Capivasertib + CDK4/6i + Fulvestrant for Advanced/Metastatic HR+/HER2- Breast Cancer (CAPItello-292)

NCT ID: NCT04862663

Last Updated: 2025-12-23

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

RECRUITING

Clinical Phase

PHASE3

Total Enrollment

895 participants

Study Classification

INTERVENTIONAL

Study Start Date

2021-05-10

Study Completion Date

2029-08-14

Brief Summary

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A Phase Ib/III Open-label, Randomised Study of Capivasertib plus CDK4/6 Inhibitors and Fulvestrant versus CDK4/6 Inhibitors and Fulvestrant in Hormone Receptor-Positive and Human Epidermal Growth Factor Receptor 2-Negative Locally Advanced, Unresectable or Metastatic Breast Cancer (CAPItello-292)

Detailed Description

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This Phase Ib/III study (CAPItello-292) aims to evaluate the efficacy, safety and the degree of added benefit of capivasertib combined with CDK4/6i and fulvestrant in participants with locally advanced (inoperable) or metastatic HR+/HER2- breast cancer. Although the dosing regimens of capivasertib + fulvestrant and of CDK4/6i + fulvestrant are established separately, the dose and schedule for the triplet combinations (capivasertib + CDK4/6i + fulvestrant) need to be confirmed. Therefore, the initial dose finding Phase Ib part of the study will determine the recommended Phase III doses (RP3D) of the triplet combinations. The Phase III part of the study will evaluate the efficacy, safety and the degree of added benefit of the triplet combinations of capivasertib and fulvestrant with investigator's choice of CDK4/6i (either palbociclib or ribociclib at safe and tolerable doses, once identified) in comparison with a control arm (fulvestrant + investigator's choice of CDK4/6i \[palbociclib or ribociclib\]) in a ER+ HER2- maC high risk population that did not receive prior endocrine therapy in the advanced setting.

Conditions

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Locally Advanced (Inoperable) or Metastatic Breast Cancer

Keywords

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Locally advanced (inoperable) or Metastatic Breast Cancer

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Phase Ib: Open, Parallel groups allowed, recruiting up to approx. 222 participants.

Phase III: open-label, randomised, recruiting approx. 794 participants.
Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Capivasertib Plus Palbociclib and Fulvestrant

Capivasertib Plus Palbociclib and Fulvestrant (Ph 1b)

Group Type EXPERIMENTAL

Capivasertib

Intervention Type DRUG

Phase Ib: Capivasertib 320 mg/ 400 mg administered PO BD 4 days on /3 days off per week for 4 weeks (28 days cycle) Phase III: : Capivasertib, administered PO BD 4 days on / 3 days off per week for 4 weeks (28 days cycle) at the dose confirmed in the phase Ib portion

Fulvestrant

Intervention Type DRUG

Phase Ib and Phase III: 500 mg (2 injections of 250 mg) on Day 1 of Weeks 1 and 3 of Cycle 1, and then on Day 1, Week 1 of each cycle thereafter

Palbociclib

Intervention Type DRUG

Phase Ib: 100 mg/ 125 mg. Once daily for 21 consecutive days followed by 7 days off treatment to comprise a complete 28-day cycle Phase III: Administered once daily for 21 days of 28-day cycle, at the dose of 125 mg.

Capivasertib Plus Ribociclib and Fulvestrant

Capivasertib Plus Ribociclib and Fulvestrant (Ph 1b)

Group Type EXPERIMENTAL

Ribociclib

Intervention Type DRUG

Phase Ib: 200 mg/ 400 mg/ 600 mg. Once daily for 21 consecutive days followed by 7 days off treatment to comprise a complete 28-day cycle Phase III: Administered once daily for 21 days of 28-day cycle, at the dose confirmed in the phase 1b portion.

