Trial Outcomes & Findings for A Study Assessing the Safety, Efficacy, and Optimum Dosage of K-161 in Subjects With Moderate to Severe Dry Eye Disease (NCT NCT04084483)

NCT ID: NCT04084483

Last Updated: 2023-03-15

Results Overview

Fluorescein Staining is measured with the Ora Calibra® Corneal and Conjunctival Staining Scale which is a 0 to 4 scale with increasing half-units and where higher numbers indicating more severe staining. K-161 compared to Vehicle. When study patients are exposed to Controlled Adverse Environment (CAE) in terms of relative humidity, temperature, airflow, and visual tasking, the ocular surface is stressed to react. This controlled environmental stress creates a consistent response that's reproducible over time.

Recruitment status

COMPLETED

Study phase

PHASE2

Target enrollment

238 participants

Primary outcome timeframe

Baseline to Day 29

Results posted on

2023-03-15

Participant Flow

During the screening period, two 90-minute exposures to the CAE® were conducted to ascertain eligibility to enter the study. Participants who qualified after the initial screening visit entered the run-in phase, where they self-administered Vehicle for approximately 14 days. Those who qualified at Visit 2 (Day 1) were randomized to receive study drug in a double-masked fashion for 28 days.

Participant milestones

Participant milestones
Measure
Placebo (BID) (Vehicle)
1 drop Ophthalmic Solution
0.025% K-161 (BID)
1 drop Ophthalmic Solution
0.1% K-161 (BID)
1 drop Ophthalmic Solution
0.1% K-161 (QID)
1 drop Ophthalmic Solution
Overall Study
STARTED
59
59
61
59
Overall Study
COMPLETED
56
57
59
57
Overall Study
NOT COMPLETED
3
2
2
2

Reasons for withdrawal

Withdrawal data not reported

Baseline Characteristics

A Study Assessing the Safety, Efficacy, and Optimum Dosage of K-161 in Subjects With Moderate to Severe Dry Eye Disease

