Beamion BCGC-1: A Study to Find a Suitable Dose of Zongertinib Used Alone and in Combination With Other Treatments to Test Whether it Helps People With Different Types of HER2+ Cancer That Has Spread

NCT ID: NCT06324357

Last Updated: 2025-11-12

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

RECRUITING

Clinical Phase

PHASE1/PHASE2

Total Enrollment

582 participants

Study Classification

INTERVENTIONAL

Study Start Date

2024-06-03

Study Completion Date

2029-09-28

Brief Summary

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This study is open to adults aged 18 years and older with different types of HER2+ cancer that has spread and cannot be removed by surgery. People can take part in this study if their tumours show HER2 aberrations and previous treatment was not successful. The purpose of this study is to find a suitable dose of zongertinib that people with different types of HER2+ cancer that has spread can tolerate best when taken together with trastuzumab deruxtecan (T-DXd), with trastuzumab emtansine (T-DM1), or with trastuzumab and capecitabine. Another purpose is to check whether zongertinib alone and in combination with other treatments can make tumours shrink. Zongertinib inhibits HER2. HER2 causes cancer cells to grow.

In this study, participants receive treatment in cycles. Study participants are treated with zongertinib alone or in combination with other treatments. This study has 2 parts. In Part 1, participants in different groups receive increasing doses of zongertinib. In Part 2, participants are put into different groups by chance. Each group receives a different dose of zongertinib. Every participant has an equal chance of being in each group.

During the study, the participants visit the study site regularly. In this study, researchers want to find the highest dose of zongertinib that participants can tolerate when taken together with other treatments. To find this out, researchers look at certain severe health problems that a number of participants have. The doctors regularly check the size of the tumour with imaging methods (CT/MRI) during the study. The doctors also regularly check participants' health and take note of any unwanted effects

Detailed Description

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Conditions

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Metastatic Breast Cancer Metastatic Gastric Adenocarcinoma Gastroesophageal Junction Adenocarcinoma Esophageal Adenocarcinoma

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

SEQUENTIAL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Phase Ib - Cohort A: zongertinib + Trastuzumab emtansine

Dose escalation (Phase Ib)

Group Type EXPERIMENTAL

Zongertinib

Intervention Type DRUG

Zongertinib

Trastuzumab emtansine

Intervention Type DRUG

Trastuzumab emtansine

Phase Ib - Cohort B: zongertinib + Trastuzumab deruxtecan

Dose escalation (Phase Ib)

Group Type EXPERIMENTAL

Zongertinib

Intervention Type DRUG

Zongertinib

Trastuzumab deruxtecan

Intervention Type DRUG

Trastuzumab deruxtecan

Phase Ib - Cohort C: zongertinib + Trastuzumab deruxtecan

Dose escalation (Phase Ib)

Group Type EXPERIMENTAL

Zongertinib

Intervention Type DRUG

Zongertinib

Trastuzumab deruxtecan

Intervention Type DRUG

Trastuzumab deruxtecan

Phase II - Cohort D: zongertinib + Trastuzumab emtansine

Dose optimization (Phase II).

Group Type EXPERIMENTAL

Zongertinib

Intervention Type DRUG

Zongertinib

Trastuzumab emtansine

Intervention Type DRUG

Trastuzumab emtansine

Phase II - Cohort E: zongertinib + Trastuzumab deruxtecan

Dose optimization (Phase II).

Group Type EXPERIMENTAL

Zongertinib

Intervention Type DRUG

Zongertinib

Trastuzumab deruxtecan

Intervention Type DRUG

Trastuzumab deruxtecan

Phase II - Cohort F: zongertinib + Trastuzumab deruxtecan

Dose optimization (Phase II).

Group Type EXPERIMENTAL

Zongertinib

Intervention Type DRUG

Zongertinib

Trastuzumab deruxtecan

Intervention Type DRUG

Trastuzumab deruxtecan

Phase Ib - Cohort G: zongertinib + trastuzumab + capecitabine

Dose escalation (Phase Ib)

Group Type EXPERIMENTAL

Zongertinib

Intervention Type DRUG

Zongertinib

Trastuzumab

Intervention Type DRUG

Herceptin®

Capecitabine

Intervention Type DRUG

Xeloda®

Phase Ib - Cohort K: zongertinib + trastuzumab

Dose escalation (Phase Ib)

Group Type EXPERIMENTAL

Zongertinib

Intervention Type DRUG

Zongertinib

Trastuzumab

Intervention Type DRUG

Herceptin®

Phase II - Cohort H: zongertinib + trastuzumab + capecitabine

Dose optimization (Phase II).

