A Bioequivalence Study Between the Proposed and Current Talazoparib Capsule Formulation and Food Effect Study for the Proposed Talazoparib Capsule Formulation in Participants With Advanced Solid Tumors

NCT ID: NCT04672460

Last Updated: 2024-09-25

Study Results

Results available

Outcome measurements, participant flow, baseline characteristics, and adverse events have been published for this study.

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

73 participants

Study Classification

INTERVENTIONAL

Study Start Date

2020-12-21

Study Completion Date

2022-07-22

Brief Summary

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This will be a Phase 1, open label, 2-sequence, crossover study to establish the BE of the current commercial formulation (Generation 3.1 talazoparib capsules) to the proposed talazoparib liquid-filled soft gelatin capsule (soft gel capsule) formulation after multiple dosing under fasting conditions in participants with advanced solid tumors. In addition, the effect of food on the PK of the proposed talazoparib soft gel capsule formulation will be evaluated in fixed sequence after the 2 BE assessment periods.

Detailed Description

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Conditions

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Advanced Solid Tumors Solid Tumors Ovarian Cancer Breast Cancer Prostate Cancer NSCLC Pancreatic Cancer Colorectal Cancer

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

CROSSOVER

Participants will be randomly assigned to 1 of 2 sequences to receive Treatment A, B and C in different order as shown below. The first 2 periods will be for BE assessment, with the first period being 28 days and the following periods being 21 days. Period 3 will be a 21 day period to evaluate the food effect on the PK of the proposed talazoparib soft gel capsule formulation that will be included in the fixed sequence after the 2 BE assessment periods (for participants who can tolerate one high-fat/high-calorie meal). Participants must have received 21 consecutive days of continuous 1mg QD drug administration to be considered as completers of a treatment period, before moving on to the next scheduled treatment.
Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Sequence 1

Participants receive Treatment B for 28 days, followed by Treatment A for 21 days, followed by Treatment C for 21 days.

Group Type EXPERIMENTAL

TALZENNA capsule

Intervention Type DRUG

Current commercial talazoparib formulation 1 mg once daily given under fasting condition

Talazoparib soft gel capsule

Intervention Type DRUG

Proposed talazoparib soft gel capsule formulation 1 mg once daily under fasting condition

Talazoparib soft gel capsule

Intervention Type DRUG

Proposed talazoparib soft gel capsule formulation 1 mg once daily under fed condition

Sequence 2

Participants receive Treatment A for 28 days, followed by Treatment B for 21 days, followed by Treatment C for 21 days.

Group Type EXPERIMENTAL

TALZENNA capsule

Intervention Type DRUG

Current commercial talazoparib formulation 1 mg once daily given under fasting condition

Talazoparib soft gel capsule

Intervention Type DRUG

Proposed talazoparib soft gel capsule formulation 1 mg once daily under fasting condition

Talazoparib soft gel capsule

Intervention Type DRUG

Proposed talazoparib soft gel capsule formulation 1 mg once daily under fed condition

Interventions

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TALZENNA capsule

Current commercial talazoparib formulation 1 mg once daily given under fasting condition

Intervention Type DRUG

Talazoparib soft gel capsule

Proposed talazoparib soft gel capsule formulation 1 mg once daily under fasting condition

Intervention Type DRUG

Talazoparib soft gel capsule

Proposed talazoparib soft gel capsule formulation 1 mg once daily under fed condition

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

1. Histological diagnosis of recurrent, locally advanced or metastatic solid tumor that is not amenable for treatment with curative intent.

* Solid tumors with known or likely pathogenic germline or somatic tumor gene defect (eg, one or more BRCA1 or BRCA2 gene defect except for ovarian cancer) that would benefit from PARPi therapy per current approvals for the tumor indication or supported by strong scientific evidence.
* Received at least 1 prior SOC regimen, if it exists, as appropriate for the respective tumor type unless deemed unsuitable or declined these therapies; ovarian cancer participants must have at least 1 prior cytotoxic chemotherapy regimen, including at least 1 course of platinum-based therapy. Participants must not have had disease progression within 6 months of initiation of platinum containing regimen.
2. ECOG performance score of 0-1.
3. Adequate bone marrow function:

* ANC ≥1500 cells/mm3
* Platelets ≥100,000 cells/mm3
* Hemoglobin ≥10.0 g/dL
4. Adequate organ functions:

* CLCR ≥60 mL/min and no documented CLCR \<60 mL/min and no change in CLCR \>25% in the past 4 weeks
* AST and ALT ≤2.5 × ULN; if liver function abnormalities are due to hepatic metastasis, then AST and ALT ≤5 × ULN;
* Total bilirubin ≤1.5 × ULN (≤3 × ULN for Gilbert's syndrome);

