A Pharmacokinetic Study to Evaluate the Drug Interaction Between HRS5091 and Probe Drugs in Healthy Volunteers

NCT ID: NCT05273775

Last Updated: 2022-12-23

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

22 participants

Study Classification

INTERVENTIONAL

Study Start Date

2022-04-29

Study Completion Date

2022-06-23

Brief Summary

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This is a drug-drug interaction study conducted in healthy volunteers to evaluate the effect of HRS5091 on CYP3A4, CYP2C9, CYP2C19, P-gp, BCRP and OATP1B1, using midazolam, s-warfarin, omeprazole, digoxin and rosuvastatin as probe drugs.

Detailed Description

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Conditions

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Chronic Hepatitis B

Study Design

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Allocation Method

NA

Intervention Model

SINGLE_GROUP

Single-center, single arm, open-label, fixed sequence, self-control
Primary Study Purpose

BASIC_SCIENCE

Blinding Strategy

NONE

Study Groups

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single arm

HRS5091 + probe drugs (Midazolam Maleate Tablets+Warfarin Sodium Tablets+ Omeprazole Enteric Capsules+ Digoxin Tablets+ Rosuvastatin Calcium) + Vitamin K1 Tablets

Group Type EXPERIMENTAL

HRS5091 Tablets

Intervention Type DRUG

HRS5091 Tablets once daily

Midazolam Maleate Tablets

Intervention Type DRUG

Midazolam Maleate Tablets single dose

Warfarin Sodium Tablets

Intervention Type DRUG

Warfarin Sodium Tablets single dose

Omeprazole Enteric Capsules

Intervention Type DRUG

Omeprazole Enteric Capsules single dose

Vitamin K1 Tablets

Intervention Type DRUG

Vitamin K1 Tablets once daily

Digoxin Tablets

Intervention Type DRUG

Digoxin Tablets single dose

Rosuvastatin Calcium Tablets

Intervention Type DRUG

Rosuvastatin Calcium Tablets single dose

Interventions

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HRS5091 Tablets

HRS5091 Tablets once daily

Intervention Type DRUG

Midazolam Maleate Tablets

Midazolam Maleate Tablets single dose

Intervention Type DRUG

Warfarin Sodium Tablets

Warfarin Sodium Tablets single dose

Intervention Type DRUG

Omeprazole Enteric Capsules

Omeprazole Enteric Capsules single dose

Intervention Type DRUG

Vitamin K1 Tablets

Vitamin K1 Tablets once daily

Intervention Type DRUG

Digoxin Tablets

Digoxin Tablets single dose

Intervention Type DRUG

Rosuvastatin Calcium Tablets

Rosuvastatin Calcium Tablets single dose

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

1. The subject can communicate well with the researcher, understand and comply with the requirements of this study, and understand and sign the informed consent;
2. Healthy subjects aged 18\~50 (including 18 and 50 years old);
3. Body weight ≥ 50 kg, body mass index (BMI) within the range of 19 \~ 26 kg /m2 (including 19 and 26 kg/m2) (BMI= weight (kg)/height2 (m2));
4. Give informed consent not to have a family plan for six months after the last dose, and agree to take effective contraception.

Exclusion Criteria

1. Has the medicine or food allergy history, or is the allergic constitution person;
2. Inability to swallow, chronic diarrhea and intestinal obstruction, or the presence of a variety of other factors affecting drug use and absorption;
3. QTCF \> 450 ms in 12-lead ECG examination or other abnormal conditions judged by the researchers to have clinical significance;
4. Hepatitis B surface Antigen (HBSAG), Hepatitis C virus antibody, human immunodeficiency virus (HIV) antibody, syphilis antibody test positive;
5. Those who smoked more than 5 cigarettes per day within 3 months before screening and could not stop using any tobacco products during the trial period;
6. Regular drinkers who had consumed more than 14 units of alcohol per week (1 unit = 285 ml of beer, 25 ml of spirits, or 100 ml of wine) during the six months prior to screening and could not stop using any alcoholic product during the trial; positive Breath test for alcohol;
7. Having a history of drug abuse, drug dependence (consultation) or positive urine drug abuse screening before drug administration;
8. Anyone who has undergone any surgery within 6 months prior to screening;
9. Clinical trial participants who have participated in any drug or medical device within 3 months prior to screening (subject to the intervention of the experimental drug or medical device);10.Blood donation (or blood loss) within 3 months before screening and the amount of blood donation (or blood loss)≥400 ml, or receiving blood transfusion.
Minimum Eligible Age

18 Years

Maximum Eligible Age

50 Years

Eligible Sex

MALE

Accepts Healthy Volunteers

Yes

Sponsors

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Jiangsu HengRui Medicine Co., Ltd.

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Locations

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The Second Affiliated Hospital of Guangzhou Medical University

Guangzhou, Guangdong, China

Site Status

Countries

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China

Other Identifiers

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HRS5091-102

Identifier Type: -

Identifier Source: org_study_id