A Study of LY3499446 in Participants With Advanced Solid Tumors With KRAS G12C Mutation

NCT ID: NCT04165031

Last Updated: 2021-11-24

Study Results

Results available

Outcome measurements, participant flow, baseline characteristics, and adverse events have been published for this study.

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Basic Information

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Recruitment Status

TERMINATED

Clinical Phase

PHASE1/PHASE2

Total Enrollment

5 participants

Study Classification

INTERVENTIONAL

Study Start Date

2019-11-28

Study Completion Date

2020-10-30

Brief Summary

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The reason for this study is to see if the study drug LY3499446 is safe and effective in participants with solid tumors with KRAS G12C mutation.

Detailed Description

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Conditions

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Advanced Solid Tumor Non-Small Cell Lung Cancer Colorectal Cancer

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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LY3499446 Phase 1 Cohort A1 High Dose

Participants received high dose LY3499446 as oral monotherapy twice daily (BID) in 21-day cycles.

Group Type EXPERIMENTAL

LY3499446

Intervention Type DRUG

Administered orally

LY3499446 Phase 1 Cohort AO Mid Dose

Participant received mid dose LY3499446 as oral monotherapy once every other day (QOD) in 21-day cycles.

Group Type EXPERIMENTAL

LY3499446

Intervention Type DRUG

Administered orally

LY3499446 Phase 1 Cohort A-2 Low Dose

Participants received low dose LY3499446 as oral monotherapy once daily (QD) in 21-Day cycles.

Group Type EXPERIMENTAL

LY3499446

Intervention Type DRUG

Administered orally

LY3499446 + Combination Drugs Phase 1

LY3499446 combined with either abemaciclib (orally), erlotinib (orally), or cetuximab (IV).

This trial was terminated prior to initiation of combination therapy cohorts.

Group Type EXPERIMENTAL

LY3499446

Intervention Type DRUG

Administered orally

Abemaciclib

Intervention Type DRUG

Administered orally

Cetuximab

Intervention Type DRUG

Administered IV

Erlotinib

Intervention Type DRUG

Administered orally

LY3499446 Monotherapy + Combination Drugs Phase 2

LY3499446 as oral monotherapy and LY3499446 combined with either abemaciclib (orally), erlotinib (orally), or cetuximab (IV).

The trial was terminated prior to initiation of Phase 2 of this study.

Group Type EXPERIMENTAL

LY3499446

Intervention Type DRUG

Administered orally

Abemaciclib

Intervention Type DRUG

Administered orally

Cetuximab

Intervention Type DRUG

Administered IV

Erlotinib

Intervention Type DRUG

Administered orally

Docetaxel Phase 2

Docetaxel IV infusion.

The trial was terminated prior to initiation of Phase 2 of this study.

Group Type ACTIVE_COMPARATOR

Docetaxel

Intervention Type DRUG

Administered IV

Interventions

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LY3499446

Administered orally

Intervention Type DRUG

Abemaciclib

Administered orally

Intervention Type DRUG

Cetuximab

Administered IV

Intervention Type DRUG

Erlotinib

Administered orally

Intervention Type DRUG

Docetaxel

Administered IV

Intervention Type DRUG

Other Intervention Names

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LY2835219

Eligibility Criteria

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Inclusion Criteria

* Participants must have diagnosis of a solid tumor with KRAS G12C mutation that did not respond to at least 1 line of standard therapy and has spread to other part(s) of the body
* For phase II, participants must be willing to have new tumor tissue biopsies (doctor removes a small amount of tissue) during the study if it does not cause undue risks to health
* Participants must be willing to use highly effective birth control
* Participants must have adequate organ function
* Participants must be able to swallow capsules

Exclusion Criteria

* Participants must not have certain infections such as hepatitis or tuberculosis or HIV that is not well controlled
* Participants must not have another serious medical condition including a serious heart condition, such as congestive heart failure, unstable angina pectoris, or heart attack within the last three months
* Participants must not have cancer of the central nervous system that is not stable
* Participants must not be pregnant or breastfeeding
* Participants must not use herbal supplements
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Eli Lilly and Company

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Call 1-877-CTLILLY (1-877-285-4559) or 1-317-615-4559 Mon - Fri 9 AM - 5 PM Eastern time (UTC/GMT - 5 hours, EST)

Role: STUDY_DIRECTOR

Eli Lilly and Company

Locations

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Indiana Univ Melvin & Bren Simon Cancer Center

Indianapolis, Indiana, United States

Site Status

Memorial Sloan Kettering Cancer Center

Middletown, New Jersey, United States

Site Status

Memorial Sloan Kettering Cancer Center

Harrison, New York, United States

Site Status

Memorial Sloan Kettering Cancer Center

New York, New York, United States

Site Status

St Vincent's Hospital

Darlinghurst, New South Wales, Australia

Site Status

Linear Clinical Research Ltd

Nedlands, Western Australia, Australia

Site Status

Countries

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Canada Italy Japan Spain United States Australia

Provided Documents

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Document Type: Study Protocol

View Document

Document Type: Statistical Analysis Plan

View Document

Related Links

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https://www.lillytrialguide.com/en-US/studies/solid-tumor/JZKA#?postal=

A Study of LY3499446 in Participants With Advanced Solid Tumors With KRAS G12C Mutation

Other Identifiers

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J2K-MC-JZKA

Identifier Type: OTHER

Identifier Source: secondary_id

2019-003070-53

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

17501

Identifier Type: -

Identifier Source: org_study_id