A Study of DZD9008 Versus Platinum-Based Doublet Chemotherapy in Local Advanced or Metastatic Non-small Cell Lung Cancer (WU-KONG28)

NCT ID: NCT05668988

Last Updated: 2025-09-30

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

ACTIVE_NOT_RECRUITING

Clinical Phase

PHASE3

Total Enrollment

324 participants

Study Classification

INTERVENTIONAL

Study Start Date

2022-12-13

Study Completion Date

2027-10-31

Brief Summary

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This is a phase 3, open-label, randomized, multi-center study assessing the efficacy and safety of DZD9008 versus platinum-based doublet chemotherapy in participants with locally advanced or metastatic NSCLC with EGFR Exon20ins mutation, who are newly diagnosed or have not received prior systemic therapy in advanced stage.

Primary objective of this study is to assess the efficacy of DZD9008 versus platinum-based doublet chemotherapy using by BICR-assessed PFS per RECIST 1.1 as primary endpoint. Approximately 320 participants are estimated to be randomized into the study. Participants enrolled will be randomized to DZD9008 or platinum-based doublet chemotherapy in a 1:1 manner, stratified by baseline brain metastasis (with/without).

Detailed Description

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Conditions

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Non-small Cell Lung Cancer

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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sunvozertinib

Group Type EXPERIMENTAL

sunvozertinib

Intervention Type DRUG

orally, 300 mg, once daily until a treatment discontinuation criterion is met.

Platinum-based Chemotherapy

Group Type ACTIVE_COMPARATOR

Pemetrexed+carboplatin

Intervention Type DRUG

Participants randomized into chemotherapy arm can receive up to 6 cycles of pemetrexed + carboplatin (pemetrexed 500 mg/m2 + carboplatin area under the plasma concentration-time curve 5 mg/ml per minute (AUC5), IV infusion, every 3 weeks) as the initial treatment. Participants whose disease has not progressed after 4 cycles of first-line platinum-based doublet chemotherapy may receive pemetrexed maintenance monotherapy until a treatment discontinuation criterion is met.

Interventions

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sunvozertinib

orally, 300 mg, once daily until a treatment discontinuation criterion is met.

Intervention Type DRUG

Pemetrexed+carboplatin

Participants randomized into chemotherapy arm can receive up to 6 cycles of pemetrexed + carboplatin (pemetrexed 500 mg/m2 + carboplatin area under the plasma concentration-time curve 5 mg/ml per minute (AUC5), IV infusion, every 3 weeks) as the initial treatment. Participants whose disease has not progressed after 4 cycles of first-line platinum-based doublet chemotherapy may receive pemetrexed maintenance monotherapy until a treatment discontinuation criterion is met.

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

1. Aged at least 18 years old (or per local regulatory/IRB requirement).
2. Histologically or cytologically confirmed diagnosis of non-squamous NSCLC, locally advanced (Stage IIIB and IIIC according to the 8th edition of the AJCC TNM staging criteria) or metastatic (Stage IV), not suitable for curative therapy.
3. Adequate tumor tissue available, for central laboratory confirmation of EGFR exon 20 insertion mutation
4. At least 1 measurable lesion per RECIST Version 1.1
5. Life expectancy ≥ 12 weeks
6. Eastern Cooperative Oncology Group (ECOG) performance status of 0 to 1
7. Adequate organ and hematologic function

Exclusion Criteria

1. Prior treatment with any systemic anti-cancer therapy for locally advanced or metastatic NSCLC.
2. Spinal cord compression or leptomeningeal metastasis.
3. Concurrent EGFR mutations: exon 19 deletion, L858R, T790M, G719X, S768I, or L861Q.
4. History of stroke or intracranial hemorrhage within 6 months before randomization.
5. As judged by the investigator, any evidence of severe or uncontrolled systemic diseases, including uncontrolled hypertension and active bleeding diatheses (i.e., hemophilia and Von Willebrand disease).
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Dizal Pharmaceuticals

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Caicun Zhou

Role: PRINCIPAL_INVESTIGATOR

Shanghai Pulmonary Hospital, Shanghai, China

Locations

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OPN Healthcare, Inc.

