Substudy 06C: A Study of Investigational Agents With Pembrolizumab (MK-3475) and Chemotherapy in Participants With First-Line Locally Advanced Unresectable/Metastatic Gastroesophageal Adenocarcinoma (MK-3475-06C/KEYMAKER-U06)

NCT ID: NCT06469944

Last Updated: 2026-01-05

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

Get a concise snapshot of the trial, including recruitment status, study phase, enrollment targets, and key timeline milestones.

Recruitment Status

RECRUITING

Clinical Phase

PHASE1/PHASE2

Total Enrollment

160 participants

Study Classification

INTERVENTIONAL

Study Start Date

2024-09-20

Study Completion Date

2029-04-12

Brief Summary

Review the sponsor-provided synopsis that highlights what the study is about and why it is being conducted.

This is a phase 1/2, multicenter, open-label umbrella platform study that will evaluate the safety and tolerability of investigational agents with pembrolizumab and fluoropyrimidine chemotherapy for the first-line (1L) treatment of participants with locally advanced unresectable or metastatic human epidermal growth factor receptor 2 (HER2)-negative gastric, gastroesophageal junction, or esophageal adenocarcinoma.

This substudy will have two phases: a safety lead-in phase and an efficacy phase. The safety lead-in phase will be used to evaluate the safety and tolerability, and to establish a recommended Phase 2 dose (RP2D) for investigational agents in combination with chemotherapy and immunotherapy. There is no formal hypothesis in this study.

Detailed Description

Dive into the extended narrative that explains the scientific background, objectives, and procedures in greater depth.

The master protocol is MK-3475-U06.

Conditions

See the medical conditions and disease areas that this research is targeting or investigating.

Gastroesophageal Junction Gastroesophageal Adenocarcinoma Esophageal Neoplasms Esophageal Cancer

Study Design

Understand how the trial is structured, including allocation methods, masking strategies, primary purpose, and other design elements.

Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

Review each arm or cohort in the study, along with the interventions and objectives associated with them.

Pembrolizumab plus Chemotherapy

Participants will receive pembrolizumab 400 mg via intravenous (IV) injection on day 1 of every 6 week cycle (Q6W) for up to 18 cycles (up to \~2 years) AND investigator's choice of CAPOX chemotherapy (capecitabine 1000 mg/m\^2 orally twice daily for 14 days every 3 weeks (Q3W) and oxaliplatin 130 mg/m\^2 via IV infusion Q3W) OR mFOLFOX6 chemotherapy (oxaliplatin 85 mg/m\^2 via IV infusion Q3W; 5-Fluorouracil (5-FU) 400 mg/\^2 via bolus IV plus 2400 mg/m\^2 continuous IV once every 2 weeks (Q2W); and leucovorin 400 mg/m\^2 via IV infusion Q2W OR levoleucovorin 200 mg/m\^2 Q2W).

Group Type ACTIVE_COMPARATOR

Pembrolizumab

Intervention Type BIOLOGICAL

Administered via intravenous (IV) infusion.

Capecitabine

Intervention Type DRUG

Administered via oral tablet.

Leucovorin

Intervention Type DRUG

Administered via IV infusion.

Levoleucovorin

Intervention Type DRUG

Administered via IV infusion.

5-Fluorouracil (5-FU)

Intervention Type DRUG

Administered via IV infusion

Oxaliplatin

Intervention Type DRUG

Administered via IV infusion

Pembrolizumab plus Sacituzumab Tirumotecan plus Chemotherapy

Participants will receive sacituzumab tirumotecan via IV infusion on Days 1, 15, and 29 Q6W until discontinuation, pembrolizumab 400 mg via IV injection on day 1 Q6W for up to 18 cycles (up to \~2 years) AND investigator's choice of capecitabine 1000 mg/m\^2 orally twice daily for 14 days Q3W OR 5-FU 400 mg/\^2 via bolus IV plus 2400 mg/m\^2 continuous IV once Q2W AND leucovorin 400 mg/m\^2 via IV infusion Q2W OR levoleucovorin 200 mg/m\^2 Q2W.

Group Type EXPERIMENTAL

Pembrolizumab

Intervention Type BIOLOGICAL

Administered via intravenous (IV) infusion.

Sacituzumab Tirumotecan (sac-TMT)

Intervention Type BIOLOGICAL

Administered via IV infusion.

Capecitabine

Intervention Type DRUG

Administered via oral tablet.

