Clinical Trial of YH25448(Lazertinib) as the First-line Treatment in Patients With EGFR Mutation Positive Locally Advanced or Metastatic NSCLC (LASER301)

NCT ID: NCT04248829

Last Updated: 2024-12-03

Study Results

Results available

Outcome measurements, participant flow, baseline characteristics, and adverse events have been published for this study.

View full results

Basic Information

Get a concise snapshot of the trial, including recruitment status, study phase, enrollment targets, and key timeline milestones.

Recruitment Status

ACTIVE_NOT_RECRUITING

Clinical Phase

PHASE3

Total Enrollment

393 participants

Study Classification

INTERVENTIONAL

Study Start Date

2020-02-13

Study Completion Date

2026-06-30

Brief Summary

Review the sponsor-provided synopsis that highlights what the study is about and why it is being conducted.

This Phase III study will be conducted to evaluate the efficacy and safety of YH25448 as first-line treatment in locally advanced or metastatic Non-small Cell Lung Cancer (NSCLC) patients with EGFR mutations

Detailed Description

Dive into the extended narrative that explains the scientific background, objectives, and procedures in greater depth.

YH25448 is an oral, highly potent, mutant-selective and irreversible EGFR Tyrosine-kinase inhibitors (TKIs) that targets both the T790M mutation and activating EGFR mutations while sparing wild type EGFR.

This is a Phase III, Randomized, Double-blind study evaluating the efficacy and safety of YH25448 (240 mg orally, once daily) versus Gefitinib (250 mg orally, once daily) in patients with locally advanced or metastatic NSCLC that is known to be EGFR sensitizing mutation (EGFRm) positive, treatment-naïve and eligible for first-line treatment with an EGFR-TKI.

Conditions

See the medical conditions and disease areas that this research is targeting or investigating.

Non-Small Cell Lung Cancer

Study Design

Understand how the trial is structured, including allocation methods, masking strategies, primary purpose, and other design elements.

Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Approximately 380 patients will be randomized in a 1:1 ratio to either lazertinib (n=190) or gefitinib (n= 190).

Following objective disease progression according to RECIST v1.1, as per investigator assessment, patients who were randomized to gefitinib arm may have the option to receive open-label lazertinib
Primary Study Purpose

TREATMENT

Blinding Strategy

QUADRUPLE

Participants Caregivers Investigators Outcome Assessors

Study Groups

Review each arm or cohort in the study, along with the interventions and objectives associated with them.

Lazertinib + Gefitinib-matching placebo

Lazertinib (240 mg or 160 mg orally, once daily) plus Gefitinib-matching placebo (250 mg orally, once daily) in accordance with the randomization schedule

Group Type EXPERIMENTAL

Lazertinib 240 mg/160 mg

Intervention Type DRUG

The initial dose of lazertinib 240 mg (3 tablets of 80 mg lazertinib) once daily can be reduced to 160 mg once daily (2 tablets of 80 mg lazertinib) under specific circumstances

Gefitinib-matching placebo 250 mg

Intervention Type DRUG

The initial dose for Gefitinib-matching placebo (250 mg once daily) cannot be reduced to a lower dose

Gefitinib + Lazertinib-matching placebo

Gefitinib (250 mg orally, once daily) plus Lazertinib-matching placebo (240 mg or 160 mg orally, once daily) in accordance with the randomization schedule

Group Type ACTIVE_COMPARATOR

Gefitinib 250 mg

Intervention Type DRUG

The initial dose for Gefitinib (250 mg once daily) cannot be reduced to a lower dose

Lazertinib-matching placebo 240 mg/160 mg

Intervention Type DRUG

The initial dose of lazertinib-matching placebo 240 mg (3 tablets of 80 mg lazertinib-matching placebo) once daily can be reduced to 160 mg once daily (2 tablets of 80 mg lazertinib-matching placebo) under specific circumstances

Interventions

Learn about the drugs, procedures, or behavioral strategies being tested and how they are applied within this trial.