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
Placebo (BID) (Vehicle)
n=59 Participants
1 drop Ophthalmic Solution
0.025% K-161 (BID)
n=59 Participants
1 drop Ophthalmic Solution
0.1% K-161 (BID)
n=61 Participants
1 drop Ophthalmic Solution
0.1% K-161 (QID)
n=59 Participants
1 drop Ophthalmic Solution
Total
n=238 Participants
Total of all reporting groups
Age, Customized
< 65 years
34 Participants
n=5 Participants
37 Participants
n=7 Participants
38 Participants
n=5 Participants
38 Participants
n=4 Participants
147 Participants
n=21 Participants
Age, Customized
≥ 65 years
25 Participants
n=5 Participants
22 Participants
n=7 Participants
23 Participants
n=5 Participants
21 Participants
n=4 Participants
91 Participants
n=21 Participants
Sex: Female, Male
Female
41 Participants
n=5 Participants
43 Participants
n=7 Participants
44 Participants
n=5 Participants
43 Participants
n=4 Participants
171 Participants
n=21 Participants
Sex: Female, Male
Male
18 Participants
n=5 Participants
16 Participants
n=7 Participants
17 Participants
n=5 Participants
16 Participants
n=4 Participants
67 Participants
n=21 Participants
Ethnicity (NIH/OMB)
Hispanic or Latino
1 Participants
n=5 Participants
1 Participants
n=7 Participants
1 Participants
n=5 Participants
1 Participants
n=4 Participants
4 Participants
n=21 Participants
Ethnicity (NIH/OMB)
Not Hispanic or Latino
58 Participants
n=5 Participants
58 Participants
n=7 Participants
60 Participants
n=5 Participants
58 Participants
n=4 Participants
234 Participants
n=21 Participants
Ethnicity (NIH/OMB)
Unknown or Not Reported
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
0 Participants
n=4 Participants
0 Participants
n=21 Participants
Race (NIH/OMB)
American Indian or Alaska Native
1 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
0 Participants
n=4 Participants
1 Participants
n=21 Participants
Race (NIH/OMB)
Asian
13 Participants
n=5 Participants
16 Participants
n=7 Participants
12 Participants
n=5 Participants
15 Participants
n=4 Participants
56 Participants
n=21 Participants
Race (NIH/OMB)
Native Hawaiian or Other Pacific Islander
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
0 Participants
n=4 Participants
0 Participants
n=21 Participants
Race (NIH/OMB)
Black or African American
15 Participants
n=5 Participants
11 Participants
n=7 Participants
10 Participants
n=5 Participants
9 Participants
n=4 Participants
45 Participants
n=21 Participants
Race (NIH/OMB)
White
29 Participants
n=5 Participants
32 Participants
n=7 Participants
37 Participants
n=5 Participants
35 Participants
n=4 Participants
133 Participants
n=21 Participants
Race (NIH/OMB)
More than one race
1 Participants
n=5 Participants
0 Participants
n=7 Participants
2 Participants
n=5 Participants
0 Participants
n=4 Participants
3 Participants
n=21 Participants
Race (NIH/OMB)
Unknown or Not Reported
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
0 Participants
n=4 Participants
0 Participants
n=21 Participants
Inferior Corneal Fluorescein Staining Score Post Controlled Adverse Environment (Post-CAE)
3.30 scores on a scale
STANDARD_DEVIATION 0.361 • n=5 Participants
3.36 scores on a scale
STANDARD_DEVIATION 0.405 • n=7 Participants
3.35 scores on a scale
STANDARD_DEVIATION 0.412 • n=5 Participants
3.33 scores on a scale
STANDARD_DEVIATION 0.378 • n=4 Participants
3.33 scores on a scale
STANDARD_DEVIATION 0.388 • n=21 Participants
Ocular Discomfort Scale Post-CAE
3.8 scores on a scale
STANDARD_DEVIATION 0.49 • n=5 Participants
3.7 scores on a scale
STANDARD_DEVIATION 0.48 • n=7 Participants
3.7 scores on a scale
STANDARD_DEVIATION 0.61 • n=5 Participants
3.6 scores on a scale
STANDARD_DEVIATION 0.72 • n=4 Participants
3.7 scores on a scale
STANDARD_DEVIATION 0.58 • n=21 Participants

PRIMARY outcome

Timeframe: Baseline to Day 29

Population: Endpoints analysis was determined by comparing 0.1% K-161 BID to its Vehicle BID

Fluorescein Staining is measured with the Ora Calibra® Corneal and Conjunctival Staining Scale which is a 0 to 4 scale with increasing half-units and where higher numbers indicating more severe staining. K-161 compared to Vehicle. When study patients are exposed to Controlled Adverse Environment (CAE) in terms of relative humidity, temperature, airflow, and visual tasking, the ocular surface is stressed to react. This controlled environmental stress creates a consistent response that's reproducible over time.

Outcome measures

Outcome measures
Measure
Placebo (BID) (Vehicle)
n=59 Participants
1 drop Ophthalmic Solution
0.1% K-161 (BID)
n=61 Participants
1 drop Ophthalmic Solution
0.1% K-161 (BID)
1 drop Ophthalmic Solution
Change in Inferior Corneal Fluorescein Staining Score Post Controlled Adverse Environment (Post-Controlled Adverse Environment (CAE))
-0.57 scores on a scale
Standard Error 0.075
-0.44 scores on a scale
Standard Error 0.073

PRIMARY outcome

Timeframe: Baseline to Day 29

Population: Endpoints analysis was determined by comparing 0.1% K-161 BID to its Vehicle BID

Ocular discomfort scores were subjectively graded by the subjects using the Ora Calibra® Ocular Discomfort Scale from 0 to 4 where 0 = No Discomfort and 4 = Constant Discomfort.

Outcome measures

Outcome measures
Measure
Placebo (BID) (Vehicle)
n=59 Participants
1 drop Ophthalmic Solution
0.1% K-161 (BID)
n=61 Participants
1 drop Ophthalmic Solution
0.1% K-161 (BID)
1 drop Ophthalmic Solution
Change in Ocular Discomfort Scale Post-CAE
0.0 score on a scale
Standard Error 0.06
0.0 score on a scale
Standard Error 0.06

SECONDARY outcome

Timeframe: Baseline to Day 29

Population: Endpoints analysis was determined by comparing 0.1% K-161 BID to its Vehicle BID

Measured with Schirmer's test strip with the length of the moistened area recorded in mm. Lower values indicate less tears produced in the eye.

