Study to Evaluate the Pharmacodynamics After Single Oral Dosing of Tegoprazan, EAPA115 and RAPA115 in Healthy Volunteers

NCT ID: NCT04231136

Last Updated: 2020-12-01

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

19 participants

Study Classification

INTERVENTIONAL

Study Start Date

2020-01-14

Study Completion Date

2020-08-03

Brief Summary

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This study aims to evaluate the pharmacodynamics after single oral dosing of tegoprazan, EAPA115 and RAPA115 in healthy volunteers.

Detailed Description

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Evaluation Criteria

* Pharmacodynamic assessments with intragastric pH
* Safety assessments with adverse event monitoring including subjective/objective symptoms, physical examination, vital signs, electrocardiogram, and laboratory test

Conditions

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Healthy

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

CROSSOVER

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Tegoprazan 50 mg

Oral administration of Tegoprazan 50 mg tablet once a day

Group Type EXPERIMENTAL

Tegoprazan 50 mg

Intervention Type DRUG

Tegoprazan 50 mg tablet

EAPA115

Oral administration of EAPA115 once a day

Group Type ACTIVE_COMPARATOR

EAPA115

Intervention Type DRUG

EAPA115

RAPA115

Oral administration of RAPA115 once a day

Group Type ACTIVE_COMPARATOR

RAPA115

Intervention Type DRUG

RAPA115

Interventions

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Tegoprazan 50 mg

Tegoprazan 50 mg tablet

Intervention Type DRUG

EAPA115

EAPA115

Intervention Type DRUG

RAPA115

RAPA115

Intervention Type DRUG

Other Intervention Names

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K-CAB

Eligibility Criteria

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Inclusion Criteria

* Healthy adults aged 19 to 65 years (not inclusive) at the time of signing the informed consent form (ICF).
* Body mass index (BMI) ≥ 17.5 and \< 30.5 kg/m\^2 with a body weight ≥ 45 kg at screening. Body mass index (kg/m\^2) = weight (kg)/height (m)\^2
* Confirmed as H. pylori negative
* A subject without any congenital or chronic disease within 3 years, and has no medical examination result as pathological symptoms or signs.
* A subject determined eligible for this study based on the screening test such as clinical laboratory tests (hematology test, chemistry test, urine test, virus/bacteria test, etc.), vital signs, and electrocardiogram.
* A subject who is fully informed of the purpose and content of the study and agrees to participate in the study on its own will and signs the consent form approved by the Institutional Review Board (IRB) of the Seoul National University Hospital, prior to participate in the study.
* A subject who has the ability and willingness to participate throughout the whole study period.

Exclusion Criteria

* A subject with clinically significant blood, renal, endocrine, respiratory, gastrointestinal, urinary, cardiovascular, hepatic, psychical, neurologic, or immunologic diseases (except for simple dental past history such as tartar, impacted tooth, or wisdom tooth) or evidence.
* A subject with a history of gastrointestinal disorders (esophageal diseases such as esophageal achalasia or esophageal stricture, Crohn's disease) or surgery (except for simple appendectomy, herniotomy, and tooth extraction surgery) that may affect the absorption of drugs.
* A subject with the \*17 allele of CYP2C19 (Ultrarapid metabolizer).
* A subject with AST and ALT levels exceeding 3 times of the upper limit of the reference range in the screening test.
* A subject with a history of excessive caffeine (\> 5 units/day) or regular alcohol consumption exceeding 210 g/week within 6 months of screening test. (1 glass of beer (5%) (250 mL) = 10 g, 1 shot of soju (20%) (50 mL) = 8 g, 1 glass of wine (12%) (125 mL) = 12 g)
* A subject who participated in other clinical trial or bioequivalence study and administered the study medication within 6 months prior to the first administration of the investigational product of this study.
* A subject with significant alcohol or drug abuse within a year of screening test.
* A subject who administered drugs that significantly induce or inhibit drug metabolizing enzymes within 30 days prior to the first administration of the investigational product of this study.
* A subject who smoked cigarettes more than 20 per day within 6 months of screening test.
* A subject who administered prescribed drug or over-the-counter drug within 10 days prior to the first administration of the investigational product of this study.
* A subject who has donated whole blood within 2 months or those who donated the component blood within 1 month prior to the first administration of the investigational product of this study.
* A subject who has hypersensitivity to the investigational product of this study, benzimidazoles, penicillin and macrolide and its related medical history.
* A subject with rare genetic problems such as fructose intolerance, glucose-galactose malabsorption, or sucrase-isomaltase deficiency.
* Pregnant or nursing women
* A subject who cannot use reliable contraception during the entire period of the clinical trial (e.g, condom use, intrauterine device, tubal ligation, cervical cap, contraceptive diaphragm, etc.).
* A subject who is judged by the investigator to be ineligible to participate in the test.
Minimum Eligible Age

19 Years

Maximum Eligible Age

64 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

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HK inno.N Corporation

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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In-Jin Jang, MD, PhD

Role: PRINCIPAL_INVESTIGATOR

Seoul National University Hospital, Dept. of Clinical Pharmacology

Locations

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Seoul National University Hospital, Clinical Trial Center

Seoul, , South Korea

Site Status

Countries

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South Korea

Other Identifiers

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CJ_APA_115

Identifier Type: -

Identifier Source: org_study_id