Capivasertib Plus Abemaciclib and Fulvestrant

Capivasertib Plus Abemaciclib and Fulvestrant (Ph 1b)

Group Type EXPERIMENTAL

Abemaciclib

Intervention Type DRUG

Phase Ib: 50 mg/ 100 mg/ 150 mg. Twice daily for 28 consecutive days to comprise a complete 28-day cycle

Capivasertib Plus Fulvestrant and Investigator's choice of CDK4/6i (palbociclib or ribociclib)

Capivasertib Plus Fulvestrant and Investigator's choice of CDK4/6i (palbociclib or ribociclib) (Ph III)

Group Type EXPERIMENTAL

Capivasertib

Intervention Type DRUG

Phase Ib: Capivasertib 320 mg/ 400 mg administered PO BD 4 days on /3 days off per week for 4 weeks (28 days cycle) Phase III: : Capivasertib, administered PO BD 4 days on / 3 days off per week for 4 weeks (28 days cycle) at the dose confirmed in the phase Ib portion

Fulvestrant and Investigator's choice of CDK4/6i (palbociclib or ribociclib)

Fulvestrant and investigator's choice of CDK4/6i (palbociclib or ribociclib) (Ph III)

Group Type ACTIVE_COMPARATOR

Fulvestrant

Intervention Type DRUG

Phase Ib and Phase III: 500 mg (2 injections of 250 mg) on Day 1 of Weeks 1 and 3 of Cycle 1, and then on Day 1, Week 1 of each cycle thereafter

Interventions

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Capivasertib

Phase Ib: Capivasertib 320 mg/ 400 mg administered PO BD 4 days on /3 days off per week for 4 weeks (28 days cycle) Phase III: : Capivasertib, administered PO BD 4 days on / 3 days off per week for 4 weeks (28 days cycle) at the dose confirmed in the phase Ib portion

Intervention Type DRUG

Fulvestrant

Phase Ib and Phase III: 500 mg (2 injections of 250 mg) on Day 1 of Weeks 1 and 3 of Cycle 1, and then on Day 1, Week 1 of each cycle thereafter

Intervention Type DRUG

Palbociclib

Phase Ib: 100 mg/ 125 mg. Once daily for 21 consecutive days followed by 7 days off treatment to comprise a complete 28-day cycle Phase III: Administered once daily for 21 days of 28-day cycle, at the dose of 125 mg.

Intervention Type DRUG

Ribociclib

Phase Ib: 200 mg/ 400 mg/ 600 mg. Once daily for 21 consecutive days followed by 7 days off treatment to comprise a complete 28-day cycle Phase III: Administered once daily for 21 days of 28-day cycle, at the dose confirmed in the phase 1b portion.

Intervention Type DRUG

Abemaciclib

Phase Ib: 50 mg/ 100 mg/ 150 mg. Twice daily for 28 consecutive days to comprise a complete 28-day cycle

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

1. Adult females (pre-/peri-/ and post-menopausal), and adult males.
2. Histologically confirmed HR+/ HER2- breast cancer determined from the most recent tumour sample (primary or metastatic) per the American Society of Clinical Oncology and College of American Pathologists guideline. To fulfil the requirement of HR+ disease, a breast cancer must express ER with or without co-expression of progesterone receptor.
3. Eligible for fulvestrant therapy and at least one of the following: palbociclib, ribociclib, or abemaciclib, as per local investigator assessment. Previous tolerance to specific CDK4/6 inhibitors and dose levels required.
4. Adequate organ and bone marrow functions.
5. Consent to provide a mandatory FFPE tumour sample.


1. Previous treatment with an ET (tamoxifen, AI, or oral SERD) as a single agent or in combination, with radiological evidence of breast cancer recurrence or progression while on, or within 12 months of, completing a (neo)adjuvant ET regimen.
2. Provision of mandatory blood samples at screening for central testing using an investigational ctDNA test to be stratified based on PIK3CA/AKT1/PTEN status.
3. Be eligible for fulvestrant and at least one out of palbociclib or ribociclib (depending on the available CDK4/6i options at time of enrolment), as per local investigator assessment.
4. Have measurable lesion(s) according to Response Evaluation Criteria in Solid Tumours version 1.1 (RECIST v1.1) or, in the absence of measurable disease, lytic or mixed bone lesions that can be assessed by computed tomography (CT) or magnetic resonance imaging (MRI).

