Trial Outcomes & Findings for Effectiveness of CRD-740 in Heart Failure (NCT NCT05409183)

NCT ID: NCT05409183

Last Updated: 2024-12-19

Results Overview

Efficacy: To assess the effect of CRD-740 compared to placebo in plasma cGMP at Week 4 in subjects with CHFrEF.

Recruitment status

TERMINATED

Study phase

PHASE2

Target enrollment

60 participants

Primary outcome timeframe

Baseline to Week 4

Results posted on

2024-12-19

Participant Flow

Participant milestones

Participant milestones
Measure
CRD-740
Part A: Participants in Part A randomly assigned to this arm will take CRD-740 at two ascending dose levels over 12 weeks. CRD-740: Tablets administered orally. Part B of the study was not conducted in favor of redesigned new studies.
Placebo
Part A: Participants in Part A randomly assigned to this arm will take placebo at two ascending dose levels over 12 weeks. Placebo: Tablets administered orally. Part B of the study was not conducted in favor of redesigned new studies.
Period 1
STARTED
40
20
Period 1
COMPLETED
40
20
Period 1
NOT COMPLETED
0
0
Period 2
STARTED
40
20
Period 2
COMPLETED
38
19
Period 2
NOT COMPLETED
2
1
Period 3
STARTED
38
19
Period 3
COMPLETED
36
19
Period 3
NOT COMPLETED
2
0
Complete Study
STARTED
40
20
Complete Study
COMPLETED
36
18
Complete Study
NOT COMPLETED
4
2

Reasons for withdrawal

Reasons for withdrawal
Measure
CRD-740
Part A: Participants in Part A randomly assigned to this arm will take CRD-740 at two ascending dose levels over 12 weeks. CRD-740: Tablets administered orally. Part B of the study was not conducted in favor of redesigned new studies.
Placebo
Part A: Participants in Part A randomly assigned to this arm will take placebo at two ascending dose levels over 12 weeks. Placebo: Tablets administered orally. Part B of the study was not conducted in favor of redesigned new studies.
Complete Study
Adverse Event
1
2
Complete Study
Withdrawal by Subject
3
0

