Trial Outcomes & Findings for A Therapeutic Equivalence Study in Subjects With Primary Open Angle Glaucoma or Ocular Hypertension (NCT NCT05022004)

NCT ID: NCT05022004

Last Updated: 2024-01-18

Results Overview

The recommended primary endpoint is the mean difference in Intraocular Pressure of both eyes between the two treatment groups at pre-specified time points.

Recruitment status

COMPLETED

Study phase

PHASE3

Target enrollment

599 participants

Primary outcome timeframe

Baseline, Week 2 & Week 6

Results posted on

2024-01-18

Participant Flow

Participant milestones

Participant milestones
Measure
BRIN-20-01
Brinzolamide ophthalmic suspension: dose: one drop of study medication; frequency: three times a day; route of administration: Topical ocular administration; duration of therapy: 6 weeks
Azopt®
Azopt®: dose: one drop of study medication; frequency: three times a day; route of administration: Topical ocular administration; duration of therapy: 6 weeks
Overall Study
STARTED
297
300
Overall Study
COMPLETED
287
289
Overall Study
NOT COMPLETED
10
11

Reasons for withdrawal

Withdrawal data not reported

Baseline Characteristics

A Therapeutic Equivalence Study in Subjects With Primary Open Angle Glaucoma or Ocular Hypertension

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
BRIN-20-01
n=297 Participants
Brinzolamide ophthalmic suspension: dose: one drop of study medication; frequency: three times a day; route of administration: Topical ocular administration; duration of therapy: 6 weeks
Azopt®
n=300 Participants
Azopt®: dose: one drop of study medication; frequency: three times a day; route of administration: Topical ocular administration; duration of therapy: 6 weeks
Total
n=597 Participants
Total of all reporting groups
Age, Continuous
61.2 years
STANDARD_DEVIATION 12.01 • n=5 Participants
61.3 years
STANDARD_DEVIATION 12.01 • n=7 Participants
61.2 years
STANDARD_DEVIATION 12.00 • n=5 Participants
Sex: Female, Male
Female
170 Participants
n=5 Participants
174 Participants
n=7 Participants
344 Participants
n=5 Participants
Sex: Female, Male
Male
127 Participants
n=5 Participants
126 Participants
n=7 Participants
253 Participants
n=5 Participants
Race (NIH/OMB)
American Indian or Alaska Native
0 Participants
n=5 Participants
1 Participants
n=7 Participants
1 Participants
n=5 Participants
Race (NIH/OMB)
Asian
99 Participants
n=5 Participants
105 Participants
n=7 Participants
204 Participants
n=5 Participants
Race (NIH/OMB)
Native Hawaiian or Other Pacific Islander
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
Race (NIH/OMB)
Black or African American
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
Race (NIH/OMB)
White
198 Participants
n=5 Participants
194 Participants
n=7 Participants
392 Participants
n=5 Participants
Race (NIH/OMB)
More than one race
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
Race (NIH/OMB)
Unknown or Not Reported
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants

PRIMARY outcome

Timeframe: Baseline, Week 2 & Week 6

The recommended primary endpoint is the mean difference in Intraocular Pressure of both eyes between the two treatment groups at pre-specified time points.

