Trial Outcomes & Findings for PET Imaging of Cyclooxygenase in Multiple Sclerosis (NCT NCT05062083)

NCT ID: NCT05062083

Last Updated: 2024-06-27

Results Overview

Standard uptake value (SUV) was measured by averaging the SUV of all lesion voxels or tissue contralateral to lesion voxels in the PET image with injection of \[11C\]PS13. The SUVR was calculated by averaging the SUV ratio between lesion or tissue contralateral to lesion voxels and the caudate from 60-90 minutes after the start of the PET scan.

Recruitment status

TERMINATED

Study phase

PHASE2

Target enrollment

7 participants

Primary outcome timeframe

60-90 minutes after the start of PET scan

Results posted on

2024-06-27

Participant Flow

Of the seven participants who were consented to the study, two participants were screen failure.

Participant milestones

Participant milestones
Measure
Participants With Multiple Sclerosis
Participants had two brain positron emission tomography (PET) scan visits. In one visit, participants had a baseline \[11C\]PS13 scan followed by a second \[11C\]PS13 scan after blockade with ketoprofen 75 mg orally. In another visit, participants had baseline \[11C\]MC1 scan followed by a second scan with \[11C\]MC1 after blockade by a dose of celecoxib 600 mg orally. Participants receive injection of up to 20 millicurie (mCi) of \[11C\]PS13 or \[11C\]MC1 during each scan.
Overall Study
STARTED
5
Overall Study
COMPLETED
5
Overall Study
NOT COMPLETED
0

Reasons for withdrawal

Withdrawal data not reported

Baseline Characteristics

PET Imaging of Cyclooxygenase in Multiple Sclerosis

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
Participants With Multiple Sclerosis
n=5 Participants
Participants had two brain positron emission tomography (PET) scan visits. In one visit, participants had a baseline \[11C\]PS13 scan followed by a second \[11C\]PS13 scan after blockade with ketoprofen 75 mg orally. In another visit, participants had baseline \[11C\]MC1 scan followed by a second scan with \[11C\]MC1 after blockade by a dose of celecoxib 600 mg orally. Participants receive injection of up to 20 millicurie (mCi) of \[11C\]PS13 or \[11C\]MC1 during each scan.
Age, Categorical
<=18 years
0 Participants
n=93 Participants
Age, Categorical
Between 18 and 65 years
5 Participants
n=93 Participants
Age, Categorical
>=65 years
0 Participants
n=93 Participants
Sex: Female, Male
Female
5 Participants
n=93 Participants
Sex: Female, Male
Male
0 Participants
n=93 Participants
Ethnicity (NIH/OMB)
Hispanic or Latino
0 Participants
n=93 Participants
Ethnicity (NIH/OMB)
Not Hispanic or Latino
5 Participants
n=93 Participants
Ethnicity (NIH/OMB)
Unknown or Not Reported
0 Participants
n=93 Participants
Race (NIH/OMB)
American Indian or Alaska Native
0 Participants
n=93 Participants
Race (NIH/OMB)
Asian
0 Participants
n=93 Participants
Race (NIH/OMB)
Native Hawaiian or Other Pacific Islander
0 Participants
n=93 Participants
Race (NIH/OMB)
Black or African American
0 Participants
n=93 Participants
Race (NIH/OMB)
White
5 Participants
n=93 Participants
Race (NIH/OMB)
More than one race
0 Participants
n=93 Participants
Race (NIH/OMB)
Unknown or Not Reported
0 Participants
n=93 Participants
Region of Enrollment
United States
5 participants
n=93 Participants

PRIMARY outcome

Timeframe: 60-90 minutes after the start of PET scan

Population: The analyses included only subjects who completed the study.

Standard uptake value (SUV) was measured by averaging the SUV of all lesion voxels or tissue contralateral to lesion voxels in the PET image with injection of \[11C\]PS13. The SUVR was calculated by averaging the SUV ratio between lesion or tissue contralateral to lesion voxels and the caudate from 60-90 minutes after the start of the PET scan.

