Study to Evaluate Loncastuximab Tesirine With Rituximab Versus Immunochemotherapy in Participants With Relapsed or Refractory Diffuse Large B-Cell Lymphoma

NCT ID: NCT04384484

Last Updated: 2025-11-05

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

ACTIVE_NOT_RECRUITING

Clinical Phase

PHASE3

Total Enrollment

440 participants

Study Classification

INTERVENTIONAL

Study Start Date

2020-09-16

Study Completion Date

2028-06-30

Brief Summary

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The purpose of this study is to evaluate the efficacy of loncastuximab tesirine (ADCT-402) combined with rituximab compared to standard immunochemotherapy.

Detailed Description

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Conditions

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Refractory Diffuse Large B-Cell Lymphoma Relapsed Diffuse Large B-Cell Lymphoma

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Part 1: Loncastuximab Tesirine + Rituximab (Lonca-R)

Part 1 consists of a non-randomized safety run-in period evaluating the study drug for the first 20 participants.

Participants will receive Lonca-R on Day 1 of each cycle for up to 8 cycles, where 1 cycle is 3 weeks. Lonca-R will be administered via an intravenous infusion of loncastuximab tesirine 150 µg/kg + rituximab 375 mg/m\^2 Q3W for 2 cycles, then loncastuximab tesirine 75 µg/kg + rituximab 375 mg/m\^2 Q3W for up to 6 additional cycles.

Group Type EXPERIMENTAL

Loncastuximab Tesirine

Intervention Type DRUG

Intravenous Infusion

Rituximab

Intervention Type DRUG

Intravenous Infusion

Part 2: Loncastuximab Tesirine + Rituximab (Lonca-R)

Randomized participants will receive Lonca-R on Day 1 of each cycle for up to 8 cycles, where 1 cycle is 3 weeks. Lonca-R will be administered via an intravenous infusion of loncastuximab tesirine 150 µg/kg + rituximab 375 mg/m\^2 every Q3W for 2 cycles, then loncastuximab tesirine 75 µg/kg + rituximab 375 mg/m\^2 Q3W for up to 6 additional cycles.

Group Type EXPERIMENTAL

Loncastuximab Tesirine

Intervention Type DRUG

Intravenous Infusion

Rituximab

Intervention Type DRUG

Intravenous Infusion

Part 2: Standard Immunochemotherapy (R-GemOx)

Randomized participants will receive R-GemOx consisting of rituximab, gemcitabine and oxaliplatin as a standard immunochemotherapy treatment on Day 1 or Day 2 of each cycle for up to 8 cycles, where 1 Cycle is 2 weeks. R-GemOx will be administered via an intravenous infusion of rituximab 375 mg/m\^2 + gemcitabine 1000 mg/m\^2 + oxaliplatin 100 mg/m\^2 every 2 weeks (Q2W) for up to 8 cycles.