Baseline Characteristics

Female population only

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
CRD-740
n=40 Participants
Part A: Participants in Part A randomly assigned to this arm will take CRD-740 at two ascending dose levels over 12 weeks. CRD-740: Tablets administered orally. Part B of the study was not conducted in favor of redesigned new studies.
Placebo
n=20 Participants
Part A: Participants in Part A randomly assigned to this arm will take placebo at two ascending dose levels over 12 weeks. Placebo: Tablets administered orally. Part B of the study was not conducted in favor of redesigned new studies.
Total
n=60 Participants
Total of all reporting groups
Age, Categorical
<=18 years
0 Participants
n=40 Participants
0 Participants
n=20 Participants
0 Participants
n=60 Participants
Age, Categorical
Between 18 and 65 years
17 Participants
n=40 Participants
9 Participants
n=20 Participants
26 Participants
n=60 Participants
Age, Categorical
>=65 years
23 Participants
n=40 Participants
11 Participants
n=20 Participants
34 Participants
n=60 Participants
Age, Continuous
68.4 years
STANDARD_DEVIATION 12.70 • n=40 Participants
65.6 years
STANDARD_DEVIATION 13.16 • n=20 Participants
67.4 years
STANDARD_DEVIATION 12.81 • n=60 Participants
Age, Customized
Median Age
70.5 years
n=40 Participants
66.0 years
n=20 Participants
69.0 years
n=60 Participants
Sex: Female, Male
Female
5 Participants
n=40 Participants
4 Participants
n=20 Participants
9 Participants
n=60 Participants
Sex: Female, Male
Male
35 Participants
n=40 Participants
16 Participants
n=20 Participants
51 Participants
n=60 Participants
Ethnicity (NIH/OMB)
Hispanic or Latino
4 Participants
n=40 Participants
2 Participants
n=20 Participants
6 Participants
n=60 Participants
Ethnicity (NIH/OMB)
Not Hispanic or Latino
36 Participants
n=40 Participants
18 Participants
n=20 Participants
54 Participants
n=60 Participants
Ethnicity (NIH/OMB)
Unknown or Not Reported
0 Participants
n=40 Participants
0 Participants
n=20 Participants
0 Participants
n=60 Participants
Race (NIH/OMB)
American Indian or Alaska Native
0 Participants
n=40 Participants
0 Participants
n=20 Participants
0 Participants
n=60 Participants
Race (NIH/OMB)
Asian
2 Participants
n=40 Participants
1 Participants
n=20 Participants
3 Participants
n=60 Participants
Race (NIH/OMB)
Native Hawaiian or Other Pacific Islander
0 Participants
n=40 Participants
0 Participants
n=20 Participants
0 Participants
n=60 Participants
Race (NIH/OMB)
Black or African American
9 Participants
n=40 Participants
4 Participants
n=20 Participants
13 Participants
n=60 Participants
Race (NIH/OMB)
White
29 Participants
n=40 Participants
15 Participants
n=20 Participants
44 Participants
n=60 Participants
Race (NIH/OMB)
More than one race
0 Participants
n=40 Participants
0 Participants
n=20 Participants
0 Participants
n=60 Participants
Race (NIH/OMB)
Unknown or Not Reported
0 Participants
n=40 Participants
0 Participants
n=20 Participants
0 Participants
n=60 Participants
Region of Enrollment
United States
27 participants
n=40 Participants
13 participants
n=20 Participants
40 participants
n=60 Participants
Region of Enrollment
United Kingdom
8 participants
n=40 Participants
4 participants
n=20 Participants
12 participants
n=60 Participants
Region of Enrollment
Israel
5 participants
n=40 Participants
3 participants
n=20 Participants
8 participants
n=60 Participants
Mean Height (cm) at Baseline
175.6 cm
STANDARD_DEVIATION 10.20 • n=40 Participants
172.5 cm
STANDARD_DEVIATION 10.65 • n=20 Participants
174.6 cm
STANDARD_DEVIATION 10.36 • n=60 Participants
Median Height (cm) at Baseline
175.0 cm
n=40 Participants
170.8 cm
n=20 Participants
173.4 cm
n=60 Participants
Reproductive System Findings Test (Female only), n (%)
Childbearing Potential
2 Participants
n=5 Participants • Female population only
0 Participants
n=4 Participants • Female population only
2 Participants
n=9 Participants • Female population only
Reproductive System Findings Test (Female only), n (%)
Menopause Status
3 Participants
n=5 Participants • Female population only
4 Participants
n=4 Participants • Female population only
7 Participants
n=9 Participants • Female population only
Mean Weight (kg) at Baseline
97.27 kg
STANDARD_DEVIATION 37.582 • n=40 Participants
84.07 kg
STANDARD_DEVIATION 16.932 • n=20 Participants
92.87 kg
STANDARD_DEVIATION 32.639 • n=60 Participants
Median Weight (kg) at Baseline
87.65 kg
n=40 Participants
81.00 kg
n=20 Participants
85.55 kg
n=60 Participants
Mean Body Mass Index (kg/m2) at Baseline
31.41 body weight (kg)/ height (m2)
STANDARD_DEVIATION 11.483 • n=40 Participants
28.38 body weight (kg)/ height (m2)
STANDARD_DEVIATION 5.953 • n=20 Participants
30.40 body weight (kg)/ height (m2)
STANDARD_DEVIATION 10.032 • n=60 Participants
Median Body Mass Index (kg/m2) at Baseline
28.92 body weight (kg)/ height (m2)
n=40 Participants
26.72 body weight (kg)/ height (m2)
n=20 Participants
27.89 body weight (kg)/ height (m2)
n=60 Participants
Echocardiogram performed during screening
Yes
40 Participants
n=40 Participants
20 Participants
n=20 Participants
60 Participants
n=60 Participants
Echocardiogram performed during screening
No
0 Participants
n=40 Participants
0 Participants
n=20 Participants
0 Participants
n=60 Participants
EF group
EF ≤ 40%
40 Participants
n=40 Participants
20 Participants
n=20 Participants
60 Participants
n=60 Participants
EF group
EF > 40%
0 Participants
n=40 Participants
0 Participants
n=20 Participants
0 Participants
n=60 Participants
Mean EF (%) for rEF (≤40%) subjects
29.16 percent
STANDARD_DEVIATION 7.191 • n=40 Participants
26.91 percent
STANDARD_DEVIATION 6.181 • n=20 Participants
28.41 percent
STANDARD_DEVIATION 6.901 • n=60 Participants
Median EF (%) for rEF (≤40%) subjects
26.50 percent
n=40 Participants
25.00 percent
n=20 Participants
25.00 percent
n=60 Participants

PRIMARY outcome

Timeframe: Baseline to Week 4

Population: The modified Intention to Treat (mITT) Population will consist of all randomized subjects who received at least one dose of CRD-740 or placebo. Subjects will be analyzed according to their randomized treatment, regardless of actual treatment received, treatment compliance, or treatment duration.

Efficacy: To assess the effect of CRD-740 compared to placebo in plasma cGMP at Week 4 in subjects with CHFrEF.