Exclusion Criteria

1. For ovarian participants: Non-epithelial tumors or ovarian tumors with low malignant potential (ie, borderline tumors) or mucinous tumors.
2. Toxicities from previous anti-cancer therapies must be resolved to NCI CTCAE \<Grade 2, except for alopecia, sensory neuropathies ≤Grade 2, or other Grade ≤2 AEs not constituting a safety risk, based on investigator's judgment, are acceptable.
3. Diagnosed with MDS or AML.
4. Active infection requiring systemic therapy within 2 weeks of enrollment.
5. Any condition in which active bleeding or pathological conditions may carry a high risk of bleeding (eg, known bleeding disorder, coagulopathy or tumor involvement with major vessels).
6. Known or suspected brain metastasis or active leptomeningeal disease undergoing or requiring treatment. Asymptomatic brain metastases currently not undergoing treatment are allowed.
7. Known history of testing positive for HIV, AIDS, positive HBV surface antigen, positive HCV RNA, or positive COVID-19 viral test. Asymptomatic patients with no active infection detected but positive antibody tests, indicating past infection, are allowed.
8. Current or anticipated use of P-gp inhibitors, BCRP inhibitors, and P-gp inducers within 2 weeks or 5 half-lives prior to randomization (whichever is longer) .
Minimum Eligible Age

18 Years

Maximum Eligible Age

70 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Pfizer

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Pfizer CT.gov Call Center

Role: STUDY_DIRECTOR

Pfizer

Locations

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California Cancer Associates for Research and Excellence, Inc (cCARE)

Encinitas, California, United States

Site Status

Cedars-Sinai Medical Center, Samuel Oschin Comprehensive Cancer Institute

Los Angeles, California, United States

Site Status

Cedars-Sinai Medical Center

Los Angeles, California, United States

Site Status

California Cancer Associates for Research and Excellence, Inc (cCARE)

San Marcos, California, United States

Site Status

Smilow Cancer Hospital at Yale New Haven

New Haven, Connecticut, United States

Site Status

Yale-New Haven Hospital

New Haven, Connecticut, United States

Site Status

Smilow Cancer Hospital Phase 1 Unit

New Haven, Connecticut, United States

Site Status

Florida Cancer Specialists

Lake Mary, Florida, United States

Site Status

Alliance for Multispecialty Research, LLC

Kansas City, Missouri, United States

Site Status

NYU Langone Hospital - Long Island Oncology

Mineola, New York, United States

Site Status

NYU Langone Hospital - Long Island

Mineola, New York, United States

Site Status

Laura & Isaac Perlmutter Cancer Center at NYU Langone Health

New York, New York, United States

Site Status

NYU Investigational Pharmacy

New York, New York, United States

Site Status

NYU Langone Medical Center (Tisch Hospital)

New York, New York, United States

Site Status

Montefiore Medical Center

The Bronx, New York, United States

Site Status

University of Cincinnati Medical Center

Cincinnati, Ohio, United States

Site Status

University Hospitals Cleveland Medical Center

Cleveland, Ohio, United States

Site Status

West Chester Hospital

West Chester, Ohio, United States

Site Status

UPCI Investigational Drug Service

Pittsburgh, Pennsylvania, United States

Site Status

UPMC Hillman Cancer Center

Pittsburgh, Pennsylvania, United States

Site Status

Upmc Shadyside

Pittsburgh, Pennsylvania, United States

Site Status

Mary Crowley Cancer Research - Medical City Hospital

Dallas, Texas, United States

Site Status

NEXT Oncology

San Antonio, Texas, United States

Site Status

Liverpool Cancer Therapy Centre

Liverpool, New South Wales, Australia

Site Status

Liverpool Hospital

Liverpool, New South Wales, Australia

Site Status

Monash Health

Clayton, Victoria, Australia

Site Status

Epworth Healthcare (Epworth Freemasons Hospital)

East Melbourne, Victoria, Australia

Site Status

Epworth Healthcare

East Melbourne, Victoria, Australia

Site Status

Epworth Healthcare

Richmond, Victoria, Australia

Site Status

Epworth Richmond Hospital (Epworth Healthcare)

Richmond, Victoria, Australia

Site Status

Epworth Healthcare

East Melbourne, , Australia

Site Status

Countries

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United States Australia

Provided Documents

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Document Type: Study Protocol

View Document

Document Type: Statistical Analysis Plan

View Document

Related Links

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https://pmiform.com/clinical-trial-info-request?StudyID=C3441037

To obtain contact information for a study center near you, click here.

Other Identifiers

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2020-006101-35

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

C3441037

Identifier Type: -

Identifier Source: org_study_id

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