Study of GS-0151 in Participants With Rheumatoid Arthritis

NCT ID: NCT06902519

Last Updated: 2025-12-23

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

RECRUITING

Clinical Phase

PHASE1

Total Enrollment

75 participants

Study Classification

INTERVENTIONAL

Study Start Date

2025-05-14

Study Completion Date

2027-03-31

Brief Summary

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The goal of this clinical study is to learn more about the study drug GS-0151. The study is done to find how safe, well-tolerated the drug is. This will also assess how the drug is absorbed, modified, distributed and cleared from the body (the pharmacokinetics (PK) of the drug), when given multiple times to participants with rheumatoid arthritis (RA).

The primary objectives of this study is to assess the safety and tolerability of multiple ascending doses of GS-0151 in participants with RA and to characterize the PK of GS-0151 following multiple doses of GS-0151 in participants with RA.

Detailed Description

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Conditions

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Rheumatoid Arthritis

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

In Part A, Cohorts 1 and 2 will be sequential, with participants receiving treatment in parallel and randomized in 6:2 ratio to either GS-0151 or placebo. In Part B, Cohort 3 will also randomized in 2:1 ratio to receive GS-0151 or placebo in parallel.
Primary Study Purpose

TREATMENT

Blinding Strategy

DOUBLE

Participants Investigators

Study Groups

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Part A: Cohort 1 (GS-0151 Dose A)

Participants with RA will be randomized to receive Dose A of GS-0151 up to 12 weeks.

Group Type EXPERIMENTAL

GS-0151

Intervention Type DRUG

Administered for 12 weeks

Part A: Cohort 1 (Placebo)

Participants with RA will be randomized to receive placebo up to 12 weeks.

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DRUG

Administered for 12 weeks

Part A: Cohort 2 (GS-0151 Dose B)

Participants with RA will be randomized to receive Dose B of GS-0151 up to 12 weeks.

Group Type EXPERIMENTAL

GS-0151

Intervention Type DRUG

Administered for 12 weeks

Part A: Cohort 2 (Placebo)

Participants with RA will be randomized to receive placebo up to 12 weeks.

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DRUG

Administered for 12 weeks

Part B: Cohort 3 (GS-0151 Dose C)

Participants with moderately to severely active RA will be randomized to receive Dose C of GS-0151.

Group Type EXPERIMENTAL

GS-0151

Intervention Type DRUG

Administered for 12 weeks

Part B: Cohort 3 (Placebo)

Participants with moderately to severely active RA will be randomized to receive placebo.

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DRUG

Administered for 12 weeks

Interventions

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GS-0151

Administered for 12 weeks

Intervention Type DRUG

Placebo

Administered for 12 weeks

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

Medical History/Physical Characteristics; All Cohorts:

* Individuals must not be on a biologic disease-modifying antirheumatic drug (b/tsDMARD) on Day 1 and must have discontinued all b/tsDMARDs (including biosimilars and generics) at least 4 weeks prior to Day 1 with the exception of B cell-depleting agents (eg, rituximab), which must be discontinued for at least 6 months prior to Day 1.
* Ongoing treatment with at least 1 but no more than 2 protocol-permitted conventional synthetic disease-modifying antirheumatic drug (csDMARDs) for at least 12 weeks, at a stable dose for at least 6 weeks prior to Day 1 and remain stable throughout the treatment period:

1. Use of oral, intramuscular (IM), or subcutaneous(ly) (SC) methotrexate 7.5 to 25 mg/week. Individuals on methotrexate must be receiving folic or folinic acid supplementation at a stable dose.
2. Oral hydroxychloroquine ≤ 400 mg/day or chloroquine ≤ 250 mg/day.
3. Oral sulfasalazine 1 to 3 g/day.
4. Oral leflunomide 10 to 20 mg/day.
* Use of oral corticosteroids of no more than 10 mg prednisone or equivalent per day is allowed if the dose is stable for at least 14 days prior to Day 1. Inhaled corticosteroids for stable medical conditions are allowed but must have been at a stable dose for at least

1 week prior to the first dose of study drug. Occasional topical corticosteroids are permitted.
* Where nonsteroidal anti-inflammatory drug (NSAIDs) or acetaminophen are used, the dose must be stable for at least 1 week prior to Day 1
* Individuals must have discontinued all high-potency opiates at least 1 week prior to Day 1.

