A Study of Inlexisertib (DCC-3116) in Combination With Anticancer Therapies in Participants With Advanced Malignancies

NCT ID: NCT05957367

Last Updated: 2026-02-04

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

RECRUITING

Clinical Phase

PHASE1/PHASE2

Total Enrollment

94 participants

Study Classification

INTERVENTIONAL

Study Start Date

2023-09-28

Study Completion Date

2029-03-31

Brief Summary

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This is a Phase 1/2, multicenter, open-label (unless otherwise specified in a combination-specific module) study of inlexisertib in combination with anticancer therapies. Modules within the master protocol are defined according to different combinations of inlexisertib with other anticancer agents.

Detailed Description

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Conditions

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GIST

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

SEQUENTIAL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Dose Escalation (Part 1, Module A)

Escalation Module A Part 1 inlexisertib combination closed on January 8, 2024, with no participants enrolled.

Group Type EXPERIMENTAL

Inlexisertib

Intervention Type DRUG

Oral Tablet Formulation

Expansion (Part 2, Module A)

Expansion Module A Part 2 inlexisertib combination closed on January 8, 2024, with no participants enrolled.

Group Type EXPERIMENTAL

Inlexisertib

Intervention Type DRUG

Oral Tablet Formulation

Dose Escalation (Part 1, Module B)

Inlexisertib tablets in escalating dose cohorts in 28-day cycles will be administered in combination with ripretinib once daily (QD).

Group Type EXPERIMENTAL

Inlexisertib

Intervention Type DRUG

Oral Tablet Formulation

Ripretinib

Intervention Type DRUG

Oral Tablet Formulation

Expansion (Part 2, Module B)

Inlexisertib tablets will be administered in combination with ripretinib in 28-day cycles to evaluate preliminary efficacy in participants with 2nd-line advanced gastrointestinal stromal tumor (GIST).

Group Type EXPERIMENTAL

Inlexisertib

Intervention Type DRUG

Oral Tablet Formulation

Ripretinib

Intervention Type DRUG

Oral Tablet Formulation

Interventions

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Inlexisertib

Oral Tablet Formulation

Intervention Type DRUG

Ripretinib

Oral Tablet Formulation

Intervention Type DRUG

Other Intervention Names

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DCC-3116 QINLOCK, DCC-2618

Eligibility Criteria

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Inclusion Criteria

* Male or female ≥18 years of age
* Module A: Part 1 and Part 2:

Module A Part 1 and Part 2 inlexisertib combination closed on January 8, 2024, with no participants enrolled.

* Module B: Only for Part 1 (Safety/Dose-finding):

* Pathologically confirmed diagnosis of GIST with a KIT or platelet-derived growth factor receptor alpha (PDGFRA) mutation
* Must have progressed on at least one approved systemic regimen given in the locally advanced or metastatic setting or have documented intolerance to it
* Must not have received prior ripretinib treatment
* Module B: Only for Part 2 (Expansion)

* Pathologically confirmed GIST with documented mutation in KIT exon 11
* Must have progressed on imatinib given in the locally advanced or metastatic setting or have been intolerant to imatinib and may not have received additional systemic therapy for GIST
* Must have at least 1 measurable lesion according to Modified Response Evaluation Criteria in Solid Tumors (mRECIST)
* Must have a life expectancy of more than 3 months and an ECOG performance status of 0-1
* Adequate organ function and bone marrow reserve based on laboratory assessments performed at Screening
* Must provide a fresh tumor biopsy, if able

Exclusion Criteria

* Must not have received the following within the specified time periods prior to the first dose of study drug:

1. Medications, including anticancer therapies, that are known strong or moderate inhibitors or inducers of CYP3A4 or P-glycoprotein (P-gp) including certain herbal medications (eg, St. John's wort): 14 days or 5×the half-life of the medication (whichever is longer)
2. Other anticancer therapies and any investigational therapies with a known safety and PK profile: 14 days or 5×the half-life of the medication (whichever is shorter)
3. Investigational therapies with unknown safety and PK profile: 28 days. If there is enough data on the investigational therapy to assess the risk for drug-drug interactions and late toxicities of prior therapy as low, the Sponsor's Medical Monitor may approve a shorter washout of 14 days
4. Grapefruit or grapefruit juice: 14 days
* Have not recovered from all clinically relevant toxicities from prior therapy
* New York Heart Association Class III or IV heart disease, active ischemia, or any other uncontrolled cardiac condition, clinically significant cardiac arrhythmia requiring therapy, uncontrolled hypertension, congestive heart failure, or myocardial infarction within 6 months prior to the first dose of study drug
* Symptomatic central nervous system (CNS) metastases or presence of leptomeningeal disease
* Malabsorption syndrome
* Radiation for indications other than bone disease must have been completed 4 weeks prior to first dose of study drug, unless it consisted of limited field palliative radiation, including whole brain radiation, which must have been completed at least 2 weeks prior to first dose of study drug
* Major surgery within 4 weeks of the first dose of study drug
* Active HIV, Hepatitis B or Hepatitis C infection
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Deciphera Pharmaceuticals, LLC

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Clinical Team

Role: STUDY_DIRECTOR

Deciphera Pharmaceuticals, LLC

Locations

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University of Southern California - Norris Comprehensive Cancer Center

Los Angeles, California, United States

Site Status RECRUITING

UCLA Department of Medicine-Hematology/Oncology

Los Angeles, California, United States

Site Status RECRUITING

Sylvester Comprehensive Cancer Center

Miami, Florida, United States

Site Status RECRUITING

University of Massachusetts Worcester

Worcester, Massachusetts, United States

Site Status RECRUITING

START Midwest

Grand Rapids, Michigan, United States

Site Status RECRUITING

Washington University School of Medicine - Siteman Cancer Center

St Louis, Missouri, United States

Site Status RECRUITING

Memorial Sloan Kettering Cancer Center - Main Campus

New York, New York, United States

Site Status RECRUITING

Cleveland Clinic Taussig Cancer Center

Cleveland, Ohio, United States

Site Status RECRUITING

Oregon Health & Science University

Portland, Oregon, United States

Site Status RECRUITING

Fox Chase Cancer Center

Philadelphia, Pennsylvania, United States

Site Status RECRUITING

Virginia Cancer Specialist, PC

Fairfax, Virginia, United States

Site Status RECRUITING

Inselspital Universitätsklinikum Bern

Bern, , Switzerland

Site Status RECRUITING

Countries

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United States Switzerland

Central Contacts

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Clinical Team

Role: CONTACT

888-724-3274

Facility Contacts

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Rabia Rehman

Role: primary

323-865-3000

Jacqueline Banuelos

Role: primary

310-869-7014 ext. 16108

Nailet Bestard

Role: primary

305-243-8173

Syliva Rollins

Role: primary

7744554454

Julie Burns

Role: primary

616-954-5559

Tori Tuma

Role: primary

314-747-9488

Pragya Khadka

Role: primary

Melessa Hardayal

Role: backup

Cancer Answer

Role: primary

216-444-7923

Knight Cancer Institute Clinical Trials

Role: primary

503-494-1080

Refiola Memushi

Role: primary

(215)-728-3564

Anthony Jones

Role: primary

571-512-3202

Other Identifiers

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2024-516476-15-00

Identifier Type: CTIS

Identifier Source: secondary_id

DCC-3116-01-002

Identifier Type: -

Identifier Source: org_study_id

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