First-In-Human Study of GFB-024 in Healthy Overweight and Obese Participants, and Participants With Type 2 Diabetes

NCT ID: NCT04880291

Last Updated: 2022-03-28

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

39 participants

Study Classification

INTERVENTIONAL

Study Start Date

2021-05-05

Study Completion Date

2022-02-08

Brief Summary

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GFB-024 is intended for use in patients with kidney disease such as diabetic nephropathy. This study is the first time GFB-024 has been used in humans. The first part of the study will assess the safety of a single dose of GFB-024 in healthy overweight and obese volunteers and the effect of GFB-024 on the body as compared to an inactive placebo medication. The second part of the study will assess the safety of repeated doses of GFB-024 in participants with Type 2 diabetes and the effect of GFB-024 on the body as compared to an inactive placebo medication.

Detailed Description

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This is a first-in-human study. It is intended to provide the initial safety, pharmacokinetics (PK), and pharmacology data for GFB-024 in humans. This study will comprise a single ascending dose (SAD) escalation component in healthy overweight and obese volunteer participants and a repeat-dose component to confirm repeat-dose safety, tolerability, PK, and immunogenicity in participants with Type 2 diabetes mellitus. It will also explore potential cannabinoid-1 receptor (CB1) activity, participant selection, pharmacodynamics, and differential response biomarkers.

Conditions

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Kidney Diseases Diabetic Nephropathies Diabetes Complications Diabetes Mellitus Endocrine System Diseases

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

SEQUENTIAL

Primary Study Purpose

TREATMENT

Blinding Strategy

DOUBLE

Participants Investigators

Study Groups

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GFB-024 SAD Active

Single ascending dose arm of GFB-024 treatment

Group Type ACTIVE_COMPARATOR

GFB-024

Intervention Type DRUG

Peripherally acting Cannabinoid-1 receptor inverse agonist monoclonal antibody

SAD Placebo

Single ascending dose arm of placebo treatment

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DRUG

Matched placebo

GFB-024 Repeat-dose Active

Repeat-dose arm of GFB-024 treatment

Group Type ACTIVE_COMPARATOR

GFB-024

Intervention Type DRUG

Peripherally acting Cannabinoid-1 receptor inverse agonist monoclonal antibody

Repeat-dose Placebo

Repeat-dose arm of placebo treatment

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DRUG

Matched placebo

Interventions

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GFB-024

Peripherally acting Cannabinoid-1 receptor inverse agonist monoclonal antibody

Intervention Type DRUG

Placebo

Matched placebo

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* 18 to 75 years of age at the time of signing informed consent.
* Body mass index (BMI) between 25.0 and 40.0 kg/m2, inclusive, at Screening.
* Female participants will be of non-childbearing potential.
* Male participants will agree to use contraception while on study intervention and for at least 6 months after the last dose of study intervention.
* SAD cohorts only: Participants must be in good health.
* Repeat-dose cohort only: Type 2 diabetes mellitus (T2DM) treated with lifestyle modification or metformin, and in otherwise good health except for well-controlled common conditions associated with T2DM, such as hypertension and dyslipidemia.

Exclusion Criteria

* History of, or treatment for, psychiatric illness, including anxiety or depression within 5 years of the Screening visit.
* Participants with a history of attempted suicide or clinically significant suicidal ideation.
* History of cardiovascular disease.
* Blood pressure \>155 mmHg systolic or \>95 mmHg diastolic.
* History of alcoholism or drug/chemical abuse within 2 years prior to Screening.
* Alcohol consumption of \>21 units per week for males and \>14 units for females. One unit of alcohol equals 12 oz (360 mL) beer, 1.5 oz (45 mL) liquor, or 5 oz (150 mL) wine.
* History of significant hypersensitivity, intolerance, or allergy to more than one class of drugs.
* Positive hepatitis panel and/or positive human immunodeficiency virus test. Participants whose results are compatible with prior immunization may be included.
* SAD cohorts only: Fasting glucose \>126 mg/dL.
Minimum Eligible Age

18 Years

Maximum Eligible Age

75 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

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Goldfinch Bio, Inc.

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Ingela Danielsson, MD, PhD, MBA

Role: PRINCIPAL_INVESTIGATOR

Worldwide Clinical Trails

Locations

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Worldwide Clinical Trials

San Antonio, Texas, United States

Site Status

Countries

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United States

Other Identifiers

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GFB-024-102

Identifier Type: -

Identifier Source: org_study_id

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