A Drug-drug Interaction Study to Evaluate the Effect of Rifampicin and Febuxostat on the Pharmacokinetics of Methotrexate in Healthy Subjects

NCT ID: NCT05575297

Last Updated: 2022-10-12

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

12 participants

Study Classification

INTERVENTIONAL

Study Start Date

2021-12-20

Study Completion Date

2022-05-09

Brief Summary

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To investigate the effect of rifampicin and febuxostat on pharmacokinetics of methotrexate in healthy volunteers

Detailed Description

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Conditions

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Drug Interaction

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

CROSSOVER

Primary Study Purpose

BASIC_SCIENCE

Blinding Strategy

NONE

Study Groups

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Methotrexate

Group Type EXPERIMENTAL

Methotrexate Sodium

Intervention Type DRUG

Methotrexate oral administration alone

Methotrexate + Rifampicin

Methotrexate + Rifampicin

Group Type EXPERIMENTAL

Methotrexate Sodium

Intervention Type DRUG

Methotrexate oral administration alone

Rifampicin Sodium

Intervention Type DRUG

Co-administration of methotrexate and rifampicin

Methotrexate + Febuxostat

Methotrexate + Febuxostat

Group Type EXPERIMENTAL

Methotrexate Sodium

Intervention Type DRUG

Methotrexate oral administration alone

Febuxostat Tablets

Intervention Type DRUG

Co-administration of methotrexate and febuxostat

Methotrexate + Rifampicin + Febuxostat

Methotrexate + Rifampicin + Febuxostat

Group Type EXPERIMENTAL

Methotrexate Sodium

Intervention Type DRUG

Methotrexate oral administration alone

Rifampicin Sodium

Intervention Type DRUG

Co-administration of methotrexate and rifampicin

Febuxostat Tablets

Intervention Type DRUG

Co-administration of methotrexate and febuxostat

Interventions

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Methotrexate Sodium

Methotrexate oral administration alone

Intervention Type DRUG

Rifampicin Sodium

Co-administration of methotrexate and rifampicin

Intervention Type DRUG

Febuxostat Tablets

Co-administration of methotrexate and febuxostat

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Age between 19 to 50, healthy male subjects (at screening)
* Body weight between 50.0 kg - 90.0 kg, BMI between 18.0 - 30.0 kg/m2
* Subject who totally understand the progress of this clinical trials, make decision by his free will, and signed a consent form to follow the progress

Exclusion Criteria

* Subject who has a past or present history of any diseases (eg. liver, kidney, neurology, immunology, pulmonary, endocrine, hematology, oncology, cardiology, mental disorder)
* Subject who had GI tract disease (Crohn's disease, ulcer, acute or chronic pancreatitis) or surgery (appendectomy, hernioplasty are excluded)
* Serum AST(SGOT), ALT(SGPT), total bilirubin \>1.5 times upper limit of normal range, MDRD eGFR \< 60mL/min/1.73m2, WBC count \< 3,500 /uL, SBP \< 90 mmHg or \> 150 mmHg, DBP \< 50 mmHg or \>100 mmHg
* Subject who had galactose intolerance, Lapplactase deficiency or glucose-galactose malabsorption
* Subject who had received drugs inhibiting or inducing metabolic enzymes/transporters such as barbiturates, statins, digoxin in 3 months
* Subject who had taken St.John's wort and food including grapefruit in 2 weeks
* Smoking in 3 months
* Subject who had whole blood donation in 2 months, or component blood donation in 1 month or transfusion in 1 month currently
Minimum Eligible Age

19 Years

Maximum Eligible Age

45 Years

Eligible Sex

MALE

Accepts Healthy Volunteers

Yes

Sponsors

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Seoul National University Hospital

OTHER

Sponsor Role lead

Responsible Party

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Jae Yong Chung, MD, PhD

Professor

Responsibility Role PRINCIPAL_INVESTIGATOR

Locations

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Seoul National University Bundang Hospital

Seoul, , South Korea

Site Status

Countries

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South Korea

Other Identifiers

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MRFI

Identifier Type: -

Identifier Source: org_study_id

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