Lazertinib 240 mg/160 mg

The initial dose of lazertinib 240 mg (3 tablets of 80 mg lazertinib) once daily can be reduced to 160 mg once daily (2 tablets of 80 mg lazertinib) under specific circumstances

Intervention Type DRUG

Gefitinib 250 mg

The initial dose for Gefitinib (250 mg once daily) cannot be reduced to a lower dose

Intervention Type DRUG

Lazertinib-matching placebo 240 mg/160 mg

The initial dose of lazertinib-matching placebo 240 mg (3 tablets of 80 mg lazertinib-matching placebo) once daily can be reduced to 160 mg once daily (2 tablets of 80 mg lazertinib-matching placebo) under specific circumstances

Intervention Type DRUG

Gefitinib-matching placebo 250 mg

The initial dose for Gefitinib-matching placebo (250 mg once daily) cannot be reduced to a lower dose

Intervention Type DRUG

Other Intervention Names

Discover alternative or legacy names that may be used to describe the listed interventions across different sources.

YH25448 240 mg/160 mg Iressa 250 mg YH25448-matching placebo 240 mg/160 mg Iressa-matching placebo 250 mg

Eligibility Criteria

Check the participation requirements, including inclusion and exclusion rules, age limits, and whether healthy volunteers are accepted.

Inclusion Criteria

* Pathologically confirmed adenocarcinoma of the lung
* Locally advanced or metastatic NSCLC, not amenable to curative surgery or radiotherapy
* At least 1 of the 2 common EGFR mutations known to be associated with EGFR TKI sensitivity (Ex19del or L858R), either alone or in combination with other EGFR mutations
* Treatment-naïve for locally advanced or metastatic NSCLC
* WHO performance status score of 0 to 1 with no clinically significant deterioration over the previous 2 weeks before randomization
* At least 1 measurable lesion, not previously irradiated and not chosen for biopsy during the study Screening period

Exclusion Criteria

* Symptomatic and unstable brain metastases
* Leptomeningeal metastases
* Symptomatic spinal cord compression
* History of interstitial lung disease (ILD), drug-induced ILD, radiation pneumonitis which required steroid treatment, or any evidence of clinically active ILD
* Any medical conditions requiring chronic continuous oxygen therapy
* History of any malignancy other than the disease under study within 3 years before randomization
* Any cardiovascular disease as follows:

* History of symptomatic chronic heart failure or serious cardiac arrhythmia requiring active treatment
* History of myocardial infarction or unstable angina within 24 weeks of randomization
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

Meet the organizations funding or collaborating on the study and learn about their roles.

Yuhan Corporation

INDUSTRY

Sponsor Role lead

Responsible Party

Identify the individual or organization who holds primary responsibility for the study information submitted to regulators.

Responsibility Role SPONSOR

Locations

Explore where the study is taking place and check the recruitment status at each participating site.

Princess Alexandra Hospital

Woolloongabba, Queensland, Australia

Site Status

Eugenideio Therapeutirio - Ongcology Department

Athens, , Greece

Site Status

Attikon Hospital

Athens, , Greece

Site Status

Theageneio Anticancer Hospital of Thessaloniki

Thessaloniki, , Greece

Site Status

Debreceni Egyetem

Debrecen, , Hungary

Site Status

Törökbálinti Tüdőgyógyintézet

Törökbálint, , Hungary

Site Status

Hospital Sultan Ismail

Johor Bahru, Johor, Malaysia

Site Status

Hospital Raja Perempuan Zainab Ii

Kota Bharu, Kelantan, Malaysia

Site Status

Hospital Tengku Ampuan Afzan

Kuantan, Pahang, Malaysia

Site Status

Hospital Pulau Pinang

George Town, Pulau Pinang, Malaysia

Site Status

Hospital Umum Sarawak

Kuching, Sarawak, Malaysia

Site Status

University Malaya Medical Centre

Kuala Lumpur, Selangor, Malaysia

Site Status

Manila Doctors Hospital - Clinical Trial Office

Manila, Quezon, Philippines

Site Status

Perpetual Succour Hospital

Cebu, , Philippines

Site Status

Philippine General Hospital

Manila, , Philippines

Site Status

Arkhangelsk Regional Clinical Oncological Dispensary

Arkhangelsk, Arkhangelskaya oblast, Russia

Site Status

GBUZ of Nizhny Novgorod region Clinical diagnostic center

Nizhny Novgorod, Nizhny Novgorod Oblast, Russia

Site Status

GAUZ Republican clinical oncology dispensary of the Ministry

Kazan', , Russia

Site Status

Republic Clinical Oncology Despensary

Kazan', , Russia

Site Status

Medincentre (GLAVUPDK)

