A Study of ZN-c3 in Participants With Solid Tumors

NCT ID: NCT04158336

Last Updated: 2023-02-01

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

UNKNOWN

Clinical Phase

PHASE1

Total Enrollment

146 participants

Study Classification

INTERVENTIONAL

Study Start Date

2019-11-01

Study Completion Date

2023-08-31

Brief Summary

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This is a Phase 1 open-label, multicenter study of ZN-c3 monotherapy which consists of Dose Escalation, a Food Effect Cohort, and Dose Expansion.

Detailed Description

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This study will evaluate the safety, tolerability, efficacy, pharmacokinetics (PK) and pharmacodynamics of ZN-c3.

In Dose Escalation, the study will identify the Maximum Tolerated Dose (MTD) of ZN-c3 monotherapy in solid tumors.

The Food Effect cohort sub-study will examine ZN-c3 PK after a single dose and determine the bioavailability of ZN-c3 under fed and fasted conditions.

In Dose Expansion, single agent ZN-c3 will be evaluated at the RP2D in subjects with recurrent or persistent uterine serous carcinoma (USC) or subjects with locally advanced or metastatic solid tumor malignancies harboring biomarkers related to deoxyribonucleic acid (DNA) damage pathways.

Conditions

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Solid Tumor

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

USC Cohort is Parallel Assignment and MOI Cohort is Single Group
Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Single Agent Dose Escalation

Subjects with solid tumors with advanced or metastatic disease who are refractory or ineligible to standard therapy(ies) or for whom no standard therapy is available.

Group Type EXPERIMENTAL

ZN-c3

Intervention Type DRUG

ZN-c3 is a study drug

Single Agent Food Effect Cohort

Subjects with solid tumors with advanced or metastatic disease who are refractory or ineligible to standard therapy(ies) or for whom no standard therapy is available. This cohort will give subjects the option to continue treatment after PK assessments are completed.

Group Type EXPERIMENTAL

ZN-c3

Intervention Type DRUG

ZN-c3 is a study drug

Single Agent Dose Expansion

Subjects with histologically confirmed recurrent or persistent USC who have had treatment with at least 1 prior platinum-based chemotherapy regimen for management of advanced or metastatic USC and subjects with locally advanced or metastatic malignancy with one or more relevant biomarkers related to DNA damage pathways.

Group Type EXPERIMENTAL

ZN-c3

Intervention Type DRUG

ZN-c3 is a study drug

Interventions

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ZN-c3

ZN-c3 is a study drug

Intervention Type DRUG

Other Intervention Names

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Study Drug

Eligibility Criteria

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Inclusion Criteria

1. Subjects must have a solid tumor with advanced or metastatic disease, refractory to standard therapy or for whom no standard therapy is available, or the subject is ineligible for standard therapy(ies).
2. Measurable or evaluable disease per RECIST version 1.1.


1. Subjects with solid tumors with advanced or metastatic disease who are refractory or ineligible to standard therapy(ies) or for whom no standard therapy is available.
2. Subjects must have no relevant dietary restrictions, and be willing to consume a high-calorie, high-fat breakfast and other standard meals provided during the study.


1. Measurable disease, defined as at least one lesion that can be accurately measured per RECIST version 1.1 criteria.
2. Recurrent or persistent USC or locally advanced or metastatic malignancy with one or more relevant biomarkers related to deoxyribonucleic acid (DNA) damage pathways.

Exclusion Criteria

1. Prior therapy with ZN-c3 or known hypersensitivity to any drugs similar to ZN-c3 in class or any inactive ingredients present in ZN-c3.
2. Prior therapy with a WEE1 inhibitor.
3. A serious illness or medical condition(s).
4. Unresolved toxicity of Grade \>1 attributed to any prior therapies (excluding Grade ≤2 neuropathy, alopecia or skin pigmentation).
5. Pregnant or lactating females (including the cessation of lactation) or females of childbearing potential who have a positive serum pregnancy test within 14 days prior to C1D1.
6. Subjects with active (uncontrolled, metastatic) second malignancies or requiring therapy.
7. 12-lead ECG demonstrating a corrected QT interval using Fridericia's formula (QTcF) of \>480 ms, except for subjects with atrioventricular pacemakers or other conditions (e.g., right bundle branch block) that render the QT measurement invalid.
8. History or current evidence of congenital or family history of long QT syndrome or Torsade de Pointes (TdP).
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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K-Group, Beta, Inc., a wholly owned subsidiary of Zentalis Pharmaceuticals, Inc

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Philippe Pultar, MD

Role: STUDY_DIRECTOR

K-Group Beta, a Zentalis Company

Locations

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Site 0102

Tucson, Arizona, United States

Site Status RECRUITING

Site 0167

Newport Beach, California, United States

Site Status RECRUITING

Site 0171

Chicago, Illinois, United States

Site Status RECRUITING

Site 0101

Detroit, Michigan, United States

Site Status RECRUITING

Site 0173

New York, New York, United States

Site Status RECRUITING

Site 0179

Pittsburgh, Pennsylvania, United States

Site Status RECRUITING

Site 0103

Houston, Texas, United States

Site Status RECRUITING

Site 0100

San Antonio, Texas, United States

Site Status RECRUITING

Countries

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United States

Central Contacts

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Project Director

Role: CONTACT

858-263-4333

Other Identifiers

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ZN-c3-001

Identifier Type: -

Identifier Source: org_study_id

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