Glendale, California, United States

Site Status

Kaiser Permanente Medical Center

Vallejo, California, United States

Site Status

University of Colorado Hospital - Anschutz Cancer Pavilion

Aurora, Colorado, United States

Site Status

D&H Cancer Research Center

Margate, Florida, United States

Site Status

Brcr Global

Plantation, Florida, United States

Site Status

H. Lee Moffitt Cancer Center

Tampa, Florida, United States

Site Status

NYU Laura & Issac Perlmutter Cancer Center

New York, New York, United States

Site Status

Columbia University Medical Center

New York, New York, United States

Site Status

Gabrail Cancer Center Research

Canton, Ohio, United States

Site Status

The Ohio State University

Columbus, Ohio, United States

Site Status

Providence Portland Medical Center

Portland, Oregon, United States

Site Status

USOR - Texas Oncology - Baylor Charles A. Sammons Cancer Center

Dallas, Texas, United States

Site Status

MD Anderson cancer center

Houston, Texas, United States

Site Status

USOR - Texas Oncology--Weslaco

Weslaco, Texas, United States

Site Status

University of Virginia Comprehensive Cancer Center

Charlottesville, Virginia, United States

Site Status

Centro de Educación Médica e Investigaciones Clínicas, CEMIC

Buenos Aires, , Argentina

Site Status

Centro Diabaid

Buenos Aires, , Argentina

Site Status

Centro Medico Austral

Buenos Aires, , Argentina

Site Status

Consultorios Medicos Dr. Doreski - Fundacion Respirar

Buenos Aires, , Argentina

Site Status

Fundacion Cenit Para El Estudio De Neurociencias

Buenos Aires, , Argentina

Site Status

Hospital Italiano de Buenos Aires (HIBA)

Buenos Aires, , Argentina

Site Status

Instituto Alexander Fleming

Buenos Aires, , Argentina

Site Status

Instituto Argentino de Diagnositco y Tratamiento S.A

Buenos Aires, , Argentina

Site Status

Fundación Estudios Clínicos

Rosario, , Argentina

Site Status

Fundación Ars Médica

San Salvador, , Argentina

Site Status

Centro de Investigación Clínicas. Clinica Viedma S.A

Viedma, , Argentina

Site Status

Concord Cancer Centre Medical Oncology Clinical Trials Unit Concord Repatriation General Hospital

Concord, , Australia

Site Status

Peter MacCallum Cancer Centre

Melbourne, , Australia

Site Status

Sir Charles Gairdner Hospital, Heart Research Insititute

Nedlands, , Australia

Site Status

Prince of Wales Hospital

Randwick, , Australia

Site Status

Ordensklinikum Linz GmbH Elisabethinen

Linz, , Austria

Site Status

Uniklinikum Salzburg

Salzburg, , Austria

Site Status

Antwerpen University Hospital (UZA)

Edegem, Antwerp, Belgium

Site Status

University Hospital Gent- Drug Research Unit Ghent (D.R.U.G.)

Ghent, Flanders, Belgium

Site Status

Grand Hopital de Charleroi (GHdC) - Hopital Notre Dame

Charleroi, Hainaut, Belgium

Site Status

Fundacao PIO XII - Hospital do Cancer de Barretos

Barretos, , Brazil

Site Status

Centro de Pesquisas Clinicas em

Cachoeiro de Itapemirim, , Brazil

Site Status

Liga Norte Riograndense Contra o Câncer

Natal, , Brazil

Site Status

Hospital São Lucas da PUCRS

Porto Alegre, , Brazil

Site Status

Santa Casa de Misericordia- Porto Alegre - Hospital Santa Rita

Porto Alegre, , Brazil

Site Status

Instituto D'Or de Pesquisa e Ensino - Recife

Recife, , Brazil

Site Status

Instituto America(COI)