Moscow, , Russia

Site Status

VitaMed LLC

Moscow, , Russia

Site Status

MBUZ City Clinical Hospital #1

Novosibirsk, , Russia

Site Status

Budgetary Healthcare Institution of Omsk Region "Clinical Oncology Dispensary"

Omsk, , Russia

Site Status

Private medical institution "Euromedservice"

Pushkin, , Russia

Site Status

First St. Petersburg State Medical University n. a. Pavlov

Saint Petersburg, , Russia

Site Status

LLC "Eurocityclinic"

Saint Petersburg, , Russia

Site Status

Limited Liability Company "AV Medical Group" - Oncology

Saint Petersburg, , Russia

Site Status

Saint-Petersburg City Clinical Oncology Dispensary

Saint Petersburg, , Russia

Site Status

GBUZ "Regional clinical oncologic dispensary of Volgograd"

Volgograd, , Russia

Site Status

Yaroslavl regional oncology hospital

Yaroslavl, , Russia

Site Status

Institute for Pulmonary Diseases of Vojvodina

Kamenitz, Vojvodina, Serbia

Site Status

Clinical Hospital Center "Bezanijska Kosa"

Belgrade, , Serbia

Site Status

Clinical Center Kragujevac

Kragujevac, , Serbia

Site Status

National University Hospital

Singapore, , Singapore

Site Status

The Catholic University of Korea, Bucheon St. Mary's Hospital

Bucheon-si, Gyeonggi-do, South Korea

Site Status

National Cancer Center

Goyang-si, Gyeonggi-do, South Korea

Site Status

CHA Bundang Medical Center, CHA University

Seongnam-si, Gyeonggi-do, South Korea

Site Status

Seoul National University Bundang Hospital

Seongnam-si, Gyeonggi-do, South Korea

Site Status

The Catholic University of Korea, St. Vincent's Hospital

Suwon, Gyeonggi-do, South Korea

Site Status

Ajou University Hospital

Suwon, Gyeonggi-do, South Korea

Site Status

Gyeongsang National University Hospital

Jinju, Gyeongsangnam-do, South Korea

Site Status

Chungbuk National University Hospital

Cheongju-si, North Chungcheong, South Korea

Site Status

Inje University Haeundae Paik Hospital

Busan, , South Korea

Site Status

Yeungnam University Medical Center

Daegu, , South Korea

Site Status

Keimyung University Dongsan Medical Center

Daegu, , South Korea

Site Status

Gachon University Gil Medical Center

Incheon, , South Korea

Site Status

Korea University Anam Hospital

Seoul, , South Korea

Site Status

Seoul National University Hospital

Seoul, , South Korea

Site Status

Kangbuk Samsung Hospital

Seoul, , South Korea

Site Status

The Catholic University of Korea, Eunpyeong St.Mary's Hospital

Seoul, , South Korea

Site Status

Severance Hospital

Seoul, , South Korea

Site Status

Asan Medical Center

Seoul, , South Korea

Site Status

Samsung Medical Center

Seoul, , South Korea

Site Status

The Catholic University of Korea, Seoul St. Mary's Hospital

Seoul, , South Korea

Site Status

SMG-SNU Boramae Medical Center

Seoul, , South Korea

Site Status

Ulsan University Hospital

Ulsan, , South Korea

Site Status

National Taiwan University Hospital

Taipei, , Taiwan

Site Status

Taipei Veterans General Hospital

Taipei, , Taiwan

Site Status

Ramathibodi Hospital, Mahidol University

Bangkok, , Thailand

Site Status

Siriraj Hospital

Bangkok, , Thailand

Site Status

Chiang Mai University - Faculty of Medicine

Chiang Mai, , Thailand

Site Status

Prince of Songkla University

Hat Yai, , Thailand

Site Status

Srinagarind Hospital, Khon Kaen University

Khon Kaen, , Thailand

Site Status

Adana Baskent Practice and Research Hospital

Adana, , Turkey (Türkiye)

Site Status

Cukurova University Medical Faculty

Adana, , Turkey (Türkiye)

Site Status

Ankara Liv Hospital

Ankara, , Turkey (Türkiye)

Site Status

Hacettepe University Medical Faculty - Medical Oncology

Ankara, , Turkey (Türkiye)

Site Status

Trakya University Medical Faculty

Edirne, , Turkey (Türkiye)

Site Status

Istanbul Medeniyet University Goztepe Training and Research Hospital - Medical Oncology