Group Type ACTIVE_COMPARATOR

Rituximab

Intervention Type DRUG

Intravenous Infusion

Gemcitabine

Intervention Type DRUG

Intravenous Infusion

Oxaliplatin

Intervention Type DRUG

Intravenous Infusion

Interventions

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Loncastuximab Tesirine

Intravenous Infusion

Intervention Type DRUG

Rituximab

Intravenous Infusion

Intervention Type DRUG

Gemcitabine

Intravenous Infusion

Intervention Type DRUG

Oxaliplatin

Intravenous Infusion

Intervention Type DRUG

Other Intervention Names

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Zynlonta ADCT-402

Eligibility Criteria

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Inclusion Criteria

* Male or female participant aged 18 years or older
* Pathologic diagnosis of DLBCL, as defined by the 2016 World Health Organization classification (including participants with DLBCL transformed from indolent lymphoma), or high-grade B-cell lymphoma, with MYC and BCL2 and/or BCL6 rearrangements
* Relapsed (disease that has recurred following a response) or refractory (disease that failed to respond to prior therapy) disease following at least one multi-agent systemic treatment regimen \[For China only: Adequate first line anti-DLBCL therapy is defined as having received at least 4 cycles of multiagent systemic treatment regimen containing rituximab and anthracycline, unless the participants are intolerant to the regimen, or had disease progression during the treatment. If disease progression occurred during the treatment period, then the disease is considered refractory where the number of treatment cycles will not be specified. For participants who are ineligible for anthracycline, anthracycline is not required.\]
* Not considered by the investigator to be a candidate for stem cell transplantation based on performance status, advanced age, and/or significant medical comorbidities such as organ dysfunction
* Measurable disease as defined by the 2014 Lugano Classification as assessed by positron-emission tomography (PET)- computed tomography (CT) or by CT or magnetic resonance imaging (MRI) if tumor is not fluorodeoxyglucose (FDG)-avid on screening PET-CT
* Availability of formalin-fixed paraffin-embedded (FFPE) tumor tissue block (or minimum 10 freshly cut unstained slides if block is not available) Note: Any biopsy since initial diagnosis is acceptable, but if several samples are available, the most recent sample is preferred \[For China only: This inclusion criterion is not applicable\]
* ECOG performance status 0-2
* Adequate organ function as defined by screening laboratory values within the following parameters:

1. Absolute neutrophil count ≥1000/μL (off growth factors for at least 72 hours)
2. Platelet count ≥100000/μL without transfusion within the past 2 weeks
3. ALT, AST, and GGT ≤2.5 × the upper limit of normal (ULN)
4. Total bilirubin ≤1.5 × ULN (participants with known Gilbert's syndrome may have a total bilirubin up to ≤3 × ULN)
5. Calculated creatinine clearance ≥30 mL/min by the Cockcroft and Gault equation

Note: A laboratory assessment may be repeated a maximum of two times during the Screening period to confirm eligibility.

* Negative beta-human chorionic gonadotropin (β-hCG) pregnancy test within 7 days prior to start of study drug (Cycle 1 Day 1) for women of childbearing potential
* Women of childbearing potential must agree to use a highly effective method of contraception from the time of giving informed consent until at least 12 months after the last dose of study treatment. Men with female partners who are of childbearing potential must agree to use a condom when sexually active or practice total abstinence from the time of giving informed consent until at least 7 months after the participant receives his last dose of study treatment.

Exclusion Criteria

* Previous treatment with loncastuximab tesirine
* Previous treatment with R-GemOx
* Known history of hypersensitivity to a CD19 antibody, loncastumiximab tesirine (including SG3249) or any of its excipients, or history of positive serum human ADA to a CD19 antibody
* Pathologic diagnosis of Burkitt lymphoma
* Active second primary malignancy other than non-melanoma skin cancers, non-metastatic prostate cancer, in situ cervical cancer, ductal or lobular carcinoma in situ of the breast, or other malignancy that the Sponsor's medical monitor and Investigator agree and document should not be exclusionary
* Autologous transplant within 30 days prior to start of study drug (Cycle 1 Day 1)
* Allogeneic transplant within 60 days prior to start of study drug (Cycle 1 Day 1)
* Active graft-versus-host disease
* Post-transplantation lymphoproliferative disorders
* Active autoimmune disease, including motor neuropathy considered of autoimmune origin and other central nervous system (CNS) autoimmune disease
* Human immunodeficiency virus (HIV) seropositive with any of the following:

1. CD4+ T-cell (CD4+) counts \<350 cells/μL
2. Acquired immunodeficiency syndrome-defining opportunistic infection within 12 months prior to screening
3. Not on anti-retroviral therapy, or on anti-retroviral therapy for \<4 weeks at the time of screening
4. HIV viral load ≥400 copies/mL
* Serologic evidence of chronic hepatitis B virus (HBV) infection and unable or unwilling to receive standard prophylactic antiviral therapy or with detectable HBV viral load
* Serologic evidence of hepatitis C virus (HCV) infection without completion of curative treatment or with detectable HCV viral load
* History of Stevens-Johnson syndrome or toxic epidermal necrolysis
* Lymphoma with active CNS involvement, including leptomeningeal disease
* Clinically significant third space fluid accumulation (i.e., ascites requiring drainage or pleural effusion that is either requiring drainage or associated with shortness of breath)
* Breastfeeding or pregnant
* Uncontrolled hypertension (blood pressure ≥160/100 mm Hg repeatedly), unstable angina, congestive heart failure (greater than New York Heart Association class II), electrocardiographic evidence of acute ischemia, coronary angioplasty or myocardial infarction within 6 months prior to screening, uncontrolled atrial or ventricular cardiac arrhythmia, poorly controlled diabetes, severe chronic pulmonary disease, or other serious medical condition which is likely to significantly impair the participant's ability to tolerate the study treatment
* Major surgery within 4 weeks prior to start of study drug (Cycle 1 Day 1); radiotherapy, chemotherapy or other antineoplastic therapy within 14 days prior to start of study drug (Cycle 1 Day 1), except shorter if approved by the Sponsor
* Use of any other experimental medication within 14 days or 5 half-lives prior to start of study drug (Cycle 1 Day 1)
* Received live vaccine within 4 weeks of Cycle 1 Day 1
* Failure to recover to ≤Grade 1 (Common Terminology Criteria for Adverse Events \[CTCAE\] version 5.0) from acute non-hematologic toxicity (except alopecia) due to previous therapy prior to screening
* Congenital long QT syndrome or a corrected QTcF interval of ≥480 ms at screening (unless secondary to pacemaker or bundle branch block)
* Any other significant medical illness, abnormality, or condition that would, in the Investigator's judgment, make the participant inappropriate for study participation or put the participant at risk
* Known history of hypersensitivity to oxaliplatin or other platinum-based drugs, or gemcitabine, or rituximab, or any of their excipients
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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ADC Therapeutics S.A.

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Locations

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University of California San Diego Moores Cancer Center

La Jolla, California, United States

Site Status

Redlands Community Hospital

Redlands, California, United States

Site Status

The Oncology Institute of Hope and Innovation

Whittier, California, United States

Site Status

Baptist MD Anderson Cancer Center

Jacksonville, Florida, United States

Site Status

UnityPoint Health - Iowa Oncology Research Association (IORA)

Des Moines, Iowa, United States

Site Status

Norton Cancer Institute

Louisville, Kentucky, United States

Site Status

Comprehensive Cancer Centers of Nevada - Henderson

Las Vegas, Nevada, United States

Site Status

Kaiser Permanente Interstate Medical Office Central

Portland, Oregon, United States

Site Status

Hollings Cancer Center

Charleston, South Carolina, United States

Site Status

Virginia Cancer Specialists

Gainesville, Virginia, United States

Site Status

Medical College of Wisconsin Cancer Center Clinical Trials Office

Milwaukee, Wisconsin, United States

Site Status

Clinica Adventista Belgrano

Belgrano, Buenos Aires, Argentina

Site Status

Clínica de Nefrología, Urología y Enfermedades Cardiovasculares S.A.