Rio de Janeiro, , Brazil

Site Status

Instituto D'Or de Pesquisa e Ensino

Rio de Janeiro, , Brazil

Site Status

Instituto Nacional de Cancer Jose Alencar Gomes da Silva

Rio de Janeiro, , Brazil

Site Status

Instituto do Cancer do Estado de Sao Paulo - ICES

São Paulo, , Brazil

Site Status

Regional Cancer Program London Health Sciences Centre

London, , Canada

Site Status

The Ottawa Hospital Cancer Center

Ottawa, , Canada

Site Status

Princess Margaret Cancer Center

Toronto, , Canada

Site Status

Beijing Cancer Hospital

Beijing, , China

Site Status

Beijing Chest Hospital, Capital Medical University

Beijing, , China

Site Status

Cancer Hospital of the Chinese Academy of Medical Sciences

Beijing, , China

Site Status

Peking Union Medical College Hospital

Beijing, , China

Site Status

Peking University Third Hospital

Beijing, , China

Site Status

Hunan Cancer Hospital

Changsha, , China

Site Status

West China Hospital of Sichuan University

Chengdu, , China

Site Status

Army Medical Center of PLA

Chongqing, , China

Site Status

Chongqing Cancer Hospital

Chongqing, , China

Site Status

Fujian Cancer Hospital

Fuzhou, , China

Site Status

Fujian Medical University Union Hospital

Fuzhou, , China

Site Status

The First Affiliated Hospital of Guangzhou Medical University

Guangzhou, , China

Site Status

The First Affiliated Hospital of Sun Yat-sen University

Guangzhou, , China

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The First Affiliated Hospital Zhejiang University School of Medicine

Hangzhou, , China

Site Status

Zhejiang Cancer Hospital

Hangzhou, , China

Site Status

Harbin Medical University Cancer Hospital

Harbin, , China

Site Status

Anhui Provincial Hospital

Hefei, , China

Site Status

The First Affiliated Hospital of Anhui Medical University

Hefei, , China

Site Status

The Affiliated Hospital of Inner Mongolia Medical University

Hohhot, , China

Site Status

Jilin Cancer Hospital

Jilin, , China

Site Status

Central Hospital Affiliated to Shandong First Medical University

Jinan, , China

Site Status

Shandong Cancer Hospital & Institution

Jinan, , China

Site Status

Yunnan Cancer Hospital

Kunming, , China

Site Status

The Second Affiliated Hospital of Nanchang University

Nanchang, , China

Site Status

Jiangsu Cancer Hospital

Nanjing, , China

Site Status

Jiangsu Provincial Hospital

Nanjing, , China

Site Status

Guangxi Medical University Cancer Hospital

Nanning, , China

Site Status

Shanghai Chest Hospital

Shanghai, , China

Site Status

Shanghai Pulmonary Hospital

Shanghai, , China

Site Status

ZhongShan Hospital Fudan University

Shanghai, , China

Site Status

The First Hospital of China Medical University

Shenyang, , China

Site Status

Cancer Hospital Chinese Academy of Medical Sciences, ShenZhen center

Shenzhen, , China

Site Status

The Fourth Hospital of Hebei Medical University

Shijiazhuang, , China

Site Status

Shanxi Provincial Cancer Hospital

Taiyuan, , China

Site Status

Taizhou Hospital of Zhejiang Province

Taizhou, , China

Site Status

Tianjin Medical University Cancer Institute & Hospital

Tianjin, , China

Site Status

Tongji Hospital affiliated to Tongji Medical College of Huazhong University of Science & Technology

Wuhan, , China

Site Status

Union Hospital, Tongji Medical College, Huazhong University of Science and Technology

Wuhan, , China

Site Status

The First Affiliated Hospital of Xi 'an Jiaotong University

Xi'an, , China

Site Status

Yantai Yuhuangding Hospital

Yantai, , China

Site Status

Henan Cancer Hospital

Zhengzhou, , China

Site Status

The First Affiliated Hospital of Zhengzhou University

Zhengzhou, , China

Site Status

Fakultni Nemocnice Olomouc (FNOL) - Onkologicka Klinika

Olomouc, , Czechia

Site Status

Vitkovicka Nemocnice a.s. - Plicni oddeleni

Ostrava, , Czechia

Site Status

Centre Hospitalier Universitaire d'Angers

Angers, , France

Site Status

Hôpital Louis Pradel

Bron, , France

Site Status

Centre Hospitalier Intercommunal de Creteil (CHIC)

Créteil, , France

Site Status

Centre Hospitalier Universitaire de Lille (CHU Lille) - Hopital Albert Calmette - Clinique des Maladies Respiratoires