Istanbul, , Turkey (Türkiye)

Site Status

Medical Point İzmir Hospital

Izmir, , Turkey (Türkiye)

Site Status

Kocaeli University Medical Faculty

Kocaeli, , Turkey (Türkiye)

Site Status

Inonu University Turgut Ozal Medical Center

Malatya, , Turkey (Türkiye)

Site Status

Komunalne nekomertsiine pidpryiemstvo Kharkivskoi oblasnoi rady "Oblasnyi klinichnyi spetsializovanyi dyspanser radiatsiinoho zakhystu naselennia" - khirurhichne viddilennia

Kharkiv, Kharkivs’ka Oblast’, Ukraine

Site Status

Tsentralna miska klinichna likarnia

Uzhhorod, Zakarpattia Oblast, Ukraine

Site Status

Oblasne komunalne nekomertsiine pidpryiemstvo "Bukovynskyi klinichnyi onkolohichnyi tsentr", strukturnyi pidrozdil klinichnoi onkolohii, m.Chernivtsi

Chernivtsi, , Ukraine

Site Status

Komunalne nekomertsiine pidpryiemstvo "Miska klinichna likarnia №4" Dniprovskoi miskoi rady", khimioterapevtychne viddilennia z dennym statsionarom, Derzhavnyi zaklad "Dnipropetrovskyi derzhavnyi medychnyi universitet", kafedra onkolohii i medychnoi radio

Dnipro, , Ukraine

Site Status

Kyiv City Clinical Oncology Center - Department of Chemotherapy

Kyiv, , Ukraine

Site Status

Komunalne nekomertsiine pidpryiemstvo Sumskoi oblasnoi rady "Sumskyi klinichnyi onkolohichnyi tsentr", onkotorakalne viddilennia, Sumskyi derzhavnyi universytet, kafedra onkolohii ta radiolohii, m. Sumy

Sumy, , Ukraine

Site Status

Podilskyi rehionalnyi tsentr onkolohii, viddilennia khimioterapii

Vinnytsia, , Ukraine

Site Status

Medychnyi tsentr Tovarystva z obmezhenoiu vidpovidalnistiu "Onkolaif"

Zaporizhzhia, , Ukraine

Site Status

Countries

Review the countries where the study has at least one active or historical site.

Australia Greece Hungary Malaysia Philippines Russia Serbia Singapore South Korea Taiwan Thailand Turkey (Türkiye) Ukraine

References

Explore related publications, articles, or registry entries linked to this study.

Soo RA, Cho BC, Kim JH, Ahn MJ, Lee KH, Zimina A, Orlov S, Bondarenko I, Lee YG, Lim YN, Lee SS, Lee KH, Pang YK, Fong CH, Kang JH, Lim CS, Danchaivijitr P, Kilickap S, Yang JC, Arslan C, Lee H, Park SN, Cicin I. Central Nervous System Outcomes of Lazertinib Versus Gefitinib in EGFR-Mutated Advanced NSCLC: A LASER301 Subset Analysis. J Thorac Oncol. 2023 Dec;18(12):1756-1766. doi: 10.1016/j.jtho.2023.08.017. Epub 2023 Oct 22.

Reference Type DERIVED
PMID: 37865896 (View on PubMed)

Cho BC, Ahn MJ, Kang JH, Soo RA, Reungwetwattana T, Yang JC, Cicin I, Kim DW, Wu YL, Lu S, Lee KH, Pang YK, Zimina A, Fong CH, Poddubskaya E, Sezer A, How SH, Danchaivijitr P, Kim Y, Lim Y, An T, Lee H, Byun HM, Zaric B. Lazertinib Versus Gefitinib as First-Line Treatment in Patients With EGFR-Mutated Advanced Non-Small-Cell Lung Cancer: Results From LASER301. J Clin Oncol. 2023 Sep 10;41(26):4208-4217. doi: 10.1200/JCO.23.00515. Epub 2023 Jun 28.

Reference Type DERIVED
PMID: 37379502 (View on PubMed)

Provided Documents

Download supplemental materials such as informed consent forms, study protocols, or participant manuals.

Document Type: Study Protocol

View Document

Document Type: Statistical Analysis Plan

View Document

Other Identifiers

Review additional registry numbers or institutional identifiers associated with this trial.

YH25448-301

Identifier Type: -

Identifier Source: org_study_id