) is a potential treatment option
* Has current visceral crisis or is at risk for impending visceral crisis that has or may cause imminent organ compromise and/or other life-threatening complications
* Has any of the following: a pulse oximeter reading \<92% at rest, or requires intermittent supplemental oxygen, or requires chronic supplemental oxygen
* Has uncontrolled, significant cardiovascular disease or cerebrovascular disease
* Has ≥Grade 2 peripheral neuropathy.
* Has clinically significant corneal disease
* Has received prior chemotherapy for unresectable locally advanced or metastatic breast cancer
* Has received prior treatment with an anti-HER3 antibody and/or antibody-drug conjugate that consists of a topoisomerase I inhibitor (eg, T-DXd) or any other topoisomerase I inhibitor therapy
* Has received prior systemic anticancer therapy within 4 weeks (or 5 half-lives, whichever is shorter) before randomization; participants previously treated with ET plus a CDK4/6 inhibitor may participate as long as at least 2 weeks have elapsed since the last dose of therapy was administered
* Has received prior radiotherapy for non-central nervous system disease, or required corticosteroids for radiation-related toxicities, within 14 days of the first dose of study intervention
* Has a diagnosis of immunodeficiency or is receiving chronic systemic steroid therapy
* Has known additional malignancy that is progressing or has required active treatment within the past 3 years
* Has history of (noninfectious) pneumonitis/interstitial lung disease (ILD) that required steroids, has current pneumonitis/interstitial lung disease, or has suspected ILD/pneumonitis that cannot be ruled out by imaging at Screening
* Has severe hypersensitivity (≥Grade 3) to HER3-DXd and/or any of its excipients
* Has severe hypersensitivity (≥Grade 3) to all the available TPC and/or any of their excipients
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Daiichi Sankyo

INDUSTRY

Sponsor Role collaborator

Merck Sharp & Dohme LLC

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Medical Director

Role: STUDY_DIRECTOR

Merck Sharp & Dohme LLC

Locations

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Los Angeles Hematology Oncology Medical Group ( Site 0026)

Los Angeles, California, United States

Site Status RECRUITING

Hoag Memorial Hospital Presbyterian ( Site 0025)

Newport Beach, California, United States

Site Status RECRUITING

St. Marys Hospital and Regional Medical Center-SCL Health Cancer Centers of Colorado ( Site 0021)

Grand Junction, Colorado, United States

Site Status RECRUITING

Comprehensive Hematology Oncology ( Site 0060)

St. Petersburg, Florida, United States

Site Status RECRUITING

Baptist Health Lexington ( Site 0050)

Lexington, Kentucky, United States

Site Status RECRUITING

Presbyterian Kaseman Hospital ( Site 0072)

Albuquerque, New Mexico, United States

Site Status RECRUITING

University of New Mexico Comprehensive Cancer Center ( Site 0047)

Albuquerque, New Mexico, United States

Site Status RECRUITING

Presbyterian Rust Jorgensen Cancer ( Site 0073)

Rio Rancho, New Mexico, United States

Site Status RECRUITING

Clinical Research Alliance ( Site 0009)

Westbury, New York, United States

Site Status RECRUITING

TriHealth Cancer Institute-Good Samaritan Hospital ( Site 0020)

Cincinnati, Ohio, United States

Site Status RECRUITING

Cancer Care Associates Of York ( Site 0063)

York, Pennsylvania, United States

Site Status RECRUITING

JPS Health Network ( Site 0067)

Fort Worth, Texas, United States

Site Status RECRUITING

Oncology Consultants P.A. ( Site 0061)

Houston, Texas, United States

Site Status RECRUITING

Mays Cancer Center ( Site 0049)

San Antonio, Texas, United States

Site Status RECRUITING

Shenandoah Oncology ( Site 8004)

Winchester, Virginia, United States

Site Status RECRUITING

Northwest Medical Specialties, PLLC ( Site 0062)

Tacoma, Washington, United States

Site Status RECRUITING

Circuit Clinical/SSM Health Dean Medical Group ( Site 0039)

Madison, Wisconsin, United States

Site Status RECRUITING

Instituto de Investigaciones Clínicas Mar del Plata ( Site 0205)

Mar del Plata, Buenos Aires, Argentina

Site Status RECRUITING

Fundación Respirar ( Site 0201)

Buenos Aires, Buenos Aires F.D., Argentina

Site Status RECRUITING

Centro Privado de RMI Rio Cuarto ( Site 0207)

Río Cuarto, Córdoba Province, Argentina

Site Status RECRUITING

Instituto de Oncología de Rosario ( Site 0208)

Rosario, Santa Fe Province, Argentina

Site Status RECRUITING

Hospital Italiano de Córdoba ( Site 0206)

Córdoba, , Argentina

Site Status RECRUITING

The Moncton Hospital ( Site 0101)

Moncton, New Brunswick, Canada

Site Status RECRUITING

The First Affiliated Hospital of Chongqing Medical University ( Site 3101)

