A Study of Selpercatinib After Surgery or Radiation in Participants With Non-Small Cell Lung Cancer (NSCLC)

NCT ID: NCT04819100

Last Updated: 2025-12-29

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

ACTIVE_NOT_RECRUITING

Clinical Phase

PHASE3

Total Enrollment

152 participants

Study Classification

INTERVENTIONAL

Study Start Date

2021-12-20

Study Completion Date

2028-04-30

Brief Summary

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The reason for this study is to see if the study drug, selpercatinib, compared to placebo is effective and safe in delaying cancer return in participants with early-stage non-small cell lung cancer (NSCLC), who have already had surgery or radiation. Participants who are assigned to placebo and stop the study drug because their disease comes back or gets worse have the option to potentially crossover to selpercatinib. Participation could last up to three years.

Detailed Description

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Conditions

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Carcinoma, Non-Small-Cell Lung

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

TRIPLE

Participants Investigators Outcome Assessors

Study Groups

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Selpercatinib

Selpercatinib administered orally.

Group Type EXPERIMENTAL

Selpercatinib

Intervention Type DRUG

Administered orally.

Placebo

Placebo administered orally.

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DRUG

Administered orally.

Interventions

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Selpercatinib

Administered orally.

Intervention Type DRUG

Placebo

Administered orally.

Intervention Type DRUG

Other Intervention Names

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LY3527723 LOXO-292

Eligibility Criteria

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Inclusion Criteria

* Must have histologically confirmed Stage IB, II, or IIIA NSCLC.
* Must have an activating RET gene fusion in tumor based on polymerase chain reaction (PCR), next generation sequencing (NGS), or another molecular test per sponsor's approval.
* Must have received definitive locoregional therapy with curative intent (surgery or radiotherapy) for Stage IB, II, or IIIA NSCLC.

\-- Must have undergone the available anti-cancer therapy (including chemotherapy or durvalumab) or not be suitable for it, based on the investigator's discretion.
* Maximum time allowed between definitive therapy completion and randomization must be:

* 10 weeks if no chemotherapy was administered
* 26 weeks if adjuvant chemotherapy was administered
* Eastern Cooperative Oncology Group (ECOG) performance status of 0-1.
* Adequate hematologic, hepatic, and renal function.
* Willingness of men and women of reproductive potential to observe conventional and highly effective birth control for the duration of the study and for at least 2 weeks after last dose of study drug.

Exclusion Criteria

* Additional oncogenic drivers in NSCLC, if known.
* Evidence of small cell lung cancer.
* Clinical or radiologic evidence of disease recurrence or progression following definitive therapy.
* Known or suspected interstitial fibrosis or interstitial lung disease or history of (noninfectious) pneumonitis that required steroids.
* Clinically significant active cardiovascular disease or history of myocardial infarction within six months prior to planned start of selpercatinib or prolongation of the QT interval corrected for heart rate using Fridericia's formula (QTcF) greater than 470 milliseconds.
* Have known uncontrolled human immunodeficiency virus (HIV)-1/2 infection.
* Have known active hepatitis B or C.
* Active uncontrolled systemic bacterial, viral, or fungal infection or serious ongoing intercurrent illness, such as hypertension or diabetes, despite optimal treatment.
* Major surgery within 4 weeks prior to planned start of selpercatinib.
* Clinically significant active malabsorption syndrome or other condition likely to affect gastrointestinal absorption of the study drug.
* Other malignancy unless nonmelanoma skin cancer, carcinoma in situ of the cervix or other in situ cancers or a malignancy diagnosed greater than or equal to two years previously and not currently active.
* Pregnancy or lactation.
* Prior treatment with a selective RET inhibitor (e.g. selpercatinib or pralsetinib).
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Loxo Oncology, Inc.