Group Type EXPERIMENTAL

Zongertinib

Intervention Type DRUG

Zongertinib

Trastuzumab

Intervention Type DRUG

Herceptin®

Capecitabine

Intervention Type DRUG

Xeloda®

Phase II - Cohort I: zongertinib

Dose optimization (Phase II).

Group Type EXPERIMENTAL

Zongertinib

Intervention Type DRUG

Zongertinib

Phase II - Cohort J: zongertinib + trastuzumab

Dose optimization (Phase II).

Group Type EXPERIMENTAL

Zongertinib

Intervention Type DRUG

Zongertinib

Trastuzumab

Intervention Type DRUG

Herceptin®

Phase II - Cohort I-ext: zongertinib

Extension Phase II

Group Type EXPERIMENTAL

Zongertinib

Intervention Type DRUG

Zongertinib

Phase II - Cohort J-ext: zongertinib + trastuzumab

Extension Phase II

Group Type EXPERIMENTAL

Zongertinib

Intervention Type DRUG

Zongertinib

Trastuzumab

Intervention Type DRUG

Herceptin®

Interventions

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Zongertinib

Zongertinib

Intervention Type DRUG

Trastuzumab deruxtecan

Trastuzumab deruxtecan

Intervention Type DRUG

Trastuzumab emtansine

Trastuzumab emtansine

Intervention Type DRUG

Trastuzumab

Herceptin®

Intervention Type DRUG

Capecitabine

Xeloda®

Intervention Type DRUG

Other Intervention Names

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BI 1810631, Hernexeos® T-DXd; Enhertu® T-DM1; Kadcyla®

Eligibility Criteria

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Inclusion Criteria

* Signed and dated written Informed consent form (ICF) in accordance with International Council for Harmonisation-Good Clinical Practice (ICH-GCP) and local legislation prior to admission to the trial.
* Patients ≥18 years of age or over the legal age of consent in countries where that is greater than 18 years at the time of signature of the ICF.
* Documented Human epidermal growth factor receptor 2 overexpressing and/or amplified (HER2+), metastatic breast cancer (mBC) or metastatic gastric adenocarcinoma, gastroesophageal junction adenocarcinoma, or esophageal adenocarcinoma (mGEAC).
* For dose optimization (Phase II): Patient must provide tumor tissue from locations not radiated prior to biopsy, if possible, collected through archival tissue.
* Documented investigator assessed progression after HER2-directed treatment (including treatment with trastuzumab deruxtecan (T-DXd) for non-T-DXd combination cohorts) for unresectable locally advanced or metastatic disease.
* Recovered from any previous therapy-related toxicity to ≤ Common Terminology Criteria for Adverse Events (CTCAE) Grade 1 at start of treatment (except for alopecia, stable sensory neuropathy, and hypothyroidism (patients on thyroid replacement therapy) which must be ≤ CTCAE Grade 2).
* Presence of at least one measurable lesion according to Response evaluation criteria in solid tumors (RECIST) 1.1, as determined by the local site investigator/radiology assessment.

Exclusion Criteria

* Previous or concomitant malignancies other than the one treated in this trial within the previous 2 years, which require current systemic therapy except:

* effectively treated non-melanoma skin cancers
* effectively treated carcinoma in situ of the cervix
* effectively treated ductal carcinoma in situ
* other effectively treated malignancy that is considered cured by local treatment
* History or presence of cardiovascular abnormalities such as uncontrolled hypertension, congestive heart failure New York Heart Association (NYHA) classification of ≥ III or IV, unstable angina or poorly controlled arrhythmia which are considered as clinically relevant by the investigator. Myocardial infarction (or troponin levels consistent with myocardial infarction within 28 days of randomization), stroke, or pulmonary embolism within 6 months prior to randomization.
* Any clinically important abnormalities (as assessed by the investigator) in rhythm, conduction, or morphology of resting electrocardiograms, e.g. complete left bundle branch block, third degree heart block.
* Mean resting corrected QT interval (QT interval corrected for heart rate by Fridericia´s formula (QTcF)) \>470 msec.
* Any factors that increase the risk of QT interval corrected for heart rate (QTc) prolongation or risk of arrhythmic events such as heart failure, hypokalemia, congenital long QT syndrome, personal or family history of long QT syndrome or unexplained sudden death under 40 years-of-age.
* Ejection fraction \<50% or the lower limit of normal of the institutional standard within 28 days prior to randomization.
* Women who are pregnant or nursing or who plan to become pregnant or nurse during the trial or within 7 months after the last dose of trial treatment with T-DXd, T-DM1, trastuzumab or capecitabine and trastuzumab.
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Boehringer Ingelheim

