A Study to Assess the Effects of Itraconazole and Rifampin on Lazertinib in Healthy Adult Participants

NCT ID: NCT04410094

Last Updated: 2021-03-01

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

32 participants

Study Classification

INTERVENTIONAL

Study Start Date

2020-09-14

Study Completion Date

2021-02-02

Brief Summary

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The purpose of this study is to evaluate the effects of multiple doses of strong cytochrome P450 (CYP) 3A4 inhibitor itraconazole and strong CYP3A4 inducer rifampin on the single dose pharmacokinetics (PK) of lazertinib in healthy adult participants.

Detailed Description

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Conditions

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Healthy

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

OTHER

Blinding Strategy

NONE

Study Groups

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Cohort 1: Lazertinib plus Itraconazole

Participants will receive a single oral dose of lazertinib tablets in Treatment Period 1 followed by itraconazole capsules orally along with a single oral dose of lazertinib tablet in Treatment Period 2.

Group Type EXPERIMENTAL

Lazertinib

Intervention Type DRUG

Lazertinib tablets will be administered orally.

Itraconazole

Intervention Type DRUG

Itraconazole capsules will be administered orally.

Cohort 2: Lazertinib plus Rifampin

Participants will receive a single oral dose of lazertinib tablets in Treatment Period 1 followed by rifampin capsules orally along with a single oral dose of lazertinib tablet in Treatment Period 2.

Group Type EXPERIMENTAL

Lazertinib

Intervention Type DRUG

Lazertinib tablets will be administered orally.

Rifampin

Intervention Type DRUG

Rifampin capsules will be administered orally.

Interventions

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Lazertinib

Lazertinib tablets will be administered orally.

Intervention Type DRUG

Itraconazole

Itraconazole capsules will be administered orally.

Intervention Type DRUG

Rifampin

Rifampin capsules will be administered orally.

Intervention Type DRUG

Other Intervention Names

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JNJ-73841937; YH25448

Eligibility Criteria

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Inclusion Criteria

* A woman must not be of childbearing potential and must have a negative serum beta-human chorionic gonadotropin (Beta HCG) pregnancy test at screening
* Hormone replacement therapy (if applicable) must have been discontinued at least 28 days prior to the first dose of study drug (Cohort 2 only)
* Participants must have a body mass index (BMI) between 18.0 and 32.0 kilogram per meter square (kg/m\^2, inclusive (BMI = weight/height\^2), and body weight not less than 50 kg at screening
* Participants must be healthy based on physical examination, medical history, and vital signs (pulse and body temperature), performed at screening
* Male participants must agree to use an adequate contraception method

Exclusion Criteria

* History of or current clinically significant medical illness that the investigator considers should exclude the participant or that could interfere with the interpretation of the study results
* History of infection suspected or confirmed to be related to Coronavirus disease 2019 (COVID-19) within 4 weeks before intake of study drug
* Participant has known allergies, hypersensitivity, or intolerance to lazertinib or its excipients or to itraconazole and rifampin
* Participant has contraindications to the use itraconazole and rifampin per local prescribing information
* Use of any cytochrome P450 (CYP) 3A4 inhibitors or inducers (other than per-protocol itraconazole/rifampin administration) within 4 weeks before the first dose of the study drug is scheduled until completion of the study
Minimum Eligible Age

18 Years

Maximum Eligible Age

60 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

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Janssen Research & Development, LLC

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Janssen Research & Development, LLC Clinical Trial

Role: STUDY_DIRECTOR

Janssen Research & Development, LLC

Locations

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Celerion

Tempe, Arizona, United States

Site Status

Countries

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United States

Other Identifiers

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73841937NSC1003

Identifier Type: OTHER

Identifier Source: secondary_id

CR108799

Identifier Type: -

Identifier Source: org_study_id

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