INDUSTRY

Sponsor Role collaborator

Eli Lilly and Company

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Call 1-877-CTLILLY (1-877-285-4559) or 1-317-615-4559 Mon - Fri 9 AM - 5 PM Eastern time (UTC/GMT - 5 hours, EST)

Role: STUDY_DIRECTOR

Eli Lilly and Company

Locations

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UCLA Hematology/Oncology - Santa Monica

Los Angeles, California, United States

Site Status

Stockton Hematology Oncology Group

Stockton, California, United States

Site Status

Lundquist Institute for Biomedical Innovation at Harbor-UCLA Medical Center

Torrance, California, United States

Site Status

GenesisCare

Aventura, Florida, United States

Site Status

GenesisCare - Boca Raton

Boca Raton, Florida, United States

Site Status

USO-Cancer Care Center of Brevard, Inc.

Palm Bay, Florida, United States

Site Status

Dana-Farber Cancer Institute

Boston, Massachusetts, United States

Site Status

Mayo Clinic in Rochester, Minnesota

Rochester, Minnesota, United States

Site Status

USO-New York Oncology Hematology, P.C

Latham, New York, United States

Site Status

Memorial Sloan Kettering Cancer Center

New York, New York, United States

Site Status

USO - Alliance Cancer Specialists, PC

Horsham, Pennsylvania, United States

Site Status

Sarah Cannon Research Institute SCRI

Nashville, Tennessee, United States

Site Status

Tennessee Oncology Nashville

Nashville, Tennessee, United States

Site Status

USO-Texas Oncology-Central/South Texas

Austin, Texas, United States

Site Status

US Oncology

The Woodlands, Texas, United States

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Sunshine Coast University Hospital

Birtinya, Queensland, Australia

Site Status

Rockhampton Hospital

Rockhampton, Queensland, Australia

Site Status

The Townsville Hospital

Townsville, Queensland, Australia

Site Status

Ballarat Health Services

Ballarat Central, Victoria, Australia

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Bendigo Health Care Group

Bendigo, Victoria, Australia

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Goulburn Valley Health

Shepparton, Victoria, Australia

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South West Healthcare

Warrnambool, Victoria, Australia

Site Status

Border Medical Oncology

Wodonga, Victoria, Australia

Site Status

Landeskrankenhaus Feldkirch

Feldkirch, Vorarlberg, Austria

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Klinik Floridsdorf

Vienna, , Austria

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Antwerp University Hospital

Edegem, Antwerpen, Belgium

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Cliniques universitaires Saint-Luc

Brussels, Bruxelles-Capitale, Région de, Belgium

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Université Catholique de Louvain-Namur - Centre Hospitalier Universitaire Dinant-Godinne - Site Godinne

Yvoir, Namur, Belgium

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Clinique Saint Pierre

Ottignies, Wallonne, Région, Belgium

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AZ Delta vzw

Roeselare, West-Vlaanderen, Belgium

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CHU UCL Namur/Site Sainte Elisabeth

Namur, , Belgium

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Nucleo de Oncologia da Bahia

Salvador, Estado de Bahia, Brazil

Site Status

Sirio-Libanes Brasilia - Centro de Oncologia - Asa Sul

Brasília, Federal District, Brazil

Site Status

Oncocentro de Minas Gerais

Belo Horizonte, Minas Gerais, Brazil

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Centro Oncológico do Triângulo

Uberlândia, Minas Gerais, Brazil

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Multihemo

Recife, Pernambuco, Brazil

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Hospital São Lucas da PUCRS

Porto Alegre, Rio Grande do Sul, Brazil

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Hospital BP

São Paulo, São Paulo, Brazil

Site Status

Instituto D'Or de Pesquisa e Ensino (IDOR)

São Paulo, São Paulo, Brazil

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Instituto de Educação, Pesquisa e Gestão em Saúde

Rio de Janeiro, , Brazil

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Centro Paulista de Oncologia Clínica

São Paulo, , Brazil

Site Status

Núcleo de Pesquisa Clínica da Rede São Camilo

São Paulo, , Brazil

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Sociedade Beneficente Israelita Brasileira Hospital Albert Einstein

São Paulo, , Brazil

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Princess Margaret Cancer Centre

Toronto, Ontario, Canada

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Beijing Friendship Hospital

Beijing, Beijing Municipality, China

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Beijing Cancer hospital

Beijing, Beijing Municipality, China

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Fujian Provincial Hospital

Fuzhou, Fujian, China

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Southern Medical University Nanfang Hospital

Guangzhou, Guangdong, China

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Guangdong Provincial People's Hospital

