Sotorasib Activity in Subjects With Advanced Solid Tumors With KRAS p.G12C Mutation (CodeBreak 101)

NCT ID: NCT04185883

Last Updated: 2025-10-22

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

ACTIVE_NOT_RECRUITING

Clinical Phase

PHASE1

Total Enrollment

610 participants

Study Classification

INTERVENTIONAL

Study Start Date

2019-12-17

Study Completion Date

2027-12-05

Brief Summary

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To evaluate the safety and tolerability of sotorasib administered in investigational regimens in adult participants with KRAS p.G12C mutant advanced solid tumors.

Detailed Description

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Conditions

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Advanced Solid Tumors Kirsten Rat Sarcoma (KRAS) pG12C Mutation

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

SEQUENTIAL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Sotorasib + palbociclib

Experimental: Sotorasib + palbociclib Dose Exploration and Dose Expansion

* Enrollment into the dose exploration cohort is for eligible participants with KRAS P.G12C advanced solid tumor.
* Upon completing the dose exploration part of the study, dose expansion may proceed consisting of participants with KRAS p.G12C mutant advanced solid tumor.

Group Type EXPERIMENTAL

Sotorasib

Intervention Type DRUG

Sotorasib administered orally as a tablet.

Palbociclib

Intervention Type DRUG

Palbociclib administered orally as a tablet.

Sotorasib + pembrolizumab

Experimental: Sotorasib + pembrolizumab Dose Exploration and Dose Expansion

* Enrollment into the dose exploration cohort is for eligible participants with KRAS P.G12C mutant non small cell lung cancer.
* Upon completing the dose exploration part of the study, dose expansion may proceed consisting of participants with KRAS P.G12C mutant non small cell lung cancer.

Group Type EXPERIMENTAL

Sotorasib

Intervention Type DRUG

Sotorasib administered orally as a tablet.

Pembrolizumab

Intervention Type DRUG

pembrolizumab administered as an intravenous (IV) infusion.

Sotorasib + trametinib + panitumumab

Experimental: Sotorasib + trametinib + panitumumab Dose Exploration and Dose Expansion

* Enrollment into the dose exploration cohort is for eligible participants with KRAS P.G12C mutant advanced solid tumors.
* Upon completing the dose exploration part of the study, dose expansion may proceed consisting of participants with KRAS p.G12C mutant advanced solid tumors.

Group Type EXPERIMENTAL

Sotorasib

Intervention Type DRUG

Sotorasib administered orally as a tablet.

Trametinib

Intervention Type DRUG

Trametinib administered orally as a tablet.

Panitumumab

Intervention Type DRUG

Panitumumab administered as an IV infusion.

Sotorasib + RMC-4630

Experimental: Sotorasib + RMC-4630 Dose Exploration and Dose Expansion

* Enrollment into the dose exploration cohort is for eligible participants with KRAS P.G12C mutant advanced solid tumors.
* Upon completing the dose exploration part of the study, dose expansion may proceed consisting of participants, with KRAS p.G12C mutant advanced solid tumors.

Group Type EXPERIMENTAL

Sotorasib

Intervention Type DRUG

Sotorasib administered orally as a tablet.

RMC-4630

Intervention Type DRUG

RMC-4630 administered orally as a capsule.

Sotorasib + afatinib

Experimental: Sotorasib + afatinib Dose Exploration and Dose Expansion

* Enrollment into the dose exploration cohort is for eligible participants with KRAS P.G12C advanced non-small cell lung cancer.
* Upon completing the dose exploration part of the study, dose expansion may proceed consisting of participants with KRAS p.G12C mutant advanced non-small cell lung cancer.

Group Type EXPERIMENTAL

Sotorasib

Intervention Type DRUG

Sotorasib administered orally as a tablet.

Afatinib

Intervention Type DRUG

afatinib administered orally as a tablet.

Sotorasib + panitumumab +/- chemotherapy

Experimental: Sotorasib + panitumumab +/- chemotherapy Dose Exploration and Dose Expansion

* Enrollment into the dose exploration cohort is for eligible participants with KRAS P.G12C mutant advanced colorectal cancer.
* Upon completing the dose exploration part of the study, dose expansion may proceed consisting of participants with KRAS p.G12C mutant advanced solid tumors.

Group Type EXPERIMENTAL

Sotorasib

Intervention Type DRUG

Sotorasib administered orally as a tablet.

