Effect of Tegoprazan on Pharmacodynamics of Clopidogrel in Healthy Subjects

NCT ID: NCT06164834

Last Updated: 2023-12-11

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

NOT_YET_RECRUITING

Clinical Phase

PHASE1

Total Enrollment

48 participants

Study Classification

INTERVENTIONAL

Study Start Date

2023-12-05

Study Completion Date

2024-11-30

Brief Summary

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This study aims to evaluate the effects of tegoprazan or esomeprazole administered in combination with clopidogrel on the pharmacodynamics/Pharmacokinetics of clopidogrel in healthy adults

Detailed Description

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Evaluation Criteria:

* Primary outcome Pharmacodynamic assessments using P2Y12 assay
* Secondary outcome Pharmacokinetics assessments on Cmax,ss, Cmin,ss, Cavg,ss, AUCτ,ss, Tmax,ss, t1/2,ss, CLss/F, Vd,ss/F, and PTF of clopidogrel
* Safety assessments with adverse event monitoring including subjective/ objective symptoms, physical examination, vital signs, electrocardiogram, and laboratory test

Conditions

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Healthy

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

CROSSOVER

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Clopidogrel 75 mg

Oral administration of clopidogrel 75 mg tablet once daily for 7 days

Group Type ACTIVE_COMPARATOR

Clopidogrel 75 mg

Intervention Type DRUG

Clopidogrel 75 mg tablet

Clopidogrel 75 mg + Tegoprazan 25 mg

Oral administration of clopidogrel 75 mg tablet and tegoprazan 25 mg tablet once daily for 7 days

Group Type EXPERIMENTAL

Clopidogrel 75 mg

Intervention Type DRUG

Clopidogrel 75 mg tablet

Tegoprazan 25 mg

Intervention Type DRUG

Tegoprazan 25 mg tablet

Clopidogrel 75 mg + Esomeprazole 20 mg

Oral administration of clopidogrel 75 mg tablet and esomeprazole 20 mg tablet once daily for 7 days

Group Type EXPERIMENTAL

Clopidogrel 75 mg

Intervention Type DRUG

Clopidogrel 75 mg tablet

Esomeprazole 20mg

Intervention Type DRUG

Esomeprazole 20 mg tablet

Interventions

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Clopidogrel 75 mg

Clopidogrel 75 mg tablet

Intervention Type DRUG

Tegoprazan 25 mg

Tegoprazan 25 mg tablet

Intervention Type DRUG

Esomeprazole 20mg

Esomeprazole 20 mg tablet

Intervention Type DRUG

Other Intervention Names

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Plavix K-CAB Nexium

Eligibility Criteria

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Inclusion Criteria

* Healthy adults aged ≥ 19 years and ≤ 50 years on the date of the written informed consent
* Body weight of ≥ 55.0 kg and ≤ 90.0 kg, with body mass index (BMI) of ≥ 18.0 kg/m2 and ≤ 27.0 kg/m2 at the time of screening
* Is given a detailed explanation and fully understood the study, then voluntarily decided to participate and provided written informed consent before any screening procedure
* Negative for serum Helicobacter pylori antibodies
* Judged by the investigator to be eligible for this study based on physical examination, laboratory test, inquiry, etc.

Exclusion Criteria

* Presence or history of clinically significant liver, kidney, nervous system, respiratory system, endocrine system, blood and tumor, cardiovascular system, urinary system or psychiatric disease
* Presence or history of gastrointestinal disorder (gastrointestinal ulcer, gastritis, gastrospasm, gastroesophageal reflux disease, Crohn's disease, etc.) that may influence the safety and pharmacodynamic assessments of the investigational product and history of gastrointestinal surgery (except simple appendectomy and hernia surgery), hemostatic disorder or hemorrhage-related disease
* Hypersensitivity to drugs including the ingredients of the investigational product and other drugs (aspirin, antibiotics, etc.) or history of clinically significant hypersensitivity
* Positive result in serology tests (Hepatitis B test, hepatitis C test, human immunodeficiency virus (HIV) test, syphilis test)
* Blood total bilirubin, AST (GOT), and ALT (GPT) \> 1.5 x upper limit of normal range at the screening test
* Platelet, PT and aPTT levels outside the upper/lower limit of normal range by 10% at the screening test
* Systolic blood pressure is \< 90 mmHg or \> 139 mmHg, diastolic blood pressure \< 50 mmHg or \> 89 mmHg, or pulse rate is \< 45 beats/minute or \> 100 beats/minute when vital signs are measured in sitting position after resting for at least 3 minutes at the screening test
* Showing the following findings on ECG at the screening test: QTc \> 450 msec, PR interval \> 210 msec, QRS interval \> 120 msec, Other clinically significant findings
* P2Y12 Reaction Unit (PRU) outside the upper/lower limit of normal range by 10% as a result of P2Y12 assay at the screening test
* History of drug abuse or positive urine screening for drug abuse
* Considered ineligible to participate in the study by the investigator based on laboratory test results or other reasons
Minimum Eligible Age

19 Years

Maximum Eligible Age

50 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

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HK inno.N Corporation

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Seung Hwan Lee

Role: PRINCIPAL_INVESTIGATOR

Seoul National University Hospital, Dept. of Clinical Pharmacology

Locations

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Seoul National University Hospital, Clinical Trial Center

Seoul, , South Korea

Site Status

Countries

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South Korea

Central Contacts

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Eun Ji Kim

Role: CONTACT

Phone: 82-2-6477-0290

Email: [email protected]

Hee Hyun Kim

Role: CONTACT

Phone: 82-2-6477-0258

Email: [email protected]

Facility Contacts

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Seung Hwan Lee, MD, PhD

Role: primary

Other Identifiers

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IN_APA_123

Identifier Type: -

Identifier Source: org_study_id