A Study to Evaluate the Safety and Efficacy of NG101 in Adult Participants With Symptomatic Diabetic or Idiopathic Gastroparesis

NCT ID: NCT04303195

Last Updated: 2025-08-28

Study Results

Results available

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE2

Total Enrollment

161 participants

Study Classification

INTERVENTIONAL

Study Start Date

2020-08-01

Study Completion Date

2023-02-25

Brief Summary

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The purpose of this study is to assess the safety and efficacy of various dose levels of NG101 compared with placebo in adult participants with gastroparesis during 12 weeks of treatment.

Detailed Description

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This is a randomized, double-blind, parallel-group , placebo-controlled, multicenter US-based study to evaluate the safety and efficacy of 3 dose levels of NG101 (Metopimazine mesylate) compared with placebo in participants with diabetic or idiopathic gastroparesis.

The study will enroll approximately 140 participants. Following the Screening Period, there is a 2-week Pretreatment Period during which participants will complete an electronic daily diary. Participants eligible for the clinical study will be randomly assigned (in a 1:1:1:1 ratio) to receive either NG101 5 mg, 10 mg, or 20 mg, or matching placebo during a 12-week Treatment Period. All participants will be asked to take one capsule 30 minutes before a meal 3 times a day and 30 minutes before bedtime for a total of 4 capsules daily (QID). The total duration of the study for each participant will be approximately 20 weeks.

Conditions

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Diabetic Gastroparesis Idiopathic Gastroparesis

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Parallel Assignment
Primary Study Purpose

OTHER

Blinding Strategy

QUADRUPLE

Participants Caregivers Investigators Outcome Assessors

Study Groups

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NG101 - 5 mg

NG101 5 mg, capsules, orally, QID (4 times a day) for up to 12 weeks

Group Type EXPERIMENTAL

NG101

Intervention Type DRUG

Capsules

NG101 - 10 mg

NG101 10 mg, capsules, orally, QID (4 times a day) for up to 12 weeks

Group Type EXPERIMENTAL

NG101

Intervention Type DRUG

Capsules

NG101 - 20 mg

NG101 20 mg, capsules, orally, QID (4 times a day) for up to 12 weeks

Group Type EXPERIMENTAL

NG101

Intervention Type DRUG

Capsules

Placebo

Placebo-matching, capsules, orally, QID (4 times a day) for up to 12 weeks

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DRUG

Capsules

Interventions

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NG101

Capsules

Intervention Type DRUG

Placebo

Capsules

Intervention Type DRUG

Other Intervention Names

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metopimazine mesylate

Eligibility Criteria

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Inclusion Criteria

* Adult patients with diabetic or idiopathic gastroparesis
* Symptoms consistent with gastroparesis (nausea, vomiting, early satiety, post-prandial fullness, and abdominal pain)
* Documented evidence of no mechanical obstruction
* Delayed gastric emptying as demonstrated by gastric scintigraphy or breath test

Exclusion Criteria

* Uncontrolled diabetes (defined as HgbA1c \> 10%)
* Severe postural symptoms or evidence of unexplained recurrent dizziness
* Participant has received and tolerated domperidone and showed no notable symptomatic improvement in gastroparesis symptoms
* Participant has had endoscopic pyloric injections of botulinum toxin within the 6 months prior to the Screening Visit.
* Participant engages in daily recreational use of marijuana
* Prolactin levels \> 2 x ULN
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Neurogastrx, Inc.

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Locations

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Digestive Health Specialists

Dothan, Alabama, United States

Site Status

G & L Research, LLC

Foley, Alabama, United States

Site Status

East View Medical Research

Mobile, Alabama, United States

Site Status

Phoenix Medical Group

Peoria, Arizona, United States

Site Status

Phoenix Clinical LLC

Phoenix, Arizona, United States

Site Status

Del Sol Research Management

Tucson, Arizona, United States

Site Status

Preferred Research Partners

Little Rock, Arkansas, United States

Site Status

GW Research, Inc

Chula Vista, California, United States

Site Status

Precision Research Institute, LLC

Chula Vista, California, United States

Site Status

Kindred Medical Institute for Clinical Trials, LLC

Corona, California, United States

Site Status

Diagnamics Inc.

Encinitas, California, United States

Site Status

Paragon Rx Clinical, Inc

Garden Grove, California, United States

Site Status

United Clinical Research

Irvine, California, United States

Site Status

Prime Care Clinical Rsearch

Laguna Hills, California, United States

Site Status

Torrance Clinical Research Institute, Inc.

Lomita, California, United States

Site Status

Angel City Research

Los Angeles, California, United States

Site Status

United Clinical Research

Murrieta, California, United States

Site Status

Diabetes Medical Center of California

Northridge, California, United States

Site Status

Precision Research Institute

San Diego, California, United States

Site Status

Peak Gastroenterology Associates

Colorado Springs, Colorado, United States

Site Status

Innovative Research of West Florida

Clearwater, Florida, United States

Site Status

Innovation Medical Group, LLC.

