A Single Dose Safety, Tolerability, Pharmacokinetic and Food Effect Study of KVD900 (Sebetralstat) in Healthy Volunteers

NCT ID: NCT04349800

Last Updated: 2025-04-29

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

84 participants

Study Classification

INTERVENTIONAL

Study Start Date

2018-01-04

Study Completion Date

2018-09-10

Brief Summary

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A safety, tolerability, pharmacokinetic and food effect study of KVD900 in healthy volunteers.

Detailed Description

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Conditions

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Hereditary Angioedema

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

DOUBLE

Participants Caregivers

Study Groups

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Single Ascending Dose - 5 mg

Group Type EXPERIMENTAL

KVD900

Intervention Type DRUG

Active

Placebo to KVD900

Intervention Type DRUG

Placebo

Single Ascending Dose - 10 mg

Group Type EXPERIMENTAL

KVD900

Intervention Type DRUG

Active

Placebo to KVD900

Intervention Type DRUG

Placebo

Single Ascending Dose - 20 mg

Group Type EXPERIMENTAL

KVD900

Intervention Type DRUG

Active

Placebo to KVD900

Intervention Type DRUG

Placebo

Single Ascending Dose - 40 mg

Group Type EXPERIMENTAL

KVD900

Intervention Type DRUG

Active

Placebo to KVD900

Intervention Type DRUG

Placebo

Single Ascending Dose - 80 mg

Group Type EXPERIMENTAL

KVD900

Intervention Type DRUG

Active

Placebo to KVD900

Intervention Type DRUG

Placebo

Single Ascending Dose - 160 mg

Group Type EXPERIMENTAL

KVD900

Intervention Type DRUG

Active

Placebo to KVD900

Intervention Type DRUG

Placebo

Single Ascending Dose - 300 mg

Group Type EXPERIMENTAL

KVD900

Intervention Type DRUG

Active

Placebo to KVD900

Intervention Type DRUG

Placebo

Single Ascending Dose - 600 mg

Group Type EXPERIMENTAL

KVD900

Intervention Type DRUG

Active

Placebo to KVD900

Intervention Type DRUG

Placebo

Formulation Screen

Group Type EXPERIMENTAL

KVD900

Intervention Type DRUG

Active

Food Effect

Group Type EXPERIMENTAL

KVD900

Intervention Type DRUG

Active

Interventions

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KVD900

Active

Intervention Type DRUG

Placebo to KVD900

Placebo

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Healthy male subjects between 18 and 55 years of age.
* Healthy subjects as determined by past medical history and as judged by the Chief Investigator or designee.
* Male subject willing to use a highly effective method of contraception.
* Subject with a body mass index (BMI) of 18-32 kg/m2.
* Subject with no clinically significant history of previous allergy or sensitivity to KVD900 or any of the excipients contained within the investigational medicinal product (IMP).
* Subject with no clinically significant abnormal serum biochemistry, haematology, clotting profiles, and urine examination values within 28 days before the first dose of IMP.
* Subject with a negative urinary drugs of abuse screen, determined within 28 days before the first dose of IMP
* Subject with negative human immunodeficiency virus (HIV) and hepatitis B surface antigen (Hep B) and hepatitis C virus antibody (Hep C) results.
* Subject with no clinically significant abnormalities in 12-lead electrocardiogram
* Subjects must not donate sperm from first dose until at least 3 months after last dose of IMP.
* Subjects without any special food restrictions that would hinder ability to consume the high fat breakfast provided during study Part C; such as lactose intolerance , vegan, low-fat, low sodium, etc.
* Subjects with no known allergy or sensitivity to lactose and/or any additional excipients contained in IMP.
* Subject must be available to complete the study (including all follow up visits).
* Subject must satisfy the Chief Investigator or designee about their fitness to participate in the study.
* Subject must provide written informed consent to participate in the study.

Exclusion Criteria

* A clinically significant history of gastrointestinal disorder likely to influence IMP absorption.
* Use of prescription or non-prescription drugs, including vitamins, herbal and dietary supplements .
* Evidence of renal, hepatic, central nervous system, respiratory, cardiovascular (no history of syncope or vasovagal events), or metabolic dysfunction.
* Subjects with a history of clotting abnormalities.
* A clinically significant history of drug or alcohol abuse in the last 5 years.
* Users of nicotine products i.e., current smokers or ex-smokers who have smoked within the 6 months prior to dosing with the study medication or users of cigarette replacements.
* Inability to communicate well with Investigators.
* Participation in a New Chemical Entity clinical study within the previous 3 months or a marketed drug clinical study within the 30 days before the first dose of IMP.
* Donation of 450 mL or more blood within the 3 months before the first dose of IMP.
Minimum Eligible Age

18 Years

Maximum Eligible Age

55 Years

Eligible Sex

MALE

Accepts Healthy Volunteers

Yes

Sponsors

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KalVista Pharmaceuticals, Ltd.

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Locations

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KalVista Investigative Site

Wales, , United Kingdom

Site Status

Countries

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United Kingdom

References

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Maetzel A, Smith MD, Duckworth EJ, Hampton SL, De Donatis GM, Murugesan N, Rushbrooke LJ, Li L, Francombe D, Feener EP, Yea CM. KVD900, an oral on-demand treatment for hereditary angioedema: Phase 1 study results. J Allergy Clin Immunol. 2022 Jun;149(6):2034-2042. doi: 10.1016/j.jaci.2021.10.038. Epub 2022 Jan 24.

Reference Type DERIVED
PMID: 35086692 (View on PubMed)

Other Identifiers

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KVD900-101

Identifier Type: -

Identifier Source: org_study_id

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