Safety and Pharmacokinetics Study of MBX 2109 in Adult Subjects With Normal and Impaired Renal Function

NCT ID: NCT06496217

Last Updated: 2025-10-28

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

Get a concise snapshot of the trial, including recruitment status, study phase, enrollment targets, and key timeline milestones.

Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

25 participants

Study Classification

INTERVENTIONAL

Study Start Date

2024-06-13

Study Completion Date

2025-09-04

Brief Summary

Review the sponsor-provided synopsis that highlights what the study is about and why it is being conducted.

Evaluate the Safety and Pharmacokinetics of MBX 2109 in Adult Subjects with Normal and Impaired Renal Function

Detailed Description

Dive into the extended narrative that explains the scientific background, objectives, and procedures in greater depth.

A Phase 1, Open-Label, Parallel-Group, Single-Dose Adaptive Study to Evaluate the Safety and Pharmacokinetics of MBX 2109 in Adult Subjects with Normal and Impaired Renal Function

Conditions

See the medical conditions and disease areas that this research is targeting or investigating.

Renal Impairment

Study Design

Understand how the trial is structured, including allocation methods, masking strategies, primary purpose, and other design elements.

Allocation Method

NA

Intervention Model

SEQUENTIAL

Primary Study Purpose

BASIC_SCIENCE

Blinding Strategy

NONE

Study Groups

Review each arm or cohort in the study, along with the interventions and objectives associated with them.

Single 900 µg dose of MBX 2109

A single, 900 µg dose of MBX 2109 will be administered subcutaneously in the abdomen

Group Type EXPERIMENTAL

MBX 2109

Intervention Type DRUG

Group 1: Subjects with mild renal impairment (eGFR ≥ 60 and \< 90 mL/min)

MBX 2109

Intervention Type DRUG

Group 2: Subjects with moderate renal impairment (eGFR ≥ 30 and \< 60 mL/min)

MBX 2109

Intervention Type DRUG

Group 3: Subjects with severe renal impairment (eGFR \< 30 mL/min), or kidney failure and not receiving dialysis

MBX 2109

Intervention Type DRUG

Group 4: Matched healthy subjects with normal renal function (eGFR ≥ 90 mL/min)

Interventions

Learn about the drugs, procedures, or behavioral strategies being tested and how they are applied within this trial.

MBX 2109

Group 1: Subjects with mild renal impairment (eGFR ≥ 60 and \< 90 mL/min)

Intervention Type DRUG

MBX 2109

Group 2: Subjects with moderate renal impairment (eGFR ≥ 30 and \< 60 mL/min)

Intervention Type DRUG

MBX 2109

Group 3: Subjects with severe renal impairment (eGFR \< 30 mL/min), or kidney failure and not receiving dialysis

Intervention Type DRUG

MBX 2109

Group 4: Matched healthy subjects with normal renal function (eGFR ≥ 90 mL/min)

Intervention Type DRUG

Eligibility Criteria

Check the participation requirements, including inclusion and exclusion rules, age limits, and whether healthy volunteers are accepted.

Inclusion Criteria

1. Willingness to adhere to the Protocol requirements as evidenced by a signed and dated informed consent form (ICF)
2. Subject is, as stated and in the opinion of the Investigator, willing and able to comply with the study drug regimen and all other study procedures and requirements, and is available for the duration of the study
3. Adult male or female, of at least 18 years of age, but not older than 80 years
4. Subject is willing to comply with the contraceptive requirements.
5. BMI ≥ 18.5 kg/m2 and \< 40.0 kg/m2 at the time of Screening.
6. Light-, non- or ex-smoker
7. Has suitable venous access for blood sampling

Subjects with Normal Renal Function (Group 4):
8. Medically healthy, in the opinion of an Investigator, with clinically insignificant Screening results (eg, laboratory profiles, medical history, vital signs, ECG, physical examination)
9. Normal renal function with eGFR ≥ 90 mL/min at Screening
10. Must match to the pooled mean age (± 10 years), BMI (within 20%) and gender (ratio should be similar) of mild, moderate, and severe (if applicable) renal impaired subjects at Screening.

Subjects with Mild, Moderate, and Severe Renal Impaired Function (Groups 1, 2, and 3):
11. Considered clinically stable in the opinion of an Investigator
12. Presence of mild renal impairment (eGFR ≥ 60 and \<90 mL/min), moderate renal impairment (eGFR ≥ 30 and \<60 mL/min), or severe renal impairment (eGFR \<30 mL/min) or kidney failure not receiving dialysis, at Screening: renal impairment should have been stable for at least 1 month prior to Screening.

