Tislelizumab in Combination With Sitravatinib in Participants With Locally Advanced or Metastatic Non-Small Cell Lung Cancer

NCT ID: NCT04921358

Last Updated: 2025-06-29

Study Results

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Basic Information

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Recruitment Status

TERMINATED

Clinical Phase

PHASE3

Total Enrollment

377 participants

Study Classification

INTERVENTIONAL

Study Start Date

2021-07-27

Study Completion Date

2023-12-20

Brief Summary

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The purpose of this study was to evaluate the efficacy and safety of tislelizumab in combination with sitravatinib compared to docetaxel in participants with locally advanced or metastatic non-small cell lung cancer (NSCLC) who experienced disease progression following platinum-based chemotherapy and anti-programmed cell death protein-1 (PD-1)/programmed cell death ligand-1 (PD-L1) antibody treatment, with the anti-PD-(L)1 antibody administered either in combination with or sequentially before or after the platinum-based chemotherapy.

Detailed Description

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Conditions

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Non-Small Cell Lung Cancer (NSCLC)

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Tislelizumab + Sitravatinib

Participants received 200 mg of intravenous tislelizumab every 3 weeks, combined with 100 mg of oral sitravatinib daily until disease progression, intolerable toxicity, death, or withdrawal of consent, whichever occurred earlier.

Group Type EXPERIMENTAL

Tislelizumab

Intervention Type DRUG

200 mg intravenously once every 3 weeks

Sitravatinib

Intervention Type DRUG

100 mg orally once daily

Docetaxel

Participants received 75 mg/m² of intravenous docetaxel once every 3 weeks until disease progression, intolerable toxicity, death, or withdrawal of consent, whichever occurred earlier.

Group Type ACTIVE_COMPARATOR

Docetaxel

Intervention Type DRUG

75 mg/m\^2 intravenously once every 3 weeks

Interventions

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Tislelizumab

200 mg intravenously once every 3 weeks

Intervention Type DRUG

Docetaxel

75 mg/m\^2 intravenously once every 3 weeks

Intervention Type DRUG

Sitravatinib

100 mg orally once daily

Intervention Type DRUG

Other Intervention Names

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BGB-A317 BGB-9468

Eligibility Criteria

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Inclusion Criteria

1. Metastatic or unresectable locally advanced histologically or cytologically confirmed Non-Small Cell Lung Cancer (NCSLC), not amenable to treatment with curative intent
2. Able to provide archival/fresh tumor tissues for biomarker analysis to assess PD-L1 expression and other biomarkers.
3. No known Epidermal Growth Factor Receptor (EGFR) or B-Raf proto-oncogene (BRAF) sensitizing mutation, or anaplastic lymphoma kinase (ALK) rearrangement or ROS proto oncogene 1 (ROS1) rearrangement
4. Radiographic progression per Response Evaluation Criteria in Solid Tumours (RECIST) v1.1 on or after anti-PD-(L)1 containing therapy for locally advanced and unresectable or metastatic NSCLC.
5. No prior anticancer therapy having the same mechanism of action as sitravatinib (eg, tyrosine kinase inhibitor with a similar target profile or vascular endothelial growth factor (VEGF)- or VEGFR inhibitor)
6. At least 1 measurable lesion as defined based on RECIST v1.1 by investigator

Exclusion Criteria

1. Has received docetaxel as monotherapy or in combination with other therapies.
2. Squamous NSCLC with central cavitation, or NSCLC with hemoptysis (\> 50 mL/day)
3. Participants with tumor shown by imaging to be located around important vascular structures or if the investigator determines that the tumor is likely to invade important blood vessels and may cause fatal bleeding.
4. Active leptomeningeal disease for metastatic NSCLC, or uncontrolled or untreated brain metastasis.
5. Active autoimmune diseases or history of autoimmune diseases that may relapse.
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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BeiGene

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Locations

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Blacktown Cancer and Haematology Centre