Leucovorin

Intervention Type DRUG

Administered via IV infusion.

Levoleucovorin

Intervention Type DRUG

Administered via IV infusion.

5-Fluorouracil (5-FU)

Intervention Type DRUG

Administered via IV infusion

Pembrolizumab plus Patritumab Deruxtecan plus Chemotherapy

Participants will receive patritumab deruxtecan via IV infusion on Days 1 and 22 Q6W until discontinuation, pembrolizumab 400 mg via IV injection on day 1 Q6W for up to 18 cycles (up to \~2 years) AND investigator's choice of capecitabine 1000 mg/m\^2 orally twice daily for 14 days Q3W OR 5-FU 400 mg/\^2 via bolus IV plus 2400 mg/m\^2 continuous IV once Q2W AND leucovorin 400 mg/m\^2 via IV infusion Q2W OR levoleucovorin 200 mg/m\^2 Q2W.

Group Type EXPERIMENTAL

Pembrolizumab

Intervention Type BIOLOGICAL

Administered via intravenous (IV) infusion.

Capecitabine

Intervention Type DRUG

Administered via oral tablet.

Leucovorin

Intervention Type DRUG

Administered via IV infusion.

Levoleucovorin

Intervention Type DRUG

Administered via IV infusion.

5-Fluorouracil (5-FU)

Intervention Type DRUG

Administered via IV infusion

Patritumab Deruxtecan

Intervention Type BIOLOGICAL

Administered via IV infusion

Interventions

Learn about the drugs, procedures, or behavioral strategies being tested and how they are applied within this trial.

Pembrolizumab

Administered via intravenous (IV) infusion.

Intervention Type BIOLOGICAL

Sacituzumab Tirumotecan (sac-TMT)

Administered via IV infusion.

Intervention Type BIOLOGICAL

Capecitabine

Administered via oral tablet.

Intervention Type DRUG

Leucovorin

Administered via IV infusion.

Intervention Type DRUG

Levoleucovorin

Administered via IV infusion.

Intervention Type DRUG

5-Fluorouracil (5-FU)

Administered via IV infusion

Intervention Type DRUG

Oxaliplatin

Administered via IV infusion

Intervention Type DRUG

Patritumab Deruxtecan

Administered via IV infusion

Intervention Type BIOLOGICAL

Other Intervention Names

Discover alternative or legacy names that may be used to describe the listed interventions across different sources.

MK-3475 Keytruda® MK-2870 SKB264 XELODA calcium folinate folinic acid WELLCOVORIN® calcium levofolinate levofolinic acid FUSILEV® ADRUCIL® HER3-DXd MK-1022 U3-1402

Eligibility Criteria

Check the participation requirements, including inclusion and exclusion rules, age limits, and whether healthy volunteers are accepted.

Inclusion Criteria

* Has histologically and/or cytologically confirmed diagnosis of previously untreated locally advanced unresectable or metastatic first-line (1L) gastroesophageal adenocarcinoma
* Is not expected to require tumor resection during the treatment course
* Tumor tissue must be confirmed as negative for human epidermal growth factor receptor 2 (HER2) expression as classified by American Society of Clinical Oncology/College of American Pathologists (ASCO-CAP) guidelines
* Core/excisional biopsy of a tumor lesion not previously irradiated has been provided
* Participants who have adverse events (AEs) due to previous anticancer therapies must have recovered to ≤Grade 1 or baseline
* Participants with endocrine-related AEs who are adequately treated with hormone replacement therapy are eligible
* Has adequate organ function
* Has measurable disease per Response Evaluation Criteria in Solid Tumors Version 1.1 (RECIST 1.1) as determined by the local site investigator/radiology assessment and verified by blinded independent central review (BICR)
* Has Eastern Cooperative Oncology Group (ECOG) performance status of 0 or 1 within 3 days prior to the first dose of study intervention
* Has a life expectancy of at least 6 months
* Participants who are hepatitis B surface antigen (HBsAg) positive are eligible if they have received Hepatitis B Virus (HBV) antiviral therapy for at least 4 weeks, and have undetectable HBV viral load prior to allocation/randomization
* Participants with history of Hepatitis C Virus (HCV) infection are eligible if HCV viral load is undetectable at screening
* Human Immunodeficiency Virus (HIV)-infected participants must have well controlled HIV on antiretroviral therapy

