Trial Outcomes & Findings for A Clinical Trial to Evaluate the Safety and Efficacy of ADX-629 in in Subjects With Elevated Ethanol Levels (NCT NCT05487404)

NCT ID: NCT05487404

Last Updated: 2025-02-28

Results Overview

Safety was assessed through serious adverse event collection.

Recruitment status

COMPLETED

Study phase

PHASE1/PHASE2

Target enrollment

26 participants

Primary outcome timeframe

The safety assessment period was approximately two days for each treatment period.

Results posted on

2025-02-28

Participant Flow

Twenty-six subjects were randomized in a crossover design. On Day 1 for each treatment period, subjects were dosed followed by ethanol consumption. Approximately three hours later, subjects were administered a second dose followed by continued ethanol consumption to reach a target blood alcohol concentration of 0.14 g/100mL, at which time assessments were conducted. On Day 2, subjects were dosed once and assessments were completed approximately two hours and five hours after dosing.

Participant milestones

Participant milestones
Measure
ADX-629 First, Then Placebo
Subjects received three oral doses of ADX-629 600mg over two consecutive days, followed by a fourteen-day washout. Subjects then received three oral doses of placebo over two consecutive days.
Placebo First, Then ADX-629
Subjects received three oral doses of placebo over two consecutive days, followed by a fourteen-day washout. Subjects then received three oral doses of ADX-629 600mg over two consecutive days.
Overall Study
STARTED
12
14
Overall Study
COMPLETED
11
11
Overall Study
NOT COMPLETED
1
3

Reasons for withdrawal

Withdrawal data not reported

Baseline Characteristics

A Clinical Trial to Evaluate the Safety and Efficacy of ADX-629 in in Subjects With Elevated Ethanol Levels

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
ADX-629 First, Then Placebo
n=12 Participants
Subjects received three oral doses of ADX-629 600mg over two consecutive days, followed by a fourteen-day washout. Subjects then received three oral doses of placebo over two consecutive days.
Placebo First, Then ADX-629
n=14 Participants
Subjects received three oral doses of placebo over two consecutive days, followed by a fourteen-day washout. Subjects then received three oral doses of ADX-629 600mg over two consecutive days.
Total
n=26 Participants
Total of all reporting groups
Age, Categorical
<=18 years
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
Age, Categorical
Between 18 and 65 years
12 Participants
n=5 Participants
14 Participants
n=7 Participants
26 Participants
n=5 Participants
Age, Categorical
>=65 years
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
Age, Continuous
44.1 years
STANDARD_DEVIATION 9.0 • n=5 Participants
41.1 years
STANDARD_DEVIATION 12.4 • n=7 Participants
42.5 years
STANDARD_DEVIATION 10.8 • n=5 Participants
Sex: Female, Male
Female
4 Participants
n=5 Participants
3 Participants
n=7 Participants
7 Participants
n=5 Participants
Sex: Female, Male
Male
8 Participants
n=5 Participants
11 Participants
n=7 Participants
19 Participants
n=5 Participants
Race (NIH/OMB)
American Indian or Alaska Native
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
Race (NIH/OMB)
Asian
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
Race (NIH/OMB)
Native Hawaiian or Other Pacific Islander
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
Race (NIH/OMB)
Black or African American
3 Participants
n=5 Participants
7 Participants
n=7 Participants
10 Participants
n=5 Participants
Race (NIH/OMB)
White
9 Participants
n=5 Participants
6 Participants
n=7 Participants
15 Participants
n=5 Participants
Race (NIH/OMB)
More than one race
0 Participants
n=5 Participants
1 Participants
n=7 Participants
1 Participants
n=5 Participants
Race (NIH/OMB)
Unknown or Not Reported
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
Body Mass Index
26.4 kg/m2
STANDARD_DEVIATION 3.0 • n=5 Participants
26.6 kg/m2
STANDARD_DEVIATION 3.5 • n=7 Participants
26.5 kg/m2
STANDARD_DEVIATION 3.2 • n=5 Participants

PRIMARY outcome

Timeframe: The safety assessment period was approximately two days for each treatment period.

Population: Safety Population

Safety was assessed through serious adverse event collection.

Outcome measures

Outcome measures
Measure
ADX-629
n=23 Participants
Three oral doses of ADX-629 600mg over two consecutive days
Placebo
n=25 Participants
Three oral doses of placebo over two consecutive days
Number of Subjects With Serious Adverse Events
0 Participants
0 Participants

SECONDARY outcome

Timeframe: The efficacy assessment period was approximately two days for each treatment period. Baseline was the last measurement prior to each treatment period.