Santa Fe, Buenos Aires, Argentina

Site Status

Instituto Médico Especializado Alexander Fleming

Buenos Aires, Distrito Federal, Argentina

Site Status

Grupo Gamma - Hospital Privado Rosario

Rosario, Santa Fe Province, Argentina

Site Status

Algemeen Ziekenhuis Sint-Jan Brugge-Oostende - Campus Sint-Jan

Bruges, , Belgium

Site Status

Cliniques Universitaires Saint-Luc

Brussels, , Belgium

Site Status

Centre Hospitalier Universitaire Universite Catholique de Louvain

Namur, , Belgium

Site Status

Algemeen Ziekenhuis Delta - Campus Rumbeke

Roeselare, , Belgium

Site Status

Hospital Erasto Gaertner - Liga Paranaense de Combate ao Câncer

Curitiba, Paraná, Brazil

Site Status

Hospital Moinhos de Vento

Porto Alegre, Rio Grande do Sul, Brazil

Site Status

Hospital de Clínicas de Porto Alegre

Porto Alegre, Rio Grande do Sul, Brazil

Site Status

Hospital Mãe de Deus - Centro Integrado de Oncologia

Porto Alegre, Rio Grande do Sul, Brazil

Site Status

Hospital do Câncer

Rio de Janeiro, , Brazil

Site Status

Hemomed Instituto de Oncologia e Hematologia

São Paulo, , Brazil

Site Status

A Beneficência Portuguesa de São Paulo - Unidade Mirante

São Paulo, , Brazil

Site Status

Hospital das Clínicas da Faculdade de Medicina da Universidade de São Paulo

São Paulo, , Brazil

Site Status

Hospital Israelita Albert Einstein

São Paulo, , Brazil

Site Status

Hospital Santa Marcelina

São Paulo, , Brazil

Site Status

Cross Cancer Institute

Edmonton, , Canada

Site Status

Research Institute of the McGill University Health Centre

Montreal, , Canada

Site Status

Hôpital Fleurimont

Sherbrooke, , Canada

Site Status

Centro de Estudios Clínicos SAGA

Santiago, Santiago Metropolitan, Chile

Site Status

Instituto Oncológico Fundación Arturo López Pérez

Santiago, Santiago Metropolitan, Chile

Site Status

CeCim - Centro de Estudios Clínicos e Investigaciones Médicas

Santiago, Santiago Metropolitan, Chile

Site Status

Peking University Third Hospital

Beijing, Beijing Municipality, China

Site Status

The First Affiliated Hospital of Xiamen University

Xiamen, Fujian, China

Site Status

Sun Yat-Sen University Cancer Center

Guangzhou, Guangdong, China

Site Status

Guangdong Provincial People's Hospital

Guangzhou, Guangdong, China

Site Status

Zhujiang Hospital of Southern Medical University

Guangzhou, Guangdong, China

Site Status

Henan Cancer Hospital - Zhengzhou University

Zhengzhou, Henan, China

Site Status

Jilin Cancer Hospital

Changchun, Jilin, China

Site Status

The First Hospital of Jilin University

Changchun, Jilin, China

Site Status

Second Affiliated Hospital of Dalian Medical University

Dalian, Liaoning, China

Site Status

Shanghai Cancer Center

Shanghai, Shanghai Municipality, China

Site Status

West China School of Medicine - West China Hospital of Sichuan University

Chengdu, Sichuan, China

Site Status

Tianjin Medical University Cancer Institute & Hospital

Tianjin, Tianjin Municipality, China

Site Status

The First Affiliated Hospital of Zhejiang University School of Medicine

Hangzhou, Zhejiang, China

Site Status

Chongqing University Cancer Hospital - Chongqing Cancer Hospital

Chongqing, , China

Site Status

Huizhou Municipal Central Hospital

Huizhou, , China

Site Status

The First Affiliated Hospital of Nanchang University

Nanchang, , China

Site Status

Institute of Hematology and Blood Diseases Hospital of CAMS - PUMC

Tianjin, , China

Site Status

Wuhan Union Hospital

Wuhan, , China

Site Status

Tongji Hospital

Wuhan, , China

Site Status

Fakultni nemocnice Ostrava

Ostrava, , Czechia

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Fakultni Nemocnice Kralovske Vinohrady

Prague, , Czechia

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Fakultni nemocnice v Motole

Prague, , Czechia

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Centre Hospitalier Regional Universitaire Brest

Brest, Brittany Region, France

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Hôpital Avicenne

Bobigny, , France

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Centre Hospitalier Regional Universitaire Brest

Brest, , France

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Hôpital François Mitterrand

Dijon, , France

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Hôpital Privé du Confluent

Nantes, , France

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Hopital Universitaire Pitie Salpetriere

Paris, , France

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Hôpital Haut-Lévêque

Pessac, , France

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Centre de Lutte Contre le Cancer - Centre Henri-Becquerel

Rouen, , France

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Heves Varmegyei Markhot Ferenc Oktatokorhaz es Rendelointezet

Heves, Budapest, Hungary

Site Status

Dél-pesti Centrumkórház - Országos Hematológiai és Infektológiai Intézet - Szent László