Panitumumab

Intervention Type DRUG

Panitumumab administered as an IV infusion.

IV Chemotherapy (Regimen 1)

Intervention Type DRUG

Chemotherapy combination of leucovorin administered as an IV injection, 5-fluorouracil (5-FU) administered as IV bolus injection or IV continuous infusion (depending on dose), and irinotecan administered as IV injection.

Sotorasib + atezolizumab

Experimental: Sotorasib + atezolizumab Dose Exploration and Dose Expansion

* Enrollment into the dose exploration cohort is for eligible participants with KRAS P.G12C advanced non-small cell lung cancer.
* Upon completing the dose exploration part of the study, dose expansion may proceed consisting of participants with KRAS p.G12C mutant advanced non-small cell lung cancer.

Group Type EXPERIMENTAL

Sotorasib

Intervention Type DRUG

Sotorasib administered orally as a tablet.

Atezolizumab

Intervention Type DRUG

Atezolizumab administered as an IV injection.

Sotorasib + carboplatin, pemetrexed, docetaxel, paclitaxel, pembrolizumab

Experimental: Sotorasib + carboplatin, pemetrexed, docetaxel, paclitaxel, pembrolizumab Dose Exploration and Dose Expansion

* Enrollment into the dose exploration cohort is for eligible participants with KRAS P.G12C advanced non-small cell lung cancer.
* Upon completing the dose exploration part of the study, dose expansion may proceed consisting of participants with KRAS p.G12C mutant advanced non-small cell lung cancer.

Group Type EXPERIMENTAL

Sotorasib

Intervention Type DRUG

Sotorasib administered orally as a tablet.

Pembrolizumab

Intervention Type DRUG

pembrolizumab administered as an intravenous (IV) infusion.

Carboplatin, pemetrexed, docetaxel, paclitaxel

Intervention Type DRUG

Carboplatin, pemetrexed, docetaxel administered as an IV infusion.

Sotorasib Monotherapy

Experimental: Sotorasib only Dose Exploration and Dose Expansion

* Enrollment into the dose exploration cohort is for eligible participants with KRAS P.G12C advanced non-small cell lung cancer with brain metastases.
* Upon completing the dose exploration part of the study, dose expansion may proceed consisting of participants with KRAS p.G12C mutant advanced non-small cell lung cancer with brain metastases.

Group Type EXPERIMENTAL

Sotorasib

Intervention Type DRUG

Sotorasib administered orally as a tablet.

Sotorasib + MVASI® (bevacizumab-awwb)+ Chemotherapy

Experimental: Sotorasib + MVASI® (bevacizumab-awwb)+ chemotherapy Dose Exploration and Dose Expansion

* Enrollment into the dose exploration cohort is for eligible participants with KRAS P.G12C mutant advanced colorectal cancer.
* Upon completing the dose exploration part of the study, dose expansion may proceed consisting of participants with KRAS p.G12C mutant advanced colorectal cancer.

Group Type EXPERIMENTAL

Sotorasib

Intervention Type DRUG

Sotorasib administered orally as a tablet.

MVASI® (bevacizumab-awwb)

Intervention Type DRUG

MVASI® (bevacizumab-awwb) administered as an IV infusion.

IV Chemotherapy (Regimen 1)

Intervention Type DRUG

Chemotherapy combination of leucovorin administered as an IV injection, 5-fluorouracil (5-FU) administered as IV bolus injection or IV continuous infusion (depending on dose), and irinotecan administered as IV injection.

IV Chemotherapy (Regimen 2)

Intervention Type DRUG

IV chemotherapy combination of leucovorin administered as an IV injection, 5-FU administered as IV bolus injection or IV continuous infusion (depending on dose), and oxaliplatin administered as IV injection.

Sotorasib + TNO155

Experimental: Sotorasib + TNO155 Dose Exploration and Dose Expansion

* Enrollment into the dose exploration cohort is for eligible participants with KRAS P.G12C mutant advanced solid tumors.
* Upon completing the dose exploration part of the study, dose expansion may proceed consisting of participants with KRAS p.G12C mutant advanced solid tumors.

Group Type EXPERIMENTAL

Sotorasib

Intervention Type DRUG

Sotorasib administered orally as a tablet.

TNO155

Intervention Type DRUG

TNO155 administered orally as a capsule.