Population: Intent-to-treat population

Dermal flushing was assessed on a 0 to 100 scale (0 = none, 100 = extremely severe). Change from baseline was analyzed using mixed model for repeated measures (MMRM), with baseline and emesis volume as covariates, and sequence, period, time point, and treatment as factors.

Outcome measures

Outcome measures
Measure
ADX-629
n=23 Participants
Three oral doses of ADX-629 600mg over two consecutive days
Placebo
n=25 Participants
Three oral doses of placebo over two consecutive days
Change From Baseline of Dermal Flushing
-4.02 score on a scale
Standard Error 0.44
1.15 score on a scale
Standard Error 1.37

SECONDARY outcome

Timeframe: The efficacy assessment period was approximately two days for each treatment period. Baseline was the last measurement prior to each treatment period.

Population: Intent-to-treat population

Romberg Test was assessed for up to 60 seconds. Subjects stood with feet together and eyes closed, and the length of time the subject was able to stand without movement was recorded. Change from baseline was analyzed using MMRM, with baseline, number of bodyweight-standardized drinks consumed, and blood alcohol concentration as covariates, and sequence, period, time point, treatment, and the interaction of treatment by time point as factors.

Outcome measures

Outcome measures
Measure
ADX-629
n=23 Participants
Three oral doses of ADX-629 600mg over two consecutive days
Placebo
n=25 Participants
Three oral doses of placebo over two consecutive days
Change From Baseline for Romberg Test
-0.04 seconds
Standard Error 1.25
-1.42 seconds
Standard Error 1.20

Adverse Events

ADX-629

Serious events: 0 serious events
Other events: 15 other events
Deaths: 0 deaths

Placebo

Serious events: 0 serious events
Other events: 21 other events
Deaths: 0 deaths

Serious adverse events

Adverse event data not reported

Other adverse events

Other adverse events
Measure
ADX-629
n=23 participants at risk
Three oral doses of ADX-629 600mg over two consecutive days
Placebo
n=25 participants at risk
Three oral doses of placebo over two consecutive days
Gastrointestinal disorders
Abdominal pain
0.00%
0/23 • Two days for each intervention
4.0%
1/25 • Number of events 1 • Two days for each intervention
Gastrointestinal disorders
Dyspepsia
8.7%
2/23 • Number of events 2 • Two days for each intervention
8.0%
2/25 • Number of events 2 • Two days for each intervention
Gastrointestinal disorders
Gastroesophageal reflux disease
4.3%
1/23 • Number of events 1 • Two days for each intervention
0.00%
0/25 • Two days for each intervention
Gastrointestinal disorders
Nausea
47.8%
11/23 • Number of events 11 • Two days for each intervention
56.0%
14/25 • Number of events 14 • Two days for each intervention
Gastrointestinal disorders
Vomiting
30.4%
7/23 • Number of events 20 • Two days for each intervention
28.0%
7/25 • Number of events 14 • Two days for each intervention
Gastrointestinal disorders
Asthenia
0.00%
0/23 • Two days for each intervention
4.0%
1/25 • Number of events 1 • Two days for each intervention
Infections and infestations
COVID-19
0.00%
0/23 • Two days for each intervention
4.0%
1/25 • Number of events 1 • Two days for each intervention
Infections and infestations
Influenza
0.00%
0/23 • Two days for each intervention
4.0%
1/25 • Number of events 1 • Two days for each intervention
Infections and infestations
Upper respiratory tract infection
0.00%
0/23 • Two days for each intervention
4.0%
1/25 • Number of events 1 • Two days for each intervention
Nervous system disorders
Dizziness
8.7%
2/23 • Number of events 2 • Two days for each intervention
12.0%
3/25 • Number of events 3 • Two days for each intervention
Nervous system disorders
Headache
52.2%
12/23 • Number of events 12 • Two days for each intervention
56.0%
14/25 • Number of events 14 • Two days for each intervention
Skin and subcutaneous tissue disorders
Dermatitis
4.3%
1/23 • Number of events 1 • Two days for each intervention
0.00%
0/25 • Two days for each intervention

Additional Information

Director of Clinical Trials

Aldeyra Therapeutics, Inc.

Phone: 781-257-3063

Results disclosure agreements

  • Principal investigator is a sponsor employee
  • Publication restrictions are in place