Cohort 3 Only:


Moderately to severely active RA defined by the following:

Screening and Day 1:

1. 6 or more tender joints on the tender joint count based on 68 joints (TJC68), AND.
2. 6 or more swollen joints on the swollen joint count based on 66 joints (SJC66). The distal interphalangeal joints should be evaluated but not included in the total count to determine eligibility.

Screening Only
3. Have a hsCRP ≥ ULN

* Inadequate response or intolerance to at least 1 but no more than 3 b/tsDMARDs with no more than 2 mechanisms of action. A lack of response is defined as documented continued or recurrent disease activity after at least 12 weeks of treatment of RA. Intolerance is defined as any documented adverse effect associated with a b/tsDMARD used according to its respective label.

Laboratory Assessments:

Cohort 3 Only:

* Anti-cyclic citrullinated peptide antibody (Anti-CCP) positive and/or rheumatoid factor (RF) positive

Exclusion Criteria

Medical Conditions; All Cohorts:

* Have a diagnosis of any generalized musculoskeletal disorder that would interfere with study procedures or assessments per the discretion of the investigator.
* History of opportunistic infection or immunodeficiency syndrome that would put the individual at risk, as per investigator's judgment.
* Active infection that is clinically significant, per investigator's judgment, or any infection requiring hospitalization or treatment with intravenous anti-infectives within 60 days of screening; or any infection requiring oral anti-infective therapy within 30 days of screening.
* History of or current moderate to severe congestive heart failure (New York Heart Association class III or IV), or within the last 6 months prior to screening.
* History of lymphoproliferative disease or possible current lymphoproliferative disease.
* History of organ or bone marrow transplant.
* Have a history of major surgery (requiring regional block or general anesthesia) within the last 12 weeks prior to screening or planned major surgery during the study.
* History of an infected joint prosthesis or other implanted device with the prosthesis or device still in situ.
* Clinically significant ECG abnormalities at screening, including electrocardiographic interval between the beginning of the Q wave and termination of the T wave, representing the time for both ventricular depolarization and repolarization to occur (QT) interval corrected for heart rate using the Fridericia formula (QTcF) \> 450 msec, or hypokalemia if recurrent or persistent \< 3.0 mmol/L, or family history of long QT syndrome

Prior/Concurrent Therapy or Clinical Study Experience:

* Administration of a live attenuated vaccine 4 weeks prior to Day 1 or planned throughout the study.
* Participation in any investigational drug/device clinical study within 4 weeks or 5 half-lives prior to screening, whichever is longer. Exposure to investigational biologics should be discussed with the sponsor.

Diagnostic Assessments; All Cohorts:

* Any positive tuberculosis (TB) test using interferon-gamma release assay (IGRA) performed by central laboratory at screening. Tests with inconclusive results may be repeated one time. If an inconclusive test is repeated and is returned with inconclusive results a second time, the individual will be excluded from the study. Individuals with a history of latent or active TB who have been treated with a full course of treatment, as per local guidelines, are eligible without the need for an IGRA at screening. Appropriate documentation of prior treatment is required.
* Evidence of active hepatitis C virus (HCV) infection. Individuals with positive HCV Ab at screening require reflex testing for HCV ribonucleic acid (RNA). Individuals with positive HCV Ab but negative HCV RNA viral load are eligible per investigator judgment and require HCV viral load monitoring on Day 85 and Day 169.
* The results of the following laboratory tests performed at the central laboratory at screening meet any of the criteria below (out-of-range laboratory values may be rechecked 1 time, per investigator's judgment, before individual is considered a screen failure):

