Study of ART0380 in Patients With Biologically Selected Solid Tumors

NCT ID: NCT05798611

Last Updated: 2025-11-06

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

Get a concise snapshot of the trial, including recruitment status, study phase, enrollment targets, and key timeline milestones.

Recruitment Status

TERMINATED

Clinical Phase

PHASE2

Total Enrollment

36 participants

Study Classification

INTERVENTIONAL

Study Start Date

2023-09-06

Study Completion Date

2025-05-27

Brief Summary

Review the sponsor-provided synopsis that highlights what the study is about and why it is being conducted.

This interventional study will evaluate the efficacy and safety of ART0380 as monotherapy in patients whose tumors have a biology to predict for sensitivity to inhibition of Ataxia-Telangiectasia Mutated and Rad3-related protein kinase (ATR).

Detailed Description

Dive into the extended narrative that explains the scientific background, objectives, and procedures in greater depth.

ART0380 is being developed as an oral anti-cancer agent for the treatment of patients with cancers that have defects in deoxyribonucleic acid (DNA) repair.

The study will recruit selected patients with advanced or metastatic solid tumors, specifically:

* Patients with persistent or recurrent endometrial cancer (EC)
* Patients with advanced or metastatic solid tumors of any histology

Above patients will be randomized in a 1:1 ratio to one of two dose regimens of ART0380.

Safety will be evaluated on a quarterly basis, at a minimum. Patients may continue to receive ART0380 as long as they are continuing to derive benefit from treatment or until disease progression, withdrawal of consent, or until they experience unacceptable drug-related toxicity.

Conditions

See the medical conditions and disease areas that this research is targeting or investigating.

Advanced Solid Tumor Recurrent Endometrial Cancer Metastatic Cancer

Keywords

Explore important study keywords that can help with search, categorization, and topic discovery.

Solid Tumors Monotherapy Cancer cell Oral anti-cancer

Study Design

Understand how the trial is structured, including allocation methods, masking strategies, primary purpose, and other design elements.

Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

Review each arm or cohort in the study, along with the interventions and objectives associated with them.

Arm 1 [ART0380 monotherapy (endometrial cancer patients)]

Patients with persistent or recurrent endometrial cancer (EC) will receive ART0380 monotherapy in one of two dose regimens for a 21-day cycle.

Group Type EXPERIMENTAL

ART0380

Intervention Type DRUG

Randomized patients will orally receive ART0380.

Arm 2 [ART0380 monotherapy (solid tumors patients)]

Patients with advanced or metastatic solid tumors will receive ART0380 monotherapy in one of two dose regimens for a 21-day cycle.

Group Type EXPERIMENTAL

ART0380

Intervention Type DRUG

Randomized patients will orally receive ART0380.

Interventions

Learn about the drugs, procedures, or behavioral strategies being tested and how they are applied within this trial.

ART0380

Randomized patients will orally receive ART0380.

Intervention Type DRUG

Eligibility Criteria

Check the participation requirements, including inclusion and exclusion rules, age limits, and whether healthy volunteers are accepted.

Inclusion Criteria

* Patients who have discontinued all previous treatments for cancer for at least 21 days or 5 half-lives (not including palliative radiotherapy at focal sites), whichever is shorter. Palliative radiotherapy must have completed 1 week prior to start of study treatment.
* Resolution of all toxicities of prior therapy or surgical procedures to baseline or Grade 1 (except for hypothyroidism requiring medication, neuropathy, and alopecia, which must have resolved to Grade ≤2).
* Have adequate organ function.
* Patients of childbearing potential and patients with partners of childbearing potential are required to use highly effective contraception.
* Have an estimated life expectancy of ≥12 weeks, in the judgment of the investigator.
* Performance status of 0-1 on the Eastern Cooperative Oncology Group scale.
* Have a non-irradiated tumor tissue sample (archival or newly obtained core biopsy of a tumor lesion) available.



* Persistent or recurrent EC with biological selection.
* Patients should have received taxane/platinum chemotherapy unless contraindicated.
* Measurable disease.


* Advanced or metastatic solid cancers of any histology with biological selection.
* If a Programmed cell death protein-1 /Programmed death-ligand-1 inhibitor (e.g., pembrolizumab) is approved and available for the patient's cancer, the patient should have received such treatment before participating in this study.
* Radiologically evaluable disease.

Exclusion Criteria

* Patients who are pregnant.
* Prior treatment with an inhibitor of ATR, WEE1, checkpoint kinase 1 or PKMYT1.
* Have a serious concomitant systemic disorder that would compromise the patient's ability to adhere to the protocol.
* Have ongoing interstitial lung disease or pneumonitis (whether symptomatic or asymptomatic).
* Patients with treated brain metastases are eligible if follow-up brain imaging after central nervous system (CNS) directed therapy shows no evidence of progression.
* Have any major gastrointestinal issues that could impact absorption of ART0380.
* Have a history of allergy or hypersensitivity to study drug components.
* Have a significant bleeding disorder or vasculitis or had a Grade ≥3 bleeding episode within 12 weeks prior to enrollment.
* Patients who plan to father a child while in the study or within 16 weeks (5 months in France) after the last administration of study treatment.
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

Meet the organizations funding or collaborating on the study and learn about their roles.

Artios Pharma Ltd

INDUSTRY

Sponsor Role lead

Responsible Party

Identify the individual or organization who holds primary responsibility for the study information submitted to regulators.

Responsibility Role SPONSOR

Locations

Explore where the study is taking place and check the recruitment status at each participating site.

University of California Los Angeles (UCLA)

Los Angeles, California, United States

Site Status

The University of Chicago

Chicago, Illinois, United States

Site Status

Dana Farber Cancer Center

Boston, Massachusetts, United States

Site Status

Northwell Health R.J. Zuckerberg Cancer Center

Lake Success, New York, United States

Site Status

Memorial Sloan Kettering Cancer Center (MSKCC) - Memorial Hospital - Oncology

New York, New York, United States

Site Status

University of Oklahoma/Sarah Cannon Research Institute

Oklahoma City, Oklahoma, United States

Site Status

Western Pennsylvania Hospital

Pittsburgh, Pennsylvania, United States

Site Status

Women and Infants Hospital

Providence, Rhode Island, United States

Site Status

Institut de Cancérologie de l'Ouest

Angers, NAP, France

Site Status

Centre Francois Baclesse - Service d'Oncologie médicale

Caen, NAP, France

Site Status

Hopital Cochin Saint Vincent De Paul

Paris, NAP, France

Site Status

Hopital Lyon Sud

Pierre-Bénite, NAP, France

Site Status

Centre Hospitalier Universitaire De Poitiers

Poitiers, NAP, France

Site Status

Hospital Universitario De Jaén

Jaén, Andalusia, Spain

Site Status

Fundación Instituto Valenciano De Oncología

Valencia, , Spain

Site Status

Countries

Review the countries where the study has at least one active or historical site.

United States France Spain

Other Identifiers

Review additional registry numbers or institutional identifiers associated with this trial.

2023-504153-12

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

ART0380C004

Identifier Type: -

Identifier Source: org_study_id