Sotorasib + BI 1701963

Experimental: Sotorasib + BI 1701963 Dose Exploration and Dose Expansion

* Enrollment into the dose exploration cohort is for eligible participants with KRAS P.G12C mutant advanced solid tumors.
* Upon completion of dose exploration part of the study the dose expansion cohort is for eligible participants with KRAS P.G12C mutant advanced non-small cell lung cancer and advanced colorectal cancer.

Group Type EXPERIMENTAL

Sotorasib

Intervention Type DRUG

Sotorasib administered orally as a tablet.

BI 1701963

Intervention Type DRUG

BI 1701963 administered orally

Sotorasib + AMG 404

Experimental: Sotorasib + AMG 404 Dose Exploration and Dose Expansion • Enrollment into the dose exploration cohort is for eligible participants with KRAS P.G12C mutant advanced solid tumors. • Upon completing the dose exploration part of the study, dose expansion may proceed consisting of participants with KRAS p.G12C mutant advanced solid tumors

Group Type EXPERIMENTAL

Sotorasib

Intervention Type DRUG

Sotorasib administered orally as a tablet.

AMG 404

Intervention Type DRUG

AMG 404 administered as an IV infusion.

Sotorasib + everolimus

Experimental: Sotorasib + everolimus Dose Exploration and Dose Expansion • Enrollment into the dose exploration cohort is for eligible participants with KRAS P.G12C advanced solid tumor. • Upon completing the dose exploration part of the study, dose expansion may proceed consisting of participants with KRAS p.G12C mutant advanced solid tumor.

Group Type EXPERIMENTAL

Sotorasib

Intervention Type DRUG

Sotorasib administered orally as a tablet.

Everolimus

Intervention Type DRUG

Everolimus administered orally.

Interventions

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Sotorasib

Sotorasib administered orally as a tablet.

Intervention Type DRUG

Trametinib

Trametinib administered orally as a tablet.

Intervention Type DRUG

RMC-4630

RMC-4630 administered orally as a capsule.

Intervention Type DRUG

Afatinib

afatinib administered orally as a tablet.

Intervention Type DRUG

Pembrolizumab

pembrolizumab administered as an intravenous (IV) infusion.

Intervention Type DRUG

Panitumumab

Panitumumab administered as an IV infusion.

Intervention Type DRUG

Carboplatin, pemetrexed, docetaxel, paclitaxel

Carboplatin, pemetrexed, docetaxel administered as an IV infusion.

Intervention Type DRUG

Atezolizumab

Atezolizumab administered as an IV injection.

Intervention Type DRUG

Palbociclib

Palbociclib administered orally as a tablet.

Intervention Type DRUG

MVASI® (bevacizumab-awwb)

MVASI® (bevacizumab-awwb) administered as an IV infusion.

Intervention Type DRUG

TNO155

TNO155 administered orally as a capsule.

Intervention Type DRUG

IV Chemotherapy (Regimen 1)

Chemotherapy combination of leucovorin administered as an IV injection, 5-fluorouracil (5-FU) administered as IV bolus injection or IV continuous infusion (depending on dose), and irinotecan administered as IV injection.

Intervention Type DRUG

IV Chemotherapy (Regimen 2)

IV chemotherapy combination of leucovorin administered as an IV injection, 5-FU administered as IV bolus injection or IV continuous infusion (depending on dose), and oxaliplatin administered as IV injection.

Intervention Type DRUG

BI 1701963

BI 1701963 administered orally

Intervention Type DRUG

AMG 404

AMG 404 administered as an IV infusion.

Intervention Type DRUG

Everolimus

Everolimus administered orally.

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Men or women greater than or equal to 18 years old.
* Pathologically documented, locally-advanced or metastatic malignancy with, KRAS p.G12C mutation identified through molecular testing performed according to in-country requirements. In the United States, this test must be performed in a Clinical Laboratory Improvement Amendments (CLIA)-certified laboratory.