Outcome measures

Outcome measures
Measure
Placebo (BID) (Vehicle)
n=59 Participants
1 drop Ophthalmic Solution
0.1% K-161 (BID)
n=61 Participants
1 drop Ophthalmic Solution
0.1% K-161 (BID)
1 drop Ophthalmic Solution
Change in Schirmer's Test Value (Unanesthetized) Pre-CAE
3.4 mm
Standard Error 0.85
2.2 mm
Standard Error 0.80

SECONDARY outcome

Timeframe: Baseline to Day 29

Population: Endpoints analysis was determined by comparing 0.1% K-161 BID to its Vehicle BID

Outcome measures

Outcome measures
Measure
Placebo (BID) (Vehicle)
n=59 Participants
1 drop Ophthalmic Solution
0.1% K-161 (BID)
n=61 Participants
1 drop Ophthalmic Solution
0.1% K-161 (BID)
1 drop Ophthalmic Solution
Change in Tear Film Break-up Time (TFBUT) Post-CAE
0.402 Seconds
Standard Error 0.1090
0.132 Seconds
Standard Error 0.1049

SECONDARY outcome

Timeframe: Baseline to Day 29

Population: Endpoints analysis was determined by comparing Vehicle BID to 0.1% K-161 BID and 0.025% K-161 BID

Fluorescein Staining is measured with the Ora Calibra® Corneal and Conjunctival Staining Scale which is a 0 to 4 scale with increasing half-units and where higher numbers indicating more severe staining.

Outcome measures

Outcome measures
Measure
Placebo (BID) (Vehicle)
n=59 Participants
1 drop Ophthalmic Solution
0.1% K-161 (BID)
n=59 Participants
1 drop Ophthalmic Solution
0.1% K-161 (BID)
n=61 Participants
1 drop Ophthalmic Solution
Change in Fluorescein Staining Scores (Pre-CAE®)
Corneal Sum
-0.28 score on a scale
Standard Error 0.184
-0.36 score on a scale
Standard Error 0.182
-0.50 score on a scale
Standard Error 0.178
Change in Fluorescein Staining Scores (Pre-CAE®)
Conjunctival Sum
-0.03 score on a scale
Standard Error 0.138
-0.22 score on a scale
Standard Error 0.136
-0.28 score on a scale
Standard Error 0.133
Change in Fluorescein Staining Scores (Pre-CAE®)
Total Eye Sum
-0.30 score on a scale
Standard Error 0.292
-0.59 score on a scale
Standard Error 0.290
-0.80 score on a scale
Standard Error 0.283

SECONDARY outcome

Timeframe: Baseline to Day 29

Population: Endpoints analysis was determined by comparing Vehicle BID to 0.1% K-161 BID and 0.025% K-161 BID

Ora Calibra Scale which is 0 to 4 scale with increasing half-units and where higher numbers indicating more severe staining.

Outcome measures

Outcome measures
Measure
Placebo (BID) (Vehicle)
n=59 Participants
1 drop Ophthalmic Solution
0.1% K-161 (BID)
n=59 Participants
1 drop Ophthalmic Solution
0.1% K-161 (BID)
n=61 Participants
1 drop Ophthalmic Solution
Change in Lissamine Green Staining (Pre-CAE) Using the Ora Calibra® Scale (Conjunctival Sum)
-0.16 score on a scale
Standard Error 0.132
-0.25 score on a scale
Standard Error 0.131
-0.39 score on a scale
Standard Error 0.127

SECONDARY outcome

Timeframe: Baseline to Day 29

Population: Endpoints analysis was determined by comparing Vehicle BID to 0.1% K-161 BID and 0.025% K-161 BID

Conjunctival Redness Scale ranges from 0 to 4, where 0 = normal, without vasodilation and 4 = Broad Ciliary and Prominent, Horizontal Conjunctival Vasodilation. Higher scores indicate worsening conjunctival redness.

