Combination Study of RMC-4630 and Sotorasib for NSCLC Subjects With KRASG12C Mutation After Failure of Prior Standard Therapies

NCT ID: NCT05054725

Last Updated: 2026-01-06

Study Results

Results available

Outcome measurements, participant flow, baseline characteristics, and adverse events have been published for this study.

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE2

Total Enrollment

47 participants

Study Classification

INTERVENTIONAL

Study Start Date

2021-12-30

Study Completion Date

2024-08-29

Brief Summary

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The purpose of this study is to evaluate the antitumor effects of sotorasib and RMC-4630 in subjects with KRASG12C mutant NSCLC

Detailed Description

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This is a phase 2 multicenter, open-label study evaluating the efficacy, safety, tolerability, and pharmacokinetics (PK) of RMC-4630 in combination with sotorasib in subjects with KRASG12C mutant NSCLC after failure of prior standard therapies.

Conditions

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Non-Small Cell Lung Cancer

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

SEQUENTIAL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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RMC-4630 and sotorasib, Safety Run-in

Safety Run-In:

RMC-4630 and sotorasib

Group Type EXPERIMENTAL

RMC-4630

Intervention Type DRUG

RMC-4630 administered orally as a capsule

Sotorasib

Intervention Type DRUG

Sotorasib administered orally as a tablet

RMC-4630 and sotorasib, Expansion

Dose Expansion:

RMC-4630 and sotorasib

Group Type EXPERIMENTAL

RMC-4630

Intervention Type DRUG

RMC-4630 administered orally as a capsule

Sotorasib

Intervention Type DRUG

Sotorasib administered orally as a tablet

Interventions

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RMC-4630

RMC-4630 administered orally as a capsule

Intervention Type DRUG

Sotorasib

Sotorasib administered orally as a tablet

Intervention Type DRUG

Other Intervention Names

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SAR442720 AMG 510 Lumakras

Eligibility Criteria

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Inclusion Criteria

* Subject must be ≥18 years of age.
* Subject must have pathologically documented, locally advanced or metastatic KRASG12C NSCLC (not amenable to curative surgery) that has progressed on prior standard therapies (no more than 3 prior lines of therapies are allowed)

Exclusion Criteria

* Primary central nervous system (CNS) tumors
* Known or suspected leptomeningeal or brain metastases or spinal cord compression
* Clinically significant cardiac disease
* Known impairment of GI function that would alter the absorption
* Active autoimmune disease requiring systemic treatment within past 2 years
* History of severe allergic reactions to any of the study intervention components
* Major surgical procedures within 28 days or non-study-related minor procedures within 7 days of treatment.
* Prior therapy with KRASG12C inhibitor and/or SHP2 inhibitor
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Sanofi

INDUSTRY

Sponsor Role collaborator

Amgen

INDUSTRY

Sponsor Role collaborator

Revolution Medicines, Inc.

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Revolution Medicines, Inc.

Role: STUDY_DIRECTOR

Revolution Medicines, Inc.

Locations

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Florida Cancer Specialists

Fort Myers, Florida, United States

Site Status

BRCR Medical Center Inc.

Plantation, Florida, United States

Site Status

Cancer Specialists of North Florida

Saint Augustine, Florida, United States

Site Status

GenHarp Clinical Solutions

Evergreen Park, Illinois, United States

Site Status

Hematology Oncology Clinic

Baton Rouge, Louisiana, United States

Site Status

New England Cancer Specialists

Scarborough, Maine, United States

Site Status

American Oncology Partners of Maryland, PA

Bethesda, Maryland, United States

Site Status

Maryland Oncology Hematology, P.A.

Columbia, Maryland, United States

Site Status

Minnesota Oncology Hematology, P.A.

Minneapolis, Minnesota, United States

Site Status

Nebraska Cancer Specialists

Omaha, Nebraska, United States

Site Status

Comprehensive Cancer Centers of Nevada

Las Vegas, Nevada, United States

Site Status

New Jersey Center for Cancer Research

Brick, New Jersey, United States

Site Status

University of New Mexico Comprehensive Cancer Center

Albuquerque, New Mexico, United States

Site Status

Roswell Park cancer Institute

Buffalo, New York, United States

Site Status

Clinical Research Alliance, Inc.

