Study of Momelotinib in Combination With Luspatercept in Participants With Transfusion Dependent Myelofibrosis

NCT ID: NCT06517875

Last Updated: 2025-12-16

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

RECRUITING

Clinical Phase

PHASE2

Total Enrollment

56 participants

Study Classification

INTERVENTIONAL

Study Start Date

2025-02-28

Study Completion Date

2026-11-13

Brief Summary

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The purpose of this Phase 2 study is to evaluate the efficacy and safety of momelotinib (MMB) in combination with luspatercept (LUSPA) in participants with transfusion dependence (TD) primary myelofibrosis (PMF) or Post-polycythemia vera (PV)/ essential thrombocythemia (ET) myelofibrosis (MF) who are either janus kinase (JAK) inhibitor (JAKi) naïve or experienced.

Detailed Description

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Conditions

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Primary Myelofibrosis Myelofibrosis; Primary Myelofibrosis; Post-polycythemia Vera Myelofibrosis; Post-essential Thrombocythemia Myelofibrosis

Study Design

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Allocation Method

NA

Intervention Model

SINGLE_GROUP

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Momelotinib + Luspatercept

Participants with transfusion dependent primary myelofibrosis or post- PV/ ET myelofibrosis that is JAKi naïve or JAKi experienced will receive momelotinib and luspatercept.

Group Type EXPERIMENTAL

Momelotinib

Intervention Type DRUG

Momelotinib will be administered orally.

Luspatercept

Intervention Type DRUG

Luspatercept will be administered subcutaneously.

Interventions

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Momelotinib

Momelotinib will be administered orally.

Intervention Type DRUG

Luspatercept

Luspatercept will be administered subcutaneously.

Intervention Type DRUG

Other Intervention Names

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Ojjaara; CYT387 REBLOZYL; ACE-536

Eligibility Criteria

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Inclusion Criteria

1. Is age ≥18 years.
2. Confirmed diagnosis of PMF in accordance with the World Health Organization (WHO) 2016 criteria, or Post-PV/ET myelofibrosis in accordance with the International Working Group-Myeloproliferative Neoplasms Research and Treatment (IWG-MRT) criteria.
3. JAKi naïve or previously treated with either ruxolitinib or fedratinib for PMF or Post-PV/ET myelofibrosis for ≥90 days, or ≥28 days if JAKi therapy is complicated by RBC transfusion requirement of ≥4 units in 8 weeks, or Grade 3/4 AEs of thrombocytopenia, anemia, or hematoma.
4. High risk, intermediate-2, or intermediate-1 risk as defined by Dynamic International Prognostic Scoring System (DIPSS) \[Passamonti, 2010\] or DIPSS-plus \[Gangat, 2011\].
5. TD defined as requiring RBC transfusion ≥4 units or HgB \< 8 g/dL in the 8 weeks prior to the first dose of study treatment. Only transfusions given when Hgb levels are ≤9.5 g/dL are counted towards TD. RBC transfusions given for clinically overt bleeding, or accident/injury (as assessed by the investigator) are not counted towards TD.

Exclusion Criteria

1. History of intestinal disease, inflammatory bowel disease, major gastric surgery, or other gastrointestinal conditions (e.g., uncontrolled nausea, vomiting, malabsorption syndrome) likely to alter absorption of study intervention or result in inability to swallow oral medications.
2. Participants with an invasive malignancy or history of invasive malignancy other than the disease under study within the last 5 years.
3. Known clinically significant anemia due to iron, vitamin B12, or folate deficiencies, or autoimmune or hereditary hemolytic anemia, gastrointestinal bleeding, or thalassemia.
4. Uncontrolled intercurrent illness:

1. Active uncontrolled infection (participants receiving outpatient antibacterial and/or antiviral treatments for infection that is under control or as infection prophylaxis may be included in the trial);
2. Uncontrolled acute and chronic liver disease (e.g., Child-Pugh score ≥10) OR has current unstable liver or biliary disease per investigator assessment defined by the presence of ascites, encephalopathy, coagulopathy, hypoalbuminemia, esophageal or gastric varices, persistent jaundice, or cirrhosis. NOTE: Stable chronic liver disease (including Gilbert's syndrome or asymptomatic gallstones) is acceptable if participant otherwise meets entry criteria.
5. Uncontrolled hypertension, defined as repeated elevations of systolic blood pressure ≥140 mmHg or diastolic blood pressure ≥90 mmHg, that is not resolved at the time of the first dose of study treatment.
6. Any of the following in conditions within 6 months prior to the first dose of study intervention:

1. Unstable angina pectoris; OR
2. Symptomatic congestive heart failure; OR
3. Uncontrolled cardiac arrhythmia
7. QTc interval \>450 msec or QTc \>480 msec for participants with bundle branch block.
8. Participants with stroke, deep venous thrombosis, pulmonary or arterial embolism within 6 months prior to the first dose of study intervention.
9. History of porphyria.
10. Presence of peripheral neuropathy ≥Grade 2 per CTCAE v5.0.
11. Use of the following treatments within the time periods noted NOTE: All active anti-MF therapy must discontinue at least 1 week prior to the start of baseline MFSAF recording (Study Day -7):

1. Active anti-MF therapy within 28 days or 5 half-lives, whichever is shorter (exception is prior JAKi therapy).
2. Steroid use for the treatment of myelofibrosis is prohibited within 14 days prior to the first dose of study treatment until discontinuation of study treatment. Supportive care including steroids for non-myelofibrosis indications may be used.
3. Potent cytochrome P450 3A4 (CYP3A4) inducers, except for rifampin and rifampicin, within 14 days prior to the first dose of study intervention.
4. Any prior investigational agent for myelofibrosis within 4 weeks prior to the first dose of study treatment.
5. Erythropoiesis stimulating agent (ESA) within 4 weeks prior to the first dose of study treatment.
6. Splenic irradiation within 3 months prior to the first dose of study treatment.
12. Prior treatment with MMB.
13. Prior treatment with luspatercept or sotatercept.
14. Prior splenectomy.
15. Inability or unwillingness to comply with the protocol restrictions on myelofibrosis therapy and other medications prior to and during study treatment.
16. Unresolved non-hematologic toxicities from prior therapies that are \>Grade 1 per CTCAE v5.0 unless otherwise specified.
17. Known positive status for human immunodeficiency virus (HIV).
18. Hepatitis A, B, or C status as defined below:

1. Chronic active or acute viral hepatitis A.
2. Active Hepatitis B infection indicated by the presence of hepatitis B surface antigen (HBsAg) at screening or within 3 months prior to the first dose of study intervention.
3. Positive hepatitis C antibody test result at screening or within 3 months before the first dose of study intervention. NOTE: Participants with positive hepatitis C antibody due to prior resolved disease can be enrolled, only if a confirmatory negative hepatitis C ribonucleic acid (RNA) test is obtained.
19. Women who are already pregnant or lactating.
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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GlaxoSmithKline

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Locations

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GSK Investigational Site

Nashville, Tennessee, United States

Site Status RECRUITING

GSK Investigational Site

Toronto, Ontario, Canada

Site Status RECRUITING

GSK Investigational Site

Montreal, Quebec, Canada

Site Status RECRUITING

GSK Investigational Site

Angers, , France

Site Status RECRUITING

GSK Investigational Site

Brest, , France

Site Status RECRUITING

GSK Investigational Site

Lyon, , France

Site Status RECRUITING

GSK Investigational Site

Nice, , France

Site Status RECRUITING

GSK Investigational Site

Nîmes, , France

Site Status RECRUITING

GSK Investigational Site

Paris, , France

Site Status RECRUITING

GSK Investigational Site

Poitiers, , France

Site Status RECRUITING

GSK Investigational Site

Florence, , Italy

Site Status RECRUITING

GSK Investigational Site

Roma, , Italy

Site Status RECRUITING

GSK Investigational Site

Málaga, , Spain

Site Status RECRUITING

GSK Investigational Site

Valencia, , Spain

Site Status RECRUITING

Countries

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United States Canada France Italy Spain

Central Contacts

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US GSK Clinical Trials Call Center

Role: CONTACT

877-379-3718

EU GSK Clinical Trials Call Center

Role: CONTACT

+44 (0) 20 89904466

Facility Contacts

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US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

Other Identifiers

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2024-518225-15

Identifier Type: REGISTRY

Identifier Source: secondary_id

220752

Identifier Type: -

Identifier Source: org_study_id