Outcome measures

Outcome measures
Measure
Participants With Multiple Sclerosis
n=5 Participants
Participants had two brain positron emission tomography (PET) scan visits. In one visit, participants had a baseline \[11C\]PS13 scan followed by a second \[11C\]PS13 scan after blockade with ketoprofen 75 mg orally. In another visit, participants had baseline \[11C\]MC1 scan followed by a second scan with \[11C\]MC1 after blockade by a dose of celecoxib 600 mg orally. Participants receive injection of up to 20 millicurie (mCi) of \[11C\]PS13 or \[11C\]MC1 during each scan.
Standard Uptake Value Ratio (SUVR) of Lesions With Injection of [11C]PS13
Brain lesions
1.380 SUV Ratio (SUVR)
Standard Deviation 0.112
Standard Uptake Value Ratio (SUVR) of Lesions With Injection of [11C]PS13
Contralateral normal appearing brain tissues
1.408 SUV Ratio (SUVR)
Standard Deviation 0.109

PRIMARY outcome

Timeframe: 60-90 minutes after the start of PET scan

Population: The analyses included only subjects who completed the study.

Standard uptake value (SUV) was measured by averaging the SUV of all lesion voxels or tissue contralateral to lesion voxels in the PET image with injection of \[11C\]MC1. The SUVR was calculated by averaging the SUV ratio between lesion or tissue contralateral to lesion voxels and the cerebellum from 60-90 minutes after the start of the PET scan.

Outcome measures

Outcome measures
Measure
Participants With Multiple Sclerosis
n=5 Participants
Participants had two brain positron emission tomography (PET) scan visits. In one visit, participants had a baseline \[11C\]PS13 scan followed by a second \[11C\]PS13 scan after blockade with ketoprofen 75 mg orally. In another visit, participants had baseline \[11C\]MC1 scan followed by a second scan with \[11C\]MC1 after blockade by a dose of celecoxib 600 mg orally. Participants receive injection of up to 20 millicurie (mCi) of \[11C\]PS13 or \[11C\]MC1 during each scan.
Standard Uptake Value Ratio (SUVR) of Lesions With Injection of [11C]MC1
Brain lesions
1.455 SUV Ratio (SUVR)
Standard Deviation 0.142
Standard Uptake Value Ratio (SUVR) of Lesions With Injection of [11C]MC1
Contralateral normal appearing brain tissues
1.594 SUV Ratio (SUVR)
Standard Deviation 0.120

PRIMARY outcome

Timeframe: 60-90 minutes after the start of PET scan

Population: The analyses included only subjects who completed the study.

Calculation of standard uptake value (SUV) by averaging the SUV of all lesion voxels or tissue contralateral to lesion voxels in the PET image with injection of \[11C\]PS13 after blockade with ketoprofen. Calculation of SUVR by averaging the SUV ratio between lesion or tissue contralateral to lesion voxels and the caudate from 60-90 minutes after the start of the PET scan.

Outcome measures

Outcome measures
Measure
Participants With Multiple Sclerosis
n=5 Participants
Participants had two brain positron emission tomography (PET) scan visits. In one visit, participants had a baseline \[11C\]PS13 scan followed by a second \[11C\]PS13 scan after blockade with ketoprofen 75 mg orally. In another visit, participants had baseline \[11C\]MC1 scan followed by a second scan with \[11C\]MC1 after blockade by a dose of celecoxib 600 mg orally. Participants receive injection of up to 20 millicurie (mCi) of \[11C\]PS13 or \[11C\]MC1 during each scan.
Standard Uptake Value Ratio (SUVR) of Lesions With Injection of [11C]PS13 After Blockade With Ketoprofen
NA SUV Ratio (SUVR)
Standard Deviation NA
Insufficient imaging signal above the lower limit of quantitation (LLOQ)

PRIMARY outcome

Timeframe: 60-90 minutes after the start of PET scan

Population: The analyses included only subjects who completed the study.

Calculation of standard uptake value (SUV) by averaging the SUV of all lesion voxels or tissue contralateral to lesion voxels in the PET image with injection of \[11C\]MC1 after blockade with celecoxib. Calculation of SUVR by averaging the SUV ratio between lesion or tissue contralateral to lesion voxels and the cerebellum from 60-90 minutes after the start of the PET scan.