New York, New York, United States

Site Status

Zangmeister Cancer Center

Columbus, Ohio, United States

Site Status

Charleston Oncology

Charleston, South Carolina, United States

Site Status

Tennessee Oncology

Chattanooga, Tennessee, United States

Site Status

Sarah Cannon Research Institute

Nashville, Tennessee, United States

Site Status

CHRISTUS St. Michael-Colom and Carney Clinic P.A

Texarkana, Texas, United States

Site Status

Virginia Cancer Specialists

Fairfax, Virginia, United States

Site Status

Virginia Oncology Associates

Norfolk, Virginia, United States

Site Status

Northwest Cancer specialists, P.C.

Vancouver, Washington, United States

Site Status

South West Oncology

Warrnambool, Victoria, Australia

Site Status

Blacktown Hospital

Blacktown, , Australia

Site Status

Goulburn Valley Health

Shepparton, , Australia

Site Status

Cross Cancer Institute

Edmonton, Alberta, Canada

Site Status

William Osler Health System

Mississauga, Ontario, Canada

Site Status

APHM Hopital Nord, Service d'Oncologie Multidisciplinaire et innovations therapeutics

Marseille, , France

Site Status

Hospital Larrey Universite Paul Sabatier

Toulouse, , France

Site Status

Klinikum Esslingen GmbH

Esslingen am Neckar, Baden-Wurttemberg, Germany

Site Status

Asklepios Fachkliniken Munchen

Gauting, Bavaria, Germany

Site Status

Lungenklinik Hemer

Hemer, North Rhine-Westphalia, Germany

Site Status

Bethanien Hospital Moers

Moers, North Rhine-Westphalia, Germany

Site Status

Comprehensive Cancer Center Mainfranken, University Wuerzburg

Homburg, Saarland, Germany

Site Status

Lung Cancer Center, University of Saarland

Homburg, Saarland, Germany

Site Status

POIS Sachsen GmbH

Leipzig, Saxony, Germany

Site Status

Charite Benjamin Franklin Comprehensive Cancer center

Berlin, , Germany

Site Status

Evangelische Lung Clinic

Berlin, , Germany

Site Status

Hamato-Onkologie Hamburg

Hamburg, , Germany

Site Status

Azienda Ospedaliera dei Colli

Napoli, Campania, Italy

Site Status

Azienda Sanitaria Ospedaliera S Luigi Gonzaga

Orbassano, Piedmont, Italy

Site Status

Istituto Europeo Di Oncologia

Milan, , Italy

Site Status

Chungbuk National University Hospital

Cheongju-si, , South Korea

Site Status

Seoul National University Hospital

Seoul, , South Korea

Site Status

Asan Medical Center

Seoul, , South Korea

Site Status

Samsung Medical Center

Seoul, , South Korea

Site Status

Hospital Universitario Virgen Macarena

Seville, Andalusia, Spain

Site Status

Hospital Clinic de Barcelona

Barcelona, Catalonia, Spain

Site Status

Complejo Hospitalario Universitario A Coruña

A Coruña, Galicia, Spain

Site Status

Clinica Universidad de Navarra

Pamplona, Navarre, Spain

Site Status

Clinica Universidad de Navarra

Madrid, , Spain

Site Status

Hospital Universitario y Politecnico La Fe

Valencia, , Spain

Site Status

Kaohsiung Medical University Chung Ho Memorial Hospital

Kaohsiung City, , Taiwan

Site Status

E-DA Hospital

Kaohsiung City, , Taiwan

Site Status

Taichung Veterans General Hospital

Taichung, , Taiwan

Site Status

National Cheng Kung University Hospital

Tainan, , Taiwan

Site Status

National Taiwan University Hospital

Taipei, , Taiwan

Site Status

The Christie NHS Foundation Trust

Manchester, Greater Manchester, United Kingdom

Site Status

The Royal Marsden NHS Foundation Trust

Sutton, Surrey, United Kingdom

Site Status

Countries

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United States Australia Canada France Germany Italy South Korea Spain Taiwan United Kingdom

Provided Documents

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Document Type: Study Protocol

View Document

Document Type: Statistical Analysis Plan

View Document

Other Identifiers

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RMC-4630-03

Identifier Type: -

Identifier Source: org_study_id

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