Hellemmes-Lille, , France

Site Status

Centre Hospitalier Universitaire Grenoble Alpes (CHU Grenoble Alpes) - Hopital Albert Michallon

La Tronche, , France

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APHM-Hôpital NORD

Marseille, , France

Site Status

Centre de Cancérologie Montpellier

Montpellier, , France

Site Status

APHP Hôpital Tenon

Paris, , France

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Cochin Hospital

Paris, , France

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Hopital Saint Joseph

Paris, , France

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Hôpital Bichat - Claude Bernard

Paris, , France

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CHU Poitiers

Poitiers, , France

Site Status

Centre Hospitalier Universitaire de Nantes (CHU de Nantes)

Saint-Herblain, , France

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Institut de Cancerologie de L'Ouest

Saint-Herblain, , France

Site Status

Hopital d'Instruction Des Armees Begin

Saint-Mandé, , France

Site Status

Hopital Foch

Suresnes, , France

Site Status

Evangelische Lungenklinik Berlin - Klinik fuer Pneumologie

Berlin, , Germany

Site Status

Asklepios Klinik Gauting GmbH - Klinik fuer Thorakale Onkologie

Gauting, , Germany

Site Status

Niels-Stensen-Kliniken - Franziskus-Hospital Harderberg

Georgsmarienhütte, , Germany

Site Status

Universitaetsklinikum Heidelberg (UKHD) - Thoraxklinik-Heidelberg gGmbH

Heidelberg, , Germany

Site Status

Universitaetsmedizin der Johannes Gutenberg-Universitaet Mainz - III. Medizinische Klinik und Poliklinik

Mainz, , Germany

Site Status

Pius-Hospital Oldenburg - Klinik fuer Haematologie und Onkologie

Oldenburg, , Germany

Site Status

Centro di Riferimento Oncologico (CRO Aviano)

Aviano, , Italy

Site Status

Azienda Ospedaliero Universitaria di Bologna - Policlinico S. Orsola-Malpighi

Bologna, , Italy

Site Status

Azienda Ospedaliero - Universitaria "Policlinico-Vittorio Emanuele" Catania

Catania, , Italy

Site Status

Università degli Studi di Firenze - Azienda Ospedaliero-Universitaria Careggi (AOUC) - SC di Oncologia MedicaI

Florence, , Italy

Site Status

Azienda USL Toscana Sud Est -Ospedale Misericordia - Grosseto

Grosseto, , Italy

Site Status

Servizio Sanitario Regionale Emilia-Romagna - Istituto Scientifico Romagnolo per lo Studio e La Cura dei Tumori Srl (IRST)

Meldola, , Italy

Site Status

Azienda Ospedaliero-Universitaria di Modena (AOU Modena) - Policlinico di Modena

Modena, , Italy

Site Status

Azienda Ospedaliera San Gerardo - Monza

Monza, , Italy

Site Status

La Maddalena Casa di Cura di Alta Specialita - Palermo

Palermo, , Italy

Site Status

Azienda Ospedaliero-Universitaria di Parma

Parma, , Italy

Site Status

Azienda Unità Sanitaria Locale Romagna

Ravenna, , Italy

Site Status

Azienda Ospedaliera di Reggio Emilia - Arcispedale S. Maria Nuova (ASMN)

Reggio Emilia, , Italy

Site Status

IRCCS Istituti Fisioterapici Ospitalieri- Istituto Nazionale tumori Regina Elena

Roma, , Italy

Site Status

Azienda Ospedaliera Universitaria Senese - Istituto Toscano Tumori (ITT) - Center for Immuno-Oncology (CIO)

Siena, , Italy

Site Status

Universiteit Maastricht (UM) - Maastricht University Medical Centre (Maastricht UMC+)

Maastricht, , Netherlands

Site Status

Uniwersyteckie Centrum Kliniczne, Klinika Onkologii i Radioterapii

Gdansk, , Poland

Site Status

MED-POLONIA Sp. z o.o.

