An Investigational Study of BGB-58067 As a Single Agent and in Combination With Anticancer Agents in Participants With Advanced Solid Tumors

NCT ID: NCT06589596

Last Updated: 2025-11-12

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

RECRUITING

Clinical Phase

PHASE1

Total Enrollment

237 participants

Study Classification

INTERVENTIONAL

Study Start Date

2024-10-11

Study Completion Date

2027-06-30

Brief Summary

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This is an open-label, multicenter, first-in-human dose escalation and dose expansion study to evaluate the safety, tolerability, pharmacokinetics, pharmacodynamics, and preliminary antitumor activity of BGB-58067 alone, in combination with BG-89894, and in combination with standard of care therapy in participants with advanced solid tumors and with methylthioadenosine phosphorylase (MTAP) deficiency.

Detailed Description

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BGB-58067 is a new drug designed to target a specific protein called protein arginine methyltransferase 5 (PRMT5). This protein is involved in many cell activities and can promote cancer growth when it is overactive. High levels of PRMT5 are linked to poor outcomes in several types of cancer.

This new study will check how safe and helpful a potential anticancer drug called BGB-58067 is. This drug will be tested alone, in combination with BG-89894, and in combination with standard of care therapy in participants with advanced solid tumors and with MTAP deficiency.

Conditions

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Advanced Solid Tumor

Keywords

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advanced solid tumor BGB-58067 MTAP deficiency BG-89894

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

SEQUENTIAL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Phase 1a: BGB-58067 Monotherapy Dose Escalation and Safety Expansion

Sequential cohorts of increasing dose levels of BGB-58067 as monotherapy will be evaluated.

Group Type EXPERIMENTAL

BGB-58067

Intervention Type DRUG

Planned doses administered on specified days per protocol.

Phase 1a: BGB-58067 + BG-89894 Combination Therapy Dose Escalation

Sequential cohorts of increasing dose levels of BGB-58067 in combination with BGB-89894 will be evaluated.

Group Type EXPERIMENTAL

BGB-58067

Intervention Type DRUG

Planned doses administered on specified days per protocol.

BG-89894

Intervention Type DRUG

Planned doses administered on specified days per protocol.

Phase 1a: BGB-58067 + Standard of Care Combination Therapy Dose Escalation

Sequential cohorts of increasing dose levels of BGB-58067 in combination with standard of care therapy will be evaluated.

Group Type EXPERIMENTAL

BGB-58067

Intervention Type DRUG

Planned doses administered on specified days per protocol.

Standard of Care Therapy

Intervention Type DRUG

Administered in accordance with relevant local guidelines and/or prescribing information.

Phase 1b: Dose Expansion and Optimization

Recommended Dose(s) for Expansion (RDFE\[s\]) of BGB-58067 alone, in combination with BG-89894, and in combination with standard of care therapy will be evaluated for selected indications and regimen(s) based on emerging data.

Group Type EXPERIMENTAL

BGB-58067

Intervention Type DRUG

Planned doses administered on specified days per protocol.

BG-89894

Intervention Type DRUG

Planned doses administered on specified days per protocol.

Standard of Care Therapy

Intervention Type DRUG

Administered in accordance with relevant local guidelines and/or prescribing information.

Interventions

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BGB-58067

Planned doses administered on specified days per protocol.

Intervention Type DRUG

BG-89894

Planned doses administered on specified days per protocol.

Intervention Type DRUG

Standard of Care Therapy

Administered in accordance with relevant local guidelines and/or prescribing information.

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Participants must sign the ICF and be capable of giving written informed consent
* Eastern Cooperative Oncology Group (ECOG) Performance Status of 0 or 1 or Karnofsky Performance Scale (KPS) ≥ 70
* Life expectancy ≥ 3 months
* Evidence of homozygous loss of MTAP or lost MTAP expression in the tumor tissue
* Able to provide tumor sample to meet the minimum tissue requirement for central MTAP deficiency testing
* Participants with histologically or cytologically confirmed advanced, metastatic, or unresectable solid tumors, whose diseases have progressed or recurred after receiving standard systemic therapy or radiotherapy, or for whom standard systemic therapy is not available or tolerated, or would be unlikely to tolerate or derive clinically meaningful benefit from appropriate standard treatment in the opinion of the investigator
* Adequate organ function

Exclusion Criteria

* Prior treatment with any methylthioadenosine (MTA)-cooperative PRMT5 inhibitor or methionine adenosyltransferase 2a (MAT2A) inhibitor
* Active leptomeningeal disease or symptomatic spinal cord compression
* Uncontrollable pleural effusion, pericardial effusion, or ascites requiring frequent drainage
* Any malignancy ≤ 2 years before first dose of study drug except for the specific cancer under investigation in this study and any locally recurring cancer that has been treated curatively
* Significantly impaired pulmonary function
* Clinically significant infections
* Serologically active hepatitis B or C infection
* Known HIV infection. Participants with treated HIV infection may be included in Phase 1b if they meet certain criteria
* High cardiovascular risk factors
* QTcF \> 470 ms based on the screening triplicate 12-lead ECG records and/or a history of additional risk factors for torsade de pointes (eg, heart failure, hypokalemia, or a family history of Long QT Syndrome)
* Toxicities (because of prior anticancer therapy) that have not recovered to baseline or stabilized
* Participants who are unable to swallow or with disease/procedure significantly affecting gastrointestinal function
* Female participants who are pregnant or are breastfeeding
* Concurrent participation in another therapeutic clinical study (participation in observational or noninterventional studies is allowed)
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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BeiGene