Exclusion Criteria

* Has squamous cell or undifferentiated gastroesophageal cancer.
* Has had previous therapy for locally advanced unresectable or metastatic gastric/gastroesophageal junction (GEJ)/esophageal adenocarcinoma
* Has experienced weight loss \>20% over 3 months before the first dose of study intervention
* Has a history of documented severe dry eye syndrome, severe Meibomian gland disease and/or blepharitis, or severe corneal disease that prevents/delays corneal healing
* Has Grade ≥2 peripheral neuropathy
* Has active inflammatory bowel disease requiring immunosuppressive medication or previous history of inflammatory bowel disease
* Has uncontrolled, significant cardiovascular disease or cerebrovascular disease within 6 months preceding study intervention
* Has accumulation of pleural, ascitic, or pericardial fluid requiring drainage or diuretic drugs within 2 weeks prior to enrollment
* Has history of human immunodeficiency virus (HIV) infection with Kaposi's sarcoma and/or Multicentric Castleman's Disease
* Has received prior treatment with a trophoblast antigen 2 (TROP2)-targeted or anti-human epidermal growth factor receptor 3 (HER3) targeted agents
* Has received prior treatment with a topoisomerase I inhibitor-based antibody-drug conjugate (ADC) and/or a topoisomerase I inhibitor-based chemotherapy
* Has received prior systemic anticancer therapy within 4 weeks before the first dose of study intervention
* Has received prior therapy with an anti-Programmed Cell Death Protein 1 (PD-1), anti-Programmed Cell Death-Ligand 1 (PD-L1), anti-Programmed Cell Death-Ligand 2 (PD-L2) agent or with an agent directed to another stimulatory or co-inhibitory T-cell receptor (TCR)
* Has received prior radiotherapy within 2 weeks of start of study intervention, or has radiation related toxicities, requiring corticosteroids
* Has received a live or live-attenuated vaccine within 30 days before the first dose of study intervention
* Has received a strong inducer/inhibitor of CYP3A4 that cannot be discontinued
* Has received an investigational agent or has used an investigational device within 4 weeks prior to study intervention administration
* Has diagnosis of immunodeficiency or is receiving chronic systemic steroid therapy or any other form of immunosuppressive therapy within 7 days prior to the first dose of study intervention
* Has known additional malignancy that is progressing or has required active treatment within the past 3 years
* Has known active central nervous system (CNS) metastases and/or carcinomatous meningitis
* Has Severe hypersensitivity (≥Grade 3) to pembrolizumab, sacituzumab tirumotecan, patritumab deruxtecan, or other biologic therapy, chemotherapy (ie, oxaliplatin, fluorouracil, capecitabine), leucovorin, levoleucovorin, or any of their excipients
* Has active autoimmune disease that has required systemic treatment in the past 2 years
* Has history of (noninfectious) pneumonitis or interstitial lung disease (ILD) that required steroids or has current pneumonitis or ILD, or where suspected ILD or pneumonitis cannot be ruled out by imaging at screening
* Has an active infection requiring systemic therapy
* Has concurrent active hepatitis B (defined as Hepatitis B surface antigen \[HBsAg\] positive and/or detectable HBV DNA) and hepatitis C virus (defined as anti-hepatitis C virus \[HCV\] Ab positive and detectable HCV ribonucleic acid \[RNA\] infection or a known history of hepatitis B and/or C infection
* Has history or current evidence of any condition, therapy, laboratory abnormality, or other circumstance that might confound the results of the study or interfere with the participant's ability to cooperate with the requirements of the study
* Has gastrointestinal (GI) obstruction, poor oral intake, or difficulty in taking oral medication
* Has poorly controlled diarrhea
* Has had a major surgery or significant traumatic injury within 4 weeks before the first dose of study intervention
* Has history of allogeneic tissue/solid organ transplant
* Has not adequately recovered from major surgery or has ongoing surgical complications
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

Meet the organizations funding or collaborating on the study and learn about their roles.

Merck Sharp & Dohme LLC

INDUSTRY

Sponsor Role lead

Responsible Party

Identify the individual or organization who holds primary responsibility for the study information submitted to regulators.

Responsibility Role SPONSOR

Principal Investigators

Learn about the lead researchers overseeing the trial and their institutional affiliations.

Medical Director

Role: STUDY_DIRECTOR

Merck Sharp & Dohme LLC

Locations

Explore where the study is taking place and check the recruitment status at each participating site.