Poznan, , Poland

Site Status

Wojewódzki Szpital im. św. Ojca Pio

Przemyśl, , Poland

Site Status

Narodowy Instytut Onkologii im. Marii Sklodowskiej-Curie Panstwowy

Warsaw, , Poland

Site Status

Institut Catala d'Oncologia Badalona (ICO Badalona) - Hospital Germans Trias i Pujol

Barcelona, Barcelona, Spain

Site Status

Complejo Hospitalario Universitario A Coruña

A Coruña, , Spain

Site Status

Hospital de la Santa Creu i Sant Pau

Barcelona, , Spain

Site Status

Hospital Universitari Vall d'Hebron

Barcelona, , Spain

Site Status

Instituto Oncológico Dr Rosell Hospital Quiron Dexeus

Barcelona, , Spain

Site Status

UOMI Cancer Center - Clinica Tres Torres

Barcelona, , Spain

Site Status

Institut Catala d'Oncologia de Girona -Hospital Universitari Dr Josep Trueta

Girona, , Spain

Site Status

Hospital Universitario de Jerez

Jerez de la Frontera, , Spain

Site Status

Clínica Universidad de Navarra - Madrid

Madrid, , Spain

Site Status

Hospital HM Sanchinarro

Madrid, , Spain

Site Status

Hospital Universitario 12 de Octubre

Madrid, , Spain

Site Status

Hospital Universitario Fundación Jiménez Diaz

Madrid, , Spain

Site Status

Hospital Universitario La Paz

Madrid, , Spain

Site Status

Hospital Regional Universitario de Málaga

Málaga, , Spain

Site Status

Hospital Universitario Virgen de Valme

Seville, , Spain

Site Status

Hospital Universitario Virgen del Rocio

Seville, , Spain

Site Status

Hospital Universitario Virgen Macarena

Seville, , Spain

Site Status

Hospital Clinico Universitario de Valencia

Valencia, , Spain

Site Status

Hospital Universitari i Politècnic La Fe

Valencia, , Spain

Site Status

Ankara Bilkent City Hospital Universiteler Mahallesi

Ankara, , Turkey (Türkiye)

Site Status

Dr. Abdurrahman Yurtaslan Ankara Oncology Training

Ankara, , Turkey (Türkiye)

Site Status

Gazi Universitesi Tip Fakultesi (Gazi University Faculty of Medicine) - Gazi Hastanesi (Gazi Hospital)

Ankara, , Turkey (Türkiye)

Site Status

Liv Hospital Ankara - Medical Oncology Clinic

Ankara, , Turkey (Türkiye)

Site Status

Trakya Universitesi Saglik Arastirma ve Uygulama Merkezi Hastane

Edirne, , Turkey (Türkiye)

Site Status

Bezmialem University Hospital

Istanbul, , Turkey (Türkiye)

Site Status

Prof. Dr. Süleyman Yalçın Şehir Hastanesi - Tibbi Onkoloji Klinigi

Kadıköy, , Turkey (Türkiye)

Site Status

Necmettin Erbakan University

Konya, , Turkey (Türkiye)

Site Status

Countries

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United States Argentina Australia Austria Belgium Brazil Canada China Czechia France Germany Italy Netherlands Poland Spain Turkey (Türkiye)

References

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Wang M, Fan Y, Sun M, Wang Y, Zhao Y, Jin B, Hu Y, Han Z, Song X, Liu A, Tang K, Ding C, Liang L, Wu L, Gao J, Wang J, Cheng Y, Zhou J, He Y, Dong X, Yao Y, Yu Y, Wang H, Sun S, Huang J, Fang J, Li W, Wang L, Ren X, Zhou C, Hu Y, Zhao D, Yang R, Xu F, Huang Y, Pan Y, Cui J, Xu Y, Yang Z, Shi Y. Sunvozertinib for patients in China with platinum-pretreated locally advanced or metastatic non-small-cell lung cancer and EGFR exon 20 insertion mutation (WU-KONG6): single-arm, open-label, multicentre, phase 2 trial. Lancet Respir Med. 2024 Mar;12(3):217-224. doi: 10.1016/S2213-2600(23)00379-X. Epub 2023 Dec 12.

Reference Type DERIVED
PMID: 38101437 (View on PubMed)

Other Identifiers

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DZ2022E0005

Identifier Type: -

Identifier Source: org_study_id

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