A Study to Learn About the Study Medicine Called PF-07220060 in Combination With Fulvestrant in People With HR-positive, HER2-negative Advanced or Metastatic Breast Cancer Who Progressed After a Prior Line of Treatment

NCT ID: NCT06105632

Last Updated: 2025-12-16

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

ACTIVE_NOT_RECRUITING

Clinical Phase

PHASE2

Total Enrollment

333 participants

Study Classification

INTERVENTIONAL

Study Start Date

2024-01-09

Study Completion Date

2028-01-21

Brief Summary

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The purpose of this study is to learn about the safety and how effective the study medicine (PF-07220060) plus fulvestrant is compared to the study doctor's choice of treatment in people with advanced or metastatic breast cancer. Advanced cancer is the one that is unlikely to be cured or taken care of with treatment. Metastatic cancer is the one that has spread to other parts of the body.

This study is seeking female and male participants who:

* are 18 years of age or older;
* are hormone receptor (HR)-positive and human epidermal growth factor receptor 2 (HER2)-negative;
* have advanced or metastatic breast cancer after taking other treatments before this study;
* have not taken or need to take medications that are not allowed by the study protocol;
* do not have any medical or mental conditions that may increase the risk of study participation.

Half of the participants will take PF-07220060 two times daily by mouth along with fulvestrant. Fulvestrant will be given as a shot into the muscle. The other half will take the study doctor's choice of treatment which can either be:

* Fulvestrant alone taken as shot into the muscle.
* Everolimus along with exemestane taken once daily by mouth.

This study will compare the experiences of participants receiving the study medicine plus fulvestrant to those who are receiving the study doctor's choice of treatment. This will help decide if the study medicine is safe and effective.

Participants will receive study treatment and/or will be in the study until:

* imaging scans (such as an MRI and/or CT) show that their cancer is getting worse.
* the study doctor thinks the participant is no longer benefitting from the study medicine.
* has side effects that become too severe. A side effect is a reaction (expected or unexpected) to a medicine or treatment you take.
* the participant chooses to stop taking part.

Detailed Description

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Conditions

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Advanced or Metastatic Breast Cancer

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Arm A

PF-07220060 to be taken by mouth as a tablet in combination with fulvestrant (a solution for injection)

Group Type EXPERIMENTAL

PF-07220060 CDK4 inhibitor

Intervention Type DRUG

Experimental

Fulvestrant

Intervention Type DRUG

Experimental and Active comparator

Arm B

Investigator's choice of therapy of either:

* Fulvestrant alone (a solution for injection), or
* Everolimus in combination with exemestane, both a tablet to be taken by mouth.

Group Type ACTIVE_COMPARATOR

Fulvestrant

Intervention Type DRUG

Experimental and Active comparator

Everolimus

Intervention Type DRUG

Active Comparator

Exemestane

Intervention Type DRUG

Active Comparator

Interventions

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PF-07220060 CDK4 inhibitor

Experimental

Intervention Type DRUG

Fulvestrant

Experimental and Active comparator

Intervention Type DRUG

Everolimus

Active Comparator

Intervention Type DRUG

Exemestane

Active Comparator

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Histological confirmation of breast cancer with evidence of locally advanced or metastatic disease, which is not amenable to surgical resection or radiation therapy with curative intent.
* Documented estrogen receptor (ER) and/or progesterone receptor (PR)- positive tumor
* Documented HER2-negative tumor
* Able to provide a sufficient amount of representative formalin fixed, paraffin embedded (FFPE) tumor tissue specimen.
* Must have received CDK4/6i plus NSAI defined per study protocol. There must be documented PD during or after CDK4/6i treatment.
* Measurable disease or non-measurable bone only disease as defined by RECIST version 1.1.
* Eastern Cooperative Oncology Group (ECOG) Performance Status (PS) ≤2.

