A Study of GFH018 in Patients With Advanced Solid Tumors

NCT ID: NCT05051241

Last Updated: 2024-03-01

Study Results

Results available

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

50 participants

Study Classification

INTERVENTIONAL

Study Start Date

2019-08-30

Study Completion Date

2022-08-11

Brief Summary

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This is the first- in human study of GFH018 comprised of a dose escalation part and a dose expansion part in subjects with advanced solid tumors after single/multiple administration. The study is designed to explore the safety/tolerability, pharmacokinetics, and MTD of GFH018 and to define a RP2D of GFH018.

Detailed Description

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Conditions

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Advanced Solid Tumor

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

SINGLE_GROUP

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Dose escalation Cohort 1

5 mg BID, 14d-on/14d-off

Group Type EXPERIMENTAL

GFH018

Intervention Type DRUG

Subjects will receive GFH018 orally at different dose levels following twice daily, 14-day on/14-day off regimen. Other dose regimens, eg 7d-on/7d-off will also be considered to be explored when the safety/tolerability is confirmed.

Dose escalation Cohort 2

10 mg BID, 14d-on/14d-off

Group Type EXPERIMENTAL

GFH018

Intervention Type DRUG

Subjects will receive GFH018 orally at different dose levels following twice daily, 14-day on/14-day off regimen. Other dose regimens, eg 7d-on/7d-off will also be considered to be explored when the safety/tolerability is confirmed.

Dose escalation Cohort 3

20 mg BID, 14d-on/14d-off

Group Type EXPERIMENTAL

GFH018

Intervention Type DRUG

Subjects will receive GFH018 orally at different dose levels following twice daily, 14-day on/14-day off regimen. Other dose regimens, eg 7d-on/7d-off will also be considered to be explored when the safety/tolerability is confirmed.

Dose escalation Cohort 4

30 mg BID, 14d-on/14d-off

Group Type EXPERIMENTAL

GFH018

Intervention Type DRUG

Subjects will receive GFH018 orally at different dose levels following twice daily, 14-day on/14-day off regimen. Other dose regimens, eg 7d-on/7d-off will also be considered to be explored when the safety/tolerability is confirmed.

Dose escalation Cohort 5

40 mg BID, 14d-on/14d-off

Group Type EXPERIMENTAL

GFH018

Intervention Type DRUG

Subjects will receive GFH018 orally at different dose levels following twice daily, 14-day on/14-day off regimen. Other dose regimens, eg 7d-on/7d-off will also be considered to be explored when the safety/tolerability is confirmed.

Dose escalation Cohort 6

50 mg BID, 14d-on/14d-off

Group Type EXPERIMENTAL

GFH018

Intervention Type DRUG

Subjects will receive GFH018 orally at different dose levels following twice daily, 14-day on/14-day off regimen. Other dose regimens, eg 7d-on/7d-off will also be considered to be explored when the safety/tolerability is confirmed.

Dose escalation Cohort 7

65 mg BID, 14d-on/14d-off

Group Type EXPERIMENTAL

GFH018

Intervention Type DRUG

Subjects will receive GFH018 orally at different dose levels following twice daily, 14-day on/14-day off regimen. Other dose regimens, eg 7d-on/7d-off will also be considered to be explored when the safety/tolerability is confirmed.

Dose escalation Cohort 8

85 mg BID, 14d-on/14d-off

Group Type EXPERIMENTAL

GFH018

Intervention Type DRUG

Subjects will receive GFH018 orally at different dose levels following twice daily, 14-day on/14-day off regimen. Other dose regimens, eg 7d-on/7d-off will also be considered to be explored when the safety/tolerability is confirmed.

Dose escalation Cohort 9

85 mg BID, 7d-on/7d-off

Group Type EXPERIMENTAL

GFH018

Intervention Type DRUG

Subjects will receive GFH018 orally at different dose levels following twice daily, 14-day on/14-day off regimen. Other dose regimens, eg 7d-on/7d-off will also be considered to be explored when the safety/tolerability is confirmed.

Dose expansion Cohort 10

85 mg BID, 14d-on/14d-off

Group Type EXPERIMENTAL

GFH018

Intervention Type DRUG

Subjects will receive GFH018 orally at different dose levels following twice daily, 14-day on/14-day off regimen. Other dose regimens, eg 7d-on/7d-off will also be considered to be explored when the safety/tolerability is confirmed.

Interventions

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GFH018

Subjects will receive GFH018 orally at different dose levels following twice daily, 14-day on/14-day off regimen. Other dose regimens, eg 7d-on/7d-off will also be considered to be explored when the safety/tolerability is confirmed.

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

1. Voluntarily participate in this clinical trial and are willing to sign informed consent forms.
2. Male or female aged from 18-75 years old (inclusive).
3. Diagnosed with histologically or cytologically confirmed advanced solid tumors.
4. Evaluable lesions defined by RECIST v1.1.
5. Eastern Cooperative Oncology Group performance status of 0 to 1.
6. Subjects or their legal representatives are able to communicate well with Investigators and are willing to comply with the protocol and complete the study.

Exclusion Criteria

1. With clinically significant cardiac diseases.
2. With clinically significant digestive disorders.
3. Other severe disease.
4. Pregnant or lactating women.
5. Other unfavorable situations for subjects to participate in the study judged by Investigators.
Minimum Eligible Age

18 Years

Maximum Eligible Age

75 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Zhejiang Genfleet Therapeutics Co., Ltd.

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Jin Li, MD

Role: PRINCIPAL_INVESTIGATOR

Leading site

Locations

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Shanghai East hospital

Shanghai, , China

Site Status

Countries

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China

References

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Guo Y, Wang Z, Zhou H, Pan H, Han W, Deng Y, Li Q, Xue J, Ge X, Wang S, Wang J, Zhang Y, Zhao C, Zhu H, Wang Y, Shen H, Liu D, Li J. First-in-human study of GFH018, a small molecule inhibitor of transforming growth factor-beta receptor I inhibitor, in patients with advanced solid tumors. BMC Cancer. 2024 Apr 10;24(1):444. doi: 10.1186/s12885-024-12216-7.

Reference Type DERIVED
PMID: 38600507 (View on PubMed)

Provided Documents

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Document Type: Study Protocol

View Document

Document Type: Statistical Analysis Plan

View Document

Other Identifiers

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GFH018X1101

Identifier Type: -

Identifier Source: org_study_id

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