Guangzhou, Guangdong, China

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Harbin Medical University Cancer Hospital

Harbin, Heilongjiang, China

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Xiangya Hospital, Central South University

Changsha, Hunan, China

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Hunan Cancer Hospital

Changsha, Hunan, China

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Jilin Cancer Hospital

Changchun, Jilin, China

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Tangdu Hospital of Fourth Military Medical University of Chinese People's Liberation Army

Xi'an, Shaanxi, China

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Jinan Central Hospital

Jinan, Shandong, China

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Shanghai Chest Hospital

Shanghai, Shanghai Municipality, China

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Zhongshan Hospital, Fudan University

Shanghai, Shanghai Municipality, China

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Shanghai Pulmonary Hospital

Shanghai, Shanghai Municipality, China

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the Third People's Hospital of Chengdu

Chengdu, Sichuan, China

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West China Hospital, Sichuan University

Chengdu, Sichuan, China

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First Affiliated Hosp of College of Med, Zhejiang University

Hangzhou, Zhejiang, China

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Zhejiang Cancer Hospital

Hangzhou, Zhejiang, China

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Tongji Medical College of Huazhong University of Science and Technology

Wuhan, , China

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Masarykuv onkologicky ustav

Brno, Brno-město, Czechia

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Nemocnice AGEL Ostrava - Vitkovice a.s.

Ostrava, Ostrava Město, Czechia

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Fakultni nemocnice Bulovka

Prague, Praha 8, Czechia

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Odense Universitetshospital

Odense, Region Syddanmark, Denmark

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Centre Leon Berard

Lyon, Auvergne-Rhône-Alpes, France

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Assistance Publique Hôpitaux de Marseille - Hôpital de la Timone

Marseille, Bouches-du-Rhône, France

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CHU Charles Nicolle

Rouen, Haute-Normandie, France

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Centre Chirurgical Marie Lannelongue

Le Plessis-Robinson, Hauts-de-Seine, France

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Hospices Civils de Lyon - Hopital Louis Pradel

Lyon, Rhône, France

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Gustave Roussy

Villejuif, Val-de-Marne, France

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Hopitaux Universitaires Paris Centre-Hopital Cochin

Paris, , France

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Thoraxklinik-Heidelberg gGmbH

Heidelberg, Baden-Wurttemberg, Germany

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Klinik Löwenstein

Löwenstein, Baden-Wurttemberg, Germany

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Asklepios Fachkliniken München-Gauting

Gauting, Bavaria, Germany

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Klinikum der Ludwig-Maximilians-Universitaet Muenchen

München, Bavaria, Germany

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Lungenfachklinik Immenhausen

Immenhausen, Hesse, Germany

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Franziskus-Hospital Harderberg

Georgsmarienhütte, Lower Saxony, Germany

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KRH, Klinikum Siloah

Hanover, Lower Saxony, Germany

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Universitätsklinikum Münster - Albert Schweitzer Campus

Münster, North Rhine-Westphalia, Germany

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LungenClinic Grosshansdorf

Großhansdorf, Schleswig-Holstein, Germany

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Charite Universitätsmedizin Berlin Campus Benjamin Franklin

Berlin, , Germany

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Evangelische Lungenklinik Berlin

Berlin, , Germany

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Asklepios Klinik Harburg

Hamburg, , Germany

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University Hospital of Patras

Pátrai, Achaḯa, Greece

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Agios Savvas Regional Cancer Hospital

Athens, Attikí, Greece

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Errikos Dunant Hospital Center

Athens, Attikí, Greece

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Sotiria Thoracic Diseases Hospital of Athens

Athens, Attikí, Greece

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University General Hospital of Heraklion

Heraklion, Irakleío, Greece

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European Interbalkan Medical Center

Thessaloniki, Thessaloníki, Greece

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G. Papanikolaou General Hospital

Thessaloniki, Thessaloníki, Greece

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Hong Kong United Oncology Centre

Hong Kong, , Hong Kong

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Princess Margaret Hospital

Lai Chi Kok, , Hong Kong

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Queen Elizabeth Hospital

Yau Ma Tei, , Hong Kong

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Regional Cancer Centre - Thiruvananthapuram

