Phase 1b/2a Study of GSBR-1290 in Adult Overweight or Obese Healthy Subjects and Subjects With Type 2 Diabetes Mellitus

NCT ID: NCT05762471

Last Updated: 2024-04-25

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1/PHASE2

Total Enrollment

142 participants

Study Classification

INTERVENTIONAL

Study Start Date

2023-01-09

Study Completion Date

2024-04-11

Brief Summary

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This study will evaluate safety, tolerability, pharmacokinetic (PK) profile, and pharmacodynamic (PD) effects on GSBR-1290 in healthy overweight/obese volunteers (HOV) and Type 2 Diabetes Mellitus on Metformin (T2DM) This study includes 5 planned cohorts. Participants will receive multiple-ascending doses of GSBR-1290 or Placebo from Day 1 to Day 84

Detailed Description

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Conditions

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Overweight or Obesity Type2 Diabetes Mellitus

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

TRIPLE

Participants Caregivers Investigators
This is a double-blind study in which the GSBR-1290 and the matching placebo are matching in appearance

Study Groups

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Cohort 1

Patients will receive once daily doses of study drug (GSBR-1290 or Placebo) for a total of 4 weeks

Group Type EXPERIMENTAL

GSBR-1290

Intervention Type DRUG

Patients will receive GSBR-1290 or matching Placebo

Placebo

Intervention Type DRUG

Patients will receive GSBR-1290 or matching Placebo

Cohort 2

Patients will receive once daily doses of study drug (GSBR-1290 or Placebo) for a total of 4 weeks

Group Type EXPERIMENTAL

GSBR-1290

Intervention Type DRUG

Patients will receive GSBR-1290 or matching Placebo

Placebo

Intervention Type DRUG

Patients will receive GSBR-1290 or matching Placebo

Cohort 3

Patients will receive once daily doses of study drug (GSBR-1290 or Placebo) for a total of 4 weeks

Group Type EXPERIMENTAL

GSBR-1290

Intervention Type DRUG

Patients will receive GSBR-1290 or matching Placebo

Placebo

Intervention Type DRUG

Patients will receive GSBR-1290 or matching Placebo

Cohort 4

HOV participants (Cohort 4) will receive multiple-ascending doses of GSBR-1290 or placebo for a total of 12 weeks

Group Type EXPERIMENTAL

GSBR-1290

Intervention Type DRUG

Patients will receive GSBR-1290 or matching Placebo

Placebo

Intervention Type DRUG

Patients will receive GSBR-1290 or matching Placebo

Cohort 5

Participants with T2DM(Cohort 5) will be randomized to placebo, low-dose, or high-dose arms. Participants in the low-dose, high-dose or placebo arms will receive multiple-ascending doses for 12 weeks

Group Type EXPERIMENTAL

GSBR-1290

Intervention Type DRUG

Patients will receive GSBR-1290 or matching Placebo

Placebo

Intervention Type DRUG

Patients will receive GSBR-1290 or matching Placebo

Interventions

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GSBR-1290

Patients will receive GSBR-1290 or matching Placebo

Intervention Type DRUG

Placebo

Patients will receive GSBR-1290 or matching Placebo

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

1. Provided evidence of a signed consent
2. Age ≥ 18 and ≤ 75 years
3. Healthy overweight/obese adult men and women with body mass index ≥ 27 and ≤ 40 kg/m2
4. No nicotine use
5. Have a suitable venous access for blood sampling


1. Men and women with T2DM of ≥6 months duration
2. Age ≥ 18 and ≤ 75 years
3. BMI ≥ 27 and ≤ 40 kg/m2
4. Treated with stable doses of ≥500 mg of metformin with a duration ≥6 months and at stable doses for ≥2 months with a screening HbA1c ≥7.0% and ≤10.5%.

Exclusion Criteria

1. History or presence of significant cardiovascular, pulmonary, hepatic, renal, hematological, gastrointestinal, endocrine, immunologic, dermatologic or neurological disease, including any acute illness or major surgery within the major 3 months
2. A sitting BP after resting for 5 minutes \> 160mm Hg systolic or \> 100 mm Hg diastolic or an apical pulse rate \<50 or \>100 beats per minute.
3. Evidence of abnormality on the screening visit ECG, or a history of known arrhythmia or prolonged QTcF pr prolonged QRS interval
4. Liver function test results elevated \> 2.0-fold above the ULN for gamma glutamyl transferase, alkaline phosphatase, aspartate aminotransferase or alanine aminotransferase. Bilirubin above the ULN
5. Estimated glomerular filtration rate \< 60mL/min/1.73 m2 body surface area
6. Known hypersensitivity to any of the study drug ingredients
7. Any other condition or prior therapy that would make the participant unsuitable for this study
Minimum Eligible Age

18 Years

Maximum Eligible Age

75 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Gasherbrum Bio, Inc., a wholly owned subsidiary of Structure Therapeutics

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Locations

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Anaheim Clinical Trials

Anaheim, California, United States

Site Status

ProSciento, Inc

Chula Vista, California, United States

Site Status

QPS Miami Research Associates

Miami, Florida, United States

Site Status

Progressive Medical Research

Port Orange, Florida, United States

Site Status

Countries

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United States

Other Identifiers

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GSBR-1290-02

Identifier Type: -

Identifier Source: org_study_id

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