Exclusion Criteria

1. History of another primary malignancy except for malignancy treated with curative intent with no known active disease ≥ 2 years before the first dose of study intervention and of low potential risk for recurrence.
2. Radiotherapy within 2 weeks prior to study treatment initiation.
3. Major surgery or significant traumatic injury within 4 weeks of the first dose of study treatment.
4. Persistent toxicities (CTCAE Grade \>1) caused by previous anticancer therapy, excluding alopecia. Participants with irreversible toxicity that is not reasonably expected to be exacerbated by study intervention may be included (eg, hearing loss or peripheral sensory neuropathy) after consultation with the AstraZeneca study physician.
5. Spinal cord compression, brain metastases or leptomeningeal metastases unless these lesions are definitively treated (eg. radiotherapy, surgery) and clinically stable off steroids for management of symptoms for at least 4 weeks prior to study treatment initiation.
6. Any of the following cardiac criteria at screening:

(a). Mean resting corrected QT interval (QTcF): (i) Participants to be treated with palbociclib:: QTcF ≥ 470 ms obtained from the average of 3 consecutive (triplicate) ECGs (ii) Participants to be treated with ribociclib: QTcF ≥ 450 ms obtained from the average of 3 consecutive (triplicate) ECGs (iii) Participants to be treated with abemaciclib (Phase Ib only): QTcF ≥ 470 ms obtained from the average of 3 consecutive (triplicate) ECGs (b). Any clinically important abnormalities in cardiac rhythm, conduction or morphology of resting ECG (eg, complete left bundle branch block, third-degree heart block) (c). Any factors that increase the risk of QTc prolongation or risk of arrhythmic events (d). Experience of any of the following procedures or conditions in the preceding 6 months: coronary artery bypass graft, angioplasty, vascular stent, myocardial infarction, unstable angina pectoris, congestive heart failure New York Heart Association (NYHA) grade ≥ 2 (e). Uncontrolled hypotension (f) uncontrolled hypertension (g). Cardiac ejection fraction outside institutional range of normal or \< 50% (whichever is higher)
7. uncontrolled or high grade or symptomatic arrhythmia and atrial fibrillation
8. Any of these clinically significant abnormalities of glucose metabolism at screening:

1. . diabetes mellitus type I or type II requiring insulin treatment
2. . Glycated haemoglobin (HbA1c) ≥ 8.0% (63.9 mmol/mol)
9. Previous allogeneic bone marrow transplant or solid organ transplant.


1. Any prior treatment with, AKT, PI3K or mTOR inhibitors.
2. Prior treatment with CDK4/6 inhibitors in the metastatic setting (prior CDK4/6 inhibitors permitted in the adjuvant setting provided there was a CDK4/6i treatment free interval of at least 12 months).
3. More than 1 line of chemotherapy for metastatic disease.
4. Any line of endocrine-based therapy for inoperable locally advanced or metastatic disease.
Minimum Eligible Age

18 Years

Maximum Eligible Age

99 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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AstraZeneca

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Locations

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Research Site

Tucson, Arizona, United States

Site Status RECRUITING

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Fountain Valley, California, United States

Site Status RECRUITING

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Glendale, California, United States

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Los Angeles, California, United States

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Los Angeles, California, United States

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Napa, California, United States

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Newport Beach, California, United States

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San Francisco, California, United States

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Santa Barbara, California, United States

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Santa Rosa, California, United States

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Aurora, Colorado, United States

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New Haven, Connecticut, United States

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Newark, Delaware, United States

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Quincy, Illinois, United States

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Fort Wayne, Indiana, United States

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Louisville, Kentucky, United States

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Louisville, Kentucky, United States

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Baton Rouge, Louisiana, United States

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Covington, Louisiana, United States

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Annapolis, Maryland, United States

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Baltimore, Maryland, United States

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Baltimore, Maryland, United States

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Boston, Massachusetts, United States

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Detroit, Michigan, United States

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Grand Rapids, Michigan, United States

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Hannibal, Missouri, United States

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St Louis, Missouri, United States

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Omaha, Nebraska, United States

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Camden, New Jersey, United States

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Brooklyn, New York, United States

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Mineola, New York, United States

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New York, New York, United States

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New York, New York, United States

