Trial Outcomes & Findings for A Study to Compare ORMD-0801 Once Daily to ORMD-0801 Three Times Daily in Subjects With Type 1 Diabetes (NCT NCT04150107)

NCT ID: NCT04150107

Last Updated: 2022-06-02

Results Overview

The least squares means difference of basal exogenous insulin between treatment A and placebo and treatment B and placebo, utilized over the final ten (10) days of each treatment period

Recruitment status

COMPLETED

Study phase

PHASE2

Target enrollment

30 participants

Primary outcome timeframe

Combined Final ten days of each treatment period. Period1 (days -8 to 1)Period 2 (days 19 to 28) ,and Period 3 (days 47 to 56)

Results posted on

2022-06-02

Participant Flow

This is a crossover study with one crossover point. There are three periods in this study: Period 1: all patients consented receive placebo (run-in period). Period 2: all patients are randomized to receive either Treatment A or Treatment B. Period 3: Crossover point. Patients receiving Treatment A in period 2 now receive Treatment B in period 3, and patients receiving Treatment B in period 2 now receive Treatment A in period 3.

Participant milestones

Participant milestones
Measure
Placebo Followed by Treatment A Followed by Treatment B
Treatment administered in the following order: 1. Placebo Fish oil capsule 2. Treatment A is 24 mg (16 mg + 8 mg capsules) Once Daily (QD) at Bedtime of ORMD-0801 ORMD-0801: Oral Insulin Capsules 3. Treatment B is 8 mg (8 mg capsule) three times a day (TID) 45-90 minutes before meals ORMD-0801: Oral Insulin Capsules
Placebo Followed by Treatment B Followed by Treatment A
Treatment administered in the following order: 1. Placebo Fish oil capsule 2. Treatment B is 8 mg (8 mg capsule) three times a day (TID) 45-90 minutes before meals ORMD-0801: Oral Insulin Capsules 3. Treatment A is 24 mg (16 mg + 8 mg capsules) Once Daily (QD) at Bedtime of ORMD-0801 ORMD-0801: Oral Insulin Capsules
Period 1- Placebo run-in (All Patients)
STARTED
14
16
Period 1- Placebo run-in (All Patients)
COMPLETED
14
16
Period 1- Placebo run-in (All Patients)
NOT COMPLETED
0
0
Period 2- Either Treatment A or B
STARTED
14
16
Period 2- Either Treatment A or B
COMPLETED
14
16
Period 2- Either Treatment A or B
NOT COMPLETED
0
0
Period 3 Crossover-Treatment B or A
STARTED
14
16
Period 3 Crossover-Treatment B or A
COMPLETED
12
15
Period 3 Crossover-Treatment B or A
NOT COMPLETED
2
1

Reasons for withdrawal

Reasons for withdrawal
Measure
Placebo Followed by Treatment A Followed by Treatment B
Treatment administered in the following order: 1. Placebo Fish oil capsule 2. Treatment A is 24 mg (16 mg + 8 mg capsules) Once Daily (QD) at Bedtime of ORMD-0801 ORMD-0801: Oral Insulin Capsules 3. Treatment B is 8 mg (8 mg capsule) three times a day (TID) 45-90 minutes before meals ORMD-0801: Oral Insulin Capsules
Placebo Followed by Treatment B Followed by Treatment A
Treatment administered in the following order: 1. Placebo Fish oil capsule 2. Treatment B is 8 mg (8 mg capsule) three times a day (TID) 45-90 minutes before meals ORMD-0801: Oral Insulin Capsules 3. Treatment A is 24 mg (16 mg + 8 mg capsules) Once Daily (QD) at Bedtime of ORMD-0801 ORMD-0801: Oral Insulin Capsules
Period 3 Crossover-Treatment B or A
Adverse Event
2
0
Period 3 Crossover-Treatment B or A
Patient non-compliance
0
1

Baseline Characteristics

This is a crossover study. All patients were administered placebo at baseline.