Outcome measures

Outcome measures
Measure
BRIN-20-01
n=273 Participants
Brinzolamide ophthalmic suspension: dose: one drop of study medication; frequency: three times a day; route of administration: Topical ocular administration; duration of therapy: 6 weeks
Azopt®
n=271 Participants
Azopt®: dose: one drop of study medication; frequency: three times a day; route of administration: Topical ocular administration; duration of therapy: 6 weeks
Mean Difference in Intraocular Pressure of Both Eyes Between the Two Treatment Groups
Baseline- Right Eye 08:00
24.87 mmHg
Standard Deviation 2.378
25.12 mmHg
Standard Deviation 2.358
Mean Difference in Intraocular Pressure of Both Eyes Between the Two Treatment Groups
Baseline - Left Eye 10:00
24.54 mmHg
Standard Deviation 2.307
24.83 mmHg
Standard Deviation 2.389
Mean Difference in Intraocular Pressure of Both Eyes Between the Two Treatment Groups
Baeline - Right Eye 10:00
24.52 mmHg
Standard Deviation 2.423
24.90 mmHg
Standard Deviation 2.365
Mean Difference in Intraocular Pressure of Both Eyes Between the Two Treatment Groups
Baseline- Left Eye 08:00
24.92 mmHg
Standard Deviation 2.290
25.06 mmHg
Standard Deviation 2.363
Mean Difference in Intraocular Pressure of Both Eyes Between the Two Treatment Groups
Week 2 - Left Eye 08:00
19.87 mmHg
Standard Deviation 3.436
19.56 mmHg
Standard Deviation 3.642
Mean Difference in Intraocular Pressure of Both Eyes Between the Two Treatment Groups
Week 2 - Right Eye 08:00
19.81 mmHg
Standard Deviation 3.400
19.62 mmHg
Standard Deviation 3.423
Mean Difference in Intraocular Pressure of Both Eyes Between the Two Treatment Groups
Week 2 - Left Eye 10:00
18.87 mmHg
Standard Deviation 3.544
18.39 mmHg
Standard Deviation 3.760
Mean Difference in Intraocular Pressure of Both Eyes Between the Two Treatment Groups
Week 2 - Right Eye 10:00
18.69 mmHg
Standard Deviation 3.572
18.47 mmHg
Standard Deviation 3.468
Mean Difference in Intraocular Pressure of Both Eyes Between the Two Treatment Groups
Week 6 - Left Eye 08:00
18.86 mmHg
Standard Deviation 3.162
18.91 mmHg
Standard Deviation 3.333
Mean Difference in Intraocular Pressure of Both Eyes Between the Two Treatment Groups
Week 6 - Right Eye 08:00
18.87 mmHg
Standard Deviation 3.067
18.99 mmHg
Standard Deviation 3.123
Mean Difference in Intraocular Pressure of Both Eyes Between the Two Treatment Groups
Week 6 - Left Eye 10:00
17.76 mmHg
Standard Deviation 3.252
17.73 mmHg
Standard Deviation 3.418
Mean Difference in Intraocular Pressure of Both Eyes Between the Two Treatment Groups
Week 6 - Right Eye 10:00
17.71 mmHg
Standard Deviation 3.190
17.70 mmHg
Standard Deviation 3.162

SECONDARY outcome

Timeframe: approximately 8:00 AM. (hour 0; before the morning drop) and 10:00 AM. (hour 2) at the Day 14 (Week 2) and Day 42 (Week 6) visits

Outcome measures

Outcome measures
Measure
BRIN-20-01
n=273 Participants
Brinzolamide ophthalmic suspension: dose: one drop of study medication; frequency: three times a day; route of administration: Topical ocular administration; duration of therapy: 6 weeks
Azopt®
n=271 Participants
Azopt®: dose: one drop of study medication; frequency: three times a day; route of administration: Topical ocular administration; duration of therapy: 6 weeks
Change From Baseline in IOP of Both Eyes Between the 2 Treatment Groups.
Week 2 - Right Eye 10:00
-5.82 mmHg
Standard Deviation 3.484
-6.43 mmHg
Standard Deviation 3.630
Change From Baseline in IOP of Both Eyes Between the 2 Treatment Groups.
Week 6- Left Eye 08:00
-5.68 mmHg
Standard Deviation 3.290
-5.92 mmHg
Standard Deviation 3.577
Change From Baseline in IOP of Both Eyes Between the 2 Treatment Groups.
Week 6- Right Eye 08:00
-5.64 mmHg
Standard Deviation 3.107
-5.91 mmHg
Standard Deviation 3.468
Change From Baseline in IOP of Both Eyes Between the 2 Treatment Groups.
Week 2- Left Eye 08:00
-4.67 mmHg
Standard Deviation 3.441
-5.27 mmHg
Standard Deviation 3.617
Change From Baseline in IOP of Both Eyes Between the 2 Treatment Groups.
Week 2- Right Eye 08:00
-4.71 mmHg
Standard Deviation 3.286
-5.28 mmHg
Standard Deviation 3.531
Change From Baseline in IOP of Both Eyes Between the 2 Treatment Groups.
Week 2- Left Eye 10:00
-5.68 mmHg
Standard Deviation 3.475
-6.44 mmHg
Standard Deviation 3.717
Change From Baseline in IOP of Both Eyes Between the 2 Treatment Groups.
Week 6 - Left Eye 10:00
-6.78 mmHg
Standard Deviation 3.329
-7.10 mmHg
Standard Deviation 3.614
Change From Baseline in IOP of Both Eyes Between the 2 Treatment Groups.
Week 6 - Right Eye 10:00
-6.81 mmHg
Standard Deviation 3.239
-7.20 mmHg
Standard Deviation 3.500

