A Study to Assess the Safety, Pharmacokinetics, and Anti-Tumor Activity of Oral HP518 in mCRPC Patients

NCT ID: NCT06155084

Last Updated: 2025-12-22

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

RECRUITING

Clinical Phase

PHASE1/PHASE2

Total Enrollment

84 participants

Study Classification

INTERVENTIONAL

Study Start Date

2023-12-26

Study Completion Date

2026-09-30

Brief Summary

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The overall objective of this Phase 1 study is to evaluate the safety, PK,and anti-tumor activity of daily oral dosing with HP518,selecting the RP2D of HP518 based on assessments of patients with progressive mCRPC in dose-escalation phase

Detailed Description

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This First in Human dose escalation and expansion study of HP518 in patients with progressive mCRPC after NHA and chemotherapy is being conducted not only to evaluate the safety and tolerability of orally administered HP518, but also to provide preliminary efficacy for the reference of future studies.

Conditions

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Metastatic Castration-resistant Prostate Cancer

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

SEQUENTIAL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Part 1 - Dose Escalation, 400mg/d (Cohort1)

Oral tablet(s), once daily in 28-day cycles

Group Type EXPERIMENTAL

HP518 - Dose Escalation

Intervention Type DRUG

Part 1: Dose escalation Daily oral dosage with the prescribed dose level based on Cohort

Part 1 - Dose Escalation 500mg/d (Cohort 2)

Oral tablet(s), once daily in 28-day cycles

Group Type EXPERIMENTAL

HP518 - Dose Escalation

Intervention Type DRUG

Part 1: Dose escalation Daily oral dosage with the prescribed dose level based on Cohort

Part 2 - Dose Expansion Oral tablet(s)

Oral tablet(s), once daily in 28-day cycles

Group Type EXPERIMENTAL

HP518 -Dose Expansion

Intervention Type DRUG

Part 2: Dose expansion Daily oral dosage with the highest dose with acceptable toxicity (RP2D) based on data from Part 1.

Interventions

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HP518 - Dose Escalation

Part 1: Dose escalation Daily oral dosage with the prescribed dose level based on Cohort

Intervention Type DRUG

HP518 - Dose Escalation

Part 1: Dose escalation Daily oral dosage with the prescribed dose level based on Cohort

Intervention Type DRUG

HP518 -Dose Expansion

Part 2: Dose expansion Daily oral dosage with the highest dose with acceptable toxicity (RP2D) based on data from Part 1.

Intervention Type DRUG

Other Intervention Names

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Part 1 - Dose Escalation Part 1 - Dose Escalation Part 2 - Dose Expansion Oral tablet(s)

Eligibility Criteria

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Inclusion Criteria

1. Male, age ≥18
2. Patients with androgen receptor (AR) ligand binding domain (LBD) activation mutations (the dose expansion part of stage II)
3. Has histologically confirmed adenocarcinoma of the prostate, but there are no known significant neuroendocrine differentiation or small cell characteristics.
4. Has metastatic disease documented by 2 or more bone lesions by bone scan or soft tissue disease progression observed by CT/MRI at the beginning of study.
5. the progression of the disease after receiving at least one new endocrine therapy and progressing with at least first-line chemotherapy.
6. Must have recovered from toxicities related to any prior treatments
7. Ongoing ADT with LHRH agonist/antagonist therapy or history of bilateral orchiectomy.
8. ECOG performance status score of 0 to 1.

Exclusion Criteria

1. Combination of research or commercially available drugs targeting AR
2. Has had any other anticancer treatments, including immunotherapy, chemotherapy, or radiotherapy (eg, 177LuPSMA-617, radium 223, PARP inhibitor) within 4 weeks prior to the first dose of HP518.
3. Has gastrointestinal disorder affecting absorption (e.g., gastrectomy).
4. Has significant cardiovascular disease.
Minimum Eligible Age

18 Years

Eligible Sex

MALE

Accepts Healthy Volunteers

No

Sponsors

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Hinova Pharmaceuticals Inc.

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Locations

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The Second Hospital Of Anhui Medical University

Hefei, Anhui, China

Site Status RECRUITING

Beijing Cancer Hospital

Beijing, Beijing Municipality, China

Site Status RECRUITING

Beijing Friendship Hospital, Capital Medical University

Beijing, Beijing Municipality, China

Site Status RECRUITING

Chongqing University Cancer Hospital

Chongqing, Chongqing Municipality, China

Site Status RECRUITING

The Second Affiliated Hospital Of Chongqing Medical University

Chongqing, Chongqing Municipality, China

Site Status RECRUITING

The First Affiliated Hospital Of Xiamen Univeristy

Xiamen, Fujian, China

Site Status NOT_YET_RECRUITING

Lanzhou University Second Hospital

Lanzhou, Gansu, China

Site Status RECRUITING

The Third Affiliated Hospital of Southern Medical University

Guangzhou, Guangdong, China

Site Status RECRUITING

The Affiliated Hospital Of Guizhou Medical University

Guiyang, Guizhou, China

Site Status RECRUITING

Henan Cancer Hospital

Zhengzhou, Henan, China

Site Status RECRUITING

Zhengzhou Central Hospital

Zhengzhou, Henan, China

Site Status RECRUITING

Tongji Hospital

Wuhan, Hubei, China

Site Status RECRUITING

Hunan Cancer Hospital

Changsha, Hunan, China

Site Status RECRUITING

The First Affiliated Hospital Of Nanchang University

Nanchang, Jiangxi, China

Site Status RECRUITING

Liaoning Cancer Hospital & Institute

Shenyang, Liaoning, China

Site Status RECRUITING

Shandong Provincial Hospital

Jinan, Shandong, China

Site Status RECRUITING

The Affiliated Hospital Of Qingdao University

Qingdao, Shandong, China

Site Status RECRUITING

Yantai Yuhuangding Hospital

Yantai, Shandong, China

Site Status RECRUITING

Shanghai Tenth People's Hospital

Shanghai, Shanghai Municipality, China

Site Status RECRUITING

The First Affiliated Hospital Of Xi'An Jiaotong Univeristy

Xi’an, Shanxi, China

Site Status RECRUITING

Sichuan Academy of Medical Science & Sichuan Provincial People's Hospital

Chengdu, Sichuan, China

Site Status RECRUITING

West China Hospital Of Sichuan University

Chengdu, Sichuan, China

Site Status RECRUITING

The Affiliated Hospital Of Southwest Medical University

Luzhou, Sichuan, China

Site Status RECRUITING

Mianyang Central Hospital

Mianyang, Sichuan, China

Site Status RECRUITING

The Second Affiliated Hospital Of Kunming Medical University

Kunming, Yunnan, China

Site Status RECRUITING

The Affiliated Hospital Of School Of Medicine Of Ningbo University

Ningbo, Zhejiang, China

Site Status RECRUITING

The First Affiliated Hospital of Wenzhou Medical University

Wenzhou, Zhejiang, China

Site Status RECRUITING

Countries

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China

Central Contacts

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Qianrong Xiang

Role: CONTACT

Phone: +86 28 8505 8465

Email: [email protected]

Other Identifiers

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HP518-01-01-03

Identifier Type: -

Identifier Source: org_study_id