Trial Outcomes & Findings for A Clinical Study to Investigate the Effect of an Investigational Drug as an Added Medication to an Antipsychotic, in Adults With Schizophrenia, as Measured Positron Emission Tomography (PET) Imaging (NCT NCT04038957)

NCT ID: NCT04038957

Last Updated: 2024-12-27

Results Overview

Dopamine synthesis capacity was assessed using 18 F-DOPA PET(positron emission tomography) scans that were performed before (baseline) and after (Week 2 \[Day 14\]) administration of SEP-363856 adjunctive to an antipsychotic medication. A repeated measures ANOVA(analysis of variance) analysis was conducted. The dependent variable was Dopamine Synthesis Capacity (Ki Values). The independent variables were Time and Striatal Subregion. The covariance matrix was unstructured for each subject's Time and Striatal Subregion.

Recruitment status

COMPLETED

Study phase

PHASE1

Target enrollment

22 participants

Primary outcome timeframe

baseline and week 2

Results posted on

2024-12-27

Participant Flow

Participant milestones

Participant milestones
Measure
SEP-363856
SEP-363856 50mg, 75mg flexible dosing, dosed once daily
Overall Study
STARTED
22
Overall Study
COMPLETED
20
Overall Study
NOT COMPLETED
2

Reasons for withdrawal

Reasons for withdrawal
Measure
SEP-363856
SEP-363856 50mg, 75mg flexible dosing, dosed once daily
Overall Study
Withdrawal by Subject
1
Overall Study
SUBJECT WAS WITHDRAWN DUE TO SAFETY REASON
1

Baseline Characteristics

A Clinical Study to Investigate the Effect of an Investigational Drug as an Added Medication to an Antipsychotic, in Adults With Schizophrenia, as Measured Positron Emission Tomography (PET) Imaging

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
SEP-363856
n=22 Participants
SEP-363856 50mg, 75mg flexible dosing, dosed once daily
Age, Categorical
<=18 years
0 Participants
n=5 Participants
Age, Categorical
Between 18 and 65 years
22 Participants
n=5 Participants
Age, Categorical
>=65 years
0 Participants
n=5 Participants
Age, Continuous
32.5 Years
STANDARD_DEVIATION 6.68 • n=5 Participants
Sex: Female, Male
Female
6 Participants
n=5 Participants
Sex: Female, Male
Male
16 Participants
n=5 Participants
Ethnicity (NIH/OMB)
Hispanic or Latino
1 Participants
n=5 Participants
Ethnicity (NIH/OMB)
Not Hispanic or Latino
21 Participants
n=5 Participants
Ethnicity (NIH/OMB)
Unknown or Not Reported
0 Participants
n=5 Participants
Race (NIH/OMB)
American Indian or Alaska Native
0 Participants
n=5 Participants
Race (NIH/OMB)
Asian
2 Participants
n=5 Participants
Race (NIH/OMB)
Native Hawaiian or Other Pacific Islander
0 Participants
n=5 Participants
Race (NIH/OMB)
Black or African American
11 Participants
n=5 Participants
Race (NIH/OMB)
White
8 Participants
n=5 Participants
Race (NIH/OMB)
More than one race
0 Participants
n=5 Participants
Race (NIH/OMB)
Unknown or Not Reported
1 Participants
n=5 Participants

PRIMARY outcome

Timeframe: baseline and week 2

Dopamine synthesis capacity was assessed using 18 F-DOPA PET(positron emission tomography) scans that were performed before (baseline) and after (Week 2 \[Day 14\]) administration of SEP-363856 adjunctive to an antipsychotic medication. A repeated measures ANOVA(analysis of variance) analysis was conducted. The dependent variable was Dopamine Synthesis Capacity (Ki Values). The independent variables were Time and Striatal Subregion. The covariance matrix was unstructured for each subject's Time and Striatal Subregion.

Outcome measures

Outcome measures
Measure
SEP-363856
n=19 Participants
SEP-363856 50mg, 75mg flexible dosing, dosed once daily
Change From Baseline in Dopamine Synthesis Capacity at Week 2 Using 18F-DOPA.
Whole Striatal Dopamine Synthesis Capacity
-0.0007 Kicer
Standard Deviation 0.00157
Change From Baseline in Dopamine Synthesis Capacity at Week 2 Using 18F-DOPA.
Limbic Striatal Dopamine Synthesis Capacity
-0.0008 Kicer
Standard Deviation 0.00118
Change From Baseline in Dopamine Synthesis Capacity at Week 2 Using 18F-DOPA.
Associative Striatal Dopamine Synthesis Capacity
-0.0006 Kicer
Standard Deviation 0.00158
Change From Baseline in Dopamine Synthesis Capacity at Week 2 Using 18F-DOPA.
Sensorimotor Striatal Dopamine Synthesis Capacity
-0.0008 Kicer
Standard Deviation 0.00207

Adverse Events

SEP-363856

Serious events: 0 serious events
Other events: 19 other events
Deaths: 0 deaths

Serious adverse events

Adverse event data not reported

Other adverse events

Other adverse events
Measure
SEP-363856
n=22 participants at risk
SEP-363856 50mg, 75mg flexible dosing, dosed once daily
Eye disorders
Vision blurred
9.1%
2/22 • Number of events 2 • Up to 36 days
Gastrointestinal disorders
Dry mouth
18.2%
4/22 • Number of events 4 • Up to 36 days
Gastrointestinal disorders
Nausea
13.6%
3/22 • Number of events 3 • Up to 36 days
General disorders
Fatigue
9.1%
2/22 • Number of events 2 • Up to 36 days
Nervous system disorders
Dizziness
36.4%
8/22 • Number of events 8 • Up to 36 days
Nervous system disorders
Headache
18.2%
4/22 • Number of events 4 • Up to 36 days
Nervous system disorders
Presyncope
9.1%
2/22 • Number of events 2 • Up to 36 days
Nervous system disorders
Somnolence
63.6%
14/22 • Number of events 15 • Up to 36 days
Psychiatric disorders
Insomnia
9.1%
2/22 • Number of events 2 • Up to 36 days

Additional Information

CNS Medical Director

Sumitomo Pharma America Inc

Phone: 1-866-503-6351

Results disclosure agreements

  • Principal investigator is a sponsor employee In the event the Study is part of a multi-center study, the first publication of the results of the Study shall be made in conjunction with the results of other participating study sites as a multi-center publication; provided however, if a multi-center publication is not forthcoming within twenty-four (24) months following completion of the Study at all sites, Institution and Investigator shall be free to publish
  • Publication restrictions are in place

Restriction type: OTHER