Exclusion Criteria

* Any medical or psychiatric condition that may increase the risk of study participation or make the participant inappropriate for the study.
* In visceral crisis at risk of immediately life-threatening complications in the short term.
* Known active uncontrolled or symptomatic central nervous system metastases, carcinomatous meningitis, or leptomeningeal disease.
* Prior treatment with any of the following:
* Everolimus or investigational anti-cancer agents in any setting
* Prior chemotherapy in the advanced setting
* Radiation within 2 weeks of randomization
* Current use or anticipated need for any prohibited food, supplements or concomitant medication(s) (ie, other anti-cancer therapies, other endocrine therapies, growth factors, chronic systemic corticosteroids, strong cytochrome P450 3A4/5 \[CYP3A4/5\] or uridine 5' diphosphate-glucuronosyltransferase 2B7 \[UGT2B7\] inhibitors and inducers, direct oral anticoagulants, proton pump inhibitors).
* Inadequate renal function, hepatic dysfunction, or hematologic abnormalities.
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Pfizer

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Pfizer CT.gov Call Center

Role: STUDY_DIRECTOR

Pfizer

Locations

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UCSF - John Muir Health Cancer Center Berkeley

Berkeley, California, United States

Site Status

Washington Hospital Healthcare System

Fremont, California, United States

Site Status

Hoag Health Center Irvine

Irvine, California, United States

Site Status

Hoag Hospital Irvine

Irvine, California, United States

Site Status

Eisenhower George and Julia Argyros Health Center

La Quinta, California, United States

Site Status

Keck Hospital of USC

Los Angeles, California, United States

Site Status

Los Angeles General Medical Center

Los Angeles, California, United States

Site Status

USC/Norris Comprehensive Cancer Center

Los Angeles, California, United States

Site Status

Hoag Memorial Hospital Presbyterian

Newport Beach, California, United States

Site Status

Eisenhower Health Center at South Palm Canyon

Palm Springs, California, United States

Site Status

Keck Medical Center of USC Pasadena

Pasadena, California, United States

Site Status

Eisenhower Medical Center

Rancho Mirage, California, United States

Site Status

Zuckerberg San Francisco General Hospital and Trauma Center

San Francisco, California, United States

Site Status

UCSF Medical Center at Mission Bay

San Francisco, California, United States

Site Status

UCSF Cancer Center San Mateo

San Mateo, California, United States

Site Status

Saint Vincent's Medical Center (SVMC)

Bridgeport, Connecticut, United States

Site Status

Danbury Hospital

Danbury, Connecticut, United States

Site Status

Hartford Hospital (HH)

Hartford, Connecticut, United States

Site Status

MidState Medical Center (MMC)

Meriden, Connecticut, United States

Site Status

Hartford Healthcare

New Britain, Connecticut, United States

Site Status

Norwalk Hospital

Norwalk, Connecticut, United States

Site Status

Hartford HealthCare Cancer Institute at The Hospital of Central Connecticut, Medical Arts Center

