Efficacy and Safety of Metformin Glycinate Compared to Metformin Hydrochloride on the Progression of Type 2 Diabetes

NCT ID: NCT04943692

Last Updated: 2021-06-29

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

SUSPENDED

Clinical Phase

PHASE3

Total Enrollment

500 participants

Study Classification

INTERVENTIONAL

Study Start Date

2021-08-31

Study Completion Date

2021-08-31

Brief Summary

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Phase III study to evaluate the efficacy and safety of the treatment. Two-arm, prospective, longitudinal, double-blind, multicenter randomized clinical trial.

Detailed Description

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Study to evaluate the efficacy and safety of treatment at 6 and 12 months with metformin glycinate at a dose of 2100 mg / day compared to metformin hydrochloride at a dose of 1700 mg / day on the progression of type 2 diabetes. To assess the change in HbA1c from baseline to 6 and 12 months of treatment (primary endpoint) in both groups. As secondary objectives, changes in fasting glucose levels from baseline, changes in results of the oral glucose tolerance test 2h from baseline, changes in HOMA-IR from baseline, changes in insulin levels, leptin, adipokines and proinflammatory cytokines, MCP-1, nitric oxide and PCr from baseline, changes in BMI from baseline and changes in lipid profile from baseline will be evaluated. A blinded interim analysis will be performed at 6 months of patient follow-up and a final analysis. Demographic data will be analyzed with mean, standard deviation, minimum and maximum. Efficacy analyzes will be carried out in the treated population (all treated patients, ATP), made up of all randomized patients who received at least one dose of the study treatment and who have a baseline measurement and at least one subsequent measurement.

Conditions

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Type 2 Diabetes

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

DOUBLE

Participants Investigators

Study Groups

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Group A: Metformin glycinate 1050 mg

Metformin glycinate 1050 mg Orally twice a day.

Group Type EXPERIMENTAL

Metformin glycinate

Intervention Type DRUG

1050 mg, tablets Administered orally, twice a day, for 12 months.

Group B: Metformin hydrochloride 850 mg

Metformin hydrochloride 850mg Orally twice a day.

Group Type ACTIVE_COMPARATOR

Metformin Hydrochloride

Intervention Type DRUG

850 mg, tablets. Administered orally, twice a day, for 12 months.

Interventions

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Metformin glycinate

1050 mg, tablets Administered orally, twice a day, for 12 months.

Intervention Type DRUG

Metformin Hydrochloride

850 mg, tablets. Administered orally, twice a day, for 12 months.

Intervention Type DRUG

Other Intervention Names

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MET GLY MET HYD

Eligibility Criteria

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Inclusion Criteria

* Subjects ≥18 years old.
* Type 2 diabetes according to ADA diagnostic criteria.
* Naive to treatment or who have previously been under oral hypoglycemic treatment (whatever it may be), as long as it has been suspended for a period of ≥6 weeks prior to the start of the study. - HbA1c ≥7.5% and \<10.0%.
* In the case of women of childbearing age and with an active sexual life, the use of birth control methods is required; any of the following are accepted: barrier (male or female condom), non-hormonal intrauterine device, or bilateral tubal obstruction.
* That you agree to participate in the study and give written informed consent.

Exclusion Criteria

* Patients with known current abuse or dependence (last 2 months) to substances such as alcohol (weekly consumption\> 21 units of alcohol in men or\> 14 units of alcohol in women) or recreational drugs.
* Body Mass Index \<20 kg / m2 and\> 35 kg / m2.
* Glomerular filtration estimated with the MDRD (Modification of Diet in Renal Disease) procedure through serum creatinine \<60 ml / min / 1.72 m2.
* History of chronic liver disease or ALT (alanine aminotransferase) and / or AST (aspartate aminotransferase) ≥ 2 times the upper limit of normal, or GGT (Gamma glutamyl transpeptidase) ≥3 times the upper limit of normal.
* Chronic lung disease, causing dyspnea equivalent to a functional class ≥3 (NYHA) or requiring oxygen supplementation.
* Use of drugs that interact with biguanides.
* Other chronic diseases that limit survival or are associated with chronic inflammation such as: cancer, leukemia, lymphoma, lupus erythematosus, asthma, rheumatoid arthritis, or HIV (human immunodeficiency virus) infection.
* Pregnancy or positive pregnancy test, as well as women who are breastfeeding.
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

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Laboratorios Silanes S.A. de C.V.

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Guillermo Fanghänel Salmón, M.D

Role: PRINCIPAL_INVESTIGATOR

Clinica integral del paciente diabético y obeso

Manuel González Ortiz, M.D

Role: PRINCIPAL_INVESTIGATOR

Instituto de terapéutica experimental y clínica (INTEC)

Joel Rodríguez Saldaña, M.D

Role: PRINCIPAL_INVESTIGATOR

Resultados médicos, desarrollo e investigación SC. (REMEDI)

María L Sánchez Aldana Robles, M.D

Role: PRINCIPAL_INVESTIGATOR

Investigación Biomédica para el Desarrollo de Fármacos, S.A de C.V. (IBIOMED-GDL)

Francisco G Padilla Padilla, M.D

Role: PRINCIPAL_INVESTIGATOR

Independent

Jorge V Yamamoto Cuevas, M.D

Role: PRINCIPAL_INVESTIGATOR

Clínica Villa Coapa La Vereda S.C.

Edmundo D Ríos Mejía, M.D

Role: PRINCIPAL_INVESTIGATOR

Investigación Biomédica para el Desarrollo de Fármacos S.A. de C.V. (IBIOMED-AGS)

Luis M Román Pintos, M.D

Role: PRINCIPAL_INVESTIGATOR

Hospital Hispanos S.A. de C.V.

Víctor Bohórquez López, M.D

Role: PRINCIPAL_INVESTIGATOR

Oaxaca Site Management Organization SC. (Red OSMO)

Santiago P Ramírez Díaz, M..D

Role: PRINCIPAL_INVESTIGATOR

Centro de Investigación Médica Aguascalientes (Red OSMO)

José De la Cruz Tun Pech, M.D

Role: PRINCIPAL_INVESTIGATOR

Mérida Investigación Clínica (Red OSMO)

Fernando J Lavalle González, M.D

Role: PRINCIPAL_INVESTIGATOR

Servicio de endocrinología Hospital Univertsitario, UANL

Locations

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Laboratorio Silanes, S.A. de C.V.

Mexico City, , Mexico

Site Status

Countries

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Mexico

References

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Other Identifiers

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SIL-30000-III-19(1)

Identifier Type: -

Identifier Source: org_study_id

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