Food Effect and Relative Bioavailability Study of Rilzabrutinib in Healthy Participants

NCT ID: NCT04748926

Last Updated: 2025-09-23

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

24 participants

Study Classification

INTERVENTIONAL

Study Start Date

2021-04-07

Study Completion Date

2021-05-21

Brief Summary

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Primary Objective:

* To evaluate the impact of food on the pharmacokinetics (PK) of rilzabrutinib following single oral doses to healthy subjects.
* To evaluate the impact of formulation on the PK of rilzabrutinib following single oral doses to healthy subjects

Secondary Objective:

\- To assess the safety and tolerability of single oral doses of rilzabrutinib administered under fasted and fed conditions

Detailed Description

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The total study duration is approximately 43 days for each participant, including a screening period of 2 to 28 days, treatment period of 12 days, and follow-up of 3 days

Conditions

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Healthy Volunteers

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

CROSSOVER

Primary Study Purpose

OTHER

Blinding Strategy

NONE

Study Groups

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Group 1

Participants will receive caplets after fast (treatment A) on Day 1 and caplets after meal (treatment B) on day 6, and then receive either oral formulation 1 tablets after fast (treatment C) or oral formulation 2 tablets after fast (treatment D) on day 11.

Group Type EXPERIMENTAL

rilzabrutinib SAR444671

Intervention Type DRUG

Pharmaceutical form: caplet Route of administration: oral

rilzabrutinib SAR444671

Intervention Type DRUG

Pharmaceutical form: Oral Formulation 1 tablets Route of administration: oral

rilzabrutinib SAR444671

Intervention Type DRUG

Pharmaceutical form: Oral Formulation 2 tablets Route of administration: oral

Group 2

Participants will receive caplets after meal (treatment B) on Day 1 and caplets after fast (treatment A) on day 6, and then receive either oral formulation 1 tablets after fast (treatment C) or oral formulation 2 tablets after fast (treatment D) on day 11.

Group Type EXPERIMENTAL

rilzabrutinib SAR444671

Intervention Type DRUG

Pharmaceutical form: caplet Route of administration: oral

rilzabrutinib SAR444671

Intervention Type DRUG

Pharmaceutical form: Oral Formulation 1 tablets Route of administration: oral

rilzabrutinib SAR444671

Intervention Type DRUG

Pharmaceutical form: Oral Formulation 2 tablets Route of administration: oral

Interventions

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rilzabrutinib SAR444671

Pharmaceutical form: caplet Route of administration: oral

Intervention Type DRUG

rilzabrutinib SAR444671

Pharmaceutical form: Oral Formulation 1 tablets Route of administration: oral

Intervention Type DRUG

rilzabrutinib SAR444671

Pharmaceutical form: Oral Formulation 2 tablets Route of administration: oral

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

\- Participants who are overtly healthy as determined by medical evaluation

* Body mass index (BMI) within the range ≥18 and ≤31 kg/m2 (inclusive) and a minimum body weight of 45 kg.
* Female participant is eligible to participate if she is not pregnant or breastfeeding
* Male participants are eligible to participate if they agree to refrain from donating sperm and use contraception/barrier or be abstinent from intercourse

Exclusion Criteria

* COVID-19 infection, positive test result for human immunodeficiency virus (HIV), hepatitis B virus or hepatitis C virus antibody
* Use of any prescription or over-the-counter (OTC) medication, herbal products, or dietary supplements within 7 days
* Participation in another clinical trial of a drug or device whereby the last investigational drug/device administration is within 30 days or 5 half-lives, whichever is longer, prior to the first dose of study drug.
* Clinically significant abnormal in vital signs. - Any specific situation during study implementation/course that may rise ethics considerations.

The above information is not intended to contain all considerations relevant to a subject's potential participation in a clinical trial.
Minimum Eligible Age

18 Years

Maximum Eligible Age

65 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

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Principia Biopharma, a Sanofi Company

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Clinical Sciences & Operations

Role: STUDY_DIRECTOR

Sanofi

Locations

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Investigational Site

Adelaide, , Australia

Site Status

Countries

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Australia

Related Links

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Other Identifiers

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U1111-1260-4526

Identifier Type: OTHER

Identifier Source: secondary_id

PRN1008-25

Identifier Type: OTHER

Identifier Source: secondary_id

PKM17098

Identifier Type: -

Identifier Source: org_study_id

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