Plainville, Connecticut, United States

Site Status

Georgetown University Medical Center

Washington D.C., District of Columbia, United States

Site Status

MedStar Washington Hospital Center

Washington D.C., District of Columbia, United States

Site Status

Northwestern Memorial Hospital

Chicago, Illinois, United States

Site Status

NorthShore University HealthSystem

Chicago, Illinois, United States

Site Status

NorthShore University HealthSystem

Evanston, Illinois, United States

Site Status

NorthShore University HealthSystem

Glenview, Illinois, United States

Site Status

NorthShore University HealthSystem

Highland Park, Illinois, United States

Site Status

Intermountain Health St. Vincent Regional Hospital

Billings, Montana, United States

Site Status

Intermountain Health St. Vincent Regional Hospital - Cancer Centers of Montana

Billings, Montana, United States

Site Status

Cancer Care Specialists

Reno, Nevada, United States

Site Status

Vassar Brothers Medical Center

Poughkeepsie, New York, United States

Site Status

Memorial Hermann Cancer Center

Houston, Texas, United States

Site Status

Baylor Scott & White Medical Center - Round Rock

Round Rock, Texas, United States

Site Status

Aurora Health Center - Southern Lakes

Burlington, Wisconsin, United States

Site Status

Aurora Medical Centers - Grafton

Grafton, Wisconsin, United States

Site Status

Aurora BayCare Medical Center

Green Bay, Wisconsin, United States

Site Status

Aurora Health Center - Kenosha

Kenosha, Wisconsin, United States

Site Status

Aurora Health Center Milwaukee - Good Hope

Milwaukee, Wisconsin, United States

Site Status

Aurora St Luke's Medical Center

Milwaukee, Wisconsin, United States

Site Status

Aurora Medical Center - Summit

Summit, Wisconsin, United States

Site Status

Aurora Cancer Care

Wauwatosa, Wisconsin, United States

Site Status

CIPREC

Buenos Aires, Buenos Aires F.D., Argentina

Site Status

Organizacion Medica de Investigacion

CABA, Buenos Aires F.D., Argentina

Site Status

Fundación Cenit Para La Investigación En Neurociencias

CABA, Buenos Aires F.D., Argentina

Site Status

Clinica Viedma S. A

Viedma, Río Negro Province, Argentina

Site Status

Instituto de Oncología de Rosario

Rosario, Santa Fe Province, Argentina

Site Status

Centro Para la Atención Integral del Paciente Oncologico (CAIPO)

San Miguel de Tucumán, Tucumán Province, Argentina

Site Status

Centro de Investigaciones Metabólicas (CINME)

Buenos Aires, , Argentina

Site Status

Clínica Universitaria Reina Fabiola

Córdoba, , Argentina

Site Status

Fundación CORI para la Investigación y Prevención del Cáncer

La Rioja, , Argentina

Site Status

COE (Centro Oncológico de Excelencia)

San Juan, , Argentina

Site Status

Sanatorio Norte

Santiago del Estero, , Argentina

Site Status

Macquarie University

North Ryde, New South Wales, Australia

Site Status

Icon Cancer Centre Townsville

Rosslea, Queensland, Australia

Site Status

Instituto D'Or de Pesquisa e Ensino (IDOR) - Filial Pernambuco

Recife, Pernambuco, Brazil

Site Status

Liga Norte Riograndense Contra o Câncer

Natal, Rio Grande do Norte, Brazil

Site Status

ONCOSITE - Centro de Pesquisa Clinica em Oncologia

Ijuí, Rio Grande do Sul, Brazil

Site Status

Hospital São Lucas da PUCRS

Porto Alegre, Rio Grande do Sul, Brazil

Site Status

Fundação Pio XII - Hospital de Câncer de Barretos

Barretos, São Paulo, Brazil

Site Status

Centro de Oncologia - CEON+ - Unidade São Caetano do Sul

São Caetano do Sul, São Paulo, Brazil

Site Status

Hospital Esperança Recife: Pronto Atendimento 24h

Pernambuco, , Brazil

Site Status

Dr. Everett Chalmers Regional Hospital

Fredericton, New Brunswick, Canada

Site Status

Royal Victoria Regional Health Centre

Barrie, Ontario, Canada

Site Status

CIUSSS- saguenay-Lac-Saint-Jean

Chicoutimi, Quebec, Canada

Site Status

Jewish General Hospital

Montreal, Quebec, Canada

Site Status

Cancer Hospital Chinese Academy of Medical Science

Beijing, Beijing Municipality, China

Site Status

Beijing Cancer hospital

Beijing, Beijing Municipality, China

Site Status

The First People's Hospital of Foshan

Foshan, Guangdong, China

Site Status

Guangdong Provincial People's Hospital

Guangzhou, Guangdong, China

Site Status

Guangxi Medical University Affiliated Tumor Hospital

Nanning, Guangxi, China

Site Status

Harbin Medical University Cancer Hospital

Harbin, Heilongjiang, China

Site Status

Henan Cancer Hospital

Zhengzhou, Henan, China

Site Status

Tongji Hospital, Tongji Medical College of Huazhong University of Science and Technology