Outcome measures

Outcome measures
Measure
Placebo (BID) (Vehicle)
n=59 Participants
1 drop Ophthalmic Solution
0.1% K-161 (BID)
n=59 Participants
1 drop Ophthalmic Solution
0.1% K-161 (BID)
n=61 Participants
1 drop Ophthalmic Solution
Change in Conjunctival Redness (Pre-CAE)
-0.21 Point
Standard Error 0.061
-0.20 Point
Standard Error 0.060
-0.22 Point
Standard Error 0.059

SECONDARY outcome

Timeframe: Baseline to Day 29

Population: Endpoints analysis was determined by comparing Vehicle BID to 0.1% K-161 BID and 0.025% K-161 BID

Outcome measures

Outcome measures
Measure
Placebo (BID) (Vehicle)
n=59 Participants
1 drop Ophthalmic Solution
0.1% K-161 (BID)
n=59 Participants
1 drop Ophthalmic Solution
0.1% K-161 (BID)
n=61 Participants
1 drop Ophthalmic Solution
Change in Tear Film Break-Up Time (Pre CAE)
0.312 Seconds
Standard Error 0.0880
0.398 Seconds
Standard Error 0.0863
0.242 Seconds
Standard Error 0.0848

SECONDARY outcome

Timeframe: Baseline to Day 29

Population: Endpoints analysis was determined by comparing Vehicle BID to 0.1% K-161 BID and 0.025% K-161 BID

Outcome measures

Outcome measures
Measure
Placebo (BID) (Vehicle)
n=59 Participants
1 drop Ophthalmic Solution
0.1% K-161 (BID)
n=59 Participants
1 drop Ophthalmic Solution
0.1% K-161 (BID)
n=61 Participants
1 drop Ophthalmic Solution
Change in Tear Osmolarity (Pre CAE)
-0.5 mOsm/L
Standard Error 2.17
1.0 mOsm/L
Standard Error 2.09
0.4 mOsm/L
Standard Error 2.03

SECONDARY outcome

Timeframe: Baseline to Day 29

Population: Endpoints analysis was determined by comparing Vehicle BID to 0.1% K-161 BID and 0.025% K-161 BID

Measured with Schirmer's test strip with the length of the moistened area recorded in mm. Lower values indicate less tears produced in the eye.

Outcome measures

Outcome measures
Measure
Placebo (BID) (Vehicle)
n=59 Participants
1 drop Ophthalmic Solution
0.1% K-161 (BID)
n=59 Participants
1 drop Ophthalmic Solution
0.1% K-161 (BID)
n=61 Participants
1 drop Ophthalmic Solution
Change in Unanesthetized Schirmer's Test (Pre CAE)
3.3 mm
Standard Error 0.82
3.1 mm
Standard Error 0.80
2.1 mm
Standard Error 0.78

SECONDARY outcome

Timeframe: Baseline to Day 29

Population: Endpoints analysis was determined by comparing Vehicle BID to 0.1% K-161 BID and 0.025% K-161 BID

Blinks per 60 seconds.

Outcome measures

Outcome measures
Measure
Placebo (BID) (Vehicle)
n=59 Participants
1 drop Ophthalmic Solution
0.1% K-161 (BID)
n=59 Participants
1 drop Ophthalmic Solution
0.1% K-161 (BID)
n=61 Participants
1 drop Ophthalmic Solution
Change in Blink Rate (Pre CAE)
0.1 Blinks per 60 seconds
Standard Error 1.41
0.1 Blinks per 60 seconds
Standard Error 1.39
-0.2 Blinks per 60 seconds
Standard Error 1.36

SECONDARY outcome

Timeframe: Baseline to Day 29

Population: Endpoints analysis was determined by comparing Vehicle BID to 0.1% K-161 BID and 0.025% K-161 BID