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Durham, North Carolina, United States

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Gresham, Oregon, United States

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Philadelphia, Pennsylvania, United States

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Pittsburgh, Pennsylvania, United States

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York, Pennsylvania, United States

Site Status TERMINATED

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Providence, Rhode Island, United States

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Greenville, South Carolina, United States

Site Status TERMINATED

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Chattanooga, Tennessee, United States

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Nashville, Tennessee, United States

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Dallas, Texas, United States

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Fort Worth, Texas, United States

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Houston, Texas, United States

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San Antonio, Texas, United States

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San Antonio, Texas, United States

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Salt Lake City, Utah, United States

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Falls Church, Virginia, United States

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Leesburg, Virginia, United States

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Midlothian, Virginia, United States

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Norfolk, Virginia, United States

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Tacoma, Washington, United States

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Buenos Aires, , Argentina

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CABA, , Argentina

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CABA, , Argentina

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CABA, , Argentina

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CABA, , Argentina

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Chivilcoy, , Argentina

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Rosario, , Argentina

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Santa Fe, , Argentina

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Darlinghurst, , Australia

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Miranda, , Australia

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Nedlands, , Australia

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Nedlands, , Australia

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Wahroonga, , Australia

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Waratah, , Australia

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Brasschaat, , Belgium

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Brussels, , Belgium

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Edegem, , Belgium

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Haine-Saint-Paul, , Belgium

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Leuven, , Belgium

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Alfenas, , Brazil

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Blumenau, , Brazil

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Natal, , Brazil

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Porto Alegre, , Brazil

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Porto Velho, , Brazil

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São Paulo, , Brazil

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Taubaté, , Brazil

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Teresina, , Brazil

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Vitória, , Brazil

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Abbotsford, British Columbia, Canada

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Kelowna, British Columbia, Canada

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Winnipeg, Manitoba, Canada

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Moncton, New Brunswick, Canada

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Halifax, Nova Scotia, Canada

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Brampton, Ontario, Canada

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Ottawa, Ontario, Canada

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Sault Ste. Marie, Ontario, Canada

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Toronto, Ontario, Canada

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Sherbrooke, Quebec, Canada

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Chicoutimi, , Canada

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Montreal, , Canada

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Beijing, , China

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Beijing, , China

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Beijing, , China

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Beijing, , China

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Bengbu, , China

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Changchun, , China

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Changsha, , China

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Chengdu, , China

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Chongqing, , China

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Guangzhou, , China

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Guangzhou, , China

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Guangzhou, , China

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Hangzhou, , China

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Hangzhou, , China

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Hangzhou, , China

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Hefei, , China

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Jinan, , China

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Nanchang, , China

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Nanchang, , China

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Nanjing, , China

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Nanning, , China

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Shandong, , China

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Shanghai, , China

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Shanghai, , China

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Shenyang, , China

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Shenyang, , China

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Ürümqi, , China

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Ürümqi, , China

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Wuhan, , China

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Xi'an, , China

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Xi'an, , China

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Xiangyang, , China

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Xuzhou, , China

Site Status ACTIVE_NOT_RECRUITING

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Zhengzhou, , China

Site Status ACTIVE_NOT_RECRUITING

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Aalborg, , Denmark

Site Status ACTIVE_NOT_RECRUITING

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Aarhus N, , Denmark

Site Status ACTIVE_NOT_RECRUITING

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Hillerød, , Denmark

Site Status ACTIVE_NOT_RECRUITING

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Odense, , Denmark

Site Status COMPLETED

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Bobigny, , France

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Clermont-Ferrand, , France

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Limoges, , France

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Lyon, , France

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Plérin, , France

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Rouen, , France

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Saint-Herblain, , France

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Villejuif, , France

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Augsburg, , Germany

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Berlin, , Germany

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Berlin, , Germany

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Bottrop, , Germany

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Dresden, , Germany

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Erlangen, , Germany

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Essen, , Germany

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Frankfurt am Main, , Germany

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Freiburg im Breisgau, , Germany

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Georgsmarienhütte, , Germany