Exclusion Criteria

* Primary brain tumor.
* Spinal cord compression, or untreated, or symptomatic, or active brain metastases, or leptomeningeal disease from non-brain tumors.
* Myocardial infarction within 6 months of study day 1.
* Gastrointestinal (GI) tract disease causing the inability to take oral medication.
Minimum Eligible Age

18 Years

Maximum Eligible Age

100 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Amgen

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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MD

Role: STUDY_DIRECTOR

Amgen

Locations

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Arizona Oncology Associates Professional Corporation

Tucson, Arizona, United States

Site Status

City of Hope National Medical Center

Duarte, California, United States

Site Status

University of California San Diego Moores Cancer Center

La Jolla, California, United States

Site Status

Loma Linda University Cancer Center

Loma Linda, California, United States

Site Status

University of Southern California, Norris Comprehensive Cancer Center

Los Angeles, California, United States

Site Status

University of California Davis Medical Center

Sacramento, California, United States

Site Status

University of California San Francisco Mission Bay Campus

San Francisco, California, United States

Site Status

University of California Los Angeles

Santa Monica, California, United States

Site Status

Rocky Mountain Cancer Centers Denver Midtown

Denver, Colorado, United States

Site Status

Sarah Cannon Research Institute

Denver, Colorado, United States

Site Status

Yale New Haven Hospital

New Haven, Connecticut, United States

Site Status

Norwalk Hospital

Norwalk, Connecticut, United States

Site Status

Memorial Cancer Institute

Pembroke Pines, Florida, United States

Site Status

Moffitt Cancer Center

Tampa, Florida, United States

Site Status

Emory University

Atlanta, Georgia, United States

Site Status

Northwestern University

Chicago, Illinois, United States

Site Status

University of Chicago

Chicago, Illinois, United States

Site Status

Indiana University

Indianapolis, Indiana, United States

Site Status

University of Iowa Hospitals and Clinics

Iowa City, Iowa, United States

Site Status

Johns Hopkins University

Baltimore, Maryland, United States

Site Status

University of Michigan

Ann Arbor, Michigan, United States

Site Status

Henry Ford Cancer Detroit (Brigitte Harris Cancer Pavilion)