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
Placebo Followed by Treatment A Followed by Treatment B
n=14 Participants
Treatment administerd in the following order: 1. Placebo, standard of care Fish oil capsules 2. Treatment A is 24 mg (16 mg + 8 mg capsules) Once Daily (QD) at Bedtime of ORMD-0801 ORMD-0801: Oral Insulin Capsules 3. Treatment B is 8 mg (8 mg capsule) three times a day (TID) 45-90 minutes before meals ORMD-0801: Oral Insulin Capsules
Placebo Followed by Treatment B Followed by Treatment A
n=16 Participants
Treatment administerd in the following order: 1. Placebo, standard of care Fish oil capsules 2. Treatment B is 8 mg (8 mg capsule) three times a day (TID) 45-90 minutes before meals ORMD-0801: Oral Insulin Capsules 3. Treatment A is 24 mg (16 mg + 8 mg capsules) Once Daily (QD) at Bedtime of ORMD-0801 ORMD-0801: Oral Insulin Capsules
Total
n=30 Participants
Total of all reporting groups
Age, Continuous
43.79285714 years
STANDARD_DEVIATION 12.67793142 • n=5 Participants • This is a crossover study. All patients were administered placebo at baseline.
42.88125 years
STANDARD_DEVIATION 16.04131614 • n=7 Participants • This is a crossover study. All patients were administered placebo at baseline.
43.30667 years
STANDARD_DEVIATION 12.22325 • n=5 Participants • This is a crossover study. All patients were administered placebo at baseline.
Sex: Female, Male
Female
7 Participants
n=5 Participants
8 Participants
n=7 Participants
15 Participants
n=5 Participants
Sex: Female, Male
Male
7 Participants
n=5 Participants
8 Participants
n=7 Participants
15 Participants
n=5 Participants
Ethnicity (NIH/OMB)
Hispanic or Latino
0 Participants
n=5 Participants
1 Participants
n=7 Participants
1 Participants
n=5 Participants
Ethnicity (NIH/OMB)
Not Hispanic or Latino
13 Participants
n=5 Participants
15 Participants
n=7 Participants
28 Participants
n=5 Participants
Ethnicity (NIH/OMB)
Unknown or Not Reported
1 Participants
n=5 Participants
0 Participants
n=7 Participants
1 Participants
n=5 Participants
Race (NIH/OMB)
American Indian or Alaska Native
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
Race (NIH/OMB)
Asian
0 Participants
n=5 Participants
2 Participants
n=7 Participants
2 Participants
n=5 Participants
Race (NIH/OMB)
Native Hawaiian or Other Pacific Islander
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
Race (NIH/OMB)
Black or African American
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
Race (NIH/OMB)
White
14 Participants
n=5 Participants
14 Participants
n=7 Participants
28 Participants
n=5 Participants
Race (NIH/OMB)
More than one race
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
Race (NIH/OMB)
Unknown or Not Reported
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
Pre-dose Hb1Ac(%)
7.735714286 percent
STANDARD_DEVIATION 0.734435569 • n=5 Participants
7.6125 percent
STANDARD_DEVIATION 0.848429922 • n=7 Participants
7.67 percent
STANDARD_DEVIATION 0.786 • n=5 Participants

PRIMARY outcome

Timeframe: Combined Final ten days of each treatment period. Period1 (days -8 to 1)Period 2 (days 19 to 28) ,and Period 3 (days 47 to 56)

Population: Information collected at the day 28 visits (Day 28 and Day 56) will be analyzed using an Analysis of Covariance model with subject as a random effect.

The least squares means difference of basal exogenous insulin between treatment A and placebo and treatment B and placebo, utilized over the final ten (10) days of each treatment period