University of Arizona Cancer Center-University of Arizona Cancer Center ( Site 6927)

Tucson, Arizona, United States

Site Status RECRUITING

UCLA Hematology/Oncology - Santa Monica ( Site 6905)

Los Angeles, California, United States

Site Status RECRUITING

Norton Hospital-Norton Cancer Institute - Downtown ( Site 6900)

Louisville, Kentucky, United States

Site Status COMPLETED

The Cancer and Hematology Centers ( Site 6912)

Grand Rapids, Michigan, United States

Site Status RECRUITING

Hematology-Oncology Associates of Central NY, P.C. ( Site 6925)

East Syracuse, New York, United States

Site Status RECRUITING

Columbia University Irving Medical Center-CUIMC Herbert Irving Comprehensive Cancer Center Clinical ( Site 6907)

New York, New York, United States

Site Status COMPLETED

UPMC Hillman Cancer Center-UPMC ( Site 6904)

Pittsburgh, Pennsylvania, United States

Site Status RECRUITING

University of Texas MD Anderson Cancer Center ( Site 6920)

Houston, Texas, United States

Site Status RECRUITING

Liga Norte Riograndense Contra o Câncer ( Site 6303)

Natal, Rio Grande do Norte, Brazil

Site Status RECRUITING

Hospital Nossa Senhora da Conceição ( Site 6301)

Porto Alegre, Rio Grande do Sul, Brazil

Site Status RECRUITING

IBCC - Instituto Brasileiro de Controle do Câncer ( Site 6304)

São Paulo, , Brazil

Site Status RECRUITING

Clínica Puerto Montt ( Site 6409)

Port Montt, Los Lagos Region, Chile

Site Status RECRUITING

Centro de Investigación del Maule ( Site 6408)

Talca, Maule Region, Chile

Site Status RECRUITING

FALP-UIDO ( Site 6400)

Santiago, Region M. de Santiago, Chile

Site Status RECRUITING

Centro de Oncología de Precisión-Oncology ( Site 6404)

Santiago, Region M. de Santiago, Chile

Site Status RECRUITING

Clínica UC San Carlos de Apoquindo ( Site 6405)

Santiago, Region M. de Santiago, Chile

Site Status RECRUITING

Bradfordhill-Clinical Area ( Site 6401)

Santiago, Region M. de Santiago, Chile

Site Status RECRUITING

Bradford Hill Norte ( Site 6407)

Antofagasta, , Chile

Site Status RECRUITING

Beijing Cancer hospital-Digestive Oncology ( Site 5500)

Beijing, Beijing Municipality, China

Site Status RECRUITING

The 900th Hospital of the Joint Logistics Support Force of the Chinese People's Liberation Army ( Site 5501)

Fuzhou, Fujian, China

Site Status RECRUITING

The First Affiliated hospital of Xiamen University ( Site 5503)

Xiamen, Fujian, China

Site Status RECRUITING

Henan Cancer Hospital ( Site 5504)

Zhengzhou, Henan, China

Site Status RECRUITING

The First Affiliated Hospital of Nanchang University ( Site 5514)

Nanchang, Jiangxi, China

Site Status RECRUITING

Fudan University Shanghai Cancer Center ( Site 5513)

Shanghai, Shanghai Municipality, China

Site Status RECRUITING

Xinjiang Medical University Cancer Hospital - Urumqi ( Site 5506)

Ürümqi, Xinjiang, China

Site Status RECRUITING

Sir Run Run Shaw Hospital of Zhejiang University School of Medicine ( Site 5510)

Hangzhou, Zhejiang, China

Site Status RECRUITING

CHU-BREST Cavale Blanche ( Site 5104)

Brest, Finistere, France

Site Status RECRUITING

CIC. ( Site 5100)

Lille, Nord, France

Site Status RECRUITING

Pitie Salpetriere University Hospital-Hepato-Gastro-Enterology ( Site 5102)

Paris, Île-de-France Region, France

Site Status RECRUITING

Universitaetsklinikum Duesseldorf-Gastroenterology, Hepatology and Infectiology ( Site 6802)

Düsseldorf, North Rhine-Westphalia, Germany

Site Status RECRUITING

Facharztzentrum Eppendorf-Facharztzentrum Eppendorf ( Site 6807)

Hamburg, , Germany

Site Status RECRUITING

IRCCS - Istituto Romagnolo per lo Studio dei Tumori (IRST) "Dino Amadori"-Oncologia Medica ( Site 5207)