Thiruvananthapuram, Kerala, India

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Tata Memorial Hospital

Mumbai, Maharashtra, India

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Rashtrasant Tukdoji Regional Cancer Hospital

Nagpur, Maharashtra, India

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HCG Manavata Cancer Centre

Nashik, Maharashtra, India

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Rajiv Gandhi Cancer Institute And Research Centre

New Delhi, National Capital Territory of Delhi, India

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Sheba Medical Center

Ramat Gan, Central District, Israel

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Hadassah Medical Center

Jerusalem, Jerusalem, Israel

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Rambam Health Care Campus

Haifa, Ḥeifā, Israel

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Instituto Tumori Giovanni Paolo II

Bari, Apulia, Italy

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ASST Grande Ospedale Metropolitano Niguarda

Milan, Milano, Italy

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Humanitas

Rozzano, Milano, Italy

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Azienda Ospedaliera Dei Colli

Naples, Napoli, Italy

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Azienda Sanitaria Ospedaliera S Luigi Gonzaga

Orbassano, Torino, Italy

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Istituto Oncologico Veneto IRCCS

Padua, , Italy

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Aichi Cancer Center Hospital

Nagoya, Aichi-ken, Japan

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National Cancer Center Hospital East

Kashiwa, Chiba, Japan

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Himeji Medical Center

Himeji, Hyōgo, Japan

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Kanagawa cancer center

Yokohama, Kanagawa, Japan

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Niigata Cancer Center Hospital

Niigata, Niigata, Japan

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Shizuoka Cancer Center

Nakatogari, Shizuoka, Japan

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Japanese Foundation for Cancer Research

Koto, Tokyo, Japan

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Tottori University Hospital

Yonago, Tottori, Japan

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Hiroshima University Hospital

Hiroshima, , Japan

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Osaka International Cancer Institute

Osaka, , Japan

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Actualidad Basada en la Investigación del Cáncer

Guadalajara, Jalisco, Mexico

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Oncare Viaducto Napoles

Mexico City, Mexico City, Mexico

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Avix Investigación Clinica, S.C.

Monterrey, Nuevo León, Mexico

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Hospital Universitario "Dr. Jose Eleuterio Gonzalez"

Monterrey, Nuevo León, Mexico

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Ziekenhuis St. Jansdal

Harderwijk, Gelderland, Netherlands

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Radboudumc

Nijmegen, Gelderland, Netherlands

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Oslo Universitetssykehus Ullevål

Oslo, , Norway

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Krakowski Szpital Specjalistyczny im. Jana Pawa II

Krakow, Lesser Poland Voivodeship, Poland

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Pan American Center for Oncology Trials

Rio Piedras, , Puerto Rico

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Institutul Oncologic

Cluj-Napoca, , Romania

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Arkhangelsk Clinical Oncological Dispensary

Arkhangelsk, Arkhangelskaya oblast, Russia

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Hadassah Medical

Moscow, Moscow, Russia

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First Pavlov State Medical University of Saint Petersburg

Saint Petersburg, Sankt-Peterburg, Russia

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Scientific research institution of oncology named after N.N. Petrov

Saint Petersburg, , Russia

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Parkway Cancer Centre - Gleneagles Hospital

Singapore, Central Singapore, Singapore

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Tan Tock Seng Hospital

Singapore, Central Singapore, Singapore

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Chonnam National University Hwasun Hospital

Hwasun, Jeonranamdo, South Korea

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National Cancer Center

Goyang-si, Kyǒnggi-do, South Korea

Site Status

Seoul National University Bundang Hospital

Seongnam, Kyǒnggi-do, South Korea

Site Status

Pusan National University Hospital

Busan, Pusan-Kwangyǒkshi, South Korea

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Seoul National University Hospital

Seoul, Seoul-teukbyeolsi [Seoul], South Korea

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Severance Hospital, Yonsei University Health System

Seoul, Seoul-teukbyeolsi [Seoul], South Korea

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Asan Medical Center

Seoul, Seoul-teukbyeolsi [Seoul], South Korea

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Samsung Medical Center

Seoul, Seoul-teukbyeolsi [Seoul], South Korea

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Korea University Guro Hospital