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Hamburg, , Germany

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Hanover, , Germany

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Heilbronn, , Germany

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Kiel, , Germany

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Leipzig, , Germany

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Mannheim, , Germany

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Mönchengladbach, , Germany

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Münster, , Germany

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Regensburg, , Germany

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Stade, , Germany

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Trier, , Germany

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Ulm, , Germany

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Bangalore, , India

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Jaipur, , India

Site Status WITHDRAWN

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Jaipur, , India

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Mohali, , India

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Mysuru, , India

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Nagpur, , India

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New Delhi, , India

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New Delhi, , India

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Puducherry, , India

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Vadodara, , India

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Varanasi, , India

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Aviano, , Italy

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Bologna, , Italy

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Catanzaro, , Italy

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Florence, , Italy

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Milan, , Italy

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Milan, , Italy

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Misterbianco, , Italy

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Napoli, , Italy

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Padua, , Italy

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Prato, , Italy

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Reggio Emilia, , Italy

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Roma, , Italy

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Rozzano, , Italy

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Chiba, , Japan

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Chūōku, , Japan

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Chūōku, , Japan

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Hidaka-shi, , Japan

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Hirakata-shi, , Japan

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Hiroshima, , Japan

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Isehara-shi, , Japan

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Kagoshima, , Japan

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Kōtoku, , Japan

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Kyoto, , Japan

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Matsuyama, , Japan

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Nagoya, , Japan

Site Status NOT_YET_RECRUITING

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Naha, , Japan

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Okayama, , Japan

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Osaka, , Japan

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Ota-shi, , Japan

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Sapporo, , Japan

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Sendai, , Japan

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Shimotsuke-shi, , Japan

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Shinagawa-ku, , Japan

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Shinjuku-ku, , Japan

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Suita-shi, , Japan

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Takasaki-shi, , Japan

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Tsu, , Japan

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Yokohama, , Japan

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George Town, , Malaysia

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Kuala Lumpur, , Malaysia

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Kuala Lumpur, , Malaysia

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Kuala Selangor, , Malaysia

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Kuala Selangor, , Malaysia

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Kuching, , Malaysia

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Pulau Pinang, , Malaysia

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Bialystok, , Poland

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Bydgoszcz, , Poland

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Gdansk, , Poland

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Koszalin, , Poland