Wuhan, Hubei, China

Site Status

Hunan Cancer Hospital

Changsha, Hunan, China

Site Status

Jilin Province Tumor Hospital

Changchun, Jilin, China

Site Status

The First Hospital of Jilin University

Changchun, Jilin, China

Site Status

The First Hospital of China Medical University

Shenyang, Liaoning, China

Site Status

Fudan University Shanghai Cancer Center

Shanghai, Shanghai Municipality, China

Site Status

West China Hospital of Sichuan University

Chengdu, Sichuan, China

Site Status

Sir Run Run Shaw Hospital of Zhejiang University School of Medicine

Hangzhou, Zhejiang, China

Site Status

Zhejiang Cancer Hospital

Hangzhou, Zhejiang, China

Site Status

Kiran Hospital - Multi Super Speciality Hospital and Research Center

Surat, Gujarat, India

Site Status

Spandana Oncology Centre (SOC)

Bangalore, Karnataka, India

Site Status

Tata Memorial Hospital

Mumbai, Maharashtra, India

Site Status

Kims Kingsway Hospital

Nagpur, Maharashtra, India

Site Status

Apex Wellness Hospital

Nashik, Maharashtra, India

Site Status

Sahyadri Super Speciality Hospital

Pune, Maharashtra, India

Site Status

Bhakti Vedanta Hospital and Research Institute

Thāne, Maharashtra, India

Site Status

Rajiv Gandhi Cancer Institute And Research Centre

New Delhi, National Capital Territory of Delhi, India

Site Status

Rabin Medical Center

Petah Tikva, Central District, Israel

Site Status

Shaare Zedek Medical Center

Jerusalem, Jerusalem, Israel

Site Status

Rambam Health Care Campus

Haifa, Northern District, Israel

Site Status

Aichi Cancer Center Hospital

Nagoya, Aichi-ken, Japan

Site Status

Nagoya University Hospital

Nagoya, Aichi-ken, Japan

Site Status

Chiba cancer center

Chiba, Chiba, Japan

Site Status

National Hospital Organization Shikoku Cancer Center

Matsuyama, Ehime, Japan

Site Status

Gunma Prefectural Cancer Center

Otashi, Gunma, Japan

Site Status

National Hospital Organization Hokkaido Cancer Center

Sapporo, Hokkaido, Japan

Site Status

Tohoku University Hospital

Sendai, Miyagi, Japan

Site Status

Osaka International Cancer Institute

Osaka, Osaka, Japan

Site Status

Osaka University Hospital

Suita, Osaka, Japan

Site Status

Saitama Medical University International Medical Center

Hidaka, Saitama, Japan

Site Status

St. Luke's International Hospital

Chuo-ku, Tokyo, Japan

Site Status

The Cancer Institute Hospital of JFCR

Koto, Tokyo, Japan

Site Status

Hiroshima City Hiroshima Citizens Hospital

Hiroshima, , Japan

Site Status

Okayama University Hospital

Okayama, , Japan

Site Status

National Hospital Organization Osaka National Hospital

Osaka, , Japan

Site Status

Boca Clinical Trials Mexico S.C.

Guadajalara, Jalisco, Mexico

Site Status

Cryptex Investigación Clínica S.A. de C.V.

Cuauhtémoc, Mexico City, Mexico

Site Status

Mexico Centre for Clinical Research S.A de C.V

Mexico City, Mexico City, Mexico

Site Status

COI Centro Oncologico Internacional S.A.P.I. de C.V.

Mexico City, Mexico City, Mexico

Site Status

Filios Alta Medicina S.A. de C.V.

Monterrey, Nuevo León, Mexico

Site Status

Unidad de Investigación en Salud de Chihuahua, S.C.

Chihuahua City, , Mexico

Site Status

Oaxaca Site Management Organization S.C.

Oaxaca City, , Mexico

Site Status

Instituto Veracruzano en Investigación Clínica S.C.