Exclusion Criteria

1. Female who is lactating or breastfeeding
2. Female who is pregnant according to the pregnancy test at Screening or prior to study drug administration or planning to become pregnant before 90 days after the last study drug administration.
3. History of significant hypersensitivity to MBX 2109 or any related products (including excipients of the formulations) as well as severe hypersensitivity reactions (like angioedema) to any drugs.
4. History of, or positive test for hepatitis B surface antigen (HbsAg), hepatitis C antibody (HCV Ab), or HIV antibody, at Screening.
5. Presence or history of any disorder that could interfere with completion of the study based on the opinion of an Investigator.
6. Intake of MBX 2109, or any investigational product (IP) in the 28 days prior to study drug administration.
7. Have urinary incontinence without catheterization
8. Receipt of blood products within 3 months prior to study drug administration.
9. Donation of 50 mL or more of blood in the 28 days prior to study drug administration
10. Donated 500 mL or more of blood within 56 days prior to study drug administration
11. Donated plasma within 2 weeks prior to Screening or donated platelets within 6 weeks prior to Screening.
12. Immunization with a Coronavirus Disease 2019 (COVID-19) vaccine in the 14 days prior to the first study drug administration.
13. Scheduled immunization with a COVID-19 vaccine during the study that, in the opinion of an Investigator, could potentially interfere with subject participation, subject safety, study results, or any other reason.
14. Use of St. John's wort in the 28 days prior to the first study drug administration.
15. Inclusion in a previous group for this clinical study
16. Any skin condition and/or tattoo that may interfere with the injection site evaluation.

Subjects with Normal Renal Function (Group 4):
17. Presence of significant gastrointestinal, liver, or kidney disease, or any other conditions known to interfere with the absorption, distribution, metabolism, or excretion of drugs or known to potentiate or predispose to undesired effects.
18. History of significant gastrointestinal, liver, or kidney disease that may affect drug bioavailability.
19. Presence of significant cardiovascular, pulmonary, hematologic, neurological, psychiatric, endocrine, immunologic, or dermatologic disease.
20. Presence of clinically significant ECG abnormalities at the Screening visit, as defined by medical judgment.
21. Positive test result for alcohol and/or drugs of abuse at Screening or prior to the first study drug administration.
22. Supine or semi-supine blood pressure below 90/50 mmHg at the Screening visit
23. Supine or semi-supine blood pressure higher than 140/90 mmHg at the Screening visit (blood pressure readings greater than 140/90 mmHg may be retested if completed thought to be influenced by stress, at the discretion of the Investigator).
24. Supine or semi-supine pulse rate less than 40 beats per minute (bpm) or more than 100 bpm at Screening.
25. Any clinically significant illness in the 28 days before Day 1 of the study
26. Use of any prescription drugs (with the exception of hormonal contraceptives or hormone replacement therapy) in the 28 days before Day 1 of the study.
27. Use of over-the-counter (OTC) drugs and natural health products (eg, herbal remedies) at least 7 days (or 5-times the half-life of the drug, if longer) prior to study drug administration.
28. Use of any enzyme-modifying drugs, or drugs with effects on membrane transporters, including any strong cytochrome P450 3A4 and P-glycoprotein inducers and inhibitors in the previous 28 days before Day 1 of the study.

Subjects with Mild, Moderate, and Severe Renal Impaired Function (Groups 1, 2, and 3):
29. History of renal transplant
30. Supine or semi-supine blood pressure below 90/50 mmHg at the Screening visit.
31. Supine or semi-supine blood pressure higher than 180/110 mmHg at the Screening visit.
32. Supine or semi-supine pulse rate less than 45 bpm or more than 110 bpm at Screening.
33. History or presence, in the opinion of an Investigator, of significant clinically unstable respiratory, cardiovascular, pulmonary, hepatic, hematologic, gastrointestinal, endocrine, immunologic, dermatologic, neurologic, or psychiatric disease.
34. Presence of poorly controlled Type 1 or Type 2 diabetes as defined by Hemoglobin A1c \> 10%.
35. Presence of clinically significant physical examination, laboratory test, or ECG finding that, in the opinion of an Investigator and/or Sponsor, may interfere with any aspect of study conduct or interpretation of results.
36. Subjects requiring treatment for renal impairment or other chronic disease (eg, well controlled diabetes, hypertension) must be on a stable treatment plan (medicines, doses, and regimens) for at least 14 days (except insulin) prior to study drug administration and during the entire study.
37. Positive Screening of alcohol and/or drugs of abuse at Screening or prior to study drug administration unless results can be explained by a prescription medication.
Minimum Eligible Age

18 Years

Maximum Eligible Age

80 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

Meet the organizations funding or collaborating on the study and learn about their roles.

MBX Biosciences

INDUSTRY

Sponsor Role lead

Responsible Party

Identify the individual or organization who holds primary responsibility for the study information submitted to regulators.

Responsibility Role SPONSOR

Locations

Explore where the study is taking place and check the recruitment status at each participating site.

MBX Biosciences Investigational Site

Miami, Florida, United States

Site Status

MBX Bioscience Investigational Site

Tampa, Florida, United States

Site Status

MBX Biosciences Investigational Site

Minneapolis, Minnesota, United States

Site Status

Countries

Review the countries where the study has at least one active or historical site.

United States

Other Identifiers

Review additional registry numbers or institutional identifiers associated with this trial.

MBX-2H1003

Identifier Type: -

Identifier Source: org_study_id