A Study to Investigate the Effects of Sisunatovir on QTc Interval in Healthy Adult Participants.

NCT ID: NCT05878522

Last Updated: 2024-12-06

Study Results

Results available

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

43 participants

Study Classification

INTERVENTIONAL

Study Start Date

2023-05-15

Study Completion Date

2023-10-30

Brief Summary

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The purpose of the study is to investigate the effects of multiple oral doses of sisunatovir on QTc Interval.

This study is seeking participants who:

* are male or female of 18 years of age or older
* are examined to be healthy All participants will receive Treatment A, B, and C in a randomized order based on 6 possible sequences. All treatments will be taken by mouth. Participants assigned to treatment A will receive 5 oral doses of sisunatovir administered Q12 hours over 3 days in a fed state. Participants assigned to treatment B will receive 5 oral doses of matching placebo administered Q12 hours over 3 days in a fed state. Participants assigned to treatment C will receive 4 oral doses of placebo administered Q12 hours for 2 days followed by a single dose of 400 mg moxifloxacin on the morning of Day 3.

All participants will remain in the study clinic for 4 days for each treatment, for safety review, laboratory collections, and to assess how the study medicine affects QTc intervals.

All participants selected in the study will be required to go through a screening period up to 28 days. A screening period is the time during which a few participants are examined to see whether they are fit for the study. During this period, the participant's medical history and past and current medications will be reviewed. A series of tests will also be performed to see if they are good to be selected for the study. If the participant meets all required criteria and are interested in continuing, the participant will be brought into the study clinic to stay overnight for 4 days for each treatment. On day 4, the participant will be discharged. About 28 to 35 days after discharge following the final treatment, the participant will be contacted for a follow up visit either in person or by telephone. This is to check up on how the participant is doing and to conclude the study.

Detailed Description

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Conditions

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Healthy

Keywords

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Healthy volunteers

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

CROSSOVER

Single Group, Crossover study
Primary Study Purpose

BASIC_SCIENCE

Blinding Strategy

TRIPLE

Participants Caregivers Investigators
Sisunatovir and placebo oral capsules will be prepared in the CRU by 2 operators, 1 of whom is an unblinded pharmacist. Sisunatovir and placebo will be administered in blinded fashion to the subject.

Moxifloxacin 400 mg tablets will be packaged in an open-label manner at the CRU in the individual dosing containers by 2 operators, 1 of whom is an appropriately qualified and experienced member of the study staff (eg, physician, nurse, physician's assistant, practitioner, or pharmacist).

Study Groups

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Treatment A

6 capsules of sisunatovir administered Q12 hours for 5 doses

Group Type EXPERIMENTAL

sisunatovir

Intervention Type DRUG

6 capsules administered Q12 hours for 5 doses

Treatment B

6 capsules of placebo administered Q12 hours for 5 doses

Group Type PLACEBO_COMPARATOR

placebo

Intervention Type DRUG

6 capsules administered Q12 hours for 5 doses

Treatment C

6 capsules of placebo administered Q12 hours for 4 doses, followed by a single tablet of moxifloxacin

Group Type ACTIVE_COMPARATOR

moxifloxacin

Intervention Type DRUG

6 capsules of placebo administered Q12 hours for 4 doses, followed by a single tablet of moxifloxacin

Treatment D

7 capsules of sisunatovir administered Q12 hours for 5 doses

Group Type EXPERIMENTAL

sisunatovir

Intervention Type DRUG

7 capsules administered Q12 hours for 5 doses

Interventions

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sisunatovir

6 capsules administered Q12 hours for 5 doses

Intervention Type DRUG

placebo

6 capsules administered Q12 hours for 5 doses

Intervention Type DRUG

moxifloxacin

6 capsules of placebo administered Q12 hours for 4 doses, followed by a single tablet of moxifloxacin

Intervention Type DRUG

sisunatovir

7 capsules administered Q12 hours for 5 doses

Intervention Type DRUG

Other Intervention Names

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PF-07923568 PF-07923568

Eligibility Criteria

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Inclusion Criteria

* Body Mass Index (BMI) of 17.5 to 32 kg/m2, inclusive, and a total body weight \>50 kg (110 lb).
* Capable of giving signed informed consent.
* At screening, no clinically relevant abnormalities identified by a detailed medical history, complete physical examination, including blood pressure (BP) and pulse rate measurement, standard 12-lead electrocardiogram (ECG) and clinical laboratory tests.

Exclusion Criteria

* Any condition or surgery possibly affecting drug absorption (eg, prior bariatric surgery, gastrectomy, ileal resection)
* Those with increased risk if dosed with moxifloxacin
* Self-reported history or risk factors for QT prolongation or torsades de pointes, congenital deafness, family history of cardiac arrest or suggest death, and family history of long QT syndrome
* Positive human immunodeficiency virus (HIV) antibodies
* Positive drug or alcohol test
* Screening supine BP ≥140 mm Hg (systolic) or ≥90 mm Hg (diastolic), following at least 5 minutes of supine rest. If BP is ≥140 mm Hg (systolic) or ≥90 mm Hg (diastolic), the BP should be repeated 2 more times and the average of the 3 BP values should be used to determine the participant's eligibility-estimated glomerular filtration rate (GFR) \<60 mL/min/1.73m2 at screening
* Standard 12-lead ECG that demonstrates clinically relevant abnormalities that may affect participant safety or interpretation of study results (eg, QTcF \>450 ms, complete LBBB, signs of an acute or indeterminate- age myocardial infarction, ST-T interval changes suggestive of myocardial ischemia, second- or third- degree AV block, or serious bradyarrhythmias or tachyarrhythmias). If the uncorrected QT interval is \>450 ms, this interval should be rate-corrected using the Fridericia method only and the resulting QTcF should be used for decision making and reporting. If QTcF exceeds 450 ms, or QRS exceeds 120 ms, the ECG should be repeated twice and the average of the 3 QTcF or QRS values used to determine the participant's eligibility. Participants with an average QTc interval \>450 milliseconds (ms) will not be allowed to participate in the study. Computer-interpreted ECGs should be overread by a physician experienced in reading ECGs before excluding a participant.
* GFR \<60 mL/min/1.73m2 based on CKD-EPI equation
* AST or ALT level ≥1.5 x upper limit normal (ULN)
* Gamma-GT\> 1.2 x ULN
* Alkaline phosphatase \> 1.2 x ULN
* Total bilirubin level ≥1.5 × ULN; participants with a history of Gilbert's syndrome may have direct bilirubin measured and would be eligible for this study provided the direct bilirubin level is ≤ ULN
* History of alcohol abuse or binge drinking and/or any other illicit drug use or dependence within 6 months of Screening. Binge drinking is defined as a pattern of 5 (male) and 4 (female) or more alcoholic drinks in about 2 hours. As a general rule, alcohol intake should not exceed 14 units per week (1 unit = 8 ounces (240 mL) beer, 1 ounce (30 mL) of 40% spirit, or 3 ounces (90 mL) of wine).
Minimum Eligible Age

18 Years

Maximum Eligible Age

65 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

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Pfizer

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Pfizer CT.gov Call Center

Role: STUDY_DIRECTOR

Pfizer

Locations

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New Haven Clinical Research Unit

New Haven, Connecticut, United States

Site Status

Countries

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United States

Provided Documents

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Document Type: Study Protocol

View Document

Document Type: Statistical Analysis Plan

View Document

Related Links

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https://pmiform.com/clinical-trial-info-request?StudyID=C5241015

To obtain contact information for a study center near you, click here.

Other Identifiers

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C5241015

Identifier Type: -

Identifier Source: org_study_id