Ora Calibra® Ocular Discomfort Scale ranging from 0 to 4

Outcome measures

Outcome measures
Measure
Placebo (BID) (Vehicle)
n=59 Participants
1 drop Ophthalmic Solution
0.1% K-161 (BID)
n=59 Participants
1 drop Ophthalmic Solution
0.1% K-161 (BID)
n=61 Participants
1 drop Ophthalmic Solution
Change in Ocular Discomfort Scale (Pre CAE)
-0.3 Score
Standard Error 0.13
-0.2 Score
Standard Error 0.13
-0.5 Score
Standard Error 0.12

SECONDARY outcome

Timeframe: Baseline to Day 29

Population: Endpoints analysis was determined by comparing Vehicle BID to 0.1% K-161 BID and 0.025% K-161 BID

Scores ranging from 0 to 5. A score of 0 indicates no discomfort/symptoms and a score of 5 indicates worst discomfort/symptoms.

Outcome measures

Outcome measures
Measure
Placebo (BID) (Vehicle)
n=59 Participants
1 drop Ophthalmic Solution
0.1% K-161 (BID)
n=59 Participants
1 drop Ophthalmic Solution
0.1% K-161 (BID)
n=61 Participants
1 drop Ophthalmic Solution
Change in Ocular Discomfort and 4-Symptom Questionnaire (Pre CAE)
Ocular Discomfort
-0.2 Point
Standard Error 0.13
-0.2 Point
Standard Error 0.13
-0.4 Point
Standard Error 0.13
Change in Ocular Discomfort and 4-Symptom Questionnaire (Pre CAE)
Burning
0.1 Point
Standard Error 0.13
0.0 Point
Standard Error 0.13
-0.1 Point
Standard Error 0.13
Change in Ocular Discomfort and 4-Symptom Questionnaire (Pre CAE)
Dryness
-0.1 Point
Standard Error 0.14
-0.2 Point
Standard Error 0.14
-0.3 Point
Standard Error 0.13
Change in Ocular Discomfort and 4-Symptom Questionnaire (Pre CAE)
Grittiness
-0.1 Point
Standard Error 0.15
-0.3 Point
Standard Error 0.15
-0.1 Point
Standard Error 0.15
Change in Ocular Discomfort and 4-Symptom Questionnaire (Pre CAE)
Stinging
-0.1 Point
Standard Error 0.15
-0.1 Point
Standard Error 0.15
-0.2 Point
Standard Error 0.14

SECONDARY outcome

Timeframe: Baseline to Day 29

Population: Endpoints analysis was determined by comparing Vehicle BID to 0.1% K-161 BID and 0.025% K-161 BID

The length of the assessment line was 100 mm; a measure of 0 mm corresponded to "no discomfort" and 100 mm corresponds to "maximal discomfort".

Outcome measures

Outcome measures
Measure
Placebo (BID) (Vehicle)
n=59 Participants
1 drop Ophthalmic Solution
0.1% K-161 (BID)
n=59 Participants
1 drop Ophthalmic Solution
0.1% K-161 (BID)
n=61 Participants
1 drop Ophthalmic Solution
Change in Visual Analog Scale (Pre CAE)
Burning/Stinging
-1.9 mm
Standard Error 2.78
-7.6 mm
Standard Error 2.76
-5.6 mm
Standard Error 2.68
Change in Visual Analog Scale (Pre CAE)
Itching
-3.1 mm
Standard Error 2.92
-9.7 mm
Standard Error 2.92
-6.1 mm
Standard Error 2.84
Change in Visual Analog Scale (Pre CAE)
Foreign Body Sensation
-1.1 mm
Standard Error 2.96
-6.9 mm
Standard Error 2.94
-5.6 mm
Standard Error 2.82
Change in Visual Analog Scale (Pre CAE)
Blurry Vision
-0.2 mm
Standard Error 2.69
-5.5 mm
Standard Error 2.67
-7.5 mm
Standard Error 2.60
Change in Visual Analog Scale (Pre CAE)
Eye Dryness
-4.1 mm
Standard Error 2.71
-6.1 mm
Standard Error 2.68
-10.7 mm
Standard Error 2.60
Change in Visual Analog Scale (Pre CAE)
Photophobia
-2.8 mm
Standard Error 2.78
-6.2 mm
Standard Error 2.75
-10.7 mm
Standard Error 2.67
Change in Visual Analog Scale (Pre CAE)
Pain
0.0 mm
Standard Error 2.37
-6.0 mm
Standard Error 2.37
-4.2 mm
Standard Error 2.28

