Study in Chinese Healthy Adults to Evaluate the Safety, Tolerability and Pharmacokinetics on ZSP0678, and the Effect of Food on ZSP0678 Pharmacokinetics

NCT ID: NCT04137055

Last Updated: 2021-07-28

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

104 participants

Study Classification

INTERVENTIONAL

Study Start Date

2019-11-19

Study Completion Date

2020-12-09

Brief Summary

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This study will evaluate the safety, tolerability and pharmacokinetics (PK) of escalating single-and multiple-oral doses of ZSP0678 on fasted condition, and characterize PK of ZSP0678 on an empty stomach (fasted condition) and following a high fat, high calorie meal (fed condition) in a 2-period, 2-sequence manner. The study will be conducted in 3 parts (Ascending single dose, multiple dose and food effect). Participants will receive either ZSP0678 or placebo .

Detailed Description

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Conditions

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Nonalcoholic Steatohepatitis

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

SEQUENTIAL

Primary Study Purpose

TREATMENT

Blinding Strategy

QUADRUPLE

Participants Caregivers Investigators Outcome Assessors

Study Groups

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ZSP0678-10mg (single dose)-Cohort 1

ZSP0678/Placebo 10mg

Group Type EXPERIMENTAL

ZSP0678-10mg

Intervention Type DRUG

ZSP0678 tablet administered orally under fasted condition

ZSP0678 Placebo

Intervention Type DRUG

Participants will receive placebo matching to ZSP0678 orally.

ZSP0678-30mg (single dose)-Cohort 2

ZSP0678/Placebo 30 mg Enrollment into Cohort 2 will begin upon assurance of safety for Cohort 1.

Group Type EXPERIMENTAL

ZSP0678-30mg

Intervention Type DRUG

ZSP0678 tablets administered orally under fasted condition

ZSP0678 Placebo

Intervention Type DRUG

Participants will receive placebo matching to ZSP0678 orally.

ZSP0678-60mg (single dose)-Cohort 3

ZSP0678/Placebo 60mg Enrollment into Cohort 3 will begin upon assurance of safety for Cohort 2.

Group Type EXPERIMENTAL

ZSP0678-60mg

Intervention Type DRUG

ZSP0678 tablets administered orally under fasted condition

ZSP0678 Placebo

Intervention Type DRUG

Participants will receive placebo matching to ZSP0678 orally.

ZSP0678-120mg (single dose)-Cohort 4

ZSP0678/Placebo 120mg Enrollment into Cohort 4 will begin upon assurance of safety for Cohort 3.

Group Type EXPERIMENTAL

ZSP0678-120mg

Intervention Type DRUG

ZSP0678 tablets administered orally under fasted condition

ZSP0678 Placebo

Intervention Type DRUG

Participants will receive placebo matching to ZSP0678 orally.

ZSP0678-180mg (single dose)-Cohort 5

ZSP0678/Placebo 180mg Enrollment into Cohort 5 will begin upon assurance of safety for Cohort 4.

Group Type EXPERIMENTAL

ZSP0678-180mg

Intervention Type DRUG

ZSP0678 tablets administered orally under fasted condition

ZSP0678 Placebo

Intervention Type DRUG

Participants will receive placebo matching to ZSP0678 orally.

ZSP0678-240mg (single dose)-Cohort 6

ZSP0678/Placebo 240mg Enrollment into Cohort 6 will begin upon assurance of safety for Cohort 5.

Group Type EXPERIMENTAL

ZSP0678-240mg

Intervention Type DRUG

ZSP0678 tablets administered orally under fasted condition

ZSP0678 Placebo

Intervention Type DRUG

Participants will receive placebo matching to ZSP0678 orally.

ZSP0678-320mg (single dose)-Cohort 7

ZSP0678/Placebo 320mg Enrollment into Cohort 7 will begin upon assurance of safety for Cohort 6.

Group Type EXPERIMENTAL

ZSP0678-320mg

Intervention Type DRUG

ZSP0678 tablets administered orally under fasted condition

ZSP0678 Placebo

Intervention Type DRUG

Participants will receive placebo matching to ZSP0678 orally.

ZSP0678 (food effect)-Cohort FE

Period 1: Group A and Group B receive ZSP0678/Placebo under the fasting or fed condition ,respectively on Day1.

Period 2: Group A and Group B receive ZSP0678/Placebo under the fed or fasting condition ,respectively on Day8.

Enrollment into Cohort FE will begin upon assurance of safety for Cohort 4.

Group Type EXPERIMENTAL

ZSP0678

Intervention Type DRUG

ZSP0678 tablets administered orally under fasted or fed condition

ZSP0678 Placebo

Intervention Type DRUG

Participants will receive placebo matching to ZSP0678 orally.

ZSP0678 Dose1 (multiple doses)-Cohort 8

ZSP0678/Placebo Dose1 will be administrated according to the results of Cohort 2\&3

Group Type EXPERIMENTAL

ZSP0678-Dose 1

Intervention Type DRUG

ZSP0678 tablets administered orally once daily for 14 Days

ZSP0678 Placebo

Intervention Type DRUG

Participants will receive placebo matching to ZSP0678 orally.

ZSP0678 Dose2 (multiple doses)-Cohort 9

ZSP0678/Placebo Dose2 will be administrated according to the results of Cohort 3\&4

Group Type EXPERIMENTAL

ZSP0678-Dose 2

Intervention Type DRUG

ZSP0678 tablets administered orally once daily for 14 Days

ZSP0678 Placebo

Intervention Type DRUG

Participants will receive placebo matching to ZSP0678 orally.

ZSP0678 Dose3 (multiple doses)-Cohort 10

ZSP0678/Placebo Dose3 will be administrated according to the results of Cohort 4\&5

Group Type EXPERIMENTAL

ZSP0678-Dose 3

Intervention Type DRUG

ZSP0678 tablets administered orally once daily for 14 Days

ZSP0678 Placebo

Intervention Type DRUG

Participants will receive placebo matching to ZSP0678 orally.

Interventions

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ZSP0678-10mg

ZSP0678 tablet administered orally under fasted condition

Intervention Type DRUG

ZSP0678-30mg

ZSP0678 tablets administered orally under fasted condition

Intervention Type DRUG

ZSP0678-60mg

ZSP0678 tablets administered orally under fasted condition

Intervention Type DRUG

ZSP0678-120mg

ZSP0678 tablets administered orally under fasted condition

Intervention Type DRUG

ZSP0678-180mg

ZSP0678 tablets administered orally under fasted condition

Intervention Type DRUG

ZSP0678-240mg

ZSP0678 tablets administered orally under fasted condition

Intervention Type DRUG

ZSP0678-320mg

ZSP0678 tablets administered orally under fasted condition

Intervention Type DRUG

ZSP0678

ZSP0678 tablets administered orally under fasted or fed condition

Intervention Type DRUG

ZSP0678-Dose 1

ZSP0678 tablets administered orally once daily for 14 Days

Intervention Type DRUG

ZSP0678-Dose 2

ZSP0678 tablets administered orally once daily for 14 Days

Intervention Type DRUG

ZSP0678-Dose 3

ZSP0678 tablets administered orally once daily for 14 Days

Intervention Type DRUG

ZSP0678 Placebo

Participants will receive placebo matching to ZSP0678 orally.

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Subjects are required to meet the following criteria in order to be included in the trial:

1. Signature signed informed consent before the trial, and fully understood the content, process and possible adverse reactions.
2. Subjects must be willing and able to complete the research according to the experimental protocol.
3. Subjects (including partners) are willing to take effective contraceptive measures and have no pregnancy plan during the whole study period until 6 months after drug withdrawal.
4. Male and female subjects aged 18-50 (including 18 and 50)
5. Body weight of male subjects should not be less than 50kg and that of female subjects should not be less than 45kg.Body mass index (BMI) = weight (kg)/height 2 (m2), the range of 19\~26kg/m2 (including the critical value);
6. Physical condition:No significant abnormalities in medical history, including cardiovascular system, liver, kidneys, gastrointestinal system, neural system, respiratory system (eg.asthma,asthma induced by exercise,chronic obstructive pulmonary disease), mental, metabolism, etc.
7. Subjects in general good health or No significant abnormalities in the opinion of the investigator as determined by vital signs and a physical examination.

Exclusion Criteria

1. Allergic constitution (allergic to many drugs, especially to ingredients similar to the test drug and food)
2. The average daily smoking are more than 5 cigarettes within 3 months prior to screening.
3. Known history of drug or alcohol abuse.(defined as consumption of more than 30g of ethanol a day for male and more than 20 g for female )
4. Subjects who donated blood or bleeding profusely(\> 400 mL)in the 3 months preceding study screening.
5. History of dysphagia or any gastrointestinal illness that affects drug absorption, including a history of frequent nausea or vomiting from any cause, irregular gastrointestinal motility, such as habitual diarrhea, constipation, or irritable bowel syndrome.
6. History or presence of any disease or condition known to increase the risk of bleeding, eg.acute gastritis, duodenal ulcer, etc.
7. Participated in another clinical research study and received any investigational products within 3 months prior to dosing.
8. Use of any prescription or over-the-counter (OTC) medications, vitamins and herbal within 14 days prior to screening.
9. History of having any special food(including dragon fruit, mango, grapefruit, etc.),strenuous exercises,or other factors may interfere with the absorption, distribution, metabolism, or excretion of drug within 14 days prior to screening.
10. Subjects who cannot tolerate standard meals (this clause only applies to subjects participating in food impact studies).
11. Presence of clinically significant abnormalities in ECG or QTcB\>450ms in males,or QTcB\>470ms in females.
12. Pregnancy or breastfeeding at screening and during the study.All female subjects of childbearing potential must have a negative urine pregnancy test at screening and during the trial.
13. Any clinically significant abnormality upon physical examination or in the clinical laboratory tests. History or presence of a clinically significant gastrointestinal, renal, hepatic, neurologic, hematic, endocrine, neoplastic, pulmonary, immune, psychiatric or cardiovascular and cerebrovascular disorder(s) (but not limited to above disorders).
14. Presence of human immunodeficiency virus (HIV), viral hepatitis(including hepatitis C virus (HCV) or hepatitis B virus (HBV) ),treponema pallidum antibodies at screening.
15. Any acute illness or concomitant medication from screening to first dosing.
16. Have chocolate, any food or beverage that contains caffeine ,xanthine and alcohol within 24 hours prior to dosing.
17. Positive for urine drug screening or history of substance abuse for a period of 5 consecutive years before screening.
18. As judged by the researcher, it is not suitable to join the clinical researcher.
Minimum Eligible Age

18 Years

Maximum Eligible Age

50 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

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Guangdong Raynovent Biotech Co., Ltd

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Locations

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Beijing Friendship Hospital Affiliated to Capital Medical Universit

Beijing, Beijing Municipality, China

Site Status

Countries

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China

Other Identifiers

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ZSP0678-19-01

Identifier Type: -

Identifier Source: org_study_id

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