Meldola, Emilia-Romagna, Italy

Site Status RECRUITING

Fondazione IRCCS Istituto Nazionale dei Tumori-Struttura Complessa Oncologia Medica 1 ( Site 5200)

Milan, Lombardy, Italy

Site Status RECRUITING

Oslo universitetssykehus, Radiumhospitalet ( Site 6501)

Oslo, , Norway

Site Status RECRUITING

Asan Medical Center-Department of Oncology ( Site 5901)

Seoul, , South Korea

Site Status RECRUITING

Samsung Medical Center-Division of Hematology/Oncology ( Site 5900)

Seoul, , South Korea

Site Status RECRUITING

Hôpitaux Universitaires de Genève (HUG) ( Site 6701)

Geneva, Canton of Geneva, Switzerland

Site Status RECRUITING

Kantonsspital Graubünden-Medizin ( Site 6700)

Chur, Kanton Graubünden, Switzerland

Site Status RECRUITING

China Medical University Hospital ( Site 6007)

Taichung, , Taiwan

Site Status RECRUITING

National Cheng Kung University Hospital ( Site 6001)

Tainan, , Taiwan

Site Status RECRUITING

National Taiwan University Hospital-Oncology ( Site 6000)

Taipei, , Taiwan

Site Status RECRUITING

Taipei Veterans General Hospital ( Site 6005)

Taipei, , Taiwan

Site Status RECRUITING

Countries

Review the countries where the study has at least one active or historical site.

United States Brazil Chile China France Germany Italy Norway South Korea Switzerland Taiwan

Central Contacts

Reach out to these primary contacts for questions about participation or study logistics.

Toll Free Number

Role: CONTACT

1-888-577-8839

Facility Contacts

Find local site contact details for specific facilities participating in the trial.

Study Coordinator

Role: primary

520-621-2449

Study Coordinator

Role: primary

310-570-1453

Study Coordinator

Role: primary

888-577-8839

Study Coordinator

Role: primary

315-472-7504

Study Coordinator

Role: primary

816-898-9413

Study Coordinator

Role: primary

888-577-8839

Study Coordinator

Role: primary

+558440095595

Study Coordinator

Role: primary

+5551993590437

Study Coordinator

Role: primary

551144500300

Study Coordinator

Role: primary

56961687093

Study Coordinator

Role: primary

56712981241

Study Coordinator

Role: primary

56224205098

Study Coordinator

Role: primary

56225189885

Study Coordinator

Role: primary

56934271024

Study Coordinator

Role: primary

56229490970

Study Coordinator

Role: primary

56442023631

Study Coordinator

Role: primary

1-888-577-8839

Study Coordinator

Role: primary

0591-22859606

Study Coordinator

Role: primary

0592-2139767

Study Coordinator

Role: primary

400-0371-818

Study Coordinator

Role: primary

0791-86427234

Study Coordinator

Role: primary

(021)6417 5590

Study Coordinator

Role: primary

(+86) 0991-7819113

Study Coordinator

Role: primary

0571 8609 0073

Study Coordinator

Role: primary

33298223428

Study Coordinator

Role: primary

+33320445461

Study Coordinator

Role: primary

+331 42 16 10 41

Study Coordinator

Role: primary

+492118108751

Study Coordinator

Role: primary

+ 4940360352246

Study Coordinator

Role: primary

0543739100

Study Coordinator

Role: primary

0223903807

Study Coordinator

Role: primary

4723026600

Study Coordinator

Role: primary

+82230103217

Study Coordinator

Role: primary

82234101795

Study Coordinator

Role: primary

1-888-577-8839

Study Coordinator

Role: primary

1-888-577-8839

Study Coordinator

Role: primary

886422052121x15057

Study Coordinator

Role: primary

+88662353535x4559

Study Coordinator

Role: primary

+88623123456x267852

Study Coordinator

Role: primary

+88628717270x131

Related Links

Access external resources that provide additional context or updates about the study.

Other Identifiers

Review additional registry numbers or institutional identifiers associated with this trial.

MK-3475-06C

Identifier Type: OTHER

Identifier Source: secondary_id

KEYMAKER-06C

Identifier Type: OTHER

Identifier Source: secondary_id

2023-509307-33-00

Identifier Type: REGISTRY

Identifier Source: secondary_id

U1111-1299-8084

Identifier Type: REGISTRY

Identifier Source: secondary_id

3475-06C

Identifier Type: -

Identifier Source: org_study_id

More Related Trials

Additional clinical trials that may be relevant based on similarity analysis.