Chongqing, Chongqing Municipality, China

Site Status RECRUITING

Chongqing Three Gorges Central Hospital's ( Site 3128)

Wanzhou, Chongqing Municipality, China

Site Status RECRUITING

Jiangmen Center Hospital ( Site 3132)

Jiangmen, Guangdong, China

Site Status RECRUITING

Guangxi Medical University Affiliated Tumor Hospital ( Site 3118)

Nanning, Guangxi, China

Site Status RECRUITING

Jiangsu Province Hospital ( Site 3105)

Nanjing, Jiangsu, China

Site Status RECRUITING

Nanchang People's Hospital ( Site 3124)

Nanchang, Jiangxi, China

Site Status RECRUITING

Sichuan Cancer Hospital. ( Site 3110)

Chengdu, Sichuan, China

Site Status RECRUITING

Taizhou Hospital of Zhejiang Province ( Site 3137)

Linhai, Zhejiang, China

Site Status RECRUITING

Instituto de Cancerología-Oncology ( Site 0503)

Medellín, Antioquia, Colombia

Site Status RECRUITING

FUNDACION CTIC CENTRO DE TRATAMIENTO E INVESTIGACION SOBRE CANCER LUIS CARLOS SARMIENTO ANGULO ( Site 0502)

Bogotá, Bogota D.C., Colombia

Site Status RECRUITING

Instituto Nacional De Cancerologia ( Site 0504)

Bogotá, Bogota D.C., Colombia

Site Status RECRUITING

Sociedad De Oncología y Hematología Del Cesar SAS ( Site 0501)

Valledupar, Cesar Department, Colombia

Site Status RECRUITING

IMAT S.A.S ( Site 0500)

Montería, Departamento de Córdoba, Colombia

Site Status RECRUITING

CHRU de Brest ( Site 0904)

Brest, Finistere, France

Site Status RECRUITING

CENTRE LEON BERARD ( Site 0900)

Lyon, Rhone, France

Site Status RECRUITING

Centre de Lutte Contre le Cancer - Centre Henri Becquerel Normandie Rouen ( Site 0901)

Rouen, Seine-Maritime, France

Site Status RECRUITING

Gustave Roussy ( Site 0903)

Villejuif, Val-de-Marne, France

Site Status RECRUITING

Aretaieio Hospital ( Site 1103)

Athens, Attica, Greece

Site Status RECRUITING

University General Hospital of Heraklion ( Site 1102)

Heraklion, Irakleio, Greece

Site Status RECRUITING

European Interbalkan Medical Center-Oncology Department ( Site 1101)

Thessaloniki, , Greece

Site Status RECRUITING

Bacs-Kiskun Varmegyei Oktatokorhaz-Onkoradiologiai Kozpont ( Site 1200)

Kecskemét, Bács-Kiskun county, Hungary

Site Status RECRUITING

Rambam Health Care Campus ( Site 1401)

Haifa, , Israel

Site Status RECRUITING

Shaare Zedek Medical Center ( Site 1406)

Jerusalem, , Israel

Site Status RECRUITING

Hadassah Medical Center ( Site 1404)

Jerusalem, , Israel

Site Status RECRUITING

Sheba Medical Center ( Site 1400)

Ramat Gan, , Israel

Site Status RECRUITING

Istituto Europeo di Oncologia IRCCS ( Site 1508)

Milan, Lombardy, Italy

Site Status RECRUITING

Istituto Nazionale Tumori IRCCS Fondazione Pascale-S.C. Oncologia Clinica Sperimentale di Senologia ( Site 1506)

Napoli, , Italy

Site Status RECRUITING

Fondazione Policlinico Universitario Agostino Gemelli IRCCS - Università Cattolica del Sacro Cuore ( Site 1500)

Roma, , Italy

Site Status RECRUITING

Nagoya City University Hospital ( Site 3210)

Nagoya, Aichi-ken, Japan

Site Status RECRUITING

National Hospital Organization Hokkaido Cancer Center ( Site 3215)

Sapporo, Hokkaido, Japan

Site Status RECRUITING

Kansai Medical University Hospital ( Site 3213)

Hirakata, Osaka, Japan

Site Status RECRUITING

Kindai University Hospital ( Site 3204)

Sakai, Osaka, Japan

Site Status RECRUITING

Shizuoka Cancer Center ( Site 3202)

Sunto-gun, Shizuoka, Japan

Site Status RECRUITING

National Cancer Center Hospital ( Site 3206)

Chūō, Tokyo, Japan

Site Status RECRUITING

Toranomon Hospital ( Site 3205)

Minato, Tokyo, Japan

Site Status RECRUITING

Showa Medical University Hospital ( Site 3209)

Shinagawa, Tokyo, Japan

Site Status RECRUITING

Akita University Hospital ( Site 3207)

Akita, , Japan

Site Status RECRUITING

Chiba Cancer Center ( Site 3203)