Outcome measures

Outcome measures
Measure
Baseline
n=30 Participants
Placebo (Fish-Oil Capsule)
Treatment A
n=27 Participants
Treatment A is 24 mg (16 mg + 8 mg capsules) Once Daily (QD) at Bedtime of ORMD-0801 ORMD-0801: Oral Insulin Capsules
Treatment B
n=27 Participants
Treatment B is 8 mg (8 mg capsule) three times a day (TID) 45-90 minutes before meals ORMD-0801: Oral Insulin Capsules
Average Exogenous Basal Insulin Compared to Baseline (Placebo)
Least Squares Mean Baseline, Treatment A, Treatment B
27.28 mg/dL
Standard Error 2.489
25.84 mg/dL
Standard Error 2.486
27.32 mg/dL
Standard Error 2.492
Average Exogenous Basal Insulin Compared to Baseline (Placebo)
Least Squares Mean Difference Treatment A minus Baseline or Treatment B minus Baseline
NA mg/dL
Standard Error NA
Calculation not applicable to this Arm/Group
-1.43 mg/dL
Standard Error 0.381
0.04 mg/dL
Standard Error 0.421

PRIMARY outcome

Timeframe: Combined Final ten days of treatment per treatment period (Days -8 to 1, Days 19 to 28, and Days 47 to 56)

Population: Safety Population

The amount of exogenous bolus insulin utilized over the final ten (10) days of each treatment period measured in mg/dL

Outcome measures

Outcome measures
Measure
Baseline
n=30 Participants
Placebo (Fish-Oil Capsule)
Treatment A
n=27 Participants
Treatment A is 24 mg (16 mg + 8 mg capsules) Once Daily (QD) at Bedtime of ORMD-0801 ORMD-0801: Oral Insulin Capsules
Treatment B
n=27 Participants
Treatment B is 8 mg (8 mg capsule) three times a day (TID) 45-90 minutes before meals ORMD-0801: Oral Insulin Capsules
Average Exogenous Bolus Insulin Compared to Baseline (Placebo)
Least Squares Means Baseline, Treatment A, Treatment B
20.63 mg/dL
Standard Error 2.033
20.77 mg/dL
Standard Error 2.045
20.54 mg/dL
Standard Error 2.049
Average Exogenous Bolus Insulin Compared to Baseline (Placebo)
Least Squares Means Difference Treatment A minus Baseline, Treatmen B minus Baseline
NA mg/dL
Standard Error NA
Calculation not applicable to this Arm/Group.
0.14 mg/dL
Standard Error 0.634
-0.09 mg/dL
Standard Error 0.645

PRIMARY outcome

Timeframe: Combined Final ten days of treatment , day -8 to 1 (Period 1) Days 19 to 28 (Period 2), Days 47 to 56 (Period 3)

Population: Safety Population The number of participants anylized is based on the the number of participants that completed at least 80% of the Continuous Glucose Montioring measurements. Participants that did not meet this criterion are not inclued in this analysis.

The Least Squares Mean Difeerence ( (mg/dL) of total exogenous insulin (the sum of basal + bolus exogenous insulin) over the final ten (10) days of treatment.

Outcome measures

Outcome measures
Measure
Baseline
n=29 Participants
Placebo (Fish-Oil Capsule)
Treatment A
n=27 Participants
Treatment A is 24 mg (16 mg + 8 mg capsules) Once Daily (QD) at Bedtime of ORMD-0801 ORMD-0801: Oral Insulin Capsules
Treatment B
n=27 Participants
Treatment B is 8 mg (8 mg capsule) three times a day (TID) 45-90 minutes before meals ORMD-0801: Oral Insulin Capsules
Average Exogenous Total Insulin Compared to Baseline
Least Squares Mean Difference Treatment A minus Baseline and Treatment B minus Baseline
NA mg/dL
Standard Error NA
Calculation not applicable to this Arm/Group.
-0.127 mg/dL
Standard Error 0.758
-0.04 mg/dL
Standard Error 0.798
Average Exogenous Total Insulin Compared to Baseline
Least Squares Mean
47.92 mg/dL
Standard Error 3.395
46.64 mg/dL
Standard Error 3.397
47.88 mg/dL
Standard Error 3.406

SECONDARY outcome

Timeframe: Combined Study days -8 to 1 (Period 1) Days 19 to 28 (Period 2), and days 47 to 56 (Period 3)

Population: Safety Population. The number of participants anylized is based on the the number of participants that completed at least 80% of the Continuous Glucose Montioring measurements. Participants that did not meet this criterion are not inclued in this analysis.

Least Squares Mean Difference from Baseline of Daytime Average Mean Glucose over the final ten (10) days of each treatment and each treatment period as measured by CGM.

Outcome measures

Outcome measures
Measure
Baseline
n=30 Participants
Placebo (Fish-Oil Capsule)
Treatment A
n=26 Participants
Treatment A is 24 mg (16 mg + 8 mg capsules) Once Daily (QD) at Bedtime of ORMD-0801 ORMD-0801: Oral Insulin Capsules
Treatment B
n=26 Participants
Treatment B is 8 mg (8 mg capsule) three times a day (TID) 45-90 minutes before meals ORMD-0801: Oral Insulin Capsules
Daytime Average Mean Glucose Compared to Baseline
Least Sqaures Mean Baseline, Treatment A, Treatment B
168.72 mg/dL
Standard Error 5.825
174.84 mg/dL
Standard Error 5.957
169.75 mg/dL
Standard Error 5.930
Daytime Average Mean Glucose Compared to Baseline
Least Squares Mean Difference between each treatment and placebo
NA mg/dL
Standard Error NA
Calculation not applicable to this Arm/Group.
6.12 mg/dL
Standard Error 3.966
1.02 mg/dL
Standard Error 3.889

SECONDARY outcome

Timeframe: Study Days -8 to 1 (Period 1), Days 19-28 (Period 2), and Days 47-56 (Period 3)

Population: Safety Population. The number of participants anylized is based on the the number of participants that completed at least 80% of the Continuous Glucose Montioring measurements. Participants that did not meet this criterion are not inclued in this analysis.

Least Squares Mean Continuous Glucose Monitor (CGM) Glucose Coefficient of Variation measured over daytime hours, compared to Baseline

Outcome measures

Outcome measures
Measure
Baseline
n=30 Participants
Placebo (Fish-Oil Capsule)
Treatment A
n=26 Participants
Treatment A is 24 mg (16 mg + 8 mg capsules) Once Daily (QD) at Bedtime of ORMD-0801 ORMD-0801: Oral Insulin Capsules
Treatment B
n=26 Participants
Treatment B is 8 mg (8 mg capsule) three times a day (TID) 45-90 minutes before meals ORMD-0801: Oral Insulin Capsules
Daytime Glucose Coefficient of Variation Compared to Baseline
Least Squares Mean
45.287 percent (%)
Standard Error 2.3191
46.550 percent (%)
Standard Error 2.3073
44.996 percent (%)
Standard Error 2.2847
Daytime Glucose Coefficient of Variation Compared to Baseline
Least Squares Mean Differece between each treatment and placebo.
NA percent (%)
Standard Error NA
Calculation not applicable to this Arm/Group.
1.64 percent (%)
Standard Error 1.949
-0.291 percent (%)
Standard Error 1.9064

SECONDARY outcome

Timeframe: Combined Study Days -8 to 1 (Period 1), Days 19-28 (Period 2), and Days 47-56 (Period 3)

Population: Safety Population. The number of participants anylized is based on the the number of participants that completed at least 80% of the Continuous Glucose Montioring measurements. Participants that did not meet this criterion are not inclued in this analysis

Least Squares Mean Daytime Low Blood Glucose Index (LBGI) measured over the last ten (10) days of the treatment period, compared to Baseline LBGI is a clinical scale that indicates the probability for hypoglycemia. Blood Glucose Variability is an important measure because it provides additional clarification for HbA1c value. The risk of hypglycemic events and the LBGI scale is defined as follows: Minimal Risk ( LBGI \< 1.1) Low Risk ( 1.1 \< LBGI \< 2.5) Moderate Risk (2.5 \< LBGI \< 5), HIgh Risk ( LBGI \> 5)

Outcome measures

Outcome measures
Measure
Baseline
n=30 Participants
Placebo (Fish-Oil Capsule)
Treatment A
n=26 Participants
Treatment A is 24 mg (16 mg + 8 mg capsules) Once Daily (QD) at Bedtime of ORMD-0801 ORMD-0801: Oral Insulin Capsules
Treatment B
n=26 Participants
Treatment B is 8 mg (8 mg capsule) three times a day (TID) 45-90 minutes before meals ORMD-0801: Oral Insulin Capsules
Daytime Low Blood Glucose Index (LBGI) Compared to Baseline
Least Squares Mean Daytime Low Blood Glucose Index (LBGI) for Baseline,
1.65 units on a scale
Standard Error 0.284
1.53 units on a scale
Standard Error 0.282
1.65 units on a scale
Standard Error 0.288
Daytime Low Blood Glucose Index (LBGI) Compared to Baseline
Least Squares Mean Difference between Treatment A and Placebo, Treatment B and Placebo.
NA units on a scale
Standard Error NA
Calculation not applicable to this Arm/Group.
-0.12 units on a scale
Standard Error 0.294
0.00 units on a scale
Standard Error 0.297

Adverse Events

Placebo

Serious events: 0 serious events
Other events: 0 other events
Deaths: 0 deaths

Treatment A ORMD-0801

Serious events: 0 serious events
Other events: 9 other events
Deaths: 0 deaths

Treatment B ORMD-0801

Serious events: 0 serious events
Other events: 6 other events
Deaths: 0 deaths

Serious adverse events

Adverse event data not reported

Other adverse events

Other adverse events
Measure
Placebo
n=30 participants at risk
Placebo - Fish Oil
Treatment A ORMD-0801
n=30 participants at risk
Treatment A is 24 mg (16 mg + 8 mg capsules) Once Daily (QD) at Bedtime of ORMD-0801 ORMD-0801 Treatment A: Treatment A: 24 mg (16 mg capsule + 8 mg capsule) Once Daily (QD) at bedtime
Treatment B ORMD-0801
n=30 participants at risk
Treatment B is 8 mg (8 mg capsule) three times a day (TID) 45-90 minutes before meals ORMD-0801 Treatment B: Treatment B: 8 mg (8 mg capsule) three times a day (TID) 45-90 minutes before meals
Infections and infestations
Nasopharangitis
0.00%
0/30 • Sixty-six (66) days
0.00%
0/30 • Sixty-six (66) days
3.3%
1/30 • Number of events 1 • Sixty-six (66) days
Infections and infestations
OTITIS EXTERNA
0.00%
0/30 • Sixty-six (66) days
0.00%
0/30 • Sixty-six (66) days
3.3%
1/30 • Number of events 1 • Sixty-six (66) days
Immune system disorders
Sinusitis
0.00%
0/30 • Sixty-six (66) days
0.00%
0/30 • Sixty-six (66) days
3.3%
1/30 • Number of events 1 • Sixty-six (66) days
Infections and infestations
UPPER RESPIRATORY TRACT INFECTION
0.00%
0/30 • Sixty-six (66) days
3.3%
1/30 • Number of events 1 • Sixty-six (66) days
3.3%
1/30 • Number of events 1 • Sixty-six (66) days
Infections and infestations
Urinary Tract Infection
0.00%
0/30 • Sixty-six (66) days
3.3%
1/30 • Number of events 1 • Sixty-six (66) days
3.3%
1/30 • Number of events 1 • Sixty-six (66) days
Metabolism and nutrition disorders
Hypoglycemia
0.00%
0/30 • Sixty-six (66) days
3.3%
1/30 • Number of events 1 • Sixty-six (66) days
3.3%
1/30 • Number of events 1 • Sixty-six (66) days
Gastrointestinal disorders
Diarrhoea
0.00%
0/30 • Sixty-six (66) days
6.7%
2/30 • Number of events 2 • Sixty-six (66) days
0.00%
0/30 • Sixty-six (66) days
Gastrointestinal disorders
Abdominal discomfort
0.00%
0/30 • Sixty-six (66) days
3.3%
1/30 • Number of events 1 • Sixty-six (66) days
0.00%
0/30 • Sixty-six (66) days

Additional Information

Miriam Kidron, PhD

Oramed, Ltd.

Phone: +972-2-566-0001

Results disclosure agreements

  • Principal investigator is a sponsor employee
  • Publication restrictions are in place

Restriction type: LTE60