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Krakow, , Poland

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Lodz, , Poland

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Lodz, , Poland

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Lublin, , Poland

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Rzeszów, , Poland

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Warsaw, , Poland

Site Status COMPLETED

Research Site

Warsaw, , Poland

Site Status RECRUITING

Research Site

Goyang-si, , South Korea

Site Status ACTIVE_NOT_RECRUITING

Research Site

Seoul, , South Korea

Site Status ACTIVE_NOT_RECRUITING

Research Site

Seoul, , South Korea

Site Status ACTIVE_NOT_RECRUITING

Research Site

Seoul, , South Korea

Site Status ACTIVE_NOT_RECRUITING

Research Site

Seoul, , South Korea

Site Status ACTIVE_NOT_RECRUITING

Research Site

Seoul, , South Korea

Site Status ACTIVE_NOT_RECRUITING

Research Site

Seoul, , South Korea

Site Status ACTIVE_NOT_RECRUITING

Research Site

Barcelona, , Spain

Site Status RECRUITING

Research Site

Granada, , Spain

Site Status RECRUITING

Research Site

Lleida, , Spain

Site Status RECRUITING

Research Site

Madrid, , Spain

Site Status RECRUITING

Research Site

Madrid, , Spain

Site Status RECRUITING

Research Site

Madrid, , Spain

Site Status WITHDRAWN

Research Site

Málaga, , Spain

Site Status RECRUITING

Research Site

Pamplona, , Spain

Site Status RECRUITING

Research Site

Santiago de Compostela, , Spain

Site Status RECRUITING

Research Site

Lund, , Sweden

Site Status RECRUITING

Research Site

Solna, , Sweden

Site Status RECRUITING

Research Site

Vaxjo, , Sweden

Site Status RECRUITING

Research Site

Kaohsiung City, , Taiwan

Site Status RECRUITING

Research Site

Kaohsiung City, , Taiwan

Site Status RECRUITING

Research Site

Taichung, , Taiwan

Site Status RECRUITING

Research Site

Tainan, , Taiwan

Site Status RECRUITING

Research Site

Taipei, , Taiwan

Site Status RECRUITING

Research Site

Taipei, , Taiwan

Site Status RECRUITING

Research Site

Taoyuan District, , Taiwan

Site Status RECRUITING

Research Site

Bangkok, , Thailand

Site Status ACTIVE_NOT_RECRUITING

Research Site

Bangkok, , Thailand

Site Status ACTIVE_NOT_RECRUITING

Research Site

Bangkok, , Thailand

Site Status WITHDRAWN

Research Site

Bangkok, , Thailand

Site Status ACTIVE_NOT_RECRUITING

Research Site

Bangkok, , Thailand

Site Status ACTIVE_NOT_RECRUITING

Research Site

Chiang Mai, , Thailand

Site Status ACTIVE_NOT_RECRUITING

Research Site

Dusit, , Thailand

Site Status ACTIVE_NOT_RECRUITING

Research Site

Hat Yai, , Thailand

Site Status ACTIVE_NOT_RECRUITING

Research Site

Khon Kaen, , Thailand

Site Status ACTIVE_NOT_RECRUITING

Research Site

Lampang, , Thailand

Site Status ACTIVE_NOT_RECRUITING

Research Site

Ratchathewi, , Thailand

Site Status ACTIVE_NOT_RECRUITING

Research Site

Ankara, , Turkey (Türkiye)

Site Status ACTIVE_NOT_RECRUITING

Research Site

Antalya, , Turkey (Türkiye)

Site Status ACTIVE_NOT_RECRUITING

Research Site

Goztepe Istanbul, , Turkey (Türkiye)

Site Status ACTIVE_NOT_RECRUITING

Research Site

Karşıyaka, , Turkey (Türkiye)

Site Status ACTIVE_NOT_RECRUITING

Research Site

Kayseri, , Turkey (Türkiye)

Site Status WITHDRAWN

Research Site

Malatya, , Turkey (Türkiye)

Site Status ACTIVE_NOT_RECRUITING

Research Site

Samsun, , Turkey (Türkiye)

Site Status ACTIVE_NOT_RECRUITING

Research Site

Guildford, , United Kingdom

Site Status ACTIVE_NOT_RECRUITING

Research Site

London, , United Kingdom

Site Status ACTIVE_NOT_RECRUITING

Research Site

Londonderry, , United Kingdom

Site Status ACTIVE_NOT_RECRUITING

Research Site

Taunton, , United Kingdom

Site Status ACTIVE_NOT_RECRUITING

Research Site

York, , United Kingdom

Site Status ACTIVE_NOT_RECRUITING

Research Site

Can Tho, , Vietnam

Site Status RECRUITING

Research Site

Hanoi, , Vietnam

Site Status RECRUITING

Research Site

Ho Chi Minh City, , Vietnam

Site Status RECRUITING

Research Site

Ho Chi Minh City, , Vietnam

Site Status RECRUITING

Research Site

Hồ Chí Minh, , Vietnam

Site Status RECRUITING

Research Site

Vinh, , Vietnam

Site Status RECRUITING

Countries

Review the countries where the study has at least one active or historical site.

United States Argentina Australia Belgium Brazil Canada China Denmark France Germany India Italy Japan Malaysia Poland South Korea Spain Sweden Taiwan Thailand Turkey (Türkiye) United Kingdom Vietnam

Central Contacts

Reach out to these primary contacts for questions about participation or study logistics.

AstraZeneca Clinical Study Information Center

Role: CONTACT

Phone: 1-877-240-9479

Email: [email protected]

AstraZeneca Breast Cancer Study Locator Service

Role: CONTACT

Phone: 1-877-400-4655

Email: [email protected]

Related Links

Access external resources that provide additional context or updates about the study.

https://www.breastcancerstudylocator.com/trial/listing/284051

Breast Cancer Study Locator details (for US)

Other Identifiers

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2020-004637-20

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

D361DC00001

Identifier Type: -

Identifier Source: org_study_id