Seoul, Seoul-teukbyeolsi [Seoul], South Korea

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Kyungpook National University Chilgok Hospital

Deagu, Taegu-Kwangyǒkshi, South Korea

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CHUS - Hospital Clinico Universitario

Santiago de Compostela, A Coruña [La Coruña], Spain

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Hospital Universitario Puerta del Mar

Cadiz, Andalusia, Spain

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Hospital Universitario Reina Sofia

Córdoba, Andalusia, Spain

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Institut Català d'Oncologia (ICO) - Badalona

Badalona, Barcelona [Barcelona], Spain

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Parc de Salut Mar - Hospital del Mar

Barcelona, Barcelona [Barcelona], Spain

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Hospital Universitari Vall d'Hebron

Barcelona, Barcelona [Barcelona], Spain

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Instituto Catalan de Oncologia - Hospital Duran i Reynals

L'Hospitalet Del Llobregat, Barcelona [Barcelona], Spain

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Hospital de Mataró

Mataró, Barcelona [Barcelona], Spain

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Complejo Asistencial Universitario de León - Hospital de León

León, Castille and León, Spain

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Hospital Universitari Dexeusa

Barcelona, Catalunya [Cataluña], Spain

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Hospital Clínic de Barcelona

Barcelona, Catalunya [Cataluña], Spain

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Hospital Son Llàtzer

Palma, Illes Balears [Islas Baleares], Spain

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Hospital Lucus Augusti

Lugo, Lugo [Lugo], Spain

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Hospital Universitario Ramón y Cajal

Madrid, Madrid, Comunidad de, Spain

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Hospital Universitario 12 de Octubre

Madrid, Madrid, Comunidad de, Spain

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Hospital Clínico Universitario Virgen de la Arrixaca

El Palmar, Murcia, Murcia, Región de, Spain

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Complexo Hospitalario Universitario de Ourense

Ourense, Ourense [Orense], Spain

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CHUVI- Hospital Alvaro Cunqueiro

Pontevedra, Pontevedra [Pontevedra], Spain

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Hospital Universitario Central de Asturias

Oviedo, Principality of Asturias, Spain

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Hospital Universitario de Canarias

San Cristóbal de La Laguna, Santa Cruz De Tenerife, Spain

Site Status

Hospital Universitari Sant Joan de Reus

Reus, Tarragona [Tarragona], Spain

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Hospital General Universitario de Albacete

Albacete, , Spain

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MD Anderson Cancer Center

Madrid, , Spain

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Hospital Clinico San Carlos

Madrid, , Spain

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H.R.U Málaga - Hospital General

Málaga, , Spain

Site Status

Hospital Universitario Virgen Macarena

Seville, , Spain

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Hospital Universitari i Politecnic La Fe

Valencia, , Spain

Site Status

Sahlgrenska Universitetssjukhuset

Gothenburg, Västra Götalands Län [se-14], Sweden

Site Status

Changhua Christian Hospital

Changhua County, Changhua, Taiwan

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Chang Gung Memorial Hospital at Kaohsiung

Kaohsiung Niao Sung Dist, Kaohsiung, Taiwan

Site Status

Chung Shan Medical University Hospital

Taichung, Taichung, Taiwan

Site Status

Chi Mei Hospital - Liouying Branch

Tainan, Tainan, Taiwan

Site Status

National Taiwan University Cancer Center (NTUCC)

Taipei City, Taipei, Taiwan

Site Status

Taipei Veterans General Hospital

Taipei City, Taipei, Taiwan

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Kaohsiung Medical University Chung-Ho Memorial Hospital

Kaohsiung City, , Taiwan

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Taichung Veterans General Hospital

Taichung, , Taiwan

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National Taiwan University Hospital

Taipei, , Taiwan

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Chang Gung Medical Foundation-Linkou Branch

Taoyuan District, , Taiwan

Site Status

Ege Universitesi Hastanesi

Bornova, İzmir, Turkey (Türkiye)

Site Status

Izmir Medical Park Hospital

Izmir, Karsiyaka, İzmir, Turkey (Türkiye)

Site Status

Baskent University Dr. Turgut Noyan Research and Training Center

Adana, , Turkey (Türkiye)