Outcome measures

Outcome measures
Measure
CRD-740
n=30 Participants
Part A: Participants in Part A randomly assigned to this arm will take CRD-740 at two ascending dose levels over 12 weeks. CRD-740: Tablets administered orally.
Placebo
n=15 Participants
Part A: Participants in Part A randomly assigned to this arm will take placebo at two ascending dose levels over 12 weeks. Placebo: Tablets administered orally.
Part A: The Mean Change From Baseline (Day 1) in Plasma cGMP at Week 4.
19.139 AUC 0-6hr (hr*nmol/L)
Standard Deviation 26.9007
-8.822 AUC 0-6hr (hr*nmol/L)
Standard Deviation 31.3357

Adverse Events

Period 1: CRD-740

Serious events: 1 serious events
Other events: 1 other events
Deaths: 0 deaths

Period 1: Placebo

Serious events: 0 serious events
Other events: 1 other events
Deaths: 0 deaths

Period 2: CRD-740

Serious events: 1 serious events
Other events: 3 other events
Deaths: 0 deaths

Period 2: Placebo

Serious events: 0 serious events
Other events: 1 other events
Deaths: 0 deaths

Period 3: CRD-740

Serious events: 0 serious events
Other events: 4 other events
Deaths: 0 deaths

Period 3: Placebo

Serious events: 1 serious events
Other events: 1 other events
Deaths: 0 deaths

Overall CRD-740

Serious events: 3 serious events
Other events: 5 other events
Deaths: 0 deaths

Overall Placebo

Serious events: 3 serious events
Other events: 3 other events
Deaths: 0 deaths

Serious adverse events

Serious adverse events
Measure
Period 1: CRD-740
n=40 participants at risk
CRD-740 10 mg was administered BID to randomly assigned participants in this period from Day 1 through Day 14.
Period 1: Placebo
n=20 participants at risk
CRD-740 10 mg matching placebo was administered BID to randomly assigned participants in this period from Day 1 through Day 14.
Period 2: CRD-740
n=38 participants at risk
CRD-740 25 mg was administered BID to randomly assigned participants in this period from Day 15 through Day 28.
Period 2: Placebo
n=19 participants at risk
CRD-740 25 mg matching placebo was administered BID to randomly assigned participants in this period from Day 15 through Day 28.
Period 3: CRD-740
n=36 participants at risk
CRD-740 25 mg was administered BID to randomly assigned participants in this period from Day 29 through Day 84.
Period 3: Placebo
n=19 participants at risk
CRD-740 25 mg matching placebo was administered BID to randomly assigned participants in this period from Day 29 through Day 84.
Overall CRD-740
n=40 participants at risk
Part A: Participants in Part A randomly assigned to this arm will take CRD-740 at two ascending dose levels over 12 weeks plus a 4-week follow-up period. CRD-740: Tablets administered orally. Part B of the study was not conducted in favor of redesigned new studies.
Overall Placebo
n=20 participants at risk
Part A: Participants in Part A randomly assigned to this arm will take placebo at two ascending dose levels over 12 weeks plus a 4-week follow-up period. Placebo: Tablets administered orally. Part B of the study was not conducted in favor of redesigned new studies.
Cardiac disorders
Ventricular tachycardia
0.00%
0/40 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/20 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/38 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/19 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/36 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
5.3%
1/19 • Number of events 1 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/40 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
5.0%
1/20 • Number of events 1 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
Respiratory, thoracic and mediastinal disorders
Acute respiratory failure
0.00%
0/40 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/20 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/38 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/19 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/36 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/19 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/40 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
5.0%
1/20 • Number of events 1 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
Infections and infestations
Pneumonia
0.00%
0/40 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/20 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
2.6%
1/38 • Number of events 1 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/19 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/36 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/19 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
2.5%
1/40 • Number of events 1 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
5.0%
1/20 • Number of events 1 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
Infections and infestations
Influenza
2.5%
1/40 • Number of events 1 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/20 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/38 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/19 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/36 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/19 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
2.5%
1/40 • Number of events 1 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/20 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
Nervous system disorders
Cerebrovascular accident
0.00%
0/40 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/20 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/38 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/19 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/36 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/19 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
2.5%
1/40 • Number of events 1 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/20 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
Cardiac disorders
Cardiac failure congestive
0.00%
0/40 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/20 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/38 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/19 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/36 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/19 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/40 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
5.0%
1/20 • Number of events 1 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
Renal and urinary disorders
Renal mass
0.00%
0/40 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/20 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/38 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/19 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/36 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/19 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/40 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
5.0%
1/20 • Number of events 1 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.