SECONDARY outcome

Timeframe: Baseline to Day 29

Population: Endpoints analysis was determined by comparing Vehicle BID to 0.1% K-161 BID and 0.025% K-161 BID

The OSDI© is comprised of 12 questions, with each question assessed on a scale ranging from 0 to 4 where 0 = none of the time, 1 = some of the time, 2 = half of the time, 3 = most of the time, and 4 = all of the time. The range of total score is "0 to 100". "Subscale" scores are not reported. Higher score represents a worsen outcome. The total score is the sum of subscales.

Outcome measures

Outcome measures
Measure
Placebo (BID) (Vehicle)
n=59 Participants
1 drop Ophthalmic Solution
0.1% K-161 (BID)
n=59 Participants
1 drop Ophthalmic Solution
0.1% K-161 (BID)
n=61 Participants
1 drop Ophthalmic Solution
Change in Ocular Surface Disease Index Score (Pre-CAE) - Total OSDI
-3.2 scores on a scale
Standard Error 2.03
-2.9 scores on a scale
Standard Error 2.00
-7.8 scores on a scale
Standard Error 1.95

Adverse Events

Placebo (BID) (Vehicle)

Serious events: 3 serious events
Other events: 2 other events
Deaths: 0 deaths

0.025% K-161 (BID)

Serious events: 0 serious events
Other events: 7 other events
Deaths: 0 deaths

0.1% K-161 (BID)

Serious events: 0 serious events
Other events: 25 other events
Deaths: 0 deaths

0.1% K-161 (QID)

