A Study of Sotorasib (AMG 510) in Participants With Stage IV NSCLC Whose Tumors Harbor a KRAS p.G12C Mutation in Need of First-line Treatment

NCT ID: NCT04933695

Last Updated: 2025-10-22

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE2

Total Enrollment

42 participants

Study Classification

INTERVENTIONAL

Study Start Date

2022-01-28

Study Completion Date

2025-05-27

Brief Summary

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The main objective of this study is to evaluate the tumor objective response rate (ORR) assessed by Response Evaluation Criteria in Solid Tumors (RECIST) 1.1 criteria in participants who receive sotorasib at either 960 mg daily or 240 mg daily whose tumors are programmed death-ligand 1 (PD-L1) Tumor Proportion Score (TPS) \< 1% and/or harbor a serine/threonine kinase 11 (STK11) co-mutation, in a subgroup of participants with PD-L1 \< 1% and in a subgroup of participants with STK11 co-mutation.

Detailed Description

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Conditions

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Non-small Cell Lung Cancer

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Sotorasib: 960 mg Daily

Participants with metastatic non-small cell lung cancer (NSCLC) with Kirsten rat sarcoma (KRAS) p.G12C mutation whose tumors express \< 1% programmed death-ligand 1 (PD-L1) and/or serine/threonine kinase 11 (STK11) mutation in need of first line treatment will be administered sotorasib 960 mg daily. Participants will be stratified by known presence of STK11 mutation.

Group Type EXPERIMENTAL

Sotorasib

Intervention Type DRUG

Oral tablet

Sotorasib: 240 mg Daily

Participants with metastatic non-small cell lung cancer (NSCLC) with Kirsten rat sarcoma (KRAS) p.G12C mutation whose tumors express \< 1% programmed death-ligand 1 (PD-L1) and/or serine/threonine kinase 11 (STK11) mutation in need of first line treatment will be administered sotorasib 240 mg daily. Participants will be stratified by known presence of STK11 mutation.

Group Type EXPERIMENTAL

Sotorasib

Intervention Type DRUG

Oral tablet

Interventions

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Sotorasib

Oral tablet

Intervention Type DRUG

Other Intervention Names

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AMG 510 LUMYKRAS LUMAKRAS

Eligibility Criteria

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Inclusion Criteria

* Adult (= or \> 18 years old) with NSCLC
* Untreated Stage IV metastatic disease. Participants who received adjuvant or neoadjuvant anti-tumor therapy are eligible if the adjuvant/neoadjuvant therapy was completed greater than 12 months prior to the development of metastatic stage IV disease
* Pathologically documented metastatic NSCLC with KRAS G12C mutation (local confirmation)
* Programmed death-ligand 1 (PD-L1) TPS Score \< 1% and/or serine/threonine kinase 11 (STK11) co-mutation (local confirmation)
* Eastern Cooperative Oncology Group (ECOG) score of 0 or 1
* No active brain metastases
* Measurable disease per investigator interpretation using Response Evaluation Criteria in Solid Tumors (RECIST) 1.1 criteria

Exclusion Criteria

* Mixed small-cell lung cancer and NSCLC histology
* Myocardial Infarction within 6 months of study Day 1
* Use of proton-pump inhibitors (PPIs), histamine (H2) receptor antagonists (H2RA), strong inducers of cytochrome P450 (CYP) 3A4 (CYP3A4) or known CYP3A4 sensitive substrates or P-gp substrates
* Therapeutic or palliative radiation therapy within 2 weeks of study day 1
* Unable to take oral medication
* Unable to receive both iodinated contrast for computed tomography (CT) scans and gadolinium contrast for magnetic resonance imagine (MRI) scans
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Amgen

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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MD