Budapest, Pest County, Hungary

Site Status

Semmelweis Egyetem

Budapest, , Hungary

Site Status

Orszagos Onkologiai Intezet

Budapest, , Hungary

Site Status

Samson Assuta Ashdod University Hospital

Ashdod, , Israel

Site Status

Soroka Medical Center

Beersheba, , Israel

Site Status

Shamir Medical Center (Assaf Harofeh)

Be’er Ya‘aqov, , Israel

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Carmel Medical Center

Haifa, , Israel

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Rabin Medical Center - Beilinson Hospital

Petah Tikva, , Israel

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The Chaim Sheba Medical Center

Tel Aviv, , Israel

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Tel Aviv Sourasky Medical Center

Tel Aviv, , Israel

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Presidio Ospedaliero Universitario Santa Maria della Misericordia

Udine, Friuli Venezia Giulia, Italy

Site Status

Azienda Socio Sanitaria Territoriale (ASST) degli Spedali Civili di Brescia

Brescia, , Italy

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Azienda Ospedaliero - Universitaria Careggi

Florence, , Italy

Site Status

Ospedale Casa Sollievo della Sofferenza

Foggia, , Italy

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Istituto Romagnolo per lo Studio dei Tumori "Dino Amadori" - IRST

Meldola, , Italy

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Istituto di Ricovero e Cura a Carattere Scientifico (IRCCS) - Istituto Clinico Humanitas

Milan, , Italy

Site Status

Istituto di Ricovero e Cura a Carattere Scientifico (IRCCS) - Ospedale San Raffaele

Milan, , Italy

Site Status

Istituto Europeo di Oncologia

Milan, , Italy

Site Status

Fondazione IRCCS Policlinico San Matteo

Pavia, , Italy

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Sanitaria Locale della Romagna