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Adana City Hospital

Adana, , Turkey (Türkiye)

Site Status

Abdurrahman Yurtaslan Ankara Oncology, education and Research Hospital

Ankara, , Turkey (Türkiye)

Site Status

Ankara Bilkent Şehir Hastanesi

Ankara, , Turkey (Türkiye)

Site Status

Memorial Antalya Hospital

Antalya, , Turkey (Türkiye)

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Uludag Universitesi

Bursa, , Turkey (Türkiye)

Site Status

Dicle Üniversitesi

Diyarbakır, , Turkey (Türkiye)

Site Status

Trakya University

Edirne, , Turkey (Türkiye)

Site Status

Medipol Mega Universite Hastanesi

Istanbul, , Turkey (Türkiye)

Site Status

Acıbadem Maslak Hastanesi

Istanbul, , Turkey (Türkiye)

Site Status

TC Saglik Bakanligi Goztepe Prof. Dr. Suleyman Yalcin Sehir Hastanesi

Istanbul, , Turkey (Türkiye)

Site Status

Izmir Katip Celebi Ataturk Egitim Arastirma Hastanesi

Izmir, , Turkey (Türkiye)

Site Status

İnönü Üniversitesi Turgut Özal Tıp Merkezi Eğitim ve Araştırma Hastanesi

Malatya, , Turkey (Türkiye)

Site Status

Medical Center "Mriya Med-Service"

Kryvyi Rih, Dnipropetrovsk Oblast, Ukraine

Site Status

CNPE "Regional Center of Oncology"

Kharkiv, Kharkivs’ka Oblast’, Ukraine

Site Status

Municipal non-profit enterprise'Odesa Regional Clinical Hospital'of Odesa Regional Council

Odesa, Odesa Oblast, Ukraine

Site Status

Sumy regional clinical oncological dispensary

Sumy, Sumska Oblast, Ukraine

Site Status

Communal Noncommercial Enterprise "Podillia Regional Oncology Center Of Vinnytsia Regional Council"

Vinnytsia, Vinnytsia Oblast, Ukraine

Site Status

"Oncolife" LLC

Zaporizhzhia, Zaporizhzhia Oblast, Ukraine

Site Status

Municipal non-profit enterprise "Kyiv City Clinical Oncology Center" of executive body of Kyiv City Counci -T

Kyiv, , Ukraine

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Chelsea and Westminster Hospital NHS Foundation Trust

London, England, United Kingdom

Site Status

Royal Brompton Hospital

London, Kensington and Chelsea, United Kingdom

Site Status

University College London Hospital

London, London, City of, United Kingdom

Site Status

City Hospital, Nottingham University Hospitals

Nottingham, , United Kingdom

Site Status

New Cross Hospital

Wolverhampton, , United Kingdom

Site Status

Countries

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United States Australia Austria Belgium Brazil Canada China Czechia Denmark France Germany Greece Hong Kong India Israel Italy Japan Mexico Netherlands Norway Poland Puerto Rico Romania Russia Singapore South Korea Spain Sweden Taiwan Turkey (Türkiye) Ukraine United Kingdom

References

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Tsuboi M, Goldman JW, Wu YL, Johnson ML, Paz-Ares L, Yang JC, Besse B, Su W, Chao BH, Drilon A. LIBRETTO-432, a phase III study of adjuvant selpercatinib or placebo in stage IB-IIIA RET fusion-positive non-small-cell lung cancer. Future Oncol. 2022 Sep;18(28):3133-3141. doi: 10.2217/fon-2022-0656. Epub 2022 Aug 11.

Reference Type DERIVED
PMID: 35950566 (View on PubMed)

Related Links

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https://trials.lilly.com/ext/trial?id=J2G-MC-JZJX

A Study of Selpercatinib After Surgery or Radiation in Participants With Non-Small Cell Lung Cancer (NSCLC) (LIBRETTO-432)

Other Identifiers

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J2G-MC-JZJX

Identifier Type: OTHER

Identifier Source: secondary_id

2020-005191-35

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

2023-506784-33-00

Identifier Type: OTHER

Identifier Source: secondary_id

18126

Identifier Type: -

Identifier Source: org_study_id