Other adverse events

Other adverse events
Measure
Period 1: CRD-740
n=40 participants at risk
CRD-740 10 mg was administered BID to randomly assigned participants in this period from Day 1 through Day 14.
Period 1: Placebo
n=20 participants at risk
CRD-740 10 mg matching placebo was administered BID to randomly assigned participants in this period from Day 1 through Day 14.
Period 2: CRD-740
n=38 participants at risk
CRD-740 25 mg was administered BID to randomly assigned participants in this period from Day 15 through Day 28.
Period 2: Placebo
n=19 participants at risk
CRD-740 25 mg matching placebo was administered BID to randomly assigned participants in this period from Day 15 through Day 28.
Period 3: CRD-740
n=36 participants at risk
CRD-740 25 mg was administered BID to randomly assigned participants in this period from Day 29 through Day 84.
Period 3: Placebo
n=19 participants at risk
CRD-740 25 mg matching placebo was administered BID to randomly assigned participants in this period from Day 29 through Day 84.
Overall CRD-740
n=40 participants at risk
Part A: Participants in Part A randomly assigned to this arm will take CRD-740 at two ascending dose levels over 12 weeks plus a 4-week follow-up period. CRD-740: Tablets administered orally. Part B of the study was not conducted in favor of redesigned new studies.
Overall Placebo
n=20 participants at risk
Part A: Participants in Part A randomly assigned to this arm will take placebo at two ascending dose levels over 12 weeks plus a 4-week follow-up period. Placebo: Tablets administered orally. Part B of the study was not conducted in favor of redesigned new studies.
Metabolism and nutrition disorders
Hypokalaemia
0.00%
0/40 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/20 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
2.6%
1/38 • Number of events 1 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/19 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/36 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/19 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
2.5%
1/40 • Number of events 1 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/20 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
Nervous system disorders
Dizziness postural
0.00%
0/40 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
5.0%
1/20 • Number of events 1 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/38 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/19 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/36 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/19 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/40 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
5.0%
1/20 • Number of events 1 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
Eye disorders
Scleritis
0.00%
0/40 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/20 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/38 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/19 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/36 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
5.3%
1/19 • Number of events 1 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/40 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
5.0%
1/20 • Number of events 1 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
Ear and labyrinth disorders
Vertigo
0.00%
0/40 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/20 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/38 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/19 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
2.8%
1/36 • Number of events 1 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/19 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
2.5%
1/40 • Number of events 1 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/20 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
Respiratory, thoracic and mediastinal disorders
Dry throat
2.5%
1/40 • Number of events 1 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/20 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/38 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/19 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/36 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/19 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
2.5%
1/40 • Number of events 1 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/20 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
Respiratory, thoracic and mediastinal disorders
Throat irritation
2.5%
1/40 • Number of events 1 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/20 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/38 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/19 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/36 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/19 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
2.5%
1/40 • Number of events 1 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/20 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
Gastrointestinal disorders
Abdominal pain
0.00%
0/40 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/20 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
2.6%
1/38 • Number of events 1 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/19 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/36 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/19 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
2.5%
1/40 • Number of events 1 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/20 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
Gastrointestinal disorders
Diarrhea
0.00%
0/40 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/20 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
2.6%
1/38 • Number of events 2 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/19 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
2.8%
1/36 • Number of events 2 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/19 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
2.5%
1/40 • Number of events 4 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/20 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
Musculoskeletal and connective tissue disorders
Bone pain
0.00%
0/40 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/20 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/38 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/19 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
2.8%
1/36 • Number of events 1 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/19 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
2.5%
1/40 • Number of events 1 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/20 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
Renal and urinary disorders
Haematuria
0.00%
0/40 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/20 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/38 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
5.3%
1/19 • Number of events 1 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/36 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/19 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/40 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
5.0%
1/20 • Number of events 1 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
Injury, poisoning and procedural complications
Overdose
0.00%
0/40 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/20 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/38 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/19 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
2.8%
1/36 • Number of events 1 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/19 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
2.5%
1/40 • Number of events 1 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.
0.00%
0/20 • Through week 12 plus a 4-week follow-up period.
For Part A, the primary safety analysis was performed by reporting the exposure-adjusted incidence rates in subject-years for AEs and SAEs defined as the number of subjects with that particular AE or SAE within an SOC or PT during the relevant period divided by the sum of the at-risk times.

Additional Information

James Udelson, MD

Tufts Medical Center

Phone: (617) 636-8066

Results disclosure agreements

  • Principal investigator is a sponsor employee
  • Publication restrictions are in place