Blacktown, New South Wales, Australia

Site Status

Campbelltown Hospital

Campbelltown, New South Wales, Australia

Site Status

The Tweed Valley Hospital

Cudgen, New South Wales, Australia

Site Status

St George Hospital

Kogarah, New South Wales, Australia

Site Status

Pindara Private Hospital

Benowa, Queensland, Australia

Site Status

Cancer Research South Australia

Adelaide, South Australia, Australia

Site Status

Monash Health

Clayton, Victoria, Australia

Site Status

St Vincents Hospital Melbourne

Fitzroy, Victoria, Australia

Site Status

Sunshine Hospital

St Albans, Victoria, Australia

Site Status

Anhui Provincial Cancer Hospital Aka West Branch of Anhui Province Hospital

Hefei, Anhui, China

Site Status

Beijing Cancer Hospital

Beijing, Beijing Municipality, China

Site Status

Peking Union Medical College Hospital

Beijing, Beijing Municipality, China

Site Status

Xinqiao Hospital Affiliated to the Army Medical University

Chongqing, Chongqing Municipality, China

Site Status

Daping Hospital, Third Military Medical University

Chongqing, Chongqing Municipality, China

Site Status

Fujian Provincial Hospital

Fuzhou, Fujian, China

Site Status

Fujian Cancer Hospital

Fuzhou, Fujian, China

Site Status

The First Affiliated Hospital of Xiamen University

Xiamen, Fujian, China

Site Status

The First Hospital of Lanzhou University

Lanzhou, Gansu, China

Site Status

Cancer Center of Guangzhou Medical University

Guangzhou, Guangdong, China

Site Status

Guangdong Provincial Peoples Hospital

Guangzhou, Guangdong, China

Site Status

Nanfang Hospital of Southern Medical University

Guangzhou, Guangdong, China

Site Status

Cancer Hospital of Shantou University Medical College

Shantou, Guangdong, China

Site Status

Cancer Hospital Chinse Academy of Medical Sciences, Shenzhen Center

Shenzhen, Guangdong, China

Site Status

The Peoples Hospital of Guangxi Zhuang Autonomous Region

Nanning, Guangxi, China

Site Status

The Tumor Hospital Affiliated to Guangxi Medical University

Nanning, Guangxi, China

Site Status

Harbin Medical University Cancer Hospital

Harbin, Heilongjiang, China

Site Status

Henan Cancer Hospital

Zhengzhou, Henan, China

Site Status

The First Affiliated Hospital of Zhengzhou University

Zhengzhou, Henan, China

Site Status

Union Hospital of Tongji Medical College, Huazhong University of Science and Technology

Wuhan, Hubei, China

Site Status

Tongji Hospital of Tongji Medical College Huazhong University of Science and Technology

Wuhan, Hubei, China

Site Status

Hubei Cancer Hospital

Wuhan, Hubei, China

Site Status

The Second Xiangya Hospital of Central South University

Changsha, Hunan, China

Site Status

The First Peoples Hospital of Chenzhou

Chenzhou, Hunan, China

Site Status

The Second Hospital, University of South China

Hengyang, Hunan, China

Site Status

Changzhou No Peoples Hospital, the Affiliated Hospital of Nanjing Medical University Branch Cheng

Changzhou, Jiangsu, China

Site Status

Nanjing First Hospital

Nanjing, Jiangsu, China

Site Status

Zhongda Hospital Southeast University

Nanjing, Jiangsu, China

Site Status

The Second Affiliated Hospital of Soochow University

Suzhou, Jiangsu, China

Site Status

The First Affiliated Hospital of Soochow University

Suzhou, Jiangsu, China

Site Status

The Affiliated Hospital of Xuzhou Medical University

Xuzhou, Jiangsu, China

Site Status

The First Affiliated Hospital of Nanchang University Branch Donghu

Nanchang, Jiangxi, China

Site Status

The Second Affiliated Hospital of Nanchang University

Nanchang, Jiangxi, China

Site Status

The First Hospital of Jilin University

Changchun, Jilin, China

Site Status

First Affiliated Hospital of Dalian Medical University

Dalian, Liaoning, China

Site Status

Liaoning Cancer Hospital and Institute

Shenyang, Liaoning, China

Site Status

General Hospital of Ningxia Medical University

Yinchuan, Ningxia, China

Site Status

Jinan Central Hospital

Jinan, Shandong, China

Site Status

Shandong Cancer Hospital

Jinan, Shandong, China

Site Status

The Affiliated Hospital of Qingdao University Branch Laoshan

Qingdao, Shandong, China

Site Status

Rui Jin Hospital Shanghai Jiao Tong University School of Medicine

Shanghai, Shanghai Municipality, China

Site Status

Affiliated Zhongshan Hospital of Fudan University

Shanghai, Shanghai Municipality, China

Site Status

Huashan Hospital Affiliated to Fudan University

Shanghai, Shanghai Municipality, China

Site Status

Sichuan Cancer Hospital and Institute

Chengdu, Sichuan, China

Site Status

West China Hospital, Sichuan University

Chengdu, Sichuan, China

Site Status

Tianjin Medical University General Hospital

Tianjin, Tianjin Municipality, China

Site Status

Tianjin Medical University Cancer Institute and Hospital

Tianjin, Tianjin Municipality, China

Site Status

Affiliated Cancer Hospital of Xinjiang Medical University

Ürümqi, Xinjiang, China

Site Status

Yunnan Cancer Hospital

Kunming, Yunnan, China

Site Status

Sir Run Run Shaw Hospital, Zhejiang University School of Medicine

Hangzhou, Zhejiang, China

Site Status

Zhejiang Cancer Hospital

Hangzhou, Zhejiang, China

Site Status

Taizhou Hospital of Zhejiang

Taizhou, Zhejiang, China

Site Status

Countries

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Australia China

References

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Zhou Q, Zhao J, Gao B, et al. SAFFRON-301: A Phase 3 Study of Tislelizumab With Sitravatinib Versus Chemotherapy in Patients With Locally Advanced or Metastatic Non-Small Cell Lung Cancer Previously Treated With Platinum-Based Chemotherapy and an Anti-PD-1/PD-L1 Antibody. Poster presented at: ESMO Congress 2022; September, 2022; Paris, France.

Reference Type BACKGROUND

Zhou Q, Gao B, et al. SAFFRON-301: Sitravatinib PLUS Tislelizumab in Advanced/Metastatic NSCLC Progressing on/after Chemotherapy and Anti-PD-(L)1.

Reference Type RESULT

Provided Documents

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Document Type: Study Protocol

View Document

Document Type: Statistical Analysis Plan

View Document

Other Identifiers

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2022-001779-15

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

SAFFRON-301

Identifier Type: OTHER

Identifier Source: secondary_id

CTR20211410/CTR20211409

Identifier Type: OTHER

Identifier Source: secondary_id

BGB-A317-Sitravatinib-301

Identifier Type: -

Identifier Source: org_study_id

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