68Ga-NOTA-PEG2-RM26 PET/CT, First in Man Study

NCT ID: NCT06147362

Last Updated: 2023-11-27

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

RECRUITING

Clinical Phase

PHASE1

Total Enrollment

50 participants

Study Classification

INTERVENTIONAL

Study Start Date

2022-06-01

Study Completion Date

2023-12-31

Brief Summary

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This is an open-label positron emission tomography/computed tomography (PET/CT) study to investigate the diagnostic performance and evaluation efficacy of 68Ga-NOTA-PEG2-RM26 in prostate cancer patients. A single dose of 2 MBq/kg of 68Ga-NOTA-PEG2-RM26 limited to 100-200 MBq per examination will be given intravenously. Visual and semiquantitative method will be used to assess PET/CT images.

Detailed Description

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The gastrin-releasing peptide receptor (GRPR), also known as bombesin receptor subtype II (BB2), is a member of the G protein-coupled receptor family of bombesin receptors. GRPR is over-expressed in various types of human tumors. RM26, a GRPR antagonist with high affinity, was discovered by peptide backbone modification of bombesin analogues.

To target gastrin-releasing peptide receptor in human neoplastic cells NOTA-PEG2-RM26 was synthesised and then labeled with 68Ga.

An open-label whole-body PET/ CT study was designed to investigate the safety and dosimetry of 68Ga-NOTA-PEG2-RM26 and to assess its clinical diagnostic value in patients with cancer.

Conditions

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Cancer

Study Design

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Allocation Method

NA

Intervention Model

SINGLE_GROUP

Approximately ten patients (with primary/recurrent or metastatic cancer) in each of the following six cancer groups, prostate cancer, breast cancer, colorectal cancer, gastrointestinal carcinoid, gastric cancer, and lung cancer, will be recruited and examined.
Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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68Ga-NOTA-PEG2-RM26

Participants will be injected with 2 MBq/kg of 68Ga-NOTA-PEG2-RM26 limited to 100-200 MBq and then undergo PET/CT examination.

Group Type EXPERIMENTAL

68Ga-NOTA-PEG2-RM26

Intervention Type DRUG

Single-dose 68Ga-NOTA-PEG2-RM26, a gastrin-releasing peptide receptor antagonist linked with a positron emitting radioisotope intravenously injected into participants before the PET/CT scans.

Interventions

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68Ga-NOTA-PEG2-RM26

Single-dose 68Ga-NOTA-PEG2-RM26, a gastrin-releasing peptide receptor antagonist linked with a positron emitting radioisotope intravenously injected into participants before the PET/CT scans.

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Primary/recurrent or metastatic cancer in: prostate cancer, breast cancer, colorectal cancer, gastrointestinal carcinoid, gastric cancer, or lung cancer
* Histopathological diagnosis
* Age 18 years or more and palliative disease OR age above 50 years
* Adequate bone marrow, hepatic and renal function, Eastern Cooperative Oncology Group Performance Status Scale 0 or 1 and a negative pregnancy test

Exclusion Criteria

* Age less than 18 years
* Less than 6 months since a clinically significant cardiovascular event such as myocardial infarction, unstable angina, angioplasty, bypass surgery, stroke or transient ischemic attack
* Congestive heart failure New York Heart Association class ≥ II
* Pregnant or breast-feeding women
* Patients with reproductive potential not implementing accepted and effective means of contraception
* Participation in any other clinical trial within the previous 4 weeks
* Unable to comply with study procedures (e.g., claustrophobia, low back pain not allowing the patient to lay down in the examination bed)
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Stockholm South General Hospital

OTHER

Sponsor Role collaborator

Uppsala University

OTHER

Sponsor Role collaborator

Karolinska University Hospital

OTHER

Sponsor Role lead

Responsible Party

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Jeffrey Yachnin M.D., PhD.

Section Head Early Clinical Trial Unit

Responsibility Role PRINCIPAL_INVESTIGATOR

Principal Investigators

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Jeffrey Yachnin, MD, PhD

Role: PRINCIPAL_INVESTIGATOR

Karolinska University Hospital

Locations

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Karolinska University Hospital

Stockholm, , Sweden

Site Status RECRUITING

Countries

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Sweden

Central Contacts

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Antonios Tzortzakakis, MD, PhD

Role: CONTACT

08-123 70 000

Annette Fransson-Andreo-Hernandez, PhD

Role: CONTACT

+468 517 753 74

Facility Contacts

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Antonios Tzortzakakis, MD, PhD

Role: primary

08-123 80 000

Other Identifiers

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EudraCT 2021-004980-28

Identifier Type: -

Identifier Source: org_study_id