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Locations

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Mayo Clinic-Arizona

Phoenix, Arizona, United States

Site Status NOT_YET_RECRUITING

The Oncology Institute of Hope and Innovation

Cerritos, California, United States

Site Status NOT_YET_RECRUITING

Ellison Medical Institute

Los Angeles, California, United States

Site Status NOT_YET_RECRUITING

Valkyrie Clinical Trials

Los Angeles, California, United States

Site Status RECRUITING

University of California Los Angeles

Los Angeles, California, United States

Site Status NOT_YET_RECRUITING

University of California Irvine

Orange, California, United States

Site Status RECRUITING

Sharp Memorial Hospital

San Diego, California, United States

Site Status NOT_YET_RECRUITING

Yale University School of Medicine

New Haven, Connecticut, United States

Site Status RECRUITING

Mayo Clinic - Florida

Jacksonville, Florida, United States

Site Status NOT_YET_RECRUITING

H. Lee Moffitt Cancer Center and Research Institute

Tampa, Florida, United States

Site Status NOT_YET_RECRUITING

Community Health Network

Indianapolis, Indiana, United States

Site Status NOT_YET_RECRUITING

University of Iowa Hospitals and Clinics

Iowa City, Iowa, United States

Site Status NOT_YET_RECRUITING

Massachusetts General Hospital

Boston, Massachusetts, United States

Site Status NOT_YET_RECRUITING

Dana-Farber Cancer Institute

Boston, Massachusetts, United States

Site Status NOT_YET_RECRUITING

Mayo Clinic, Rochester

Rochester, Minnesota, United States

Site Status NOT_YET_RECRUITING

Memorial Sloan-Kettering Cancer Center

New York, New York, United States

Site Status NOT_YET_RECRUITING

Penn State Milton S. Hershey Medical Center

Hershey, Pennsylvania, United States

Site Status NOT_YET_RECRUITING

Avera Cancer Institute

Sioux Falls, South Dakota, United States

Site Status NOT_YET_RECRUITING

Baptist Cancer Center - Memphis

Memphis, Tennessee, United States

Site Status NOT_YET_RECRUITING

SCRI Oncology Partners

Nashville, Tennessee, United States

Site Status RECRUITING

Tennessee Oncology, Pllc

Nashville, Tennessee, United States

Site Status RECRUITING

The Methodist Hospital Research Institute

Houston, Texas, United States

Site Status NOT_YET_RECRUITING

Inova Schar Cancer Institute

Fairfax, Virginia, United States

Site Status NOT_YET_RECRUITING

Virginia Cancer Specialists, PC

Fairfax, Virginia, United States

Site Status RECRUITING

Fred Hutchinson Cancer Research Center

Seattle, Washington, United States

Site Status NOT_YET_RECRUITING

Cliniques Universitaires Saint-Luc

Brussels, , Belgium

Site Status NOT_YET_RECRUITING

Edegem - UNIV UZ Antwerpen

Edegem, , Belgium

Site Status RECRUITING

UZ Leuven

Leuven, , Belgium

Site Status RECRUITING

Hôpital Vivalia De Libramont

Libramont-Chevigny, , Belgium

Site Status RECRUITING

Centre Hospitalier Universitaire de Liège

Liège, , Belgium

Site Status RECRUITING

CHU UCL Namur

Namur, , Belgium

Site Status RECRUITING

Jilin Province Cancer Hospital

Changchun, , China

Site Status RECRUITING

The First Hospital of Jilin University

Changchun, , China

Site Status NOT_YET_RECRUITING

Sir Run Run Shaw Hospital, Zhejiang University, School of Medicine

Hangzhou, , China

Site Status RECRUITING

Harbin Medical University Cancer Hospital

Harbin, , China

Site Status RECRUITING

Jiangsu Province Hospital

Nanjing, , China

Site Status RECRUITING

Fudan University Shanghai Cancer Center

Shanghai, , China

Site Status RECRUITING

Tianjin Cancer Hospital

Tianjin, , China

Site Status RECRUITING

Henan Cancer Hospital

Zhengzhou, , China

Site Status RECRUITING

INS Bergonie

Bordeaux, , France

Site Status NOT_YET_RECRUITING

CTR François Baclesse

Caen, , France

Site Status NOT_YET_RECRUITING

CTR Georges-François Leclerc

Dijon, , France

Site Status NOT_YET_RECRUITING

CTR Leon Berard

Lyon, , France

Site Status NOT_YET_RECRUITING

INS Paoli-Calmettes

Marseille, , France

Site Status NOT_YET_RECRUITING

HOP Tenon

Paris, , France

Site Status NOT_YET_RECRUITING

CTR Eugène Marquis

Rennes, , France

Site Status NOT_YET_RECRUITING

Institut de Cancérologie de l'Ouest

Saint-Herblain, , France

Site Status NOT_YET_RECRUITING

Institut de Cancérologie de Strasbourg

Strasbourg, , France

Site Status NOT_YET_RECRUITING

INS Claudius Regaud IUCT-Oncopole

Toulouse, , France

Site Status NOT_YET_RECRUITING

INS Gustave Roussy

Villejuif, , France

Site Status NOT_YET_RECRUITING

Universitätsklinikum Carl Gustav Carus Dresden

Dresden, , Germany

Site Status NOT_YET_RECRUITING

Universitätsklinikum Erlangen

Erlangen, , Germany

Site Status NOT_YET_RECRUITING

Evang. Kliniken Essen-Mitte gGmbh

Essen, , Germany

Site Status NOT_YET_RECRUITING

Asklepios Kliniken GmbH & Co. KGaA

Hamburg, , Germany

Site Status NOT_YET_RECRUITING

Universitätsklinikum Mannheim GmbH

Mannheim, , Germany

Site Status NOT_YET_RECRUITING

Universitätsklinikum Ulm

Ulm, , Germany

Site Status NOT_YET_RECRUITING

Istituto Di Candiolo

Candiolo (TO), , Italy

Site Status NOT_YET_RECRUITING

Az.Osp. Universitaria "Ospedali Riuniti"

Foggia, , Italy

Site Status NOT_YET_RECRUITING

Istituto Scientifico Romagnolo

Meldola (FC), , Italy

Site Status NOT_YET_RECRUITING

Ospedale San Raffaele S.r.l.

Milan, , Italy

Site Status RECRUITING

Istituto Europeo di Oncologia

Milan, , Italy

Site Status RECRUITING

Humanitas Istituto Clinico Catanese S.p.A.