Fort Lauderdale, Florida, United States

Site Status

ENCORE Borland-Grover Clinical Research

Jacksonville, Florida, United States

Site Status

ClinCloud, LLC

Maitland, Florida, United States

Site Status

Verus Clinical Research, Corp

Miami, Florida, United States

Site Status

APF Research, LLC

Miami, Florida, United States

Site Status

Panax Clinical Research

Miami, Florida, United States

Site Status

International Research Associates LLC

Miami, Florida, United States

Site Status

PharmaSouth Research

Miami, Florida, United States

Site Status

Sensible Healthcare

Ocoee, Florida, United States

Site Status

Innovation Medical Research Center

Palmetto Bay, Florida, United States

Site Status

AES - DRS - Synexus Clinical Research US, Inc. - St. Petersburg

Pinellas Park, Florida, United States

Site Status

Avita Clinical Research

Tampa, Florida, United States

Site Status

Agile Clinical Research Trials, LLC

Atlanta, Georgia, United States

Site Status

IResearch Atlanta LLC

Decatur, Georgia, United States

Site Status

Claude Mandel Medical Center

Chicago, Illinois, United States

Site Status

Medisphere Medical Research Center LLC

Evansville, Indiana, United States

Site Status

Indiana University Hospital

Indianapolis, Indiana, United States

Site Status

Integrated Clinical Trial Services, Inc.

West Des Moines, Iowa, United States

Site Status

West Glen GI

Shawnee Mission, Kansas, United States

Site Status

Kansas Medical Clinic

Topeka, Kansas, United States

Site Status

University of Louisville

Louisville, Kentucky, United States

Site Status

Tandem Clinical Research GI, LLC

Marrero, Louisiana, United States

Site Status

Clinical Trials of America

West Monroe, Louisiana, United States

Site Status

Johns Hopkins Bayview Medical Center

Baltimore, Maryland, United States

Site Status

Beth Israel Deaconess Medical Center

Boston, Massachusetts, United States

Site Status

Henry Ford Health System

Detroit, Michigan, United States

Site Status

Aa Mrc Llc

Flint, Michigan, United States

Site Status

West Michigan Clinical Research Center

Wyoming, Michigan, United States

Site Status

KLEO Health & Research

Missoula, Montana, United States

Site Status

Clinical Research of South Nevada

Las Vegas, Nevada, United States

Site Status

Advanced Biomedical Research of America

Las Vegas, Nevada, United States

Site Status

Digestive Disease Specialists

Las Vegas, Nevada, United States

Site Status

Lovelace Respiratory Rsearch Institute

Albuquerque, New Mexico, United States

Site Status

Synexus Clinical Research

New York, New York, United States

Site Status

Tandem Clinical Research GI, LLC

New York, New York, United States

Site Status

Javara Research

Charlotte, North Carolina, United States

Site Status

Cumberland Research Associates

Fayetteville, North Carolina, United States

Site Status

Triad Clinical Trials

Greensboro, North Carolina, United States

Site Status

Carolina Digestive Diseases

Greenville, North Carolina, United States

Site Status

Dayton Gastroenterology Inc.

Beavercreek, Ohio, United States

Site Status

Hometown Urgent Care and Research

Cincinnati, Ohio, United States

Site Status

Hometown Urgent Care and Research

Columbus, Ohio, United States

Site Status

Hometown Urgent Care and Research

Dayton, Ohio, United States

Site Status

Draelos Metabolic Center

Edmond, Oklahoma, United States

Site Status

Options Health Research

Tulsa, Oklahoma, United States

Site Status

Transsouth Healthcare PC

Jackson, Tennessee, United States

Site Status

Quality Medical Research

Nashville, Tennessee, United States

Site Status

Avant Research Associates

Austin, Texas, United States

Site Status

Texas Tech University Health Sciences Center

El Paso, Texas, United States

Site Status

Biopharma Informatic, LLC

Houston, Texas, United States

Site Status

Biopharma Informatic, LLC

Houston, Texas, United States

Site Status

Sante Clinical Research

Kerville, Texas, United States

Site Status

Rio Grande Gastroenterology

McAllen, Texas, United States

Site Status

DM Clinical Research Solutions PC

Pearland, Texas, United States

Site Status

AES - DRS - Synexus Clinical Research US, Inc. - Plano

Plano, Texas, United States

Site Status

Sun Research

San Antonio, Texas, United States

Site Status

Southern Star Research Institute

San Antonio, Texas, United States

Site Status

Synexus Clinical Research

San Antonio, Texas, United States

Site Status

Horizon Clinical Research- Tomball

Tomball, Texas, United States

Site Status

Manassas Clinical Research Center

Manassas, Virginia, United States

Site Status

Digestive and Liver Disease Specialists

Norfolk, Virginia, United States

Site Status

Velocity Clinical Research Spokane

Spokane, Washington, United States

Site Status

Countries

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United States

References

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Loesch J, Hamza E, Pasricha PJ, Nee J, Cline M, MacDougall J, Simons M, Brown JT, Garg S, Hoscheit M, Gabbard S, De Colle C, Lembo A. A Phase 2 Randomized, Double-Blind, Placebo-Controlled Study of the Safety and Efficacy of Metopimazine Mesylate (NG101) in Participants With Gastroparesis. Am J Gastroenterol. 2025 May 14. doi: 10.14309/ajg.0000000000003534. Online ahead of print.

Reference Type DERIVED
PMID: 40367443 (View on PubMed)

Provided Documents

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Document Type: Study Protocol and Statistical Analysis Plan

View Document

Other Identifiers

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NG101-201

Identifier Type: -

Identifier Source: org_study_id

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