1. Hemoglobin \< 10.0 g/dL (SI: \< 100 g/L)
2. White blood cells \< 3.0 x 10\^3 cells/mm\^3 (SI: \< 3.0 x 10\^9 cells/L)
3. Neutrophils \< 1.5 x 10\^3 cells/mm\^3 (SI: \< 1.5 x 10\^9 cells/L)
4. Lymphocytes \< 1.0 x 10\^3 cells/mm\^3 (SI: \< 1.0 x 10\^9 cells/L)
5. Platelets \< 100 x 10\^3 cells/mm\^3 (SI: \< 100 x 10\^9 cells/L)
6. Alanine aminotransferase (ALT) or aspartate aminotransferase (AST) ≥ 1.5 x upper limit of normal (ULN)
7. Total bilirubin level ≥ 2 x ULN unless the individual has been diagnosed with Gilbert's disease and this is clearly documented
8. Creatinine clearance \< 50 mL/min (SI: \< 0.83 mL/s) based on the Cockcroft-Gault formula
Minimum Eligible Age

18 Years

Maximum Eligible Age

75 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Gilead Sciences

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Gilead Study Director

Role: STUDY_DIRECTOR

Gilead Sciences

Locations

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Pinnacle Research Group, LLC

Anniston, Alabama, United States

Site Status RECRUITING

University of California, San Diego

La Jolla, California, United States

Site Status RECRUITING

Stanford University School of Medicine

Palo Alto, California, United States

Site Status RECRUITING

Medvin Clinical Research

Tujunga, California, United States

Site Status RECRUITING

Medvin Clinical Research

Whittier, California, United States

Site Status RECRUITING

Clinical Research of West Florida, Inc

Clearwater, Florida, United States

Site Status RECRUITING

Great Lakes Clinical Trials dba Flourish Research Chicago

Chicago, Illinois, United States

Site Status RECRUITING

DM Clinical Research

Melrose Park, Illinois, United States

Site Status RECRUITING

Accurate Clinical Research, Inc

Lake Charles, Louisiana, United States

Site Status RECRUITING

Lynn Health Science Institute

Oklahoma City, Oklahoma, United States

Site Status RECRUITING

Altoona Center for Clinical Research

Duncansville, Pennsylvania, United States

Site Status RECRUITING

Accurate Clinical Management, LLC

Baytown, Texas, United States

Site Status RECRUITING

Accurate Clinical Research, Inc

Houston, Texas, United States

Site Status RECRUITING

Clinical Trials of Texas LLC, dba Flourish Research

San Antonio, Texas, United States

Site Status RECRUITING

Tidewater Clinical Research, LLC/ Virginia Rheumatology Clinic

Virginia Beach, Virginia, United States

Site Status RECRUITING

ARENSIA Exploratory Medicine, LLC

Tbilisi, , Georgia

Site Status RECRUITING

Universitatsklinikum Koln

Cologne, , Germany

Site Status RECRUITING

Hamburger Rheuma Forschungszentrum II

Hamburg, , Germany

Site Status RECRUITING

Republican Clinical Hospital "Timofei Mosneaga," Arensia EM

Chisinau, , Moldova

Site Status RECRUITING

Clinicmed Daniluk

Bialystok, , Poland

Site Status RECRUITING

FutureMeds Gydinia

Gdynia, , Poland

Site Status RECRUITING

FutureMeds Lodz

Lodz, , Poland

Site Status RECRUITING

MICS Centrum Medyczne Torun

Torun, , Poland

Site Status RECRUITING

FutureMeds Targowek

Warszawa Targówek, , Poland

Site Status RECRUITING

FutureMeds Wroclaw

Wroclaw, , Poland

Site Status RECRUITING

Complejo Hospitalario Universitario A Coruna

A Coruña, , Spain

Site Status RECRUITING

Hospital del Mar

Barcelona, , Spain

Site Status RECRUITING

Hospital Universitario Ramon y Cajal

Madrid, , Spain

Site Status RECRUITING

Hospital Universitari Parc Tauli

Sabadell, , Spain

Site Status RECRUITING

Hospital Infanta Luisa

Seville, , Spain

Site Status RECRUITING

Countries

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United States Georgia Germany Moldova Poland Spain

Central Contacts

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Gilead Clinical Study Information Center

Role: CONTACT

Phone: 1-833-445-3230 (GILEAD-0)

Email: [email protected]

Related Links

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Other Identifiers

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GS-US-667-6882

Identifier Type: -

Identifier Source: org_study_id

2024-516520-34

Identifier Type: OTHER

Identifier Source: secondary_id