Misterbianco (CT), , Italy

Site Status NOT_YET_RECRUITING

Istituto Nazionale IRCCS Tumori Fondazione Pascale

Napoli, , Italy

Site Status NOT_YET_RECRUITING

Istituto Clinico Humanitas

Rozzano, , Italy

Site Status RECRUITING

Aichi Cancer Center Hospital

Aichi, Nagoya, , Japan

Site Status NOT_YET_RECRUITING

Hakuaikai Sagara Hospital

Kagoshima, , Japan

Site Status NOT_YET_RECRUITING

Tokai University Hospital

Kanagawa, Isehara, , Japan

Site Status NOT_YET_RECRUITING

Kanagawa Cancer Center

Kanagawa, Yokohama, , Japan

Site Status RECRUITING

National Cancer Center Hospital East

Kashiwa-shi, , Japan

Site Status RECRUITING

Kyoto University Hospital

Kyoto, Kyoto, , Japan

Site Status RECRUITING

Osaka International Cancer Institute

Osaka, , Japan

Site Status RECRUITING

Japanese Foundation for Cancer Research

Tokyo, Koto-ku, , Japan

Site Status RECRUITING

CHA Bundang Medical Center

Seongnam-si, , South Korea

Site Status NOT_YET_RECRUITING

Seoul National University Bundang Hospital

Seongnam-si, , South Korea

Site Status NOT_YET_RECRUITING

Severance Hospital, Yonsei University Health System

Seoul, , South Korea

Site Status NOT_YET_RECRUITING

Asan Medical Center

Seoul, , South Korea

Site Status NOT_YET_RECRUITING

Korea University Anam Hospital

Seoul, , South Korea

Site Status NOT_YET_RECRUITING

Seoul National University Hospital

Seoul, , South Korea

Site Status NOT_YET_RECRUITING

The Catholic University of Korea, Seoul St.Mary's Hospital

Seoul, , South Korea

Site Status NOT_YET_RECRUITING

Severance Hospital, Yonsei University Health System

Seoul, , South Korea

Site Status NOT_YET_RECRUITING

Hospital Teresa Herrera

A Coruña, , Spain

Site Status NOT_YET_RECRUITING

Hospital del Mar

Barcelona, , Spain

Site Status NOT_YET_RECRUITING

Hospital Universitari Vall D Hebron

Barcelona, , Spain

Site Status RECRUITING

Hospital Clínic de Barcelona

Barcelona, , Spain

Site Status RECRUITING

Hospital Duran i Reynals

L'Hospitalet de Llobregat, , Spain

Site Status NOT_YET_RECRUITING

Hospital General Universitario Gregorio Marañón

Madrid, , Spain

Site Status NOT_YET_RECRUITING

Clínica Universidad de Navarra - Madrid

Madrid, , Spain

Site Status RECRUITING

Fundación Jiménez Díaz

Madrid, , Spain

Site Status RECRUITING

Hospital Clínico San Carlos

Madrid, , Spain

Site Status NOT_YET_RECRUITING

Hospital Universitario 12 de Octubre

Madrid, , Spain

Site Status NOT_YET_RECRUITING

Hospital Universitario La Paz

Madrid, , Spain

Site Status NOT_YET_RECRUITING

CIO Clara Campal

Madrid, , Spain

Site Status RECRUITING

Hospital Universitario Virgen De La Macarena

Seville, , Spain

Site Status NOT_YET_RECRUITING

Instituto Valenciano de Oncología

Valencia, , Spain

Site Status NOT_YET_RECRUITING

Velindre Cancer Centre

Cardiff, , United Kingdom

Site Status NOT_YET_RECRUITING

St James's University Hospital

Leeds, , United Kingdom

Site Status NOT_YET_RECRUITING

St Bartholomew's Hospital

London, , United Kingdom

Site Status NOT_YET_RECRUITING

University College Hospital

London, , United Kingdom

Site Status NOT_YET_RECRUITING

Royal Free Hospital

London, , United Kingdom

Site Status NOT_YET_RECRUITING

The Christie

Manchester, , United Kingdom

Site Status NOT_YET_RECRUITING

Nottingham University Hospitals NHS Trust

Nottingham, , United Kingdom

Site Status NOT_YET_RECRUITING

Countries

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United States Belgium China France Germany Italy Japan South Korea Spain United Kingdom

Central Contacts

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Boehringer Ingelheim

Role: CONTACT

Phone: 1-800-243-0127

Email: [email protected]

Facility Contacts

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Boehringer Ingelheim

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References

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Hurvitz S, Simonelli M, Yarza R, Berz D, Kitano S, Del Conte G, Acosta Eyzaguirre D, Doger de Speville Uribe BG, Maier D, Erzen D, Aykut Yazgili S, Curigliano G, Deng T, Yan M, Zhang Q, Wang X, Nakayama I, Shitara K. Beamion BCGC-1: phase Ib/II trial of zongertinib for advanced HER2-positive breast or gastroesophageal cancers. Future Oncol. 2025 Oct 17:1-9. doi: 10.1080/14796694.2025.2569553. Online ahead of print.

Reference Type DERIVED
PMID: 41108088 (View on PubMed)

Other Identifiers

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1479-0012

Identifier Type: -

Identifier Source: org_study_id