Trial Outcomes & Findings for Single Dose ADME Study of [14C]-Rencofilstat in Healthy Male Subjects (NCT NCT05737433)

NCT ID: NCT05737433

Last Updated: 2024-10-03

Results Overview

Cumulative percentage of total radioactivity recovered after a single oral dose of \[14C\]-rencofilstat.

Recruitment status

COMPLETED

Study phase

EARLY_PHASE1

Target enrollment

6 participants

Primary outcome timeframe

22 Days

Results posted on

2024-10-03

Participant Flow

After subjects consented for study, they went through the screening process. Subjects that qualified for study were assigned to the single treatment arm.

Participant milestones

Participant milestones
Measure
[14C]-RCF 225mg
\[14C\]-rencofilstat, 225mg oral dose, self-micro-emulsifying drug delivery system, single dose
Overall Study
STARTED
6
Overall Study
COMPLETED
6
Overall Study
NOT COMPLETED
0

Reasons for withdrawal

Withdrawal data not reported

Baseline Characteristics

Single Dose ADME Study of [14C]-Rencofilstat in Healthy Male Subjects

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
[14C]-RCF 225mg
n=6 Participants
\[14C\]-rencofilstat, 225mg oral dose, self-micro-emulsifying drug delivery system, single dose \[14C\]-rencofilstat 225mg: radio-labelled 225mg oral dose of rencofilstat
Age, Categorical
<=18 years
0 Participants
n=5 Participants
Age, Categorical
Between 18 and 65 years
6 Participants
n=5 Participants
Age, Categorical
>=65 years
0 Participants
n=5 Participants
Sex: Female, Male
Female
0 Participants
n=5 Participants
Sex: Female, Male
Male
6 Participants
n=5 Participants
Ethnicity (NIH/OMB)
Hispanic or Latino
0 Participants
n=5 Participants
Ethnicity (NIH/OMB)
Not Hispanic or Latino
6 Participants
n=5 Participants
Ethnicity (NIH/OMB)
Unknown or Not Reported
0 Participants
n=5 Participants
Race (NIH/OMB)
American Indian or Alaska Native
0 Participants
n=5 Participants
Race (NIH/OMB)
Asian
0 Participants
n=5 Participants
Race (NIH/OMB)
Native Hawaiian or Other Pacific Islander
0 Participants
n=5 Participants
Race (NIH/OMB)
Black or African American
0 Participants
n=5 Participants
Race (NIH/OMB)
White
6 Participants
n=5 Participants
Race (NIH/OMB)
More than one race
0 Participants
n=5 Participants
Race (NIH/OMB)
Unknown or Not Reported
0 Participants
n=5 Participants
Region of Enrollment
United Kingdom
6 Participants
n=5 Participants
% of [14C]-RCF recovered
0 %
n=5 Participants

PRIMARY outcome

Timeframe: 22 Days

Population: Mass balance population

Cumulative percentage of total radioactivity recovered after a single oral dose of \[14C\]-rencofilstat.

Outcome measures

Outcome measures
Measure
[14C]-RCF 225mg
n=6 Participants
\[14C\]-rencofilstat, 225mg oral dose, self-micro-emulsifying drug delivery system, single dose
To Determine the Mass Balance Recovery After a Single Oral Dose of [14C]-Rencofilstat
91 percentage of total radioactivity

Adverse Events

[14C]-RCF 225mg

Serious events: 0 serious events
Other events: 3 other events
Deaths: 0 deaths

Serious adverse events

Adverse event data not reported

Other adverse events

Other adverse events
Measure
[14C]-RCF 225mg
n=6 participants at risk
\[14C\]-rencofilstat, 225mg oral dose, self-micro-emulsifying drug delivery system, single dose
Gastrointestinal disorders
Abdominal Pain
16.7%
1/6 • Number of events 1 • 63 days, screening period to on study last visit.
Gastrointestinal disorders
Diarrhoea
16.7%
1/6 • Number of events 1 • 63 days, screening period to on study last visit.
Gastrointestinal disorders
Nausea
16.7%
1/6 • Number of events 1 • 63 days, screening period to on study last visit.
Nervous system disorders
Headache
33.3%
2/6 • Number of events 2 • 63 days, screening period to on study last visit.
Renal and urinary disorders
Pollakiuria
16.7%
1/6 • Number of events 1 • 63 days, screening period to on study last visit.
Respiratory, thoracic and mediastinal disorders
Oropharyngeal pain
16.7%
1/6 • Number of events 1 • 63 days, screening period to on study last visit.

Additional Information

Jill Greytok

Hepion Pharmaceuticals Inc

Phone: 732-902-4000

Results disclosure agreements

  • Principal investigator is a sponsor employee
  • Publication restrictions are in place