Study of Bitopertin in Participants With EPP or XLP (APOLLO)

NCT ID: NCT06910358

Last Updated: 2025-11-13

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

RECRUITING

Clinical Phase

PHASE3

Total Enrollment

150 participants

Study Classification

INTERVENTIONAL

Study Start Date

2025-04-04

Study Completion Date

2026-11-30

Brief Summary

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The goal of this clinical trial is to learn if bitopertin works and is safe to treat EPP or XLP in participants 12 years or older. The main questions it aims to answer are:

* Whether bitopertin increases pain-free sunlight exposure after 6 months of treatment in participants with EPP or XLP.
* How PPIX concentration levels change from before bitopertin treatment to after 6 months of treatment.

Researchers will compare bitopertin to a placebo look-alike substance that contains no drug.

Participants will complete daily questionnaires and attend study visits for assessments.

Detailed Description

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Conditions

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Erythropoietic Protoporphyria (EPP) X-Linked Protoporphyria (XLP)

Keywords

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EPP XLP DISC-1459 RO4917838 porphyria

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

QUADRUPLE

Participants Caregivers Investigators Outcome Assessors

Study Groups

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Placebo

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DRUG

Oral dose, once a day for 24 weeks

DISC-1459 oral dose

Group Type EXPERIMENTAL

DISC-1459

Intervention Type DRUG

Oral dose, once a day for 24 weeks

Interventions

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Placebo

Oral dose, once a day for 24 weeks

Intervention Type DRUG

DISC-1459

Oral dose, once a day for 24 weeks

Intervention Type DRUG

Other Intervention Names

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Bitopertin RO4917838

Eligibility Criteria

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Inclusion Criteria

1. Aged 12 years or older at the time of study consent.
2. Diagnosis of EPP or XLP, based on medical history by ferrochelatase (FECH) or aminolevulinic acid synthase 2 (ALAS2) genotyping or by biochemical porphyrin analysis.
3. Minimum daily Sun Exposure Diary compliance ≥85% on Days -14 through Day -1, inclusive, during screening, and at least 1 successfully completed Sun Exposure Challenge (adults only, as this assessment is optional for adolescents) or historical recall of time to prodrome
4. Body weight ≥32 kg (ages 12 to \<18 years), body mass index ≥18.5 kg/m2 (ages ≥18 years) at screening.
5. Washout of at least 2 months prior to screening of afamelanotide and dersimelagon, if applicable.
6. Aspartate aminotransferase and alanine transaminase \<3× upper limit of normal (ULN)and total bilirubin \<2× ULN (unless documented Gilbert syndrome) at screening. Albumin \>lower limit of normal (LLN).
7. Willing to practice highly effective methods of birth control (both males who have partners of childbearing potential and females of childbearing potential during screening, while taking study drug, and for at least 30 days after the last dose of study drug).

Exclusion Criteria

1. Major surgery within 8 weeks before screening or incomplete recovery from any previous surgery.
2. Other than EPP or XLP, an inherited intrinsic or extrinsic red cell disease associated with anemia.
3. Known hypersensitivity to any component of the study drug.
4. History of liver transplantation or anticipated need for liver transplantation.
5. History of alcohol dependence or excessive alcohol consumption, as assessed by the Investigator.
6. Active human immunodeficiency virus (HIV), active hepatitis B or C.
7. Other medical or psychiatric condition or laboratory finding not specifically noted above that, in the judgment of the Investigator or Sponsor, would put the participant at unacceptable risk or otherwise preclude the participant from participating in the study.
8. Condition or concomitant medication that would confound the ability to interpret clinical, clinical laboratory, or participant diary data, including a major psychiatric condition that has had an exacerbation or required hospitalization in the last 6 months.

Treatment History:
9. Prior exposure to bitopertin.
10. Concurrent or planned treatment with afamelanotide or dersimelagon during the study period.
11. Treatment with opioids for any period \>7 days in the 2 months prior to screening or anticipated to require opioid use for \>7 days at any point during the study.
12. New treatment for anemia, including initiation of iron supplementation, within 1 month of screening.
13. Current or planned use of any drugs or herbal remedies known to be strong or moderate inhibitors or inducers of cytochrome P450 (CYP)3A4 enzymes for 28 days prior to the first dose and throughout the study.
14. Current or planned treatment with antipsychotic medication.

Laboratory Exclusions:
15. Hemoglobin \<10 g/dL at screening.

Miscellaneous:
16. Participation in other interventional clinical studies within 30 days prior to screening.
17. If female, pregnant or breastfeeding.
Minimum Eligible Age

12 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Disc Medicine, Inc

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Will Savage, MD, PhD

Role: STUDY_DIRECTOR

Disc Medicine

Locations

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Marvel Clinical Research

Huntington Beach, California, United States

Site Status RECRUITING

University of California San Francisco

San Francisco, California, United States

Site Status RECRUITING

University of Miami Miller School of Medicine

Miami, Florida, United States

Site Status RECRUITING

Massachusetts General Hospital

Boston, Massachusetts, United States

Site Status RECRUITING

MetroBoston Clinical Partners

Boston, Massachusetts, United States

Site Status RECRUITING

Henry Ford Health System

Detroit, Michigan, United States

Site Status RECRUITING

Mount Sinai Hospital

New York, New York, United States

Site Status RECRUITING

Wake Forest University

Winston-Salem, North Carolina, United States

Site Status RECRUITING

Remington-Davis Clinical Research

Columbus, Ohio, United States

Site Status RECRUITING

University of Texas Medical Branch

Galveston, Texas, United States

Site Status RECRUITING

University of Washington

Seattle, Washington, United States

Site Status RECRUITING

Royal Prince Alfred Hospital

Camperdown, New South Wales, Australia

Site Status RECRUITING

The Royal Melbourne Hospital

Parkville, Victoria, Australia

Site Status RECRUITING

University of Alberta

Edmonton, Alberta, Canada

Site Status NOT_YET_RECRUITING

Helse Bergen

Bergen, Norway, Norway

Site Status RECRUITING

Countries

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United States Australia Canada Norway

Central Contacts

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Disc Medicine Clinical Trials

Role: CONTACT

Phone: (617) 674 9274

Email: [email protected]

Facility Contacts

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Matthew Campos

Role: primary

Jackie Lam

Role: primary

Felisa Padilla

Role: primary

Narmene Bensaber

Role: primary

Stella Schandorf

Role: primary

Jennifer Creasor

Role: primary

Georgia MacDonald

Role: primary

Dee Faust

Role: primary

Imani Ramos

Role: primary

Role: backup

Rochelle Simmons

Role: primary

Ryan Donnelly

Role: primary

Darcie Kavanagh

Role: primary

Dermatology Research

Role: primary

Samridhi Dhand

Role: primary

Study Coordinator

Role: primary

Other Identifiers

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2024-520407-27-00

Identifier Type: CTIS

Identifier Source: secondary_id

DISC-1459-301

Identifier Type: -

Identifier Source: org_study_id