Role: STUDY_DIRECTOR

Amgen

Locations

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Alabama Oncology

Birmingham, Alabama, United States

Site Status

Arizona Oncology Associates Professional Corporation

Tucson, Arizona, United States

Site Status

City of Hope at Long Beach Elm

Duarte, California, United States

Site Status

City of Hope National Medical Center

Duarte, California, United States

Site Status

Baptist MD Anderson Cancer Center

Jacksonville, Florida, United States

Site Status

Northwest Georgia Oncology Centers PC

Marietta, Georgia, United States

Site Status

Indiana University Melvin and Bren Simon Cancer Center

Indianapolis, Indiana, United States

Site Status

Baptist Health Lexington

Lexington, Kentucky, United States

Site Status

Frederick Memorial Hospital

Frederick, Maryland, United States

Site Status

Englewood Hospital and Medical Center

Englewood, New Jersey, United States

Site Status

Rutgers Cancer Institute of New Jersey

New Brunswick, New Jersey, United States

Site Status

Laura and Isaac Perlmutter Cancer Center at New York University Langone

New York, New York, United States

Site Status

Northport Veterans Affairs Medical Center

Northport, New York, United States

Site Status

State University of New York Upstate Medical University

Syracuse, New York, United States

Site Status

James J Peters VA Medical Center

The Bronx, New York, United States

Site Status

Duke University Medical Center, Morris Cancer Clinic

Durham, North Carolina, United States

Site Status

Allegheny Health Network Cancer Institute at Allegheny General Hospital

Pittsburgh, Pennsylvania, United States

Site Status

University of Pittsburgh Medical Center Cancer Pavillion

Pittsburgh, Pennsylvania, United States

Site Status

Medical University of South Carolina, Hollings Cancer Center

Charleston, South Carolina, United States

Site Status

Texas Oncology - Medical City Dallas

Dallas, Texas, United States

Site Status

Texas Oncology - Plano East

Dallas, Texas, United States

Site Status

Texas Oncology-Dallas Presbyterian Hospital

Dallas, Texas, United States

Site Status

Texas Oncology - Flower Mound

Dallas, Texas, United States

Site Status

Texas Oncology - Baylor

Dallas, Texas, United States

Site Status

Texas Oncology-Denton

Denton, Texas, United States

Site Status

Oncology Consultants PA

Houston, Texas, United States

Site Status

University of Texas MD Anderson Cancer Center

Houston, Texas, United States

Site Status

Texas Oncology- Mckinney

McKinney, Texas, United States

Site Status

Texas Oncology - Northeast Texas

Paris, Texas, United States

Site Status

Gundersen Health System

La Crosse, Wisconsin, United States

Site Status

Universite Catholique de Louvain Cliniques Universitaires Saint Luc

Brussels, , Belgium

Site Status

Universitair Ziekenhuis Antwerpen

Edegem, , Belgium

Site Status

Jessa Ziekenhuis - Campus Virga Jesse

Hasselt, , Belgium

Site Status

Centre Hospitalier Universitaire de Liege - Sart Tilman

Liège, , Belgium

Site Status

Odense Universitetshospital

Odense C, , Denmark

Site Status

Institut Sainte Catherine

Avignon, , France

Site Status

Centre Hospitalier Universitaire Régional de Lille - Hôpital Albert Calmette

Lille, , France

Site Status

Centre Hospitalier Universitaire de Limoges - Hopital Dupuytren

Limoges, , France

Site Status

Centre Hospitalier Universitaire de Montpellier - Val d Aurelle

Montpellier, , France

Site Status

Hopital Cochin

Paris, , France

Site Status

Centre Hospitalier Universitaire de Bordeaux - Hopital Haut Leveque

Pessac, , France

Site Status

Centre Hospitalier Universitaire de Rennes - Hopital Pontchaillou

Rennes, , France

Site Status

Centre Hospitalier de Nantes - Hôpital Nord Laënnec

Saint-Herblain, , France

Site Status

Hôpital Sainte Musse

Toulon, , France

Site Status

Centre Hospitalier Universitaire de Toulouse - Hopital Larrey

Toulouse, , France

Site Status

Universitätsklinikum Köln

Cologne, , Germany

Site Status

Klinikum und Fachbereich Medizin Johann Wolfgang Goethe-Universität Frankfurt am Main

Frankfurt am Main, , Germany

Site Status

Asklepios - Fachkliniken München-Gauting

Gauting, , Germany

Site Status

Azienda Socio Sanitaria Territoriale di Monza Ospedale San Gerardo

Monza (MB), , Italy

Site Status

Azienda Ospedaliera di Rilievo Nazionale Specialistica dei Colli Monaldi

Napoli, , Italy

Site Status

Azienda Ospedaliera Universitaria San Luigi Gonzaga

Orbassano (TO), , Italy

Site Status

Istituti Fisioterapici Ospitalieri Regina Elena San Gallicano

Rome, , Italy

Site Status

Nederlands Kanker Instituut Antoni van Leeuwenhoekziekenhuis

Amsterdam, , Netherlands

Site Status

Hospital del Mar

Barcelona, Catalonia, Spain

Site Status

Hospital de la Santa Creu i Sant Pau

Barcelona, Catalonia, Spain

Site Status

Hospital Clinico Universitario de Santiago

Santiago de Compostela, Galicia, Spain

Site Status

Hospital Universitario Puerta de Hierro Majadahonda

Majadahonda, Madrid, Spain

Site Status

Hospital Universitari i Politecnic La Fe

Valencia, Valencia, Spain

Site Status

Hospital Universitario La Paz

Madrid, , Spain

Site Status

Gavle Sjukhus

Gävle, , Sweden

Site Status

Sahlgrenska Universitetssjukhuset

Gothenburg, , Sweden

Site Status

Universitetssjukhuset i Linkoping

Linköping, , Sweden

Site Status

Skanes Universitetssjukhus

Lund, , Sweden

Site Status

Norrlands Universitetssjukhus

Umeå, , Sweden

Site Status

Gazi Universitesi Saglik Arastirma ve Uygulama Merkezi Gazi Hastanesi

Ankara, , Turkey (Türkiye)

Site Status

Trakya Universitesi Saglik Arastirma ve Uygulama Merkezi

Edirne, , Turkey (Türkiye)

Site Status

Koc Universitesi Hastanesi

Istanbul, , Turkey (Türkiye)

Site Status

Countries

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United States Belgium Denmark France Germany Italy Netherlands Spain Sweden Turkey (Türkiye)

Related Links

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http://www.amgentrials.com

AmgenTrials clinical trials website

Other Identifiers

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2021-002638-18

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

20190288

Identifier Type: -

Identifier Source: org_study_id

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