Detroit, Michigan, United States

Site Status

Washington University

St Louis, Missouri, United States

Site Status

Roswell Park Cancer Institute

Buffalo, New York, United States

Site Status

Icahn School of Medicine at Mount Sinai

New York, New York, United States

Site Status

Columbia University Irving Medical Center

New York, New York, United States

Site Status

Memorial Sloan Kettering Cancer Center

New York, New York, United States

Site Status

Montefiore Medical Center

The Bronx, New York, United States

Site Status

Levine Cancer Institute

Charlotte, North Carolina, United States

Site Status

Duke University

Durham, North Carolina, United States

Site Status

University of Cincinnati Medical Center

Cincinnati, Ohio, United States

Site Status

Cleveland Clinic Foundation

Cleveland, Ohio, United States

Site Status

Providence Portland Medical Center

Portland, Oregon, United States

Site Status

Oregon Health and Science University

Portland, Oregon, United States

Site Status

Thomas Jefferson University

Philadelphia, Pennsylvania, United States

Site Status

Fox Chase Cancer Center

Philadelphia, Pennsylvania, United States

Site Status

University of Pennsylvania

Philadelphia, Pennsylvania, United States

Site Status

University of Pittsburgh Medical Center

Pittsburgh, Pennsylvania, United States

Site Status

Gibbs Cancer Center and Research Institute - Spartanburg

Spartanburg, South Carolina, United States

Site Status

Avera Cancer Institute

Sioux Falls, South Dakota, United States

Site Status

United States Oncology Regulatory Affairs Corporate Office

Nashville, Tennessee, United States

Site Status

Vanderbilt University Medical Center

Nashville, Tennessee, United States

Site Status

Texas Oncology Central-South

Austin, Texas, United States

Site Status

Mary Crowley Cancer Research

Dallas, Texas, United States

Site Status

University of Texas Southwestern Medical Center

Dallas, Texas, United States

Site Status

Oncology Consultants

Houston, Texas, United States

Site Status

University of Texas MD Anderson Cancer Center

Houston, Texas, United States

Site Status

US Oncology Research Investigational Products Center

The Woodlands, Texas, United States

Site Status

Texas Oncology Northeast Texas

Tyler, Texas, United States

Site Status

Huntsman Cancer Institute

Salt Lake City, Utah, United States

Site Status

University of Virginia Cancer Center

Charlottesville, Virginia, United States

Site Status

Virginia Cancer Specialists, PC

Fairfax, Virginia, United States

Site Status

Fred Hutchinson Cancer Center

Seattle, Washington, United States

Site Status

Northwest Medical Specialties, PLLC

Tacoma, Washington, United States

Site Status

Northwest Cancer Specialists - Vancouver

Vancouver, Washington, United States

Site Status

Nepean Cancer Centre

Kingswood, New South Wales, Australia

Site Status

GenesisCare -North Shore Oncology

St Leonards, New South Wales, Australia

Site Status

Icon Cancer Care South Brisbane

South Brisbane, Queensland, Australia

Site Status

The Queen Elizabeth Hospital

Woodville South, South Australia, Australia

Site Status

St John of God Healthcare

Subiaco, Western Australia, Australia

Site Status

Medizinische Universitaet Graz

Graz, , Austria

Site Status

Landeskrankenhaus Salzburg

Salzburg, , Austria

Site Status

Universite Catholique de Louvain Cliniques Universitaires Saint Luc

Brussels, , Belgium

Site Status

Universitair Ziekenhuis Antwerpen

Edegem, , Belgium

Site Status

CHU de Quebec Hopital de l Enfant Jesus

Québec, Quebec, Canada

Site Status

Charite Universitaetsmedizin Berlin, Campus Virchow

Berlin, , Germany

Site Status

Universitatsklinikum Koln

Cologne, , Germany

Site Status

Universitaetsklinikum Dresden

Dresden, , Germany

Site Status

Universitaetsklinikum Essen

Essen, , Germany

Site Status

Azienda Socio Sanitaria Territoriale Grande Ospedale Metropolitano Niguarda

Milan, , Italy

Site Status

Azienda Ospedaliero Universitaria Pisana

Pisa, , Italy

Site Status

Centro Ricerche Cliniche Di Verona Societa responsabilita limitata

Verona, , Italy

Site Status

Aichi Cancer Center

Nagoya, Aichi-ken, Japan

Site Status

National Cancer Center Hospital East

Kashiwa-shi, Chiba, Japan

Site Status

The Cancer Institute Hospital of Japanese Foundation for Cancer Research

Koto-ku, Tokyo, Japan

Site Status

Universitair Medisch Centrum Utrecht

Utrecht, , Netherlands

Site Status

Seoul National University Hospital

Seoul, , South Korea

Site Status

The Catholic University of Korea Seoul St Marys Hospital

Seoul, , South Korea

Site Status

Asan Medical Center

Seoul, , South Korea

Site Status

Hospital Universitari Vall d Hebron

Barcelona, Catalonia, Spain

Site Status

Hospital Clinic i Provincial de Barcelona

Barcelona, Catalonia, Spain

Site Status

Institut Catala d Oncologia Hospitalet Hospital Duran i Reynals

L'Hospitalet de Llobregat, Catalonia, Spain

Site Status

Hospital Universitario Puerta de Hierro Majadahonda

Majadahonda, Madrid, Spain

Site Status

Hospital Universitario Ramon y Cajal

Madrid, , Spain

Site Status

Hospital Universitario 12 de Octubre

Madrid, , Spain

Site Status

National Cheng Kung University Hospital

Tainan City, , Taiwan

Site Status

National Taiwan University Hospital

Taipei, , Taiwan

Site Status

Taipei Veterans General Hospital

Taipei, , Taiwan

Site Status

Linkou Chang Gung Memorial Hospital of Chang Gung Medical Foundation

Taoyuan District, , Taiwan

Site Status

Sarah Cannon Research Institute UK

London, , United Kingdom

Site Status

Countries

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United States Australia Austria Belgium Canada Germany Italy Japan Netherlands South Korea Spain Taiwan United Kingdom

References

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Kuboki Y, Fakih M, Strickler J, Yaeger R, Masuishi T, Kim EJ, Bestvina CM, Kopetz S, Falchook GS, Langer C, Krauss J, Puri S, Cardona P, Chan E, Varrieur T, Mukundan L, Anderson A, Tran Q, Hong DS. Sotorasib with panitumumab in chemotherapy-refractory KRASG12C-mutated colorectal cancer: a phase 1b trial. Nat Med. 2024 Jan;30(1):265-270. doi: 10.1038/s41591-023-02717-6. Epub 2024 Jan 4.

Reference Type BACKGROUND
PMID: 38177853 (View on PubMed)

Related Links

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http://www.amgentrials.com

AmgenTrials clinical trials website

Other Identifiers

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2023-506794-35

Identifier Type: OTHER

Identifier Source: secondary_id

20190135

Identifier Type: -

Identifier Source: org_study_id

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