Veracruz, , Mexico

Site Status

National Cancer Center

Goyang-si, Kyǒnggi-do, South Korea

Site Status

Seoul National University Bundang Hospital

Seongnam, Kyǒnggi-do, South Korea

Site Status

Ajou University Hospital

Suwon, Kyǒnggi-do, South Korea

Site Status

Pusan National University Hospital

Busan, Pusan-kwangyǒkshi, South Korea

Site Status

Seoul National University Hospital

Seoul, Seoul-teukbyeolsi [seoul], South Korea

Site Status

Kangbuk Samsung Hospital

Seoul, Seoul-teukbyeolsi [seoul], South Korea

Site Status

Asan Medical Center

Seoul, Seoul-teukbyeolsi [seoul], South Korea

Site Status

Gangnam Severance Hospital, Yonsei University Health System

Seoul, Seoul-teukbyeolsi [seoul], South Korea

Site Status

Samsung Medical Center

Seoul, Seoul-teukbyeolsi [seoul], South Korea

Site Status

Korea University Guro Hospital

Seoul, Seoul-teukbyeolsi [seoul], South Korea

Site Status

Keimyung University Dongsan Hospital

Daegu, Taegu-kwangyǒkshi, South Korea

Site Status

China Medical University Hospital

Taichung, , Taiwan

Site Status

National Cheng Kung University Hospital

Tainan, , Taiwan

Site Status

National Taiwan University Hospital

Taipei, , Taiwan

Site Status

Mackay Memorial Hospital

Taipei, , Taiwan

Site Status

Taipei Veterans General Hospital

Taipei, , Taiwan

Site Status

Koo Foundation Sun Yat-Sen Cancer Center

Taipei, , Taiwan

Site Status

Chang Gung Medical Foundation-Linkou Branch

Taoyuan District, , Taiwan

Site Status

Medipol Mega Universite Hastanesi

Stanbul, İ̇stanbul, Turkey (Türkiye)

Site Status

Acibadem Altunizade Hospital

Üsküdar / Stanbul, İ̇stanbul, Turkey (Türkiye)

Site Status

Gulhane Egitim Arastirma Hastanesi

Ankara, , Turkey (Türkiye)

Site Status

Dr. Abdurrahman Yurtaslan Ankara Onkoloji Egitim ve Arastırma Hastanesi

Ankara, , Turkey (Türkiye)

Site Status

Hacettepe Universite Hastaneleri

Ankara, , Turkey (Türkiye)

Site Status

Ultramar Medical Imaging Center

Ankara, , Turkey (Türkiye)

Site Status

Memorial Ankara Hastanesi

Ankara, , Turkey (Türkiye)

Site Status

Ultramar Medical Imaging Center

Ankara, , Turkey (Türkiye)

Site Status

Ankara Bilkent Şehir Hastanesi

Ankara, , Turkey (Türkiye)

Site Status

Ultramar Medical Imaging Center

Ankara, , Turkey (Türkiye)

Site Status

Dicle Üniversitesi

Diyarbakır, , Turkey (Türkiye)

Site Status

Marmara Universitesi Pendik Egitim Arastirma Hastanesi

Istanbul, , Turkey (Türkiye)

Site Status

Erciyes Universitesi Tıp Fakultesi Hastaneleri

Kayseri, , Turkey (Türkiye)

Site Status

Kocaeli Üniversitesi

Kocaeli, , Turkey (Türkiye)

Site Status

Necmettin Erbakan Meram Medical Fac.

Konya, , Turkey (Türkiye)

Site Status

Samsun Medical Park Hastanesi

Samsun, , Turkey (Türkiye)

Site Status

Imperial College Healthcare NHS Trust, Charing Cross Hospital

London, Hammersmith and Fulham, United Kingdom

Site Status

Sarah Cannon Research Institute UK

London, London, CITY of, United Kingdom

Site Status

The Royal Surrey County Hospital

Guildford, , United Kingdom

Site Status

The Christie NHS Foundation Trust

Manchester, , United Kingdom

Site Status

Countries

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United States Argentina Australia Brazil Canada China India Israel Japan Mexico South Korea Taiwan Turkey (Türkiye) United Kingdom

Related Links

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https://pmiform.com/clinical-trial-info-request?StudyID=C4391022

To obtain contact information for a study center near you, click here.

Other Identifiers

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2023-506487-13-00

Identifier Type: REGISTRY

Identifier Source: secondary_id

C4391022

Identifier Type: -

Identifier Source: org_study_id