Chiba, , Japan

Site Status RECRUITING

National Hospital Organization Kyushu Cancer Center ( Site 3208)

Fukuoka, , Japan

Site Status RECRUITING

Fukushima Medical University Hospital ( Site 3212)

Fukushima, , Japan

Site Status RECRUITING

Hiroshima City Hiroshima Citizens Hospital ( Site 3214)

Hiroshima, , Japan

Site Status RECRUITING

National Hospital Organization Osaka National Hospital ( Site 3201)

Osaka, , Japan

Site Status RECRUITING

Narodowy Instytut Onkologii im. Marii Sklodowskiej-Curie ( Site 1600)

Warsaw, Masovian Voivodeship, Poland

Site Status RECRUITING

Szpital Kliniczny Ministerstwa Spraw Wewnętrznych i Administracji z Warmińsko-Mazurskim Centrum Onko ( Site 1614)

Olsztyn, Warmian-Masurian Voivodeship, Poland

Site Status RECRUITING

Seoul National University Bundang Hospital ( Site 2703)

Seongnam, Kyonggi-do, South Korea

Site Status RECRUITING

Gangnam Severance Hospital, Yonsei University Health System ( Site 2701)

Gangnam-gu, Seoul, South Korea

Site Status RECRUITING

Samsung Medical Center ( Site 2704)

Gangnam-gu, Seoul, South Korea

Site Status RECRUITING

Seoul National University Hospital ( Site 2702)

Jongno-Gu, Seoul, South Korea

Site Status RECRUITING

Severance Hospital Yonsei University Health System ( Site 2700)

Seoul, , South Korea

Site Status RECRUITING

Asan Medical Center ( Site 2705)

Seoul, , South Korea

Site Status RECRUITING

Hospital Universitario Marques de Valdecilla ( Site 1825)

Santander, Cantabria, Spain

Site Status RECRUITING

CHUAC-Complejo Hospitalario Universitario A Coruña ( Site 1820)

A Coruña, La Coruna, Spain

Site Status RECRUITING

Hospital Clinic de Barcelona ( Site 1821)

Barcelona, , Spain

Site Status RECRUITING

Institut Català d'Oncologia (ICO) - Badalona ( Site 1823)

Barcelona, , Spain

Site Status RECRUITING

Hospital Universitario Ramon y Cajal ( Site 1824)

Madrid, , Spain

Site Status RECRUITING

Hospital Clinico San Carlos... ( Site 1822)

Madrid, , Spain

Site Status RECRUITING

Hospital Universitario Virgen de Valme ( Site 1826)

Seville, , Spain

Site Status RECRUITING

Ditmanson Medical Foundation Chia-Yi Christian Hospital ( Site 2806)

Chiayi City, Chiayi, Taiwan

Site Status RECRUITING

Taichung Veterans General Hospital ( Site 2803)

Taichung, , Taiwan

Site Status RECRUITING

National Cheng Kung University Hospital ( Site 2804)

Tainan, , Taiwan

Site Status RECRUITING

Chi-Mei Medical Center ( Site 2805)

Tainan, , Taiwan

Site Status RECRUITING

National Taiwan University Hospital ( Site 2800)

Taipei, , Taiwan

Site Status RECRUITING

MacKay Memorial Hospital ( Site 2802)

Taipei, , Taiwan

Site Status RECRUITING

National Taiwan University Cancer Center (NTUCC) ( Site 2801)

Taipei, , Taiwan

Site Status RECRUITING

Hacettepe Universite Hastaneleri ( Site 2100)

Ankara, , Turkey (Türkiye)

Site Status RECRUITING

Memorial Ankara Hastanesi ( Site 2106)

Ankara, , Turkey (Türkiye)

Site Status RECRUITING

Ankara Bilkent Şehir Hastanesi ( Site 2105)

Ankara, , Turkey (Türkiye)

Site Status RECRUITING

Koç Üniversitesi Hastanesi ( Site 2104)

Istanbul, , Turkey (Türkiye)

Site Status RECRUITING

Samsun Medical Park Hastanesi ( Site 2109)

Samsun, , Turkey (Türkiye)

Site Status RECRUITING

Countries

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United States Argentina Canada China Colombia France Greece Hungary Israel Italy Japan Poland South Korea Spain Taiwan Turkey (Türkiye)

Central Contacts

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Toll Free Number

Role: CONTACT

Phone: 1-888-577-8839

Email: [email protected]

Facility Contacts

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Study Coordinator

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Related Links

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http://www.merckclinicaltrials.com

Merck Clinical Trials Information

Other Identifiers

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U1111-1317-5490

Identifier Type: REGISTRY

Identifier Source: secondary_id

2025-520582-51-00

Identifier Type: REGISTRY

Identifier Source: secondary_id

jRCT2031250297

Identifier Type: REGISTRY

Identifier Source: secondary_id

1022-016

Identifier Type: -

Identifier Source: org_study_id