Adverse Events

BRIN-20-01

Serious events: 0 serious events
Other events: 49 other events
Deaths: 0 deaths

Azopt®

Serious events: 1 serious events
Other events: 38 other events
Deaths: 0 deaths

Serious adverse events

Serious adverse events
Measure
BRIN-20-01
n=297 participants at risk
Brinzolamide ophthalmic suspension: dose: one drop of study medication; frequency: three times a day; route of administration: Topical ocular administration; duration of therapy: 6 weeks
Azopt®
n=300 participants at risk
Azopt®: dose: one drop of study medication; frequency: three times a day; route of administration: Topical ocular administration; duration of therapy: 6 weeks
Vascular disorders
Hypertensive Crisis
0.00%
0/297 • 7 Weeks
0.33%
1/300 • 7 Weeks

Other adverse events

Other adverse events
Measure
BRIN-20-01
n=297 participants at risk
Brinzolamide ophthalmic suspension: dose: one drop of study medication; frequency: three times a day; route of administration: Topical ocular administration; duration of therapy: 6 weeks
Azopt®
n=300 participants at risk
Azopt®: dose: one drop of study medication; frequency: three times a day; route of administration: Topical ocular administration; duration of therapy: 6 weeks
Cardiac disorders
Arrhythmia
0.34%
1/297 • 7 Weeks
0.00%
0/300 • 7 Weeks
Eye disorders
Abnormal Sensation in Eye
0.34%
1/297 • 7 Weeks
0.00%
0/300 • 7 Weeks
Eye disorders
Blepharitis
0.34%
1/297 • 7 Weeks
0.33%
1/300 • 7 Weeks
Eye disorders
Cataract
0.34%
1/297 • 7 Weeks
0.00%
0/300 • 7 Weeks
Eye disorders
Conjunctival Hyperemia
1.0%
3/297 • 7 Weeks
0.67%
2/300 • 7 Weeks
Eye disorders
Conjunctival Oedema
0.00%
0/297 • 7 Weeks
0.33%
1/300 • 7 Weeks
Eye disorders
Conjunctivitis Allergic
0.00%
0/297 • 7 Weeks
0.67%
2/300 • 7 Weeks
Eye disorders
Dry Eye
0.67%
2/297 • 7 Weeks
0.00%
0/300 • 7 Weeks
Eye disorders
Eye Irritation
1.0%
3/297 • 7 Weeks
0.67%
2/300 • 7 Weeks
Eye disorders
Eye Pain
0.00%
0/297 • 7 Weeks
0.67%
2/300 • 7 Weeks
Eye disorders
Eye Pruritus
0.67%
2/297 • 7 Weeks
0.67%
2/300 • 7 Weeks
Eye disorders
Foreign Body Sensation in Eyes
1.3%
4/297 • 7 Weeks
0.67%
2/300 • 7 Weeks
Eye disorders
Keratitis
0.34%
1/297 • 7 Weeks
0.00%
0/300 • 7 Weeks
Eye disorders
Lacrimation Increased
0.34%
1/297 • 7 Weeks
0.00%
0/300 • 7 Weeks
Eye disorders
Ocular Hyperemia
1.0%
3/297 • 7 Weeks
0.67%
2/300 • 7 Weeks
Eye disorders
Swelling of Eyelid
0.34%
1/297 • 7 Weeks
0.00%
0/300 • 7 Weeks
Eye disorders
Vision Blurred
2.7%
8/297 • 7 Weeks
1.3%
4/300 • 7 Weeks
Eye disorders
Visual Acuity Reduced
0.00%
0/297 • 7 Weeks
0.33%
1/300 • 7 Weeks
Eye disorders
Visual Impairment
0.67%
2/297 • 7 Weeks
0.00%
0/300 • 7 Weeks
Gastrointestinal disorders
Diarrhoea
0.00%
0/297 • 7 Weeks
0.67%
2/300 • 7 Weeks
Gastrointestinal disorders
Dry Mouth
0.34%
1/297 • 7 Weeks
0.00%
0/300 • 7 Weeks
Gastrointestinal disorders
Flatulence
0.00%
0/297 • 7 Weeks
0.33%
1/300 • 7 Weeks
Gastrointestinal disorders
Toothache
0.34%
1/297 • 7 Weeks
0.00%
0/300 • 7 Weeks
General disorders
Asthenia
0.34%
1/297 • 7 Weeks
0.00%
0/300 • 7 Weeks
General disorders