Ravenna, , Italy

Site Status

National Hospital Organization - Nagoya Medical Center

Nagoya, Aichi-ken, Japan

Site Status

Toyohashi Municipal Hospital

Toyohashi, Aichi-ken, Japan

Site Status

National Cancer Center Hospital East

Kashiwa, Chiba, Japan

Site Status

Matsuyama Red Cross Hospital

Matsuyama, Ehime, Japan

Site Status

Gunma Prefectural Cancer Center

Ōta, Gunma, Japan

Site Status

Sapporo Hokuyu Hospital

Sapporo, Hokkaido, Japan

Site Status

Hokkaido Cancer Center

Sapporo, Hokkaido, Japan

Site Status

Kobe City Medical Center General Hospital

Kobe, Hyōgo, Japan

Site Status

Kanagawa Cancer Center

Yokohama, Kanagawa, Japan

Site Status

Tohoku University Hospital

Sendai, Miyagi, Japan

Site Status

Nagasaki University Hospital

Nagasaki, Nagasaki, Japan

Site Status

Saitama Medical University - International Medical Center

Hidaka-Shi, Saitama, Japan

Site Status

Tokyo Metropolitan Cancer and Infectious Diseases Center Komagome Hospital

Bunkyo-ku, Tokyo, Japan

Site Status

National Hospital Organization Disaster Medical Center

Tachikawa, Tokyo, Japan

Site Status

Fukushima Medical University Hospital

Fukushima, , Japan

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Gifu Municipal Hospital

Gifu, , Japan

Site Status

Kagoshima University Hospital

Kagoshima, , Japan

Site Status

Niigata University Medical and Dental Hospital

Niigata, , Japan

Site Status

National Hospital Organization Okayama Medical Center

Okayama, , Japan

Site Status

Osaka Prefectural Hospital Organization - Osaka International Cancer Institute

Osaka, , Japan

Site Status

Boca Raton Clinical Research (BRCR) Global Mexico - Guadalajara

Guadalajara, Jalisco, Mexico

Site Status

PanAmerican Clinical Research Mexico - Guadalajara

Guadalajara, Jalisco, Mexico

Site Status

PanAmerican Clinical Research Mexico - Cuernavaca

Cuernavaca, Morelos, Mexico

Site Status

Hospital Universitario Dr. José Eleuterio González

Monterrey, Nuevo León, Mexico

Site Status

Hematológica Alta Especialidad

Huixquilucan, , Mexico

Site Status

Boca Raton Clinical Research (BRCR) Global Mexico - Ciudad de México

Mexico City, , Mexico

Site Status

Hagaziekenhuis Van Den Haag - Leyweg

The Hague, South Holland, Netherlands

Site Status

Elisabeth-TweeSteden Ziekenhuis - Elisabeth

Tilburg, , Netherlands

Site Status

Pratia MCM Kraków

Krakow, Lesser Poland Voivodeship, Poland

Site Status

Uniwersytecki Szpital Kliniczny im. Jana Mikulicza-Radeckiego we Wrocławiu

Wroclaw, Lower Silesian Voivodeship, Poland

Site Status

Szpitale Pomorskie Spółka Z Ograniczoną Odpowiedzialnością

Gdynia, , Poland

Site Status

Pratia Onkologia Katowice

Katowice, , Poland

Site Status

Wojewodzkie Wielospecjalistyczne Centrum Onkologii i Traumatologii im. M. Kopernika w Lodzi

Lodz, , Poland

Site Status

Szpital Wojewódzki w Opolu

Opole, , Poland

Site Status

Centrum Medyczne Pratia Poznań

Skorzewo, , Poland

Site Status

Instytut Hematologii I Transfuzjologii

Warsaw, , Poland

Site Status

Hospital Español Auxilio Mutuo

San Juan, , Puerto Rico

Site Status

Hospital del Mar - Parc de Salut Mar

Barcelona, , Spain

Site Status

Institut Català d'Oncologia - Hospital Duran i Reynals (ICO L'Hospitalet)

Barcelona, , Spain

Site Status

Hospital San Pedro de Alcantara

Cáceres, , Spain

Site Status

Hospital Universitario Ramón y Cajal

Madrid, , Spain

Site Status

Hospital Universitario Fundación Jiménez Díaz

Madrid, , Spain

Site Status

Hospital Universitario 12 de Octubre

Madrid, , Spain

Site Status

Hospital Universitario La Paz

Madrid, , Spain

Site Status

Hospital Universitario Marqués de Valdecilla

Santander, , Spain

Site Status

Hospital Universitario Virgen del Rocío

Seville, , Spain

Site Status

Hospital Arnau de Vilanova

Valencia, , Spain

Site Status

Istituto Oncologico della Svizzera Italiana

Bellinzona, , Switzerland

Site Status

Özel Koru Hastanesi

Çukurambar, Ankara, Turkey (Türkiye)

Site Status

VKV Amerikan Hastanesi

Şişli, Istanbul, Turkey (Türkiye)

Site Status

Ege Universitesi Tip Fakultesi Hastanesi

Bornova, İzmir, Turkey (Türkiye)

Site Status

Ondokuz Mayis Üniversitesi

Kurupelit, Samsun, Turkey (Türkiye)

Site Status

Karadeniz Teknik Üniversitesi Tip Fakültesi

Ortahisar, Trabzon, Turkey (Türkiye)

Site Status

Ankara Universitesi Tip Fakultesi - Cebeci Arastirma ve Uygulama Hastanesi

Ankara, , Turkey (Türkiye)

Site Status

Mehmet Kemal Dedeman Hematoloji Hastanesi

Kayseri, , Turkey (Türkiye)

Site Status

The Royal Marsden NHS Foundation Trust

Sutton, England, United Kingdom

Site Status

NHS Greater Glasgow and Clyde

Glasgow, , United Kingdom

Site Status

The Christie NHS Foundation Trust

Manchester, , United Kingdom

Site Status

Countries

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United States Argentina Belgium Brazil Canada Chile China Czechia France Hungary Israel Italy Japan Mexico Netherlands Poland Puerto Rico Spain Switzerland Turkey (Türkiye) United Kingdom

Other Identifiers

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2020-000241-14

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

ADCT-402-311

Identifier Type: -

Identifier Source: org_study_id

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