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Study Director

Role: STUDY_DIRECTOR

BeiGene

Locations

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Usc Norris Comprehensive Cancer Center (Nccc)

Los Angeles, California, United States

Site Status RECRUITING

Adventhealth

Celebration, Florida, United States

Site Status RECRUITING

Dana Farber Cancer Institute

Boston, Massachusetts, United States

Site Status RECRUITING

Washington University School of Medicine

St Louis, Missouri, United States

Site Status RECRUITING

Nyu Langone Health

New York, New York, United States

Site Status RECRUITING

Sidney Kimmel Cancer Center

Philadelphia, Pennsylvania, United States

Site Status RECRUITING

The University of Texas Md Anderson Cancer Center

Houston, Texas, United States

Site Status RECRUITING

Next Dallas

Irving, Texas, United States

Site Status RECRUITING

Next Virginia

Fairfax, Virginia, United States

Site Status RECRUITING

Blacktown Cancer and Haematology Centre

Blacktown, New South Wales, Australia

Site Status RECRUITING

Monash Health

Clayton, Victoria, Australia

Site Status RECRUITING

Austin Health

Heidelberg, Victoria, Australia

Site Status RECRUITING

Linear Clinical Research

Nedlands, Western Australia, Australia

Site Status RECRUITING

Cancer Hospital Chinese Academy of Medical Sciences

Beijing, Beijing Municipality, China

Site Status RECRUITING

Beijing Cancer Hospital

Beijing, Beijing Municipality, China

Site Status RECRUITING

Fujian Cancer Hospital

Fuzhou, Fujian, China

Site Status RECRUITING

Sun Yat Sen University Cancer Center

Guangzhou, Guangdong, China

Site Status RECRUITING

Harbin Medical University Cancer Hospital

Harbin, Heilongjiang, China

Site Status RECRUITING

Henan Cancer Hospital

Zhengzhou, Henan, China

Site Status RECRUITING

The First Affiliated Hospital of Zhengzhou University

Zhengzhou, Henan, China

Site Status RECRUITING

Union Hospital of Tongji Medical College, Huazhong University of Science and Technology

Wuhan, Hubei, China

Site Status RECRUITING

Jiangsu Province Hospital

Nanjing, Jiangsu, China

Site Status RECRUITING

Jiangxi Cancer Hospital

Nanchang, Jiangxi, China

Site Status RECRUITING

The First Hospital of China Medical University

Shenyang, Liaoning, China

Site Status RECRUITING

Shanghai East Hospital Branch Hospital

Shanghai, Shanghai Municipality, China

Site Status RECRUITING

Shanghai Pulmonary Hospital

Shanghai, Shanghai Municipality, China

Site Status RECRUITING

Fudan University Shanghai Cancer Centerpudong

Shanghai, Shanghai Municipality, China

Site Status RECRUITING

West China Hospital, Sichuan University

Chengdu, Sichuan, China

Site Status RECRUITING

Zhejiang Cancer Hospital

Hangzhou, Zhejiang, China

Site Status RECRUITING

Rigshospitalet

Copenhagen, , Denmark

Site Status RECRUITING

Centre de Lutte Contre Le Cancer Institut Bergonie

Bordeaux, , France

Site Status RECRUITING

Institut Curie Paris

Paris, , France

Site Status RECRUITING

Institut Gustave Roussy

Villejuif, , France

Site Status RECRUITING

Samsung Medical Center

GangnamGu, Seoul Teugbyeolsi, South Korea

Site Status RECRUITING

Severance Hospital Yonsei University Health System

SeodaemunGu, Seoul Teugbyeolsi, South Korea

Site Status RECRUITING

Seoul National University Hospital

Seoul, Seoul Teugbyeolsi, South Korea

Site Status RECRUITING

Asan Medical Center

SongpaGu, Seoul Teugbyeolsi, South Korea

Site Status RECRUITING

Hospital Universitario Vall Dhebron

Barcelona, , Spain

Site Status RECRUITING

Hospital Clinico San Carlos

Madrid, , Spain

Site Status RECRUITING

Start Madrid Fundacion Jimenez Diaz

Madrid, , Spain

Site Status RECRUITING

Hospital Universitario Hm Madrid Sanchinarro

Madrid, , Spain

Site Status RECRUITING

Countries

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United States Australia China Denmark France South Korea Spain

Central Contacts

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Study Director

Role: CONTACT

Phone: 1.877.828.5568

Email: [email protected]

Other Identifiers

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2024-515307-19-00

Identifier Type: CTIS

Identifier Source: secondary_id

CTR20244451

Identifier Type: REGISTRY

Identifier Source: secondary_id

BGB-58067-101

Identifier Type: -

Identifier Source: org_study_id