Instillation Site Dryness
0.34%
1/297 • 7 Weeks
0.00%
0/300 • 7 Weeks
General disorders
Instillation Site Pain
0.67%
2/297 • 7 Weeks
0.00%
0/300 • 7 Weeks
General disorders
Instillation Site Pruritus
0.34%
1/297 • 7 Weeks
0.00%
0/300 • 7 Weeks
General disorders
Instillation Site Reaction
0.34%
1/297 • 7 Weeks
0.00%
0/300 • 7 Weeks
General disorders
Malaise
0.34%
1/297 • 7 Weeks
0.00%
0/300 • 7 Weeks
General disorders
Pyrexia
0.34%
1/297 • 7 Weeks
0.33%
1/300 • 7 Weeks
Infections and infestations
Conjunctivitis
0.34%
1/297 • 7 Weeks
0.00%
0/300 • 7 Weeks
Infections and infestations
Nasopharyngitis
0.34%
1/297 • 7 Weeks
0.00%
0/300 • 7 Weeks
Infections and infestations
Respiratory Tract Infection Viral
0.34%
1/297 • 7 Weeks
0.67%
2/300 • 7 Weeks
Injury, poisoning and procedural complications
Ligament Sprain
0.00%
0/297 • 7 Weeks
0.33%
1/300 • 7 Weeks
Investigations
Blood Pressure Increased
0.67%
2/297 • 7 Weeks
0.33%
1/300 • 7 Weeks
Investigations
Intraocular Pressure Increased
0.00%
0/297 • 7 Weeks
0.33%
1/300 • 7 Weeks
Metabolism and nutrition disorders
Hypercholesterolemia
0.34%
1/297 • 7 Weeks
0.00%
0/300 • 7 Weeks
Musculoskeletal and connective tissue disorders
Back Pain
0.00%
0/297 • 7 Weeks
0.33%
1/300 • 7 Weeks
Musculoskeletal and connective tissue disorders
Myalgia
0.34%
1/297 • 7 Weeks
0.00%
0/300 • 7 Weeks
Musculoskeletal and connective tissue disorders
Neck Pain
0.00%
0/297 • 7 Weeks
0.33%
1/300 • 7 Weeks
Musculoskeletal and connective tissue disorders
Osteochondrosis
0.00%
0/297 • 7 Weeks
0.33%
1/300 • 7 Weeks
Nervous system disorders
Dizziness
0.34%
1/297 • 7 Weeks
0.33%
1/300 • 7 Weeks
Nervous system disorders
Dysgeusia
2.0%
6/297 • 7 Weeks
2.7%
8/300 • 7 Weeks
Nervous system disorders
Headache
1.0%
3/297 • 7 Weeks
1.0%
3/300 • 7 Weeks
Reproductive system and breast disorders
Breast Cyst
0.34%
1/297 • 7 Weeks
0.00%
0/300 • 7 Weeks
Respiratory, thoracic and mediastinal disorders
Cough
0.67%
2/297 • 7 Weeks
1.0%
3/300 • 7 Weeks
Respiratory, thoracic and mediastinal disorders
Dyspnoea
0.34%
1/297 • 7 Weeks
0.33%
1/300 • 7 Weeks
Respiratory, thoracic and mediastinal disorders
Respiratory Disorder
0.00%
0/297 • 7 Weeks
0.33%
1/300 • 7 Weeks
Skin and subcutaneous tissue disorders
Alopecia
0.34%
1/297 • 7 Weeks
0.00%
0/300 • 7 Weeks
Vascular disorders
Hypertensive Crisis
0.00%
0/297 • 7 Weeks
0.67%
2/300 • 7 Weeks

Additional Information

Head-Clinical Development

Sun Pharmaceutical Industries Limited

Phone: 2266455645

Results disclosure agreements

  • Principal investigator is a sponsor employee The Sponsor has exclusive rights, including the right of authorship, to all publications concerning Study data and findings. The Institution, the Investigator, and the Co-Investigators are contractually bound not to make any publications, public statements, oral presentations concerning the Study data and findings. The Sponsor shall have the sole right to review, use, publish, and disclose any data, information, or results developed without limitation.
  • Publication restrictions are in place

Restriction type: OTHER