Serious events: 0 serious events
Other events: 24 other events
Deaths: 0 deaths

Serious adverse events

Serious adverse events
Measure
Placebo (BID) (Vehicle)
n=59 participants at risk
1 drop Ophthalmic Solution
0.025% K-161 (BID)
n=59 participants at risk
1 drop Ophthalmic Solution
0.1% K-161 (BID)
n=61 participants at risk
1 drop Ophthalmic Solution
0.1% K-161 (QID)
n=59 participants at risk
1 drop Ophthalmic Solution
Injury, poisoning and procedural complications
Pelvic fracture
1.7%
1/59 • 36 Days
Treatment emergent adverse events (TEAE) were any adverse event that occurred or worsened after the first dose of study treatment.
0.00%
0/59 • 36 Days
Treatment emergent adverse events (TEAE) were any adverse event that occurred or worsened after the first dose of study treatment.
0.00%
0/61 • 36 Days
Treatment emergent adverse events (TEAE) were any adverse event that occurred or worsened after the first dose of study treatment.
0.00%
0/59 • 36 Days
Treatment emergent adverse events (TEAE) were any adverse event that occurred or worsened after the first dose of study treatment.
Injury, poisoning and procedural complications
Upper limb fracture
1.7%
1/59 • 36 Days
Treatment emergent adverse events (TEAE) were any adverse event that occurred or worsened after the first dose of study treatment.
0.00%
0/59 • 36 Days
Treatment emergent adverse events (TEAE) were any adverse event that occurred or worsened after the first dose of study treatment.
0.00%
0/61 • 36 Days
Treatment emergent adverse events (TEAE) were any adverse event that occurred or worsened after the first dose of study treatment.
0.00%
0/59 • 36 Days
Treatment emergent adverse events (TEAE) were any adverse event that occurred or worsened after the first dose of study treatment.
Infections and infestations
Pneumonia
1.7%
1/59 • 36 Days
Treatment emergent adverse events (TEAE) were any adverse event that occurred or worsened after the first dose of study treatment.
0.00%
0/59 • 36 Days
Treatment emergent adverse events (TEAE) were any adverse event that occurred or worsened after the first dose of study treatment.
0.00%
0/61 • 36 Days
Treatment emergent adverse events (TEAE) were any adverse event that occurred or worsened after the first dose of study treatment.
0.00%
0/59 • 36 Days
Treatment emergent adverse events (TEAE) were any adverse event that occurred or worsened after the first dose of study treatment.
Renal and urinary disorders
Acute kidney injury
1.7%
1/59 • 36 Days
Treatment emergent adverse events (TEAE) were any adverse event that occurred or worsened after the first dose of study treatment.
0.00%
0/59 • 36 Days
Treatment emergent adverse events (TEAE) were any adverse event that occurred or worsened after the first dose of study treatment.
0.00%
0/61 • 36 Days
Treatment emergent adverse events (TEAE) were any adverse event that occurred or worsened after the first dose of study treatment.
0.00%
0/59 • 36 Days
Treatment emergent adverse events (TEAE) were any adverse event that occurred or worsened after the first dose of study treatment.
Nervous system disorders
Toxic encephalopathy
1.7%
1/59 • 36 Days
Treatment emergent adverse events (TEAE) were any adverse event that occurred or worsened after the first dose of study treatment.
0.00%
0/59 • 36 Days
Treatment emergent adverse events (TEAE) were any adverse event that occurred or worsened after the first dose of study treatment.
0.00%
0/61 • 36 Days
Treatment emergent adverse events (TEAE) were any adverse event that occurred or worsened after the first dose of study treatment.
0.00%
0/59 • 36 Days
Treatment emergent adverse events (TEAE) were any adverse event that occurred or worsened after the first dose of study treatment.
Neoplasms benign, malignant and unspecified (incl cysts and polyps)
Chronic lymphocytic leukaemia
1.7%
1/59 • 36 Days
Treatment emergent adverse events (TEAE) were any adverse event that occurred or worsened after the first dose of study treatment.
0.00%
0/59 • 36 Days
Treatment emergent adverse events (TEAE) were any adverse event that occurred or worsened after the first dose of study treatment.
0.00%
0/61 • 36 Days
Treatment emergent adverse events (TEAE) were any adverse event that occurred or worsened after the first dose of study treatment.
0.00%
0/59 • 36 Days
Treatment emergent adverse events (TEAE) were any adverse event that occurred or worsened after the first dose of study treatment.

Other adverse events

Other adverse events
Measure
Placebo (BID) (Vehicle)
n=59 participants at risk
1 drop Ophthalmic Solution
0.025% K-161 (BID)
n=59 participants at risk
1 drop Ophthalmic Solution
0.1% K-161 (BID)
n=61 participants at risk
1 drop Ophthalmic Solution
0.1% K-161 (QID)
n=59 participants at risk
1 drop Ophthalmic Solution
General disorders
Instillation site pain
3.4%
2/59 • 36 Days
Treatment emergent adverse events (TEAE) were any adverse event that occurred or worsened after the first dose of study treatment.
10.2%
6/59 • 36 Days
Treatment emergent adverse events (TEAE) were any adverse event that occurred or worsened after the first dose of study treatment.
37.7%
23/61 • 36 Days
Treatment emergent adverse events (TEAE) were any adverse event that occurred or worsened after the first dose of study treatment.
35.6%
21/59 • 36 Days
Treatment emergent adverse events (TEAE) were any adverse event that occurred or worsened after the first dose of study treatment.
Nervous system disorders
Dysgeusia
0.00%
0/59 • 36 Days
Treatment emergent adverse events (TEAE) were any adverse event that occurred or worsened after the first dose of study treatment.
1.7%
1/59 • 36 Days
Treatment emergent adverse events (TEAE) were any adverse event that occurred or worsened after the first dose of study treatment.
3.3%
2/61 • 36 Days
Treatment emergent adverse events (TEAE) were any adverse event that occurred or worsened after the first dose of study treatment.
5.1%
3/59 • 36 Days
Treatment emergent adverse events (TEAE) were any adverse event that occurred or worsened after the first dose of study treatment.

Additional Information

Director, Clinical Operations

Kowa Research Institute, Inc.

Phone: 919-433-1600

Results disclosure agreements

  • Principal investigator is a sponsor employee
  • Publication restrictions are in place