Effect of Tegoprazan or RAPA114 on Pharmacokinetic of Atorvastatin in Healthy Adult Volunteers

NCT ID: NCT04221321

Last Updated: 2020-12-01

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

Get a concise snapshot of the trial, including recruitment status, study phase, enrollment targets, and key timeline milestones.

Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

32 participants

Study Classification

INTERVENTIONAL

Study Start Date

2020-01-07

Study Completion Date

2020-04-20

Brief Summary

Review the sponsor-provided synopsis that highlights what the study is about and why it is being conducted.

This study aims to evaluate the influence of tegoprazan or RAPA114 on the Pharmacokinetic characteristics of atorvastatin following co-administration of tegoprazan or RAPA114 in healthy adult volunteers.

Detailed Description

Dive into the extended narrative that explains the scientific background, objectives, and procedures in greater depth.

\[Pharmacokinetic Assessments\] : Blood concentration of atorvastatin, 2-OH atorvastatin

* Primary outcome: AUCτ, Css,max of atorvastatin
* Secondary outcome: Tss,max of atorvastatin, AUCτ, Css,max of 2-OH atorvastatin, metabolic ratio

\[Sefety Assessments\]

: Safety assessments with adverse event monitoring including subjective/objective symptoms, physical examination, vital signs, electrocardiogram, and laboratory test

Conditions

See the medical conditions and disease areas that this research is targeting or investigating.

Healthy

Study Design

Understand how the trial is structured, including allocation methods, masking strategies, primary purpose, and other design elements.

Allocation Method

RANDOMIZED

Intervention Model

CROSSOVER

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

Review each arm or cohort in the study, along with the interventions and objectives associated with them.

Atorvastatin 40 mg

Oral administration of Atorvastatin 40 mg tablet once daily for 7 days

Group Type PLACEBO_COMPARATOR

Atorvastatin 40 mg

Intervention Type DRUG

Atorvastatin 40 mg

Atorvastatin 40 mg + Tegoprazan 50 mg

Oral administration of Atorvastatin 40 mg tablet and Tegoprazan 50 mg tablet once daily for 7 days

Group Type EXPERIMENTAL

Atorvastatin 40 mg

Intervention Type DRUG

Atorvastatin 40 mg

Tegoprazan 50 mg

Intervention Type DRUG

Tegoprazan 50 mg tablet

Atorvastatin 40 mg + RAPA114

Oral administration of Atorvastatin 40 mg tablet and RAPA114 tablet once daily for 7 days

Group Type ACTIVE_COMPARATOR

Atorvastatin 40 mg

Intervention Type DRUG

Atorvastatin 40 mg

RAPA114

Intervention Type DRUG

RAPA114 tablet

Interventions

Learn about the drugs, procedures, or behavioral strategies being tested and how they are applied within this trial.

Atorvastatin 40 mg

Atorvastatin 40 mg

Intervention Type DRUG

Tegoprazan 50 mg

Tegoprazan 50 mg tablet

Intervention Type DRUG

RAPA114

RAPA114 tablet

Intervention Type DRUG

Other Intervention Names

Discover alternative or legacy names that may be used to describe the listed interventions across different sources.

Lipitor K-CAB

Eligibility Criteria

Check the participation requirements, including inclusion and exclusion rules, age limits, and whether healthy volunteers are accepted.

Inclusion Criteria

* Healthy male adults aged 19 to 55 years (inclusive) at the time of his consent.
* Body mass index (BMI) ≥ 19.0 and ≤ 27.0 kg/m2 at screening.
* Decides to participate voluntarily in the trial after being fully informed of and understanding the study completely, and provides the written informed consent to participate in the trial and to comply with the trial-specific requirements.
* Has the ability and willingness to participate in the entire period of clinical trial.

Exclusion Criteria

* A subject with clinically significant disease or history of hepatobiliary, renal, gastrointestinal, cardiovascular, musculoskeletal, endocrine, respiratory, neuropsychiatry or hemato-oncologic system, etc.
* A subject with a history of hypersensitivity reactions to main constituents of or identical affiliation of the investigational products (ex, HMG-CoA reductase inhibitor, gastric acid suppressants), or have allergic diseases that require treatment.
* A subject with a history of genetic myopathy or family history.
* A subject who has participated in other clinical trials and received the investigational products within 180 days prior to the randomization.
* A subject who received any medications or foods that could significantly affect the absorption, distribution, metabolism, or excretion of an investigational product within 30 days prior to the randomization.
* A subject with history of whole blood donation within 60 days, or with blood components or received transfusion within 30 days prior to the randomization.
* A subject with continued consumption of alcohol more than 140 g per week.
* A subject with AST, ALT, or γ-GT levels exceeding 1.5 times of the upper limit of the reference range in the screening test.
* A subject with a calculated glomerular filtration rate of less than 60 mL / min / 1.73 m2 in the screening test.
* A subject with any positive result on serology tests for hepatitis B, hepatitis C, HIV or syphilis in the screening test.
* A subject with galactose intolerance, Lapp lactose dehydrogenase deficiency or glucose-galactose malabsorption, etc.
* Male subject who don't have willing to accept medically acceptable contraceptive methods during the course of clinical trial, or who plan to provide sperm.
* A subject who is determined to be ineligible to participate in the clinical trial by the investigator for other reasons.
Minimum Eligible Age

19 Years

Maximum Eligible Age

55 Years

Eligible Sex

MALE

Accepts Healthy Volunteers

Yes

Sponsors

Meet the organizations funding or collaborating on the study and learn about their roles.

HK inno.N Corporation

INDUSTRY

Sponsor Role lead

Responsible Party

Identify the individual or organization who holds primary responsibility for the study information submitted to regulators.

Responsibility Role SPONSOR

Principal Investigators

Learn about the lead researchers overseeing the trial and their institutional affiliations.

Jung-ryul Kim

Role: PRINCIPAL_INVESTIGATOR

Samsung Medical Center

Locations

Explore where the study is taking place and check the recruitment status at each participating site.

Samsung Medical Center

Seoul, , South Korea

Site Status

Countries

Review the countries where the study has at least one active or historical site.

South Korea

Other Identifiers

Review additional registry numbers or institutional identifiers associated with this trial.

IN_APA_114

Identifier Type: -

Identifier Source: org_study_id