Outcome measures

Outcome measures
Measure
Participants With Multiple Sclerosis
n=5 Participants
Participants had two brain positron emission tomography (PET) scan visits. In one visit, participants had a baseline \[11C\]PS13 scan followed by a second \[11C\]PS13 scan after blockade with ketoprofen 75 mg orally. In another visit, participants had baseline \[11C\]MC1 scan followed by a second scan with \[11C\]MC1 after blockade by a dose of celecoxib 600 mg orally. Participants receive injection of up to 20 millicurie (mCi) of \[11C\]PS13 or \[11C\]MC1 during each scan.
Standard Uptake Value Ratio (SUVR) of Lesions With Injection of [11C]MC1 After Blockade With Celecoxib
NA SUV Ratio (SUVR)
Standard Deviation NA
Insufficient imaging signal above the lower limit of quantitation (LLOQ)

SECONDARY outcome

Timeframe: 60-90 minutes after the start of PET scan

Population: The analyses included only subjects who completed the study.

Chronic active lesion is defined as the white matter lesion with paramagnetic outer rim in quantitative susceptibility maps (QSM). Standard uptake value (SUV) was measured by averaging the SUV of chronic active lesion voxels or contralateral normal appearing brain tissues in the \[11C\]PS13 PET image. The SUVR was calculated by averaging the SUV ratio between chronic active lesion or tissue contralateral to lesion voxels and the caudate from 60-90 minutes after the start of the PET scan.

Outcome measures

Outcome measures
Measure
Participants With Multiple Sclerosis
n=5 Participants
Participants had two brain positron emission tomography (PET) scan visits. In one visit, participants had a baseline \[11C\]PS13 scan followed by a second \[11C\]PS13 scan after blockade with ketoprofen 75 mg orally. In another visit, participants had baseline \[11C\]MC1 scan followed by a second scan with \[11C\]MC1 after blockade by a dose of celecoxib 600 mg orally. Participants receive injection of up to 20 millicurie (mCi) of \[11C\]PS13 or \[11C\]MC1 during each scan.
Standard Uptake Value Ratio (SUVR) of Chronic Active Lesions With Injection of [11C]PS13
Chronic active lesion
1.424 SUV Ratio (SUVR)
Standard Deviation 0.033
Standard Uptake Value Ratio (SUVR) of Chronic Active Lesions With Injection of [11C]PS13
Contralateral normal appearing brain tissues
1.455 SUV Ratio (SUVR)
Standard Deviation 0.196

SECONDARY outcome

Timeframe: 60-90 minutes after the start of PET scan

Population: The analyses included only subjects who completed the study.

Chronic active lesion is defined as the white matter lesion with paramagnetic outer rim in quantitative susceptibility maps (QSM). Standard uptake value (SUV) was measured by averaging the SUV of chronic active lesion voxels or contralateral normal appearing brain tissues in the \[11C\]MC1 PET image. The SUVR was calculated by averaging the SUV ratio between chronic active lesion or tissue contralateral to lesion voxels and the cerebellum from 60-90 minutes after the start of the PET scan.

Outcome measures

Outcome measures
Measure
Participants With Multiple Sclerosis
n=5 Participants
Participants had two brain positron emission tomography (PET) scan visits. In one visit, participants had a baseline \[11C\]PS13 scan followed by a second \[11C\]PS13 scan after blockade with ketoprofen 75 mg orally. In another visit, participants had baseline \[11C\]MC1 scan followed by a second scan with \[11C\]MC1 after blockade by a dose of celecoxib 600 mg orally. Participants receive injection of up to 20 millicurie (mCi) of \[11C\]PS13 or \[11C\]MC1 during each scan.
Standard Uptake Value Ratio (SUVR) of Chronic Active Lesions With Injection of [11C]MC1
Chronic active lesion
1.562 SUV Ratio (SUVR)
Standard Deviation 0.080
Standard Uptake Value Ratio (SUVR) of Chronic Active Lesions With Injection of [11C]MC1
Contralateral normal appearing brain tissues
1.724 SUV Ratio (SUVR)
Standard Deviation 0.143

Adverse Events

Participants With Multiple Sclerosis

Serious events: 0 serious events
Other events: 0 other events
Deaths: 0 deaths

Serious adverse events

Adverse event data not reported

Other adverse events

Adverse event data not reported

Additional Information

Dr. Robert Innis

National Institute of Mental Health (NIMH)

Phone: 301-594-1368

Results disclosure agreements

  • Principal investigator is a sponsor employee
  • Publication restrictions are in place