An Extension Study of Ublituximab in Participants With Relapsing Multiple Sclerosis

NCT ID: NCT04130997

Last Updated: 2025-12-30

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

ACTIVE_NOT_RECRUITING

Clinical Phase

PHASE3

Total Enrollment

1100 participants

Study Classification

INTERVENTIONAL

Study Start Date

2019-11-18

Study Completion Date

2030-02-01

Brief Summary

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The purpose of this study is to evaluate long-term safety and efficacy of ublituximab therapy in participants with relapsing multiple sclerosis (RMS).

Detailed Description

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TG1101-RMS303 is an open-label, single-arm extension study designed to evaluate long-term safety and efficacy of ublituximab in participants with RMS. Participants who complete the 96-week, double-blind treatment period of TG1101-RMS301 (RMS301 \[NCT03277261\]) or TG1101-RMS302 (RMS302 \[NCT03277248\]) are eligible for participation in this Open Label Extension (OLE) study. Participants may also be eligible for TG1101-RMS303 if they have completed Week 208 of TG1101-RMS201E (RMS201E \[NCT03381170\]) (United States of America \[USA\] participants only).

Conditions

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Relapsing Multiple Sclerosis (RMS)

Study Design

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Allocation Method

NA

Intervention Model

SINGLE_GROUP

open-label, single-arm, extension study
Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Ublituximab Infusions

RMS301/RMS302: All participants transferring from RMS301/RMS302 who sign consent for this study will receive an initial 4-hour infusion of 150 mg ublituximab on Week 1 (Day 1) followed by a 1-hour infusion of 450 mg ublituximab 14 days later Week 3 (Day 15). Subsequent infusions of ublituximab will be administered at 450 mg for 1-hour every 24 weeks from Weeks 24 to 312.

RMS201E: All participants transferring from RMS201E who sign consent for this study will receive a 1-hour infusion of 450 mg ublituximab on Week 1 (Day 1) and subsequent infusions of ublituximab will be administered at 450 mg for 1-hour every 24 weeks from Weeks 24 to 312.

For all participants (RMS301/RMS302/RMS201E), infusion treatment will continue for 312 weeks, or until physician or participant decision to withdraw from the study.

Group Type EXPERIMENTAL

Ublituximab

Intervention Type BIOLOGICAL

Ublituximab (TG-1101) is a recombinant chimeric monoclonal antibody targeting CD20, available as a 25 mg/mL concentrate for intravenous use, supplied by TG Therapeutics, Inc.

Interventions

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Ublituximab

Ublituximab (TG-1101) is a recombinant chimeric monoclonal antibody targeting CD20, available as a 25 mg/mL concentrate for intravenous use, supplied by TG Therapeutics, Inc.

Intervention Type BIOLOGICAL

Other Intervention Names

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TG-1101

Eligibility Criteria

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Inclusion Criteria

Participants must meet the following criteria:

1. Complete the 96-week double-blind TG1101-RMS301 (NCT03277261) or TG1101-RMS302 (NCT03277248) study or complete the final Week 208 visit of the TG1101-RMS201E (NCT03381170) study
2. Investigator believes may benefit from treatment with ublituximab
3. Are able and willing to provide written informed consent (e.g., before the first infusion) and to comply with the study protocol
4. Female participants of child-bearing potential, and male partners must consent to use a medically acceptable method of contraception from consent, throughout the study period, and for 20 weeks after the last dose of ublituximab

Exclusion Criteria

1. Any significant or uncontrolled medical condition or treatment-emergent, clinically significant laboratory abnormality such as:

1. Absolute neutrophil count \< 1.5 x 10e3/µL
2. Hematocrit \< 24%
3. Platelet count \< 150,000 cell/mm\^3
4. Hypogammaglobulinemia immunoglobulin G (IgG) \< 4.0g/L
2. Active infection
3. Ongoing pregnancy (female participants)
4. Participants who discontinued ublituximab treatment or withdrew consent from the TG1101-RMS301 or TG1101-RMS302 study during the 96-week evaluation period or prior to completing the final Week 208 visit of the TG1101-RMS201E study
5. Participants who have started any disease modifying therapy (DMT), stem cell transplantation, or participation in any other interventional clinical trial after completion of the 96-week visit in the TG1101-RMS301, TG1101-RMS302, or after completing the final Week 208 visit of the TG1101-RMS201E study
6. Participants who have had a confirmed multiple sclerosis (MS) relapse within the past 30 days prior to Week 1 Day 1 (W1D1). Following a relapse, participants must be neurologically stable for at least 30 days prior to screening or W1D1 of the OLE
7. Participants with unstable disease activity
8. Presence of malignancy, except for surgically excised basal or squamous cell skin lesions
9. Vaccination with live virus within 2 months of randomization
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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TG Therapeutics, Inc.

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Locations

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TG Therapeutics Investigational Trial Site

Pasadena, California, United States

Site Status

TG Therapeutics Investigational Trial Site

Denver, Colorado, United States

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TG Therapeutics Investigational Trial Site

Miami, Florida, United States

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TG Therapeutics Investigational Trial Site

Tampa, Florida, United States

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TG Therapeutics Investigational Trial Site

Northbrook, Illinois, United States

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TG Therapeutics Investigational Trial Site

Kansas City, Kansas, United States

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TG Therapeutics Investigational Trial Site

Detroit, Michigan, United States

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TG Therapeutics Investigational Trial Site

Las Vegas, Nevada, United States

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TG Therapeutics Investigational Trial Site

Teaneck, New Jersey, United States

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TG Therapeutics Investigational Trial Site

Albuquerque, New Mexico, United States

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TG Therapeutics Investigational Trial Site

Amherst, New York, United States

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TG Therapeutics Investigational Trial Site

Columbus, Ohio, United States

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TG Therapeutics Investigational Trial Site

Westerville, Ohio, United States

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TG Therapeutics Investigational Trial Site

Knoxville, Tennessee, United States

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TG Therapeutics Investigational Trial Site

Dallas, Texas, United States

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TG Therapeutics Investigational Trial Site

Frisco, Texas, United States

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TG Therapeutics Investigational Trial Site

Round Rock, Texas, United States

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TG Therapeutics Investigational Trial Site

San Antonio, Texas, United States

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TG Therapeutics Investigational Trial Site

Seattle, Washington, United States

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TG Therapeutics Investigational Trial Site

Grodno, , Belarus

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TG Therapeutics Investigational Trial Site

Grodno, , Belarus

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TG Therapeutics Investigational Trial Site

Minsk, , Belarus

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TG Therapeutics Investigational Trial Site

Minsk, , Belarus

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TG Therapeutics Investigational Trial Site

Minsk, , Belarus

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TG Therapeutics Investigational Trial Site

Osijek, , Croatia

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TG Therapeutics Investigational Trial Site

Varaždin, , Croatia

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TG Investigational Trial Site

Zagreb, , Croatia

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TG Therapeutics Investigational Trial Site

Tbilisi, , Georgia

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TG Therapeutics Investigational Trial Site

Tbilisi, , Georgia

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TG Therapeutics Investigational Trial Site

Tbilisi, , Georgia

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TG Therapeutics Investigational Trial Site

Tbilisi, , Georgia

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TG Therapeutics Investigational Trial Site

Tbilisi, , Georgia

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TG Therapeutics Investigational Trial Site

Tbilisi, , Georgia

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TG Therapeutics Investigational Trial Site

Katowice, , Poland

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TG Therapeutics Investigational Trial Site

Katowice, , Poland

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TG Therapeutics Investigational Trial Site

Katowice, , Poland

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TG Therapeutics Investigational Trial Site

Krakow, , Poland

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TG Therapeutics Investigational Trial Site

Lodz, , Poland

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TG Therapeutics Investigational Trial Site

Olsztyn, , Poland

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TG Therapeutics Investigational Trial Site

Poznan, , Poland

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TG Therapeutics Investigational Trial Site

Warsaw, , Poland

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TG Therapeutics Investigational Trial Site

Zabrze, , Poland

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TG Therapeutics Investigational Trial Site

Arkhangelsk, , Russia

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TG Therapeutics Investigational Trial Site

Barnaul, , Russia

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TG Therapeutics Investigational Trial Site

Bryansk, , Russia

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TG Therapeutics Investigational Trial Site

Chelyabinsk, , Russia

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TG Therapeutics Investigational Trial Site

Kemerovo, , Russia

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TG Therapeutics Investigational Trial Site

Krasnoyarsk, , Russia

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TG Therapeutics Investigational Trial Site

Kursk, , Russia

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TG Therapeutics Investigational Trial Site

Moscow, , Russia

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TG Therapeutics Investigational Trial Site

Moscow, , Russia

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TG Therapeutics Investigational Trial Site

Nizhny Novgorod, , Russia

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TG Therapeutics Investigational Trial Site

Novosibirsk, , Russia

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TG Therapeutics Investigational Trial Site

Novosibirsk, , Russia

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TG Therapeutics Investigational Trial Site

Pyatigorsk, , Russia

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TG Therapeutics Investigational Trial Site

Saint Petersburg, , Russia

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TG Therapeutics Investigational Trial Site

Saint Petersburg, , Russia

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TG Therapeutics Investigational Trial Site

Saint Petersburg, , Russia

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TG Therapeutics Investigational Trial Site

Saransk, , Russia

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TG Therapeutics Investigational Trial Site

Smolensk, , Russia

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TG Therapeutics Investigational Trial Site

Tomsk, , Russia

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TG Therapeutics Investigational Trial Site

Tyumen, , Russia

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TG Therapeutics Investigational Trial Site

Ufa, , Russia

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TG Therapeutics Investigational Trial Site

Yekaterinburg, , Russia

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TG Therapeutics Investigational Trial Site

Belgrade, , Serbia

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TG Therapeutics Investigational Trial Site

Kragujevac, , Serbia

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TG Therapeutics Investigational Trial Site

Cherkasy, , Ukraine

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TG Therapeutics Investigational Trial Site

Chernihiv, , Ukraine

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TG Therapeutics Investigational Trial Site

Chernihiv, , Ukraine

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TG Therapeutics Investigational Trial Site

Chernivtsi, , Ukraine

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TG Therapeutics Investigational Trial Site

Ivano-Frankivsk, , Ukraine

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TG Therapeutics Investigational Trial Site

Kharkiv, , Ukraine

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TG Therapeutics Investigational Trial Site

Kharkiv, , Ukraine

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TG Therapeutics Investigational Trial Site

Kharkiv, , Ukraine

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TG Therapeutics Investigational Trial Site

Kyiv, , Ukraine

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TG Therapeutics Investigational Trial Site

Kyiv, , Ukraine

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TG Therapeutics Investigational Trial Site

Lviv, , Ukraine

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TG Therapeutics Investigational Trial Site

Lviv, , Ukraine

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TG Therapeutics Investigational Trial Site

Odesa, , Ukraine

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TG Therapeutics Investigational Trial Site

Poltava, , Ukraine

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TG Therapeutics Investigational Trial Site

Ternopil, , Ukraine

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TG Therapeutics Investigational Trial Site

Uzhhorod, , Ukraine

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TG Therapeutics Investigational Trial Site

Vinnytsia, , Ukraine

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TG Therapeutics Investigational Trial Site

Zaporizhia, , Ukraine

Site Status

TG Therapeutics Investigational Trial Site

Zaporizhia, , Ukraine

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TG Therapeutics Investigational Trial Site

Zhytomyr, , Ukraine

Site Status

Countries

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United States Belarus Croatia Georgia Poland Russia Serbia Ukraine

Other Identifiers

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2019-003625-16

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

